Nucleosides, Nucleotides and Nucleic Acids (1982-2011)

Volume 30, Issue 1 (2011)

1-11	Oligonucleotide Labeling Using BODIPY Phosphoramidite	Kha Tram; Daniel Twohig; Hongbin Yan
12-19	Further Optimization of Detritylation in Solid-Phase Oligodeoxyribonucleotide Synthesis	Kha Tram; Yogesh S. Sanghvi; Hongbin Yan
20-30	An Extracellullar Nuclease from Bacillus Firmus VKPACU-1: Specificity and Mode of Action	Periasamy Ashok Kumar; Vijayaraghavan Kannan
31-48	Oligonucleotide Analogs with Peptide Internucleotide Linkages	Anna Varizhuk; Svetlana Kochetkova; Natalia Kolganova; Edward Timofeev; Vladimir Florentiev
49-62	Synthesis and DNA Binding Studies of Mg(II) Complex of Schiff Base Derived from Vanillin and L-Tryptophan	Yan Zhang; Xingming Wang; Lisheng Ding
63-81	Interrupted 2′-O,4′-C-Aminomethylene Bridged Nucleic Acid Modification Enhances Pyrimidine Motif Triplex-Forming Ability and Nuclease Resistance Under Physiological Condition	Hidetaka Torigoe; S. M. Abdur Rahman; Hiroko Takuma; Norihiro Sato; Takeshi Imanishi; Satoshi Obika; Kiyomi Sasaki
82	Call For Papers

Volume 29, Issue 11-12 (2010)

801-808	G-Octamer Formation from N⁹-Modified Guanine Derivatives	Jeremy McCallum; Solomon Amare; Rebecca Nolan
809-820	A Facile Synthesis and Anti-Avian Influenza Virus (H5N1) Screening of Some Novel Pyrazolopyrimidine Nucleoside Derivatives	Aymn E. Rashad; Ahmed H. Shamroukh; Randa E. Abdel-Megeid; Ahmed Mostafa; Mohamed A. Ali; Klaus Banert
821-830	Synthesis and Substrate Validation of Cap Analogs Containing 7-Deazaguanosine Moiety by RNA Polymerase	Anilkumar R. Kore; Muthian Shanmugasundaram; Timothy J. Barta
831-840	Semisynthesis of 6-Chloropurine-2′-deoxyriboside 5′-Dimethoxytrityl 3′-(2-Cyanoethyl-N,N-diisopropylamino)Phosphoramidite and its Use in the Synthesis of Fluorescently Labeled Oligonucleotides	Md. Jashim Uddin; Michael I. Schulte; Leena Maddukuri; Joel Harp; Lawrence J. Marnett
841-853	Quadruplex-Duplex Motifs as New Topoisomerase I Inhibitors	Li Shuai; Minggang Deng; Dan Zhang; Yangyang Zhou; Xiang Zhou
854-866	Study on the Interaction between the Inclusion Complex of Hematoxylin with β-Cyclodextrin and DNA	Dongling Xu; Xingming Wang; Dan Fei; Lisheng Ding
867-878	Gas-Phase Cleavage and Dephosphorylation of Universal Linker-Bound Oligodeoxynucleotides	Michael A. Jensen; Keith M. Anderson; Ronald W. Davis
879-895	Labeled Nucleoside Triphosphates with Reversibly Terminating Aminoalkoxyl Groups	Daniel Hutter; Myong-Jung Kim; Nilesh Karalkar; Nicole A. Leal; Fei Chen; Evan Guggenheim; Visa Visalakshi; Jerzy Olejnik; Steven Gordon; Steven A. Benner
896-904	Simple and Rapid Enzymatic Method for the Synthesis of Single-Strand Oligonucleotides Containing Trifluorothymidine	Norihiko Suzuki; Masakazu Fukushima
905-919	Synthesis of Novel 4′-Cyclopropyl-5′-norcarbocyclic Adenosine Phosphonic Acid Analogues	Guang Huan Shen; Joon Hee Hong
920	Call For Papers

Volume 29, Issue 10 (2010)

721-733	Design and Synthesis of Dually Branched 5′-Norcarbocyclic Adenosine Phosphonodiester Analogue as a New Anti-HIV Prodrug	Chang Hyun Oh; Lian Jin Liu; Joon Hee Hong
734-747	Hydroxyl-Functionalized DNAs with Different Linkers and Their Complmentary Duplex Stability	Di Zhang; Yamin Li; Liang Xu; Maosheng Cheng; Ying Zhou; Junlin He; Keliang Liu
748-759	DNA Staining in Agarose Gels with ZN²⁺-Cyclen-Pyrene	Florian Schmidt; Jennifer Schmidt; Alexander Riechers; Susann Haase; Anja-Katrin Bosserhoff; Jörg Heilmann; Burkhard König
760-767	Cinnamic Esters of Acyclovir-Synthesis and Biological Activity	Ivanka Stankova; Kiril Chuchkov; Peter Wutzler; Michaela Schmidtke
768-785	Studies on the Synthesis of N′-Acetyl AZA-Analogues of Ganciclovir—Unexpected Liability of N′-(2-Hydroxyethyl)-Azanucleosides Under Basic Conditions	Mariola Koszytkowska-Stawińska
786-799	Antioxidative and Radiation Modulating Properties of Guanosine-5′-Monophosphate	N. R. Asadullina; A. M. Usacheva; V. S. Smirnova; S. V. Gudkov

Volume 29, Issue 9 (2010)

647-657	Extracellular-Purine Metabolism in Blood Vessels (Part I). Extracellular-Purine Level in Blood of Patients with Abdominal Aortic Aneurysm	Joanna Lecka; Stanislaw Molski; Michal Komoszynski
658-675	Antimicrobial and DNA-Cleavage Studies of 22-Membered N₄ Tetraaza Macrocyclic Triazoles: Template Synthesis and Physicochemical Characterization	Sangamesh A. Patil; Udaykumar V. Kamble; Prema S. Badami
676-683	Design of fMet-tRNA and Calculation of its Bonding Properties by Quantum Mechanics	M. Monajjemi; M. Noei; F. Mollaamin
684-697	The Spontaneous Rearrangement of 2,4-Dinitrophenyl Substituent in Ribonucleosides Under Neutral Conditions	Anna Olejnik; Zofia Gdaniec; Elzbieta Kierzek; Ryszard Kierzek
698-706	Revisit to the Reaction of O-Phenylene Diamine with Thiosemicarbazide to Give Benzimidazole-2-Thione Rather than Benzotriazine-2-Thione and its Glycosylation	El Sayed H. El Ashry; Aly A. Aly; Mohamed R. Aouad; Mohammed R. Amer
707-720	Synthesis of Novel Acyclic Nucleoside Analogues with Anti-Retroviral Activity	A. Paju; M. Päri; A. Selyutina; E. Žusinaite; A. Merits; T. Pehk; K. Siirde; A. -M. Müürisepp; T. Kailas; M. Lopp

Volume 29, Issue 8 (2010)

581-590	Synthesis and Anti-HIV Evaluation of New Acyclic Phosphonate Nucleotide Analogues and Their Bis(SATE) Derivatives	Hua Li; Joon Hee Hong
591-605	Synthesis, Antitumor, and DNA Binding Behavior of Novel 4-(2-Hydroxyquinolin-3-yl)-6-Phenyl-5, 6 Dihydropyrimidin Derivatives in Aqueous Medium	Devappa S. Lamani; K. R. Venugopala Reddy; H. S. Bhojya Naik; K. S. R. Pai; Ravishankar Kumar; Fasiulla; H. R. Prakash Naik; L. R. Naik
606-615	Effects of Chloride, Bromide, and Iodide Upon Decomposition of Nucleosides Induced by Ultrasound in Neutral Solution	Toshinori Suzuki; Kenji Yamada; Michiyo Inukai
616-627	Solvent-Free Synthesis of Pyrimidine Nucleoside-Aminophosphonate Hybrids and Their Biological Activity Evaluation	Xinying Zhang; Yingying Qu; Xuesen Fan; C. Bores; Dong Feng; Graciela Andrei; Robert Snoeck; Erik De Clercq; Philippe M. Loiseau
628-645	Stereochemistry of Internucleotide Bond Formation by the H-Phosphonate Method. 5. The Role of Brønsted and H-Bonding Base Catalysis in Ribonucleoside H-Phosphonate Condensation—Chemical and Stereochemical Consequences	Michal Sobkowski; Jacek Stawinski; Adam Kraszewski

Volume 29, Issue 7 (2010)

523-534	Reinvestigation of the Synthesis of 1-Deazauridine	Cheng-Hung Jen; Tun-Cheng Chien
535-541	Synthesis of Novel 6-Azapyrimidine Acyclic Nucleoside Analogues and Antiviral Evaluation	Malina Jasamai; Claire Simons; Jan Balzarini
542-546	Highly Efficient and Facile Synthesis of 5-Azido-2′-Deoxyuridine	Stéphanie Gourdain; Christian Petermann; Dominique Harakat; Pascale Clivio
547-561	cDNA, Genomic Sequence Cloning, and Overexpression of EIF1 from the Giant Panda (Ailuropoda Melanoleuca) and the Black Bear (Ursus Thibetanus Mupinensis)	Wan-ru Hou; Yun Tang; Yi-ling Hou; Yan Song; Tian Zhang; Guang-fu Wu
562-573	Stereoselective Nucleoside Deuteration for NMR Studies of DNA	Mark Lukin; Carlos de los Santos
574-579	The Effect of Testosterone Upon the Urate Reabsorptive Transport System in Mouse Kidney	M. Hosoyamada; Y. Takiue; T. Shibasaki; H. Saito

Volume 29, Issue 4-6 (2010)

i-bl-iii-bl	Proceedings of the 13th International Symposium on Purine and Pyrimidine Metabolism in Man	S. Eriksson; G. J. Peters
i-xi	Purine and Pyrimidine Metabolism in the Fist Decade of the 21st Century—Highlights and Perspectives	Staffan Eriksson; Godefridus J. Peters
xii-xvii	In Memoriam: Dr. Hermione Anne Simmonds December 6, 1927 –April 2, 2010	David Perrett
267-277	Novel Strategies in the Thiopurine Treatment of Inflammatory Bowel Disease	S. Almer
278-283	How Should Thiopurine Treatment be Monitored?— Methodological Aspects	S. Vikingsson; B. Carlsson; S. Almer; C. Peterson
284-290	Limited Intra-Individual Variability in Hypoxanthine-Guanine Phosphoribosyl Transferase, Thiopurine S-Methyl Transferase, and Xanthine Oxidase Activity in Inflammatory Bowel Disease Patients During 6-Thioguanine Therapy	D. P. van Asseldonk; N. K. H. de Boer; K. Smid; C. J. Mulder; A. A. van Bodegraven; G. J. Peters
291-294	Molecular Analysis of Two Enzyme Genes, HPRT1 and PRPS1, Causing X-Linked Inborn Errors of Purine Metabolism	Y. Yamada; K. Yamada; N. Nomura; A. Yamano; R. Kimura; S. Tomida; M. Naiki; N. Wakamatsu
295-300	Partial HPRT Deficiency Phenotype and Incomplete Splicing Mutation	R. J. Torres; M. G. Garcia; J. G. Puig
301-305	Methylation Status of HPRT1 Promoter in HPRT Deficiency with Normal Coding Region	M. G. Garcia; R. J. Torres; J. G. Puig
306-313	Delayed Treatment Effects of Xanthine Oxidase Inhibition on Systolic Overload-Induced Left Ventricular Hypertrophy and Dysfunction	X. Xu; L. Zhao; X. Hu; P. Zhang; J. Wessale; R. Bache; Y. Chen
314-320	Establishment and Analysis of SLC22A12 (URAT1) Knockout Mouse	M. Hosoyamada; Y. Takiue; H. Morisaki; J. Cheng; M. Ikawa; M. Okabe; T. Morisaki; K. Ichida; T. Hosoya; T. Shibasaki
321-324	Effects of Three Strong Statins (Atorvastatin, Pitavastatin, and Rosuvastatin) on Serum Uric Acid Levels in Dyslipidemic Patients	N. Ogata; S. Fujimori; Y. Oka; K. Kaneko
325-329	Metabolic Syndrome Characteristics in Gout Patients	J. M. Fraile; R. J. Torres; Mendieta E. de Miguel; P. Martínez; K. J. Lundelin; J. J. Vázquez; J. G. Puig
330-334	Uric Acid Metabolism in Patients with Primary Gout and the Metabolic Syndrome	J. M. Fraile; J. G. Puig; Rosa J. Torres; Eugenio de Miguel; Pedro Martínez; J. J. Vázquez
335-346	Role of Nucleoside Transporters in Nucleoside-Derived Drug Sensitivity	M. Molina-Arcas; M. Pastor-Anglada
347-351	Thymidine Kinase 1 Deficient Cells Show Increased Survival Rate After UV-Induced DNA Damage	T. Skovgaard; L. J. Rasmussen; B. Munch-Petersen
352-358	Thymidine Kinase 1 is a Potential Marker for Prognosis and Monitoring the Response to Treatment of Patients with Breast, Lung, and Esophageal Cancer and Non-Hodgkin's Lymphoma	E. He; X. H. Xu; H. Guan; Y. Chen; Z. H. Chen; Z. L. Pan; L. L. Tang; G. Z. Hu; Y. Li; M. Zhang; J. Zhou; S. Eriksson; T. Fornander; S. Skog
359-362	Pasteurella Multocida Thymidine Kinase 1 Efficiently Activates Pyrimidine Nucleoside Analogs	A. R. Clausen; S.A. L. Al Meani; J. Piškur
363-369	Enzymatic Regulation of Cytosolic Thymidine Kinase 1 and Mitochondrial Thymidine Kinase 2: A Mini Review	B. Munch-Petersen
370-381	Deoxynucleoside Salvage Enzymes and Tissue Specific Mitochondrial DNA Depletion	L. Wang
382-385	Identification and Characterization of Mitochondrial Factors Modulating Thymidine Kinase 2 Activity	R. Sun; S. Eriksson; L. Wang
386-393	The Activity of the Lipophilic Nucleoside Derivatives Elacytarabine and CP-4126 in a Panel of Tumor Cell Lines Resistant to Nucleoside Analogues	Marit Liland Sandvold; Carlos Galmarini; Finn Myhren; Godefridus Peters
394-399	Induction of Resistance to the Lipophilic Cytarabine Prodrug Elacytarabine (CP-4055) in CEM Leukemic Cells	A. D. Adema; N. Losekoot; K. Smid; I. Kathmann; F. Myhren; M. L. Sandvold; G. J. Peters
400-403	Tissue Specific Distribution of Pyrimidine Deoxynucleoside Salvage Enzymes Shed Light on the Mechanism of Mitochondrial DNA Depletion	L. Wang; S. Eriksson

Volume 29, Issue 4-6 (2010)

404-407	Influence of Phosphorylation of THR-3, SER-11, and SER-15 on Deoxycytidine Kinase Activity and Stability	C. Smal; S. Ntamashimikiro; A. Arts; E. Van Den Neste; F. Bontemps
408-413	Methylation Specific PCR to Characterize Methylation of the Promoter of Deoxycytidine Kinase	G. J. Peters; J. Hodzic; B. Ortega; E. Giovannetti; A. D. Adema; R. Broekhuizen; G. J. Kaspers; I. Hubeek
414-418	Effect of Clofarabine on Apoptosis and DNA Synthesis in Human Epithelial Colon Cancer Cells	X. Wang; F. Albertioni
419-426	Study of Apoptosis Induction and Deoxycytidine Kinase/Cytidine Deaminase Modulation in the Synergistic Interaction of a Novel Ceramide Analog and Gemcitabine in Pancreatic Cancer Cells	E. Giovannetti; L. G. Leon; S. Bertini; M. Macchia; F. Minutolo; N. Funel; C. Alecci; F. Giancola; R. Danesi; G. J. Peters
427-432	How to Use the Computing Environment R to Analyze ATP-Induced Ribonucleotide Reductase R1 Hexamerization Data	T. Radivoyevitch
433-437	Ribosylurea Accumulates in Yeast urc4 Mutants	O. Björnberg; M. Vodnala; V. Domkin; A. Hofer; A. Rasmussen; G. Andersen; J. Piškur
438-444	Synthesis, Biological Properties and Anti-HIV-1 Activity of New Pyrimidine P₁,P₂-Dinucleotides	A. Miazga; P. Ziemkowski; M. A. Siwecka; A. Lipniacki; A. Piasek; T. Kulikowski
445-448	Nucleoside Phosphorylases from Clostridium Perfringens in the Synthesis of 2′,3′-Dideoxyinosine	S. Christoffersen; I. Serra; M. Terreni; J. Piškur
449-452	Protection of Mouse Heart Against Hypoxic Damage by AMP Deaminase Inhibition	T. Borkowski; E. M. Slominska; C. Orlewska; S. Chlopicki; P. Siondalski; M. H. Yacoub; R. T. Smolenski
453-456	Cardiac Muscle AMP-Deaminase from a 10-Year-Old Male Heterozygous for the AMPD1 C34T Mutation	I. Rybakowska; S. Bakuła; J. Klimek; R. Milczarek; R. T. Smolenski; K. Kaletha
457-460	Biological Efficiency of AMP Deaminase Inhibitor: 3-[2-(3-CARBOXY-4-BROMO-5,6,7,8-Tetrahydronaphthyl)Ethyl]-3,6,7,8-Tetrahydroimidazo[4,5]-[1,3]Diazepin-8-OL	T. Borkowski; E. M. Slominska; C. Orlewska; A. H. Y. Yuen; S. Al-Ayoubi; P. Siondalski; M. H. Yacoub; R. T. Smolenski
461-465	Determination of Adenosine Deaminase Activity in Dried Blood Spots by a Nonradiochemical Assay Using Reversed-Phase High-Performance Liquid Chromatography	A. B. P. van Kuilenburg; L. Zoetekouw; J. Meijer; T. W. Kuijpers
466-470	Identification of Purine Nucleoside Phosphorylase Deficiency in Dried Blood Spots by a Non-Radiochemical Assay Using Reversed-Phase High-Performance Liquid Chromatography	A. B. P. van Kuilenburg; L. Zoetekouw; J. Meijer; T. W. Kuijpers
471-475	PARP Activity and NAD Concentration in PMC from Patients Affected by Systemic Sclerosis and Lupus Erythematosus	B. Cerboni; A. Di Stefano; V. Micheli; G. Morozzi; G. Pompucci; S. Sestini
476-481	Region-Specific Distribution of Dihydroorotate Dehydrogenase in the Rat Central Nervous System Points to Pyrimidine De Novo Synthesis in Neurons	Ch. M. Schaefer; M. K. -H. Schäfer; M. Löffler
482-487	Increased Migration by Stimulation of Thymidine Phosphorylase in Endothelial Cells of Different Origin	I. V. Bijnsdorp; K. Vrijland; L. Vroling; M. Fukushima; G. J. Peters
488-503	Activation of Stat1, IRF-1, and NF-κB is Required for the Induction of Uridine Phosphorylase by Tumor Necrosis Factor-α and Interferon-γ	Laxiang Wan; Deliang Cao; Jianmin Zeng; Amy Ziemba; Giuseppe Pizzorno
504-508	Relationship Between Plasma Uridine and Insulin Resistance in Patients with Non-Insulin-Dependent Diabetes Mellitus	Tetsuya Yamamoto; Taku Inokuchi; Tuneyoshi Ka; Asako Yamamoto; Sumio Takahashi; Zenta Tsutsumi; Daisuke Tamada; Chiharu Okuda; Yuji Moriwaki
509-514	Dihydropyrimidine Dehydrogenase Deficiency Caused by a Novel Genomic Deletion c.505_513del of DPYD	A. B. P. van Kuilenburg; J. Meijer; G. Gökcay; T. Baykal; M. E. Rubio-Gozalbo; A. N. P. M. Mul; C. E. M. de Die-Smulders; P. Weber; A. Capone Mori; J. Bierau; B. Fowler; K. Macke; J. O. Sass; R. Meinsma; J. B. Hennermann; P. Miny; L. Zoetekouw; J. Roelofsen; R. Vijzelaar; J. Nicolai; R. C. M. Hennekam
515-517	Development of LC-MS Method for Detection of Mutant Uromodulin Protein	M. Yasuda; K. Kaneko; H. Hachisu; M. Ochiai; T. Yamanobe; K. Mawatari; K. Nakagomi; N. Minoura; M. Hosoyamada
518-521	Analysis of Purine in Purine-Rich Cauliflower	N. Yamaoka; K. Kaneko; Y. Kudo; M. Aoki; M. Yasuda; K. Mawatari; K. Nakagomi; Y. Yamada; T. Yamamoto

Volume 29, Issue 3 (2010)

155-167	Synthesis of a Fluorescent Cationic Phosphorus Dendrimer and Preliminary Biological Studies of Its Interaction with DNA	Julia Kazmierczak-Baranska; Aleksandra Pietkiewicz; Magdalena Janicka; Yiqian Wei; Cédric-Olivier Turrin; Jean-Pierre Majoral; Barbara Nawrot; Anne-Marie Caminade
168-177	Pyrimidine-Purine and Pyrimidine Heterodinucleosides Synthesis Containing a Triazole Linkage	R. Lucas; P. H. Elchinger; P. A. Faugeras; R. Zerrouki
178-189	Synthesis, Spectral Characterization, and Biological Activity of Some New Substituted 10H-Phenothiazines, Its Ribofuranosides, and Sulfones	Naveen Gautam; Neha Ajmera; Shikha Gupta; D. C. Gautam
190-199	Inducement of G-Quadruplex DNA Forming and Down-Regulation of Oncogene C-MYC by Bile Acid-Amino Acid Conjugate—BAA	Mingyue Tian; Xiufeng Zhang; Yan Li; Yong Ju; Junfeng Xiang; Changqi Zhao; Yalin Tang
200-215	Dna Interactions and Promotion in Antibacterial Activities of Ciprofloxacin Drug Due to Formation of Mixed-Ligand Complexes of Oxovanadium(IV)	M. N. Patel; S. H. Patel; M. R. Chhasatia; C. R. Desai
216-227	Synthesis of 2′-Fluoro and 2′,4′-Dimethyl Pyrimidine C-Nucleoside Analogues as Potential Anti-HCV Agents	Lian Jin Liu; Joon Hee Hong
228-236	Assessment of Cell-Free DNA with Microvascular Complication of Type II Diabetes Mellitus, Using PCR and Elisa	Shereen A. El Tarhouny; Khaled M. Hadhoud; Magdy M. Ebrahem; Nashwa M. Al Azizi
237-244	Frequency of Thiopurine S-Methyltransferase (TPMT) Alleles in Southeast Iranian Population	Ali Bahari; Mohammad Hashemi; Zohreh Bari; Abdolkarim Moazeni-Roodi; Mahmoud-Ali Kaykhaei; Behzad Narouie
245-256	An Improved One-Pot Synthesis of Nucleoside 5′-Triphosphate Analogues	Irina Gillerman; Bilha Fischer
257-266	Design and Synthesis of Novel Sate Derivatives of Acyclic Isocytosine and 9-Deazaadenine C-Nucleosides	Lian Jin Liu; Joon Hee Hong

Volume 29, Issue 2 (2010)

81-90	Characterization of Insulin Ilpr Sequences for Their Ability to Adopt a G-Quadruplex Structure	Hanumantharao Paritala; Steven M. Firestine
91-96	Synthesis of β-Hydroxyphosphonate and 1,2-Dihydroxy Acyclic Nucleoside Analogs via 1,3-Dipolar Cycloaddition Strategy	M. Ganesan; K. M. Muraleedharan
97-112	Down-Modulation of Survivin Expression and Inhibition of Tumor Growth In Vivo by EZN-3042, A Locked Nucleic Acid Antisense Oligonucleotide	Puja Sapra; Maoliang Wang; Raj Bandaru; Hong Zhao; Lee M. Greenberger; Ivan D. Horak
113-122	Efficient Syntheses of Clofarabine and Gemcitabine From 2-Deoxyribonolactone	Yana Cen; Anthony A. Sauve
123-131	Analysis of Similarity/Dissimilarity of DNA Sequences Based on Convolutional Code Model	Xiao Liu; Feng Chun Tian; Shi Yuan Wang
132-143	An Efficient Deprotection of N-Trimethylsilylethoxymethyl (SEM) Groups From Dinucleosides and Dinucleotides	Tilak Chandra; William E. Broderick; Joan B. Broderick
144-154	Solid-Phase Synthesis of Oligodeoxyribonucleotides without Base Protection Utilizing O-Selective Reaction of Oxazaphospholidine Derivatives	Natsuhisa Oka; Yukihiro Maizuru; Mamoru Shimizu; Takeshi Wada

Volume 29, Issue 1 (2010)

1-13	Retained Sensitivity to Cytotoxic Pyrimidine Nucleoside Analogs in Thymidine Kinase 2 Deficient Human Fibroblasts	Mia Bjerke; Nicola Solaroli; Nicole Lesko; Jan Balzarini; Magnus Johansson; Anna Karlsson
14-26	Facile Small Scale Synthesis of Nucleoside 5′-Phosphate Mixtures	Robert S. Jansen; Hilde Rosing; Jan HM Schellens; Jos H. Beijnen
27-38	Silver(I)-Mediated Cytosine Self-Pairing is Preferred Over Hoogsteen-Type Base Pairs with the Artificial Nucleobase 1,3-Dideaza-6-Nitropurine	Dominik A. Megger; Jens Müller
39-48	Synthesis, Characterization, and Photoactivated DNA Cleavage by Copper (II)/Cobalt (II) Mediated Macrocyclic Complexes	H. R. Prakash Naik; H. S. Bhojya Naik; T. Aravinda; D. S. Lamani
49-54	Synthesis and in Vitro Evaluation of 5-Fluoro-6-[(2-Iminopyrrolidin-1-YL)Methyl]Uracil, TPI(F): An Inhibitor of Human Thymidine Phosphorylase (TP)	John R. Grierson; J. Scott Brockenbrough; Janet S. Rasey; Linda Wiens; Hubert Vesselle
55-71	Glycosylation, Sugar Hydrazones, and Antimicrobial Evaluation of Some 6-Substituted-1,2,4-Triazines	A. A. El-Barbary; Y. A. Hafiz; M. S. Abdel-Wahed
72-80	Synthesis of 1H-Indole-2,3-Dione-3-Thiosemicarbazone Ribonucleosides as Antibacterial Agents	Shaymaa E. Kassab; Gehan H. Hegazy; Nahed M. Eid; Kamelia M. Amin; Adel A. El-Gendy

Volume 28, Issue 11-12 (2009)

989-997	Study on the Interaction Between Nucleic Acids and Imidacloprid and Its Application	Shicong Hou; Xiaofeng Jiang; Fengpei Du; Huifang Cong; Ying Li; Nianqin Jie
998-1006	Synthesis and Antimicrobial Activities of Novel Biologically Active Heterocycles: 10H-Phenothiazines, Their Ribofuranosides, and Sulfone Derivatives	Yogesh Dixit; Rahul Dixit; Naveen Gautam; D. C. Gautam
1007-1015	Synthesis and Anti-Hepatitis C Virus Activity of 2′(β)-Hydroxyethyl and 4′(α)-Hydroxymethyl Carbodine Analogues	Lian Jin Liu; Joon Hee Hong
1016-1029	Chemoselective Deprotection of Triethylsilyl Ethers	Tilak Chandra; William E. Broderick; Joan B. Broderick
1030-1041	Cyclic Enzymatic Solid Phase Synthesis of Isotopically Labeled DNA Oligonucleotides	Ahmed M. Khan; Subrata H. Mishra; Markus W. Germann
1042-1050	Synthesis of 2′-N-Formamido Nucleosides and Biological Evaluation	Mikhail Abramov; Marleen Renders; Piet Herdewijn
1051-1067	An Electrochemical Assay of β-1,3-Glucanase Gene from Transgenic Capsicum Using Asymmetric PCR	Guofan Wu; Zhihua Wang; Huini Zhang; Ning Yang; Jie Du; Xiaoquan Lu; Jingwan Kang
1068-1075	Bacterial Deoxyribonucleoside Kinases are Poor Suicide Genes in Mammalian Cells	Claire Hébrard; Emeline Cros-Perrial; Anders Ranegaard Clausen; Charles Dumontet; Jure Piškur; Lars Petter Jordheim
1076-1094	Synthesis of Guanosine and Deoxyguanosine Phosphoramidites with Cross-Linkable Thioalkyl Tethers for Direct Incorporation into RNA and DNA	Xiaorong Hou; Gang Wang; Barbara L. Gaffney; Roger A. Jones
1095-1103	Nucleosides 5¹⁵: Synthesis of Novel 1,2,4-Triazolo[3,4-c]-1,2,4-Triazole Nucleosides	M. A. N. Mosselhi; R. Neidlein
1104-1116	Synthesis and In Vitro Activity of 4′ and 5′-Modified Analogues of Apiosyl Nucleosides as Potent Anti-HCV Agents	Hua Li; Wonjae Lee; Joon Hee Hong
1117-1130	Stereoselective Synthesis of 2-Deoxy-2-Fluoroarabinofuranosyl-α-1-Phosphate and Its Application to the Synthesis of 2′-Deoxy-2′-Fluoroarabinofuranosyl Purine Nucleosides by a Chemo-Enzymatic Method	Kohei Yamada; Noritake Matsumoto; Hiroyuki Hayakawa
1131-1143	Labeling of an Antisense Oligonucleotide with [¹⁸F]FPy5yne	James A. H. Inkster; Michael J. Adam; Tim Storr; Thomas J. Ruth

Volume 28, Issue 10 (2009)

875-901	D-Arbinose-Based Synthesis of homo-C-d4T and homo-C-thymidine	Bogdan Doboszewski
902-910	Activity of siRNAs with 2-Thio-2′-O-Methyluridine Modification in Mammalian Cells	Thazha P. Prakash; Nishant Naik; Namir Sioufi; Balkrishen Bhat; Eric E. Swayze
911-923	Synthesis of Novel 5′-Uridine-Head Amphiphiles as Model for DNA Molecular Recognition	Matteo Tiecco; Pietro Di Profio; Raimondo Germani; Gianfranco Savelli
924-942	Hydroxyl-Functionalized DNA: An Efficient Orthogonal Protecting Strategy and Duplex Stability	Di Zhang; Liang Xu; Xia Wei; Yaming Li; Junlin He; Keliang Liu
943-952	Synthesis and Properties of Oligodeoxyribonucleotides Bearing a Polyamino Group at the 2′ Position via 2′-O-Carbamoylmethyl and 2′-S-Carbamoylmethyl groups	Hiroaki Ozaki; Shingo Nomura; Shingo Momiyama; Kazuyuki Yokotsuka; Masayasu Kuwahara; Hiroaki Sawai
953-968	DNA-Binding and Photocleavage Properties of Ru(II) Polypyridyl Complexes with DNA and Their Toxicity Studies on Eukaryotic Microorganisms	Kotha Laxma Reddy; Y. Harish Kumar Reddy; S. Satyanarayana
969-986	Synthesis of 3′-Amino-3′-Deoxyguanosine and 3′-Amino-3′-Deoxyxyloguanosine Monophosphate Hepdirect Prodrugs from Guanosine	Brett C. Bookser; Nicholas B. Raffaele; K. Raja Reddy; Kevin Fan; Wenjian Huang; Mark D. Erion
987	Erratum

Volume 28, Issue 9 (2009)

795-808	Synthesis and Enantioselectivity of Cyclopropavir Phosphates for Cellular GMP Kinase	Chengwei Li; Brian G. Gentry; John C. Drach; Jiri Zemlicka
809-820	Synthesis and anti-HCV Evaluation of 4′(α)-ethyl and 2′(β)-methyl-carbodine Analogues	Hua Li; Jin Cheol Yoo; Joon Hee Hong
821-834	Ionic Liquid Mediated Synthesis of 5-Halouracil Nucleosides: Key Precursors for Potential Antiviral Drugs	Vineet Kumar; Sanjay V. Malhotra
835-845	Synthesis and Antimicrobial Activity of Some S-β-D-Glucosides of 4-Mercaptopyrimidine	A. H. Moustafa; H. A. Morsy; M. G. Assy; A. Z. Haikal
846-865	Synthesis Of RNA by the Rapid Phosphotriester Method Using Azido-Based 2′-O-Protecting Groups	V. A. Efimov; A. V. Aralov; V. N. Klykov; O. G. Chakhmakhcheva
866-873	3-Substituted Pyrazinone Nucleosides—A New Family of D4T Analogues	Nathalie Batoux; Robert Granet; Rachida Zerrouki; Pierre Krausz

Volume 28, Issue 8 (2009)

725-735	Method to Improve DNA Condensation Efficiency by Alkali Treatment	Sen Hou; Xinxin Li; Xi-Zeng Feng
736-751	Novel Isopentenyladenosine Analogues: Synthesis, Characterization, and Evaluation of Antiproliferative Activity on Bladder Carcinoma Cells	Roberta Ottria; Silvana Casati; Jeanette A. M. Maier; Massimo Mariotti; Pierangela Ciuffreda
752-760	A New Odorless Procedure for the Synthesis of 2′-Deoxy-6-Thioguanosine and Its Incorporation into Oligodeoxynucleotides	Kazumitsu Onizuka; Yosuke Taniguchi; Shigeki Sasaki
761-771	Synthesis and In Vitro Activity Evaluation of 2′,3′-C-Dimethyl Carbocyclic Nucleoside Analogues as Potential Anti-HCV Agents	Ok Hyun Ko; Joon Hee Hong
772-775	A Proposed Structure of Modified Nucleosides Expected to Have High Antiviral Activity and Low Toxicity	Hiroshi Ohrui
776-792	Nucleoside Diphosphate Kinase and the Activation of Antiviral Phosphonate Analogs of Nucleotides: Binding Mode and Phosphorylation of Tenofovir Derivatives	Kerstin Koch; Yuxing Chen; Joy Y. Feng; Katyna Borroto-Esoda; Dominique Deville-Bonne; Joël Janin; Solange Moréra
793	Editorial Retraction

Volume 28, Issue 5-7 (2009)

Commemorating the 70th Birthday of Morris J. Robins

333-336	Foreword: Morris J. Robins—Teacher, Mentor, Scientist, Colleague, and Friend	Stanislaw F. Wnuk
337-351	Synthesis of 3′-O-Phosphonoethyl Nucleosides with an Adenine and a Thymine Base Moiety	Qiuya Huang; Piet Herdewijn
352-378	Thiophosphate Analogs of c-di-GMP: Impact on Polymorphism	Jianwei Zhao; Elizabeth Veliath; Seho Kim; Barbara L. Gaffney; Roger A. Jones
379-393	Biodistribution and Imaging of 1-(2-Deoxy-β-D-Ribofuranosyl)-2,4-Difluoro-5-[^123/125I]Iodobenzene (dRF[^123/125I]IB), A Nonpolar Thymidine-Mimetic Nucleoside, in Rats and Tumor-Bearing Mice	Anke Stahlschmidt; Panteha Khalili; William Sun; Hans-Jürgen Machulla; Edward E. Knaus; Leonard I. Wiebe
394-407	Antiproliferative and Protein Kinase Binding Activities of Some N⁶, 5′-bis-ureido 5′-Amino-5′-Deoxyadenosine Derivatives	Matt A. Peterson; Marcelio Oliveira; Michael A. Christiansen
408-423	Base-Functionalized Carbocyclic Nucleosides: Design, Synthesis, and Mechanism of Antiviral Activity	Vasu Nair; Fan Zhang; Xiaohui Ma; Eric Bonsu
424-434	Modulation of RNA Metal Binding by Flanking Bases: ¹⁵N NMR Evaluation of GC, Tandem GU, and Tandem GA Sites	Weimin Wang; Jianwei Zhao; Qianwei Han; Gang Wang; Gengcheng Yang; Anthony J. Shallop; Jane Liu; Barbara L. Gaffney; Roger A. Jones
435-449	Synthesis and Antiviral Evaluation of 4′-C-Azidomethyl-β-D-Ribofuranosyl Purine and Pyrimidine Nucleosides	Jean-François Griffon; Audrey Dumas; Richard Storer; Jean-Pierre Sommadossi; Gilles Gosselin
450-463	Human Nucleoside Transporters: Biomarkers for Response to Nucleoside Drugs	Vijaya L. Damaraju; Michael B. Sawyer; John R. Mackey; James D. Young; Carol E. Cass
464-472	The “Corey's Reagent,” 3,5-di-tert-butyl-1,2-Benzoquinone, as a Modifying Agent in the Synthesis of Fluorescent and Double-Headed Nucleosides	Victor A. Timoshchuk; Richard I. Hogrefe
473-484	Evaluation of NAD(H) Analogues as Selective Inhibitors for Trypanosoma Cruzi S-Adenosylhomocysteine Hydrolase	Qing-Shan Li; Sumin Cai; Jianwen Fang; Ronald T. Borchardt; Krzysztof Kuczera; C. Russell Middaugh; Richard L. Schowen
485-503	The Rationale for Targeting the NAD/NADH Cofactor Binding Site of Parasitic S-Adenosyl-L-Homocysteine Hydrolase for the Design of Anti-Parasitic Drugs	Sumin Cai; Qing-Shan Li; Jianwen Fang; Ronald T. Borchardt; Krzysztof Kuczera; C. Russell Middaugh; Richard L. Schowen
504-518	A Convergent Approach for the Synthesis of Ara-Neplanocin a Analogues Under Subzero Microwave Assisted Conditions	Marco Radi; Jagadeeshwar R. Rao; Ashok K. Jha; Chung K. Chu
519-536	Synthesis and Antiviral Activity of Purine 2′,3′-Dideoxy-2′,3′-Difluoro-D-Arabinofuranosyl Nucleosides	Grigorii G. Sivets; Elena N. Kalinichenko; Igor A. Mikhailopulo; Mervi A. Detorio; Tami R. McBrayer; Tony Whitaker; Raymond F. Schinazi
537-549	Application of Germyldesulfonylation Reactions to the Synthesis of Germanium-Containing Nucleoside Analogues	Stanislaw F. Wnuk; Pablo R. Sacasa; Jorge Restrepo
550-585	Nucleosides Part LXVI I^[¹^]: Synthesis of 4-Amino-7(8H)Pteridinone-N₈-Nucleosides—Structural Analogs of Adenosine	Oliver Jungmann; Wolfgang Pfleiderer
586-600	The Unabated Synthesis of New Nucleoside Analogues with Antiviral Potential: A Tribute to Morris J. Robins	Erik De Clercq
601-613	Truncated Fluorocyclopentenyl Pyrimidines as S-Adenosylhomocysteine Hydrolase Inhibitors	Yeon Hee Park; Won Jun Choi; Amol S. Tipnis; Kang Man Lee; Lak Shin Jeong
614-632	Contrasting Behavior of Conformationally Locked Carbocyclic Nucleosides of Adenosine and Cytidine as Substrates for Deaminases	Victor E. Marquez; Gottfried K. Schroeder; Olaf R. Ludek; Maqbool A. Siddiqui; Abdallah Ezzitouni; Richard Wolfenden

Volume 28, Issue 5-7 (2009)

Commemorating the 70th Birthday of Morris J. Robins

633-641	Carbocyclic Thymidine Analogues for Use as Potential Therapeutic Agents	Katherine L. Seley-Radtke; Naresh K. Sunkara
642-656	Regioselective Metalation of 6-Methylpurines: Synthesis of Fluoromethyl Purines and Related Nucleosides for Suicide Gene Therapy of Cancer	Abdalla E. A. Hassan; William B. Parker; Paula W. Allan; John A. Secrist III
657-677	Synthesis and Anticancer Evaluation of 4′-C-Methyl-2′-Fluoro Arabino Nucleosides	Kamal N. Tiwari; Anita T. Shortnacy-Fowler; William B. Parker; William R. Waud; John A. Secrist III
678-694	Studies on the Glycosylation of Pyrrolo[2,3-d] Pyrimidines with 1-O-Acetyl-2,3,5-Tri-O-Benzoyl-β-D-Ribofuranose: The Formation of Regioisomers During Toyocamycin and 7-Deazainosine Syntheses	Peter Leonard; Sachin A. Ingale; Ping Ding; Xin Ming; Frank Seela
695-712	Synthesis of Ansa¹-Cytidines	Konrad Krolikiewicz; Martina Schäfer; Helmut Vorbrüggen
713-723	Synthesis and Antiviral Evaluation of 2′-C-Methyl Analogues of 5-Alkynyl- and 6-Alkylfurano- and Pyrrolo[2,3-d]Pyrimidine Ribonucleosides	Piotr Januszczyk; Joanna Fogt; Jerzy Boryski; Kunisuke Izawa; Tomoyuki Onishi; Johan Neyts; Erik De Clercq

Volume 28, Issue 4 (2009)

261-274	Synthesis and In Vitro Antitumor Activity of New Substituted Thiopyrimidine Acyclic Nucleosides and Their Thioglycoside Analogs	Wael A. El-Sayed; Aymn E. Rashad; Samir M. Awad; Mamdouh M. Ali
275-291	A Convenient Synthesis of N,N′-dibenzyl-2,4-diaminopyrimidine-2′-deoxyribonucleoside and 1-Methyl-2′-Deoxypseudoisocytidine	Kevin W. Wellington; Hua Chee Ooi; Steven A. Benner
292-302	Synthesis and Activity of Modified Cytidine 5′-Monophosphate Probes for T4 RNA Ligase 1	Anilkumar R. Kore; Irudaya Charles; Litao Yang; Scott Kuersten
303-314	Synthesis and Anti-Hiv Activity of 4′-Modified Cyclopentenyl Pyrimidine C-Nucleosides	Lian Jin Liu; Joon Hee Hong
315-323	Very Stable End-Sealed Double Stranded DNA by Click Chemistry	Afaf H. El-Sagheer
324-330	High GC Contents of Primer 5′-End Increases Reaction Efficiency in Polymerase Chain Reaction	Naoki Shinoda; Tomotaro Yoshida; Toyoko Kusama; Masami Takagi; Toshiaki Hayakawa; Takashi Onodera; Katsuaki Sugiura
331	Erratum

Volume 28, Issue 3 (2009)

165-174	Stereoselective Approach to the Z-Isomers of Methylenecyclopropane Analogues of Nucleosides: A New Synthesis of Antiviral Synguanol	Zhimeng Wu; Shaoman Zhou; Jiri Zemlicka
175-183	Microwave-Assisted Synthesis of Acyclic C-Nucleosides from 1,2- and 1,3-Diketones	Najim A. Al-Masoudi; Bahjat. A. Saeed; Ali H. Essa; Yaseen A. Al-Soud
184-192	Synthesis and Antibacterial Activity of Some Glucosyl- and Ribosyl-Pyridazin-3-ones	H. A. El-Sayed; A. H. Moustafa; A. Z. Haikal; E. S. H. El-Ashry
193-203	Purine Nucleotide Catabolism in Rat Liver. Certain Preliminary Aspects of Uricase Reaction	Lucia Terzuoli; Brunetta Porcelli; Fabio Ponticelli; Enrico Marinello
204-219	Synthesis, Characterization, DNA-Binding, and DNA-Photocleavage Properties of [Co(bpy)₂(7-NO₂-dppz)]³⁺, [Co(dmb)₂(7-NO₂-dppz)]³⁺, and [Co(phen)₂(7-NO₂-dppz)]³⁺ Complexes: (7-Nitro-dppz = 7-Nitro dipyrido[3,2-a:2′-3′-c]phenazine; bpy = 2,2′-bipyridine; dmb = 4,4′-dimethyl-2,2′-bipyridine; phen = 1,10-phenanthroline) and their Toxicity on Different Microorganisms	Kotha Laxma Reddy; Y.Harish Kumar Reddy; K. Ashwini Kumar; S. Vidhisha; S. Satyanarayana
220-237	Synthesis of a Novel, Optically Active Uridine Analog Containing a 1,4-Dioxane Sugar Moiety. Synthesis of the Corresponding Dinucleotide	Qiang Yu; Per Carlsen
238-259	β-1,2,3-Triazolyl-Nucleosides as Nicotinamide Riboside Mimics	E. J. Amigues; E. Armstrong; M. Dvorakova; M. E. Migaud; M. Huang

Volume 28, Issue 2 (2009)

67-77	Synthesis of Oligonucleotides Containing 2′-Deoxyguanosine Adducts of Nitropyrenes	Laureen C. Colis; Debasis Chakraborti; Pablo Hilario; Christopher McCarty; Ashis K. Basu
78-88	Synthesis and Evaluation of an RNA Editing Substrate Bearing 2′-Deoxy-2′-Mercaptoadenosine	Prasanna Jayalath; Subhash Pokharel; Eduardo Véliz; Peter A. Beal
89-102	Synthesis of Zidovudine Derivatives with Anti-HIV-1 and Antibacterial Activities	Palaniappan Senthilkumar; Jing Long; Raparla Swetha; Vaidyanathan Shruthi; Rui-Rui Wang; Srinivasan Preethi; Perumal Yogeeswari; Yong-Tang Zheng; Dharmarajan Sriram
103-117	Novel Acyclic Amide-Conjugated Nucleosides and Their Analogues	Slawomir Boncel; Krzysztof Walczak
118-149	Reactions of Peroxynitrite with Uric Acid: Formation of Reactive Intermediates, Alkylated Products and Triuret, and In Vivo Production of Triuret Under Conditions of Oxidative Stress	Christine Gersch; Sergiu P. Palii; Witcha Imaram; Kyung Mee Kim; S. Ananth Karumanchi; Alexander Angerhofer; Richard J. Johnson; George N. Henderson
150-164	Short Synthesis and Antiviral Activity of Acyclic Phosphonic Acid Nucleoside Analogues	Lian Jin Liu; Jin Cheol Yoo; Joon Hee Hong

Volume 28, Issue 1 (2009)

1-11	Downregulation of Human Telomerase Reverse Transcriptase Through Anti-C-Myc Sirna in Human Colon Cancer Colo 320 Cells	Xiaoyun Hu; Nancai Yu; Lei Fu; Wen Su; Guofu Huang; Yanxia Wu; Hanju Huang; Hao Huang
12-28	Visible-Light Photocontrol of (E)/(Z) Isomerization of the 4-(Dimethylamino)azobenzene Pseudo-Nucleotide Unit Incorporated into an Oligonucleotide and DNA Hybridization in Aqueous Media	Takashi Kamei; Haruhisa Akiyama; Hisayuki Morii; Nobuyuki Tamaoki; Taro Q. P. Uyeda
29-42	A Proposal for a Convenient Notation for P-Chiral Nucleotide Analogues. Part 4. A Relationship Between the D_P/L_P Notation and Stereochemistry of Reactions	Michal Sobkowski; Jacek Stawinski; Adam Kraszewski
43-55	5′-O-D-Valyl ara A, A Potential Prodrug for Improving Oral Bioavailability of the Antiviral Agent Vidarabine	Wei Shen; Jae-Seung Kim; Stefanie Mitchell; Phil Kish; Paul Kijek; John Hilfinger
56-66	Facile Synthesis and Anti-Tumor Cell Activity of Se-Containing Nucleosides	Lina Lin; Jia Sheng; Razin K. Momin; Quan Du; Zhen Huang

Volume 27, Issue 12 (2008)

1211-1214	Substrate Specificity of Thymidine Phosphorylase of E. Coli: Role of Hydroxyl Groups	Natalya G. Panova; Cyril S. Alexeev; Konstantin M. Polyakov; Sergei A. Gavryushov; Anatoliy M. Kritzyn; Sergey N. Mikhailov
1215-1226	Ring-Opening of 3-β-D-Ribofuranosyl-3,7,8,9-Tetrahydropyrimido [1,2-i]Purin-8-ol and Preparation of 2-Thio- and 2-aza-Adenosine Derivatives	Pernilla Sund; Leif Kronberg
1227-1237	An Expeditious Synthesis of Benzoxazine-2-Thione c-Nucleosides Via Cu(OTf)₂-Mediated Dehydrazinative β-Glycosylation	Lal Dhar S. Yadav; Vijai K. Rai
1238-1249	Novel Synthesis and Anti-HIV Activity of 4′-Branched Exomethylene Carbocyclic Nucleosides Using a Ring-Closing Metathesis of Triene	Hua Li; Jin Cheol Yoo; Joon Hee Hong
1250-1256	Simultaneous Removal of Benzyl and Benzyloxycarbonyl Protective Groups in 5′-O-(2-Deoxy-α-D-Glucopyranosyl)Uridine by Catalytic Transfer Hydrogenolysis	Ilona Wandzik; Tadeusz Bieg; Monika Kadela
1257-1271	Synthesis and Antiviral Evaluation of Novel 2,3-Dihydroxypropyl Nucleosides from 2- and 4-Thiouracils	Adel A. -H. Abdel-Rahman; Abd-Allah SH. El-Etrawy; Ahmed E. -S. Abdel-Megied; Ibrahim F. Zeid; El Sayed H. El Ashry
1272-1281	Study on Disulfur-Backboned Nucleic Acids: Part 3. Efficient Synthesis of 3′,5′-Dithio-2′-Deoxyuridine and Deoxycytidine	Peihua Shang; Hua Wang; Changmei Cheng; Hongchao Zheng; Yufen Zhao
1282-1300	Design and Synthesis of bis-carbamate Analogs of Cyclic bis-(3′-5′)-Diguanylic Acid (c-di-GMP) and the Acyclic Dimer PGPG	Toni Kline; Stona R. Jackson; Wei Deng; Christophe L. M. J. Verlinde; Samuel I. Miller

Volume 27, Issue 10-11 (2008)

1097-1106	Synthesis of Novel Bicyclic Nucleosides with 3,6-Anhydro Sugar Moiety	Myong Jung Kim
1107-1112	One-Pot Synthesis of Antiviral Acyclovir and Other Nucleosides Derivatives Using Doped Natural Phosphate as Lewis Acid Catalyst	Hassan B. Lazrek; Laila Baddi; Michael Smietana; Jean-Jacques Vasseur; Saïd Sebti; Mohamed Zahouily
1113-1126	Structure and Conformation of 1-β-D-Ribo Furanosyl Pyridin-2-one-5-Carboxamide: An Anti-Inflammatory Agent	Manju Rajeswaran; Thamarapu Srikrishnan
1127-1143	Synthesis of Simple Adenosine Diphosphate Ribose Analogues	Olivier P. Chevallier; Marie E. Migaud
1144-1152	First Synthesis and Anti-HIV Evaluation of 4′-Methyl-Cyclopentanyl 9-Deazaadenosine	Chang Hyun Oh; Lian Jin Liu; Joon Hee Hong
1153-1157	Synthesis of Carbocyclic 2-Substituted Adenine Nucleoside and Related Analogs	Fazila Zulfiqar; Hiroharu Kojima; Masayuki Nakanishi; Takayuki Ando; Yukio Kitade
1158-1174	Conformational Preferences of Hypermodified Nucleoside Lysidine (k²C) Occurring at “Wobble” Position in Anticodon Loop of tRNA^Ile	Kailas D. Sonawane; Ravindra Tewari
1175-1185	Synthesis of Photo-Responsive Acridine-Modified DNA and Its Application to Site-Selective RNA Scission	Keita Tanaka; Yoji Yamamoto; Akinori Kuzuya; Makoto Komiyama
1186-1196	Efficient Synthesis of 4′-Cyclopropylated Carbovir Analogues with Use of Ring-Closing Metathesis from Glycolate	Lian Jin Liu; Jin Cheol Yoo; Joon Hee Hong
1197-1210	Synthesis and DNA Binding Studies of Novel Heterocyclic Substituted Quinoline Schiff Bases: A Potent Antimicrobial Agent	Devappa. S. Lamani; Kallam. R. Venugopala Reddy; H.S. Bhojya Naik; A. Savyasachi; H. Raja. Naik

Volume 27, Issue 9 (2008)

1011-1023	Studies on the Inhibition of Moloney Murine Leukemia Virus Reverse Transcriptase by N-Tritylamino Acids and N-Tritylamino Acid-Nucleotide Compounds	Arthur Hawtrey; Anton Pieterse; Johann van Zyl; Pieter Van der Bijl; Marichen Van der Merwe; William Nel; Mario Ariatti
1024-1033	Process Research on the Preparation of DMT Protected 2′-O-Methoxyethylguanosine for Oligonucleotide Synthesis in Therapeutic Applications	Shabbir Ali S. Taj; S. Narayanan; S. Suman Meenakshi; Yogesh S. Sanghvi; Bruce S. Ross; Vasulinga T. Ravikumar
1034-1044	New Sulphonamide and Carboxamide Derivatives of Acyclic C-Nucleosides of Triazolo-Thiadiazole and the Thiadiazine Analogues. Synthesis, Anti-HIV, and Antitumor Activities. Part 2	Najim A. Al-Masoudi; Yaseen A. Al-Soud
1045-1060	Novel Enamine Derivatives of 5,6-Dihydro-2′-Deoxyuridine Formed in Reductive Amination of 5-Formyl-2′-Deoxyuridine	Elzbieta Sochacka; Damian Smuga
1061-1071	Synthesis and Evaluation of Antimicrobial Activity of Some Pyrimidine Glycosides	H. A. El-Sayed; A. H. Moustafa; A. Z. Haikal; I. M. Abdou; E. S. H. El-Ashry
1072-1082	Long, Processive Enzymatic DNA Synthesis Using 100% Dye-Labeled Terminal Phosphate-Linked Nucleotides	Jonas Korlach; Arek Bibillo; Jeffrey Wegener; Paul Peluso; Thang T. Pham; Insil Park; Sonya Clark; Geoff A. Otto; Stephen W. Turner
1084-1096	Metalloregulation of Triple Helix Formation by Control of the Loop Conformation	Toshihiro Ihara; Yoshinobu Sato; Hiroshi Shimada; Akinori Jyo

Volume 27, Issue 8 (2008)

901-913	Synthetic Studies on Formamidopyrimidines Related to Clofarabine	William R. Cantrell Jr.; Dennis Lovett; Tracy Engles; Bruce Anderson; William E. Bauta; Paul C. Wolstenholme-Hogg
914-930	A Rapid Synthetic Route to Conformationally Restricted [5,5]-Bicyclic Nucleoside-Amino Acid Conjugates	Kevin W. C. Poon; Apurba Datta
931-948	Protecting Groups Transfer: Unusual Method of Removal of Tr and Tbdms Groups by Transetherification	Nadia L. D. Cabral; Luciano Hoeltgebaum Thiessen; Bogdan Doboszewski
949-966	In Vitro Selection and Characterization of Cellulose-Binding RNA Aptamers Using isothermal Amplification	B. J. Boese; K. Corbino; R. R. Breaker
967-978	Inactivation of Nitric Oxide by Uric Acid	Christine Gersch; Sergiu P. Palii; Kyung Mee Kim; Alexander Angerhofer; Richard J. Johnson; George N. Henderson
979-991	Synthesis of the Fully Protected Phosphoramidite of the Benzene-DNA Adduct, N²-(4-Hydroxyphenyl)-2′-Deoxyguanosine and Incorporation of the Later into DNA Oligomers	Ahmed Chenna; Ramesh C. Gupta; Radha R. Bonala; Francis Johnson; Bo Hang
992-1000	Mineral Supported Facile Synthesis of Novel 4-Hydroxybenzoxazin-2-Thione N-Nucleosides	Ibadur R. Siddiqui; Vishal Srivastava; Pravin K. Singh
1001-1008	Synthesis and Biological Evaluation of Novel Selenonucleosides	Yao Chen; Yingdan Peng; Jiancun Zhang; Lei Fu
1009	Erratum

Volume 27, Issue 6-7 (2008)

547-553	PP07: New Approaches, New Knowledge, New Challenges in Human Purine and Pyrimidine Metabolism	Michael A. Becker; Richard L. Sabina
554-556	In Memoriam: J. Edwin Seegmiller, M.D. (1920–2006)	Michael A. Becker; Theodore Friedmann; Kari O. Raivio; Michael S. Hershfield; George Nuki
557-558	In Memoriam: Albert van Gennip (1943–2007)	Andre van Kuilenburg; Ronney de Abreu
559-563	Lesch-Nyhan Disease	W. L. Nyhan
564-569	The Diagnosis Of HPRT Deficiency in the 21St Century	R. J. Torres; J. G. Puig
570-574	Molecular Analysis of Hypoxanthine Guanine Phosphoribosyltransferase (HPRT) Deficiencies: Novel Mutations and the Spectrum of Japanese Mutations	Yasukazu Yamada; Noriko Nomura; Kenichro Yamada; Nobuaki Wakamatsu; Kiyoko Kaneko; Shin Fujimori
575-577	Urinary Guanidinoacetate and Creatine Levels in Patients with HPRT Deficiency	A. Verdú; R. J. Torres; B. Merinero; J. G. Puig
578-584	Urate Transport Across the Apical Membrane of Renal Proximal Tubules	Hitoshi Endou; Naohiko Anzai
585-591	Determinants of the Clinical Outcomes of Gout During the First Year of Urate-Lowering Therapy	Michael A. Becker; Patricia A. MacDonald; Barbara J. Hunt; Christopher Lademacher; Nancy Joseph-Ridge
592-595	Asymptomatic Hyperuricemia: Impact of Ultrasonography	J. G. Puig; E. de Miguel; M. C. Castillo; A. López Rocha; M. A. Martínez; R. J. Torres
596-600	Production and Characterization of Transgenic Mice Harboring Mutant Human UMOD Gene	Yuichi Takiue; Makoto Hosoyamada; Takuya Yokoo; Masaki Kimura; Manami Ochiai; Kiyoko Kaneko; Kimiyoshi Ichida; Tatsuo Hosoya; Toshiaki Shibasaki
601-603	Effects of Allopurinol on Beer-Induced Increases in Plasma Concentrations of Purine Bases and Uridine	Taku Inokuchi; Tuneyoshi Ka; Asako Yamamoto; Sumio Takahashi; Zenta Tsutsumi; Yuji Moriwaki; Tetsuya Yamamoto
604-607	An Unusual Patient with Hypothyroidism, Tophaceous Gout, and Marked Joint Destruction	F. Montoya; R. J. Torres; J. M. Fraile; J. G. Puig
608-619	Uric Acid: The Oxidant-Antioxidant Paradox	Yuri Y. Sautin; Richard J. Johnson
620-623	Serum Urate, Metabolic Syndrome, and Cardiovascular Risk Factors. A Population-Based Study	J. G. Puig; M. A. Martínez; M. Mora; J. M. Fraile; F. Montoya; R. J. Torres
624-627	Antioxidant Status and Purine Bases in Carotid Artery Plaque	I. Ciari; L. Terzuoli; B. Porcelli; M. G. Coppola; E. Marinello
628-630	Purine Contents of Soybean-Derived Foods and Selected Japanese Vegetables and Mushrooms	K. Kaneko; Y. Kudo; T. Yamanobe; K. Mawatari; M. Yasuda; K. Nakagomi; S. Fujimori
631-633	Effect of Acarbose on the Increased Plasma Concentration of Uric Acid Induced by Sucrose Ingestion	Y. Moriwaki; T. Inokuchi; T. Ka; A. Yamamoto; Z. Tsutsumi; S. Takahashi; T. Yamamoto
634-640	Fludarabine Induces Differential Expression of Proteins in Human Leukemia and Lymphoma Cells	S. Henrich; S. Gez; B. Crossett; S. P. Mulligan; R. I. Christopherson

Volume 27, Issue 6-7 (2008)

641-647	Application of Metabolomic Principles to Disorders of Nucleotide Metabolism Reveals New Metabolic Perturbations	Floyd F. Snyder; Robert J. Carter; Ernest Fung; Stephen D. Hodges; Kevin B. Mantik
648-655	Unusual Presentation of Kelley-Seegmiller Syndrome	I. Sebesta; B. StibÅrková; L. Dvorakova; M. Hrebicek; J. Minks; L. Stolnaja; Z. Vernerova; I. Rychlik
656-660	ITPase Activity in Dry Blood Spots is Comparable with That in Fresh Erythrocytes	J. Tomkova; D. Friedecky; P. Vyskocilova; T. Adam
661-665	Fatal Myelotoxicity After Azathioprine Treatment	O. Slanař; P. Chalupná; A. Novotný; M. Bortlík; Z. Krška; M. Lukáš
666-672	Neurotrophic Effects of Extracellular Guanosine	Michel Rathbone; Lara Pilutti; Francesco Caciagli; Shucui Jiang
673-680	Metabolism and Distribution of Guanosine Given Intraperitoneally: Implications for Spinal Cord Injury	Shucui Jiang; Gemma Fischione; Patricia Guiliani; Silvia Romano; Francesco Caciagli; Patrizia DiIorio
681-691	The Role of Platelet-Derived Endothelial Cell Growth Factor/Thymidine Phosphorylase in Tumor Behavior	I. V. Bijnsdorp; M. de Bruin; A. C. Laan; M. Fukushima; G. J. Peters
692-698	Pharmacokinetics of 5-Fluorouracil in Patients Heterozygous for the IVS14+1G > A Mutation in the Dihydropyrimidine Dehydrogenase Gene	A. B. P. van Kuilenburg; J. G. Maring; A. Schalhorn; C. Terborg; H. Schmalenberg; D. Behnke; W. Schwabe; K. Jabschinsky; P. Hausler
699-703	Trifluorothymidine Induces Cell Death Independently of p53	I. V. Bijnsdorp; F. A. Kruyt; M. Fukushima; G. J. Peters
704-711	Guanine Nucleotide Depletion Mediates Translocation of Nucleolar Proteins, Including RNA Helicase A (DHX-9)	Min Huang; Beverly S. Mitchell
712-719	RNAi Depletion of Deoxycytidine and Deoxyguanosine Kinase in Human Leukemic CEM Cells	Anna Fyrberg; Freidoun Albertioni; Kourosh Lotfi
720-725	Correlation Between Cytidine Deaminase Genotype and Gemcitabine Deamination in Blood Samples	E. Giovannetti; A. C. Laan; E. Vasile; C. Tibaldi; S. Nannizzi; S. Ricciardi; A. Falcone; R. Danesi; G. J. Peters
726-732	Altered Dihydropyrimidine Dehydrogenase Activity Associated with Mild Toxicity in Patients Treated with 5-Fluorouracil Containing Chemotherapy	André B. P. van Kuilenburg; Heinz-Josef Klumpen; Anneke M. Westermann; Lida Zoetekouw; Piet J. M. Bakker; Henk-Jan Guchelaar; Dick J. Richel
733-739	Selective Protection by Uridine of Growth Inhibition by 5-Fluorouracil (5FU) Mediated by 5FU Incorporation into RNA, But Not the Thymidylate Synthase Mediated Growth Inhibition by 5FU-Leucovorin	G. Codacci-Pisanelli; P. Noordhuis; C. L. van der Wilt; G. J. Peters
740-745	Functional Inactivity and Mutations of p53 Differentially Affect Sensitivity to 5-Fluorouracil and Antifolate Inhibitors of Thymidylate Synthase (TS) by Altering TS Levels in Colorectal Cancer Cells	E. Giovannetti; H. H. J. Backus; D. Wouters; G. J. Peters
746-749	Reduced Levels of Mitochondrial DNA Increases the Toxicity of 9-ß-D-Arabinofuranosylguanine (araG)	M. Bjerke; J. Balzarini; A. Karlsson
750-754	Adenosine Kinase Gene Expression in Human Colorectal Cancer	S. Giglioni; R. Leoncini; E. Aceto; A. Chessa; S. Civitelli; A. Bernini; G. Tanzini; F. Carraro; A. Pucci; D. Vannoni
755-760	Regulation of Leukocyte Migration Across Endothelial Barriers by ECTO-5′-Nucleotidase-Generated Adenosine	Linda F. Thompson; Masahide Takedachi; Yukihiko Ebisuno; Toshiyuki Tanaka; Masayuki Miyasaka; Jeffery H. Mills; Margaret S. Bynoe
761-768	Decreased Ecto-Ntpdase1/Cd39 Activity Leads to Desensitization of P2 Purinoceptors Regulating Tonus of Corpora Cavernosa in Impotent Men with Endothelial Dysfunction	M. Faria; T. Magalhães-Cardoso; J. -M. Lafuente-de-Carvalho; P. Correia-de Sá
769-778	Physiological and Pharmacological Roles of Nucleoside Transporter Proteins	Míriam Molina-Arcas; Laia Trigueros-Motos; F. Javier Casado; Marçal Pastor-Anglada

Volume 27, Issue 6-7 (2008)

779-786	Imatinib-Resistant CML Cells Have Low ENT Activity But Maintain Sensitivity to Gemcitabine	Andrea V. Leisewitz; Eric I. Zimmerman; Shannon Z. Jones; Jing Yang; Lee M. Graves
787-793	Immunocytochemical Detection of hENT1 and hCNT1 in Normal Tissues, Lung Cancer Cell Lines, and NSCLC Patient Samples	I. Hubeek; E. Giovannetti; A. J. F. Broekhuizen; M. Pastor-Anglada; G. J. L. Kaspers; G. J. Peters
794-799	Degradation of Pyrimidines in Saccharomyces Kluyveri: Transamination of β-Alanine	K. D. Schnackerz; G. Andersen; D. Dobritzsch; J. Piškur
800-808	Molecular Mechanisms of Mitochondrial DNA Depletion Diseases Caused by Deficiencies in Enzymes in Purine and Pyrimidine Metabolism	Staffan Eriksson; Liya Wang
809-815	Identification of Two Novel Mutations C79X and R235Q in the Dihydropyrimidine Dehydrogenase Gene in a Patient Presenting With Hematuria	A. B. P. van Kuilenburg; J. Meijer; D. Dobritzsch; B. Lohkamp; W. Ruitenbeek; J. Roelofsen; N. G. G. M. Abeling; M. Duran; C. Buzing
816-820	Inhibition of Deoxynucleoside Kinases in Human Thymocytes Prevents dATP Accumulation and Induction of Apoptosis	Michelle L. Joachims; Patrick Marble; Christopher Knott-Craig; Peter Pastuszko; Michael R. Blackburn; Linda F. Thompson
821-824	Ecto-5′-Nucleotidase (Cd73)-Mediated Extracellular Adenosine Production Plays a Critical Role in Hepatic Fibrosis	Zhongsheng Peng; Patricia Fernandez; Tuere Wilder; Herman Yee; Luis Chiriboga; Edwin S. L. Chan; Bruce N. Cronstein
825-829	ß-Alanine and ß-Aminoisobutyric Acid Levels in Two Siblings With Dihydropyrimidinase Deficiency	A. B. P. van Kuilenburg; A. E. M. Stroomer; A. M. Bosch; M. Duran
830-834	Metabolism of 4-Pyridone-3-Carboxamide-1-ß-D- Ribonucleoside Triphosphate and Its Nucleoside Precursor in the Erythrocytes	E. M. Slominska; C. Orlewska; A. Yuen; L. Osman; P. Romaszko; E. Sokolowska; H. Foks; H. A. Simmonds; M. H. Yacoub; R. T. Smolenski
835-838	Polymorphisms of the TPMT Gene in the Czech Healthy Population and Patients with Inflammatory Bowel Disease	Ondřej Slanař; Martin Bortlík; Helena Buzková; Robert Donoval; Kristina Pechandová; Ivan Šebesta; Milan Lukáš; František Perlík
839-849	IMP Dehydrogenase-Linked Retinitis Pigmentosa	Lizbeth Hedstrom
850-857	Human Cytidine Triphosphate Synthetase 1 Interacting Proteins	M. J. Higgins; D. Loiselle; T. A. Haystead; L. M. Graves
858-862	5-Bromovinyl 2′-Deoxyuridine Phosphorylation by Mitochondrial and Cytosolic Thymidine Kinase (TK2 and TK1) and Its Use in Selective Measurement of TK2 Activity in Crude Extracts	Liya Wang; Staffan Eriksson
863-866	Cytoprotective Effects of Nicotinamide Derivatives in Endothelial Cells	E. M. Slominska; A. Yuen; L. Osman; J. Gebicki; M. H. Yacoub; R. T. Smolenski
867-871	Pharmacological Inhibition of AMP-Deaminase in Rat Cardiac Myocytes	T. Borkowski; C. Orlewska; E. M. Slominska; A. Yuen; M. Lipinski; I. Rybakowska; H. Foks; K. K. Kaletha; M. H. Yacoub; R. T. Smolenski
872-875	A Kinetic Study of the Rat Liver Adenosine Kinase Reverse Reaction	D. Vannoni; S. Giglioni; A. Santoro; E. Aceto; E. Marinello; R. Leoncini
876-880	Modulation of AMP Deaminase in Rat Hearts Subjected to Ischemia and Reperfusion by Purine Riboside	T. Borkowski; M. Lipinski; R. Kaminski; E. Krzyminska-Stasiuk; M. Langowska; G. Raczak; E. M. Slominska; R. T. Smolenski
881-887	Mechanism of Transition from Xanthine Dehydrogenase to Xanthine Oxidase: Effect of Guanidine-HCL or Urea on the Activity	Atsuko Tsujii; Takeshi Nishino
888-893	Mechanism of Inhibition of Xanthine Oxidoreductase by Allopurinol: Crystal Structure of Reduced Bovine Milk Xanthine Oxidoreductase Bound with Oxipurinol	Ken Okamoto; Bryan T. Eger; Tomoko Nishino; Emil F. Pai; Takeshi Nishino
894-899	The Role for Glutamic Acid at Position 196 in Human Hypoxanthine Phosphoribosyltransferase (HPRT) as Investigated Using Site-Directed Mutagenesis	B. Canyuk; A. E-Wan; W. Keawwijit; T. Nualnoi; L. Sirisatean; P. Tansakul; C. Tanthana

Volume 27, Issue 5 (2008)

433-438	Association of Nuclear Membrane Protein Lamin B1 with Necrosis and Apoptosis in Cell Death Induced by 5-Fluoro-2′-Deoxyuridine	Akira Sato; Akiko Hiramoto; Akito Satake; Eriko Miyazaki; Tomoharu Naito; Yusuke Wataya; Hye-Sook Kim
439-448	Synthesis and Biological Activity of Mustard Derivatives of Thymine	Amel Hadj-Bouazza; Karine Teste; Ludovic Colombeau; Vincent Chaleix; Rachida Zerrouki; Michel Kraemer; Odile Sainte Catherine
449-459	Synthesis of 2′-([1,2,3]Triazol-1-yl)-2′-deoxyadenosines	Gavin O′Mahony; Sara Svensson; Andreas Sundgren; Morten Grøtli
460-468	Synthesis and Antitumor Activity of a Heterodinucleotide of BVDU and Gemcitabine	L. Cappellacci; P. Franchetti; P. Vita; R. Petrelli; M. Grifantini
469-483	Microwave-Assisted Synthesis and Anti-HIV Activity of New Acyclic C-Nucleosides of 3-(D-Ribo-Tetritol-1-yl)-5-Mercapto-1,2,4-Triazoles. Part 1	Yaseen A. Al-Soud; Najim A. Al-Masoudi; Thilo Schuppler; Erik De Clercq; Christophe Pannecouque
484-494	Bicyclic Nucleoside Synthesis—A Photochemical Approach	E. Lee-Ruff; D. Wells
495-505	Inhibitors Interacting with the Magnesium Binding Site of Reverse Transcriptase: Synthesis and Biological Activity Studies of 3′-(Ω-Amino-Acyl) Amino-3′-Deoxy-Thymidine	Thirumani Venkateshwar Goud; Anne-Marie Aubertin; Jean-François Biellmann
506-524	The Electron Affinities of Deprotonated Adenine, Guanine, Cytosine, Uracil, and Thymine	Edward C. M. Chen; John R. Wiley; Edward S. Chen
525-533	7-Deazainosine Derivatives: Synthesis and Characterization of 7- and 7,8-Substituted Pyrrolo [2,3-d]Pyrimidine Ribonucleosides	Nunzia Ciliberti; Elisa Durini; Stefano Manfredini; Silvia Vertuani
534-545	Tailoring the Peptide-Binding Specificity Of An RNA by Combinations of Specificity-Altering Mutations	Maki Sugaya; Futoshi Nishimura; Akira Katoh; Kazuo Harada

Volume 27, Issue 4 (2008)

319-331	Acyclic Phosphonate Nucleotides and Human Adenylate Kinases: Impact of a Borano Group on α-P Position	D. Topalis; K. Alvarez; K. Barral; H. Munier-Lehmann; B. Schneider; M. Véron; C. Guerreiro; L. Mulard; C. El-Amri; B. Canard; D. Deville-Bonne
332-350	Diastereomer Separation of Azobenzene-Tethered Oligodeoxyribonucleotides and Determination of Their Absolute Configurations by Enzymatic Digestion	Xingguo Liang; Makoto Komiyama; Hiroyuki Asanuma
351-367	Novel N-3 Substituted TSAO-T Derivatives: Synthesis and Anti-HIV-Evaluation	María-Cruz Bonache; Ernesto Quesada; Chih-Wei Sheen; Jan Balzarini; Nicolas Sluis-Cremer; María Jesús Pérez-Pérez; María-José Camarasa; Ana San-Félix
368-375	A Highly Efficient and Selective Synthesis of 1,2,3-Triazole Linked Saccharide Nucleosides Via “Click Chemistry”	Haixin Ding; Ruchun Yang; Yang Song; Qiang Xiao; Jun Wu
376-388	ChipcheckII—Predicting Binding Curves for Multiple Analyte Strands on Small DNA Microarrays	Karsten Siegmund; Carolin Ahlborn; Clemens Richert
389-407	De Novo Synthetic Route to a Combinatorial Library of Peptidyl Nucleosides	Kevin W. C. Poon; Ningning Liang; Apurba Datta
408-420	Synthesis of 3′-Acetamidoadenosine Derivatives as Potential A₃ Adenosine Receptor Agonists	Moon Woo Chun; Sung Wook Choi; Tae Kyung Kang; Won Jun Choi; Hea Ok Kim; Zhan-Guo Gao; Kenneth A. Jacobson; Lak Shin Jeong
421-430	Regio- and Diastereo-Selectivity of Montmorillonite-Catalyzed Oligomerization of Racemic Adenosine 5′-Phosphorimidazolide	Hidehito Urata; Mami Fujimori; Chie Aono; Tomomi Yamakawa; Emi Harada; Masao Akagi
431	Erratum

Volume 27, Issue 3 (2008)

213-223	Selective Synthesis and Application to the Synthesis of (E)-Fluorovinyl Nucleosides	Qingbo Shen; Joon Hee Hong
224-243	Nucleic Acid Isothermal Amplification Technologies—A Review	Pooria Gill; Amir Ghaemi
244-260	Synthesis and Biological Evaluation of Inhibitors of Thymidine Monophosphate Kinase from Bacillus Anthracis	Youngjoo Byun; Susan R. Vogel; Andrew J. Phipps; Cecilia Carnrot; Staffan Eriksson; Rohit Tiwari; Werner Tjarks
261-278	Incorporation of Multiple Sequential Pseudothymidines by DNA Polymerases and Their Impact on DNA Duplex Structure	Stephanie A. Havemann; Shuichi Hoshika; Daniel Hutter; Steven A. Benner
279-291	Synthesis of Ethyl (1S,2R,3S,4S,5S)-2,3-O-(Isopropylidene)-4-Hydroxy-Bicyclo[3.1.0]Hexane-Carboxylate from L-Ribose: A Versatile Chiral Synthon for Preparation of Adenosine and P2 Receptor Ligands	Bhalchandra V. Joshi; Artem Melman; Richard L. Mackman; Kenneth A. Jacobson
292-308	Recognition of a Flipped Base in a Hairpinloop DNA by a Small Peptide	Junji Kawakami; Shinji Okabe; Yoshiatsu Tanabe; Naoki Sugimoto
309-317	Synthesis and Activity Against HBV of Novel Tetra-Seconucleoside Analogues of Dyphlline Having the Acyclic Chains of ACV and HBG	El Sayed H. El Ashry; Laila F. Awad; Nagwa Rashed; Adel AbdelRahman; Hana A. Rasheed

Volume 27, Issue 2 (2008)

103-109	“One-Pot” Syntheses of Malondialdehyde Adducts of Nucleosides	Jozsef Szekely; Hao Wang; Katherine M. Peplowski; Charles G. Knutson; Lawrence J. Marnett; Carmelo J. Rizzo
110-120	Synthesis and Biological Activity of Chloroethyl Pyrimidine Nucleosides	Ludovic Colombeau; Karine Teste; Amel Hadj-Bouazza; Vincent Chaleix; Rachida Zerrouki; Michel Kraemer; Odile Sainte Catherine
121-130	Synthesis and anti-HIV Study of Novel Acyclic Guanine Derivatives	Aihong Kim; Joon Hee Hong
131-145	Incorporation of Zebularine from its 2′-Deoxyribonucleoside Triphosphate Derivative and Activity as a Template-Coding Nucleobase	Casimir L. Dowd; Brian T. Sutch; Ian S. Haworth; Ramón Eritja; Victor E. Marquez; Allen S. Yang
146-156	New Acyclic Quinoxaline Nucleosides. Synthesis and Anti-Hiv Activity	Ibrahim A. I. Ali; Iman A. Al-Masoudi; Nazik M. Aziz; Najim A. Al-Masoudi
157-172	A Novel Thymidine Phosphoramidite Synthon for Incorporation of Internucleoside Phosphate Linkers During Automated Oligodeoxynucleotide Synthesis	David Tabatadze; Paul Zamecnik; Ivan Yanachkov; George Wright; Katherine Pierson; Surong Zhang; Alexei Bogdanov Jr.; Valeri Metelev
173-185	Synthesis, Characterization, and In Vitro Assay of Folic Acid Conjugates of 3′-Azido-3′-Deoxythymidine (AZT): Toward Targeted AZT Based Anticancer Therapeutics	Anthony R. Vortherms; Robert P. Doyle; Dayuan Gao; Olivia Debrah; Patrick J. Sinko
186-195	Design, Synthesis and Anti-HIV Activity of Homologous PMEA Derivatives	Chang Hyun Oh; Joon Hee Hong
196-212	Steric Block High Affinity Oligonucleotide Analogues: A New Tool for Mapping RNA-Protein Binding Sites	Douglas Brown; Emily Joy; Jane Greatorex; Michael J. Gait; Andrew M. L. Lever

Volume 27, Issue 1 (2007)

1-17	Chemical Synthesis of LNA-mCTP and Its Application for MicroRNA Detection	Anilkumar Kore; Melissa Hodeib; Zhongting Hu
18-30	Synthesis and Stability of Novel Terminal Phosphate-Labeled Nucleotides	Bambi Reynolds; Rachel Miller; John Williams; Jon Anderson
31-36	Activity of Adenosine Deaminase and Adenylate Deaminase on Adenosine and 2', 3'-Isopropylidene Adenosine: Role of the Protecting Group at Different pH Values	Laura Alessandrini; Pierangela Ciuffreda; Radmila Pavlovic; Enzo Santaniello
37-42	Synthesis and Biological Evaluation of LNA Phosphoramidates	Jacob Jensen; Gitte Sjøgren; Jens Bo Hansen; Christoph Rosenbohm; Troels Koch
43-56	Synthesis of Pyrophosphates for In Vitro Selection of Catalytic RNA Molecules	Hyo-Joong Kim; Myong Jung Kim; Nilesh Karalkar; Daniel Hutter; Steven A. Benner
57-66	In Vivo Evaluation of the Uptake of [123I]FIAU, [123I]IVFRU and [123I]IVFAU by Normal Mouse Brain: Potential For Noninvasive Assessment of HSV-1 Thymidine Kinase Gene Expression in Gliomas	H. -F. Li; A. Winkeler; S. Moharram; E. E. Knaus; K. Dittmar; M. Stockle; W. D. Heiss; L. I. Wiebe; A. J. Jacob
67-69	An Efficient and Scalable Synthesis of 2,6-Diaminopurine Riboside	Bruce Ross; Robert Springer; Vasulinga Ravikumar
70-83	Plasmid Loss in Plasmid-carrying Strains of Escherichia coli Treated with Phenoxazines and an Approach to Study Their DNA Binding Properties	K. H. Chandramouli; Cletus D'Souza; K. N. Thimmaiah
84-100	Application of Chiral Cyclic Nitrones to the Diastereoselective Synthesis of Bicyclic Isoxazolidine Nucleoside Analogues	Evdoxia Coutouli-Argyropoulou; Christos Xatzis; Nikolaos Argyropoulos
101	Erratum	Hyuk Woo Lee; Dae Hong Shin; Ji Young Jung; Hea Ok Kim; Moon Woo Chun; N. Melman; Z. -G. Gao; Kenneth Jacobson; Lak Shin Jeong

Volume 26, Issue 10-12 (2007)

1211-1215	Kinetics of C. Elegans DcpS Cap Hydrolysis Studied by Fluorescence Spectroscopy	J. Wierzchowski; M. Pietrzak; J. Stepinski; J. Jemielity; M. Kalek; E. Bojarska; M. Jankowska-Anyszka; R. E. Davis; E. Darzynkiewicz
1217-1220	Synthesis of C8-Modified 2″-Deoxyadenosine with Carcinogenic Arylamines	M. I. Jacobsen; C. Meier
1221-1224	Polyaza Crown Ether as Non-Nucleosidic Building Blocks in DNA-Conjugates	Ulla Jakobsen; Katja Rohr; Rasmus K. Madsen; Stefan Vogel
1225-1229	Synthesis and Biophysical Characterization of G-Rich Oligonucleotides Conjugated with Sugar-Phosphate Tails	J. D'Onofrio; E. Erra; G. Di Fabio; A. Iadonisi; L. Petraccone; L. De Napoli; G. Barone; J. Balzarini; C. Giancola; D. Montesarchio
1231-1236	Synthesis and Characterization of Tetra-End Linked Oligonucleotides Capable of Forming Monomolecular G-Quadruplexes	Nicola Borbone; Giorgia Oliviero; Jussara Amato; Stefano D'Errico; Aldo Galeone; Gennaro Piccialli; Luciano Mayol
1237-1240	Synthesis Study of 2′-O-(2-Methoxyethyl)-Purine Derivatives	Grigorii G. Sivets
1241-1244	Synthesis of L-2′-Deoxypentofuranonucleoside Derivatives of Thymine From D-Glucose	Grigorii G. Sivets
1245-1248	Novel CoA-Polyamine Conjugates for Effective Inhibition of Spermine/Spermidine-N¹-Acetyltransferase	Alina Simonian; Alex Khomutov; Tapani Hyvonen; Nikolay Grigorenko; Tuomo Keinanen; Jouko Vepsalainen; Leena Alhonen; Juhani Janne
1249-1253	Efficient Synthesis of Benzamide Riboside, a Potential Anticancer Agent	Laurent F. Bonnac; Guang-Yao Gao; Liqiang Chen; Steven E. Patterson; Hiremagalur N. Jayaram; Krzysztof W. Pankiewicz
1255-1260	Fission Yeast Telomeric DNA Binding Protein Pot1 Has The Ability To Unfold Tetraplex Structure of Telomeric DNA	Hidetaka Torigoe
1261-1263	Dual-Probe System Using Pyrenylmethyl-Modified Amino-Lna for Mismatch Detection	Tadashi Umemoto; Patrick J. Hrdlicka; B. Ravindra Babu; Jesper Wengel
1265-1268	Development of Artificial Restriction DNA Cutter Composed of Ce(Iv)/EDTA and PNA	Yoji Yamamoto; Akihiko Uehara; Kazuyuki Miura; Akira Watanabe; Hiroyuki Aburatani; Makoto Komiyama
1269-1271	Sulfur Containing Acyclovir Derivatives: Synthesis, Cytotoxic Activity, and Cell Phenotype Studies	Martins Ikaunieks; Irina Shestakova; Ilona Domracheva; Sergey Belyakov; Marina Madre
1273-1276	A Convenient Solid-Phase Method for the Synthesis of Novel Oligonucleotide-Folate Conjugates	Eugenia V. Kazanova; Eugeny M. Zubin; Anna V. Kachalova; Eugeny M. Volkov; Tatiana S. Oretskaya; Dmitry A. Stetsenko; Marina B. Gottikh
1277-1281	Stepwise Functionalization of Ribonucleopeptides: Optimization of the Response of Fluorescent Ribonucleopeptide Sensors for ATP	Tetsuya Hasegawa; Masaki Hagihara; Masatora Fukuda; Takashi Morii
1283-1286	2′-O-Dimethylaminoethoxyuridine and 5-Dimethylaminopropargyl Deoxyuridine for at Base Pair Recognition in Triple Helices	Lavinia Brennan; Guomei Peng; Natarajan Srinivasan; Keith R. Fox; Tom Brown
1287-1293	Oligonucleotide Synthesis Using Ionic Liquids as Soluble Supports	Robert A. Donga; Matthew Hassler; Tak-Hang Chan; Masad J. Damha
1295-1299	Optical Tweezers as a Probe for Oligodeoxyribonucleotide Structuration	Nicola Borbone; Giorgia Oliviero; Jussara Amato; Gennaro Piccialli; Luciano Mayol; Lisa Miccio; Giuseppe Pescen; Antonio Sasso
1301-1305	Assignment of the Absolute Configuration of P-Chiral 5′Mrna Cap Analogues Containing Phosphorothioate Moiety	Joanna Kowalska; Magdalena Lewdorowicz; Joanna Zuberek; Elzbieta Bojarska; Janusz Stepinski; Ryszard Stolarski; Edward Darzynkiewicz; Jacek Jemielity

Volume 26, Issue 10-12 (2007)

1307-1310	dabPna: Design, Synthesis, And Dna Binding Studies	Giovanni N. Roviello; Domenica Musumeci; Maria Moccia; Mariangela Castiglione; Roberto Sapio; Margherita Valente; Enrico M. Bucci; Giuseppe Perretta; Carlo Pedone
1311-1313	2′,3′-Isopropylidene Group, A Molecular Scaffold to Study the Activity of Adenosine and Adenylate Deaminase on Adenosine Analogues Modified in the Ribose Moiety	Pierangela Ciuffreda; Laura Alessandrini; Enzo Santaniello
1315-1319	Synthesis of ³H and ¹³C Labeled Mrna Cap Dinucleotides—Useful Tools for Nmr, Biochemical, and Biological Studies	Jacek Jemielity; Ryszard Stolarski; Edward Darzynkiewicz
1321-1324	Synthesis of A New Ribose Modified Analogue of Cyclic Inosine Diphosphate Ribose	Giorgia Oliviero; Nicola Borbone; Jussara Amato; Stefano D'Errico; Gennaro Piccialli; Michela Varra; Luciano Mayol
1325-1328	New Developments of the “Lock-in” Modified *cyclo*Sal-d4TMPs	Dalibor Vukadinović-Tenter; Jan Balzarini; Chris Meier
1329-1333	Solid-Supported Synthesis of 5′-mRNA CAP-4 from Trypanosomatids	Magdalena Lewdorowicz; Jacek Jemielity; Ryszard Kierzek; Michal Shapira; Janusz Stepinski; Edward Darzynkiewicz
1335-1338	A Pyrimidopyrimidoindole Nucleoside (dC^PPI): Photophysical Properties and Thermal Stability of the Modified Dna Duplexes	Masahiro Mizuta; Kohji Seio; Kenichi Miyata; Akihiro Ohkubo; Haruhiko Taguchi; Mitsuo Sekine
1339-1348	Synthesis of *Leishmania* Cap-4 Intermediates, Cap-2 and Cap-3	Magdalena Lewdorowicz; Janusz Stepinski; Ryszard Kierzek; Jacek Jemielity; Joanna Zuberek; Yael Yoffe; Michal Shapira; Ryszard Stolarski; Edward Darzynkiewicz
1349-1352	Affinity of Dinucleotide Cap Analogues for Human Decapping Scavenger (hDcpS)	Zbigniew M. Darzynkiewicz; Elzbieta Bojarska; Janusz Stepinski; Jacek Jemielity; Marzena Jankowska-Anyszka; Richard E. Davis; Edward Darzynkiewicz
1353-1357	Evaluation of Different Chemical Strategies for Conjugation of Oligonucleotides to Peptides	Igor A. Kozlov; Peter C. Melnyk; John P. Hachmann; David L. Barker; Michal Lebl; Chanfeng Zhao
1359-1362	Synthesis and Incorporation of a Simple Acyclic Furan Containing Phosphoramidite	K. Stevens; A. Madder
1363-1367	Cg Base Pair Recognition Within Dna Triple Helices Using N-Methyl-3H-Pyrrolo[2,3-d]Pyrimidin-2(7H)-One Nucleoside Analogues	Simon R. Gerrard; Natarajan Srinivasan; Keith R. Fox; Tom Brown
1369-1373	Looking for New Pyrimidine Acyclic Nucleotide Analogues Designed for Phosphorylation by Human Ump-Cmp Kinase	Dimitri Topalis; Hiroki Kumamoto; Julie A. C. Alexandre; Laurence Dugué; Sylvie Pochet; Sabine Berteina-Raboin; Luigi A. Agrofoglio; Dominique Deville-Bonne
1375-1379	Enantio-Selectivity of Human Nucleoside Monophosphate Kinases	J. A. C. Alexandre; B. Roy; D. Topalis; C. Périgaud; D. Deville-Bonne
1381-1386	Synthesis of Pyrene Labeled Rna for Fluorescence Measurements	Taewoo Kwon; Nelly Piton; Christian Grünewald; Joachim W. Engels
1387-1389	Synthesis of 9-(2,3-Dideoxy-2,3-Difluoro-β-D- Arabinofuranosyl)Adenine	Grigorii G. Sivets; Elena N. Kalinichenko; Igor A. Mikhailopulo
1391-1394	Alkyne-Azide Click Chemistry Mediated Carbanucleosides Synthesis	Julie Broggi; Nicolas Joubert; Vincent Aucagne; Sabine Berteina-Raboin; S. Diez-Gonzalez; Steve Nolan; Dimitri Topalis; Dominique Deville-Bonne; Jan Balzarini; Johan Neyts; Graciela Andrei; Robert Snoeck; Luigi A. Agrofoglio
1395-1398	Supported Synthesis and Functionnalization of 2″-Deoxyuridine by Suzuki-Miyaura Cross-Coupling	Saïd El Kazzouli; Sabine Berteina-Raboin; Luigi A. Agrofoglio
1399-1402	Cross-Metathesis Mediated Synthesis of New Acyclic Nucleoside Phosphonates	Vincent Roy; Hiroki Kumamoto; Sabine Berteina-Raboin; Steven P. Nolan; Dimitri Topalis; Dominique Deville-Bonne; Jan Balzarini; Johan Neyts; Gracelia Andrei; Robert Snoeck; Luigi A. Agrofoglio
1403-1405	Synthesis and Biophysical Studies of N2′-Functionalized 2′-Amino-α-L-LNA	T. Santhosh Kumar; Andreas S. Madsen; Jesper Wengel; Patrick J. Hrdlicka

Volume 26, Issue 10-12 (2007)

1407-1409	Pyrene-Functionalized 2 ′-Amino-α-L-LNA as Potential Diagnostic Probes	T. Santhosh Kumar; Jesper Wengel; Patrick J. Hrdlicka
1411-1414	Triplex-Forming Ability of Modified Oligonucleotides	Torben Højland; B. Ravindra Babu; Torsten Bryld; Jesper Wengel
1415-1417	N2′-Functionalized 2′-Amino-α-L-LNA Adenine Derivatives—Efficient Targeting of Single Stranded DNA	Nicolai K. Andersen; Jesper Wengel; Patrick J. Hrdlicka
1419-1422	Toward a Catalytic Site in DNA: Polyaza Crown Ether as Non-Nucleosidic Building Blocks in DNA Conjugates	Ulla Jakobsen; Katja Rohr; Stefan Vogel
1423-1426	Cu²⁺TerPy Complexes as Catalysts of the Cleavage of the 5′-*cap* Structure of mRNA	Leena Maanpää; Sharmin Taherpour; Zhibo Zhang; Clemence Guillaume; Istvan Szilagy; Esa Mäki; Satu Mikkola
1427-1430	Survivin mRNA Antagonists Using Locked Nucleic Acid, Potential for Molecular Cancer Therapy	Niels Fisker; Majken Westergaard; Henrik Frydenlund Hansen; Jens Bo Hansen
1431-1434	Synthesis of 1′-C-Fluoromethyladenosine	Annelaure Damont; David Dukhan; Gilles Gosselin; Jérôme Peyronnet; Richard Storer
1435-1438	Synthesis of Nucleosides with Additional Nucleobases	Charlotte Andersen; Søren L. Pedersen; Poul Nielsen
1439-1442	Synthesis and Stability Studies of 2′,3′,5′-tri-O-Acetyl-2-Amino(-N⁶-Cyclopentyl)-1-Deazaadenosines	Sauro Vittori; Ram Chandra Mishra; Diego Dal Ben; Dhuldeo Kachare; Catia Lambertucci; Rosaria Volpini; Gloria Cristalli
1443-1446	Synthesis and Biological Activity of Trisubstituted Adenines as A_2A Adenosine Receptor Antagonists	Catia Lambertucci; Sauro Vittori; Ram Chandra Mishra; Diego Dal Ben; Karl-Norbert Klotz; Rosaria Volpini; Gloria Cristalli
1447-1450	Bent Oligonucleotide Duplexes as HMGB1 Inhibitors: a Comparative Study	D. Musumeci; G. N. Roviello; M. Moccia; C. Pedone; E. M. Bucci; R. Sapio; M. Valente; S. Fumero
1451-1454	Solid-Phase Synthesis of Modified RNAs Containing Amide-Linked Oligoribonucleosides at Their 3′-End and Their Application to siRNA	Reiko Iwase; Takaaki Toyama; Kengo Nishimori
1455-1457	Synthesis of 9-Fluorenemethyl Boranophosphonodiphosphate Via an H-Phosphonate Approach	Hongyan Liu; Syed N. Hashmi; Barbara Ramsay Shaw
1459-1462	Labeling of Oligonucleotides with DTPA and DOTA on Solid Phase	Jari Hovinen
1463-1466	Triplex Formation-Based Artificial Transcription Factor to Regulate Target Gene Expression	Hidetaka Torigoe; Takuma Katayama; Yusuke Tsukamoto
1467-1470	Synthesis of Aminomethyl- and Bis-Aminomethyl-Fluorescein Energy Transfer Terminators	Sudhakar Rao Takkellapati; Chung Y. Chen; Vladimir Neschadimenko; Satyam Nampalli; Haiguang Xiao; Jeffrey Wegener; Prasad Dhulipala; Shiv Kumar; Carl Fuller
1471-1477	2-5A Ligands—A New Concept for the Treatment of Prostate Cancer	Hagen Cramer; James R. Okicki; Taikyun Rho; Xinning Wang; Robert H. Silverman; Warren D. W. Heston
1479-1483	RNA Cleavage by 2,9-Diamino-1,10-Phenanthroline PNA Conjugates	Merita Murtola; Dimitri Ossipov; Jessica Sandbrink; Roger Strömberg
1485-1489	Solid Support Post-Conjugation of Amino Acids and a Phenanthroline Derivative to a Central Position in Peptide Nucleic Acids	Jessica Sandbrink; Merita Murtola; Roger Strömberg
1491-1493	Evaluation of Lactam Protection for Synthesis of 2′-O-Alkylated Uridines	Stefan Milton; Roger Strömberg

Volume 26, Issue 10-12 (2007)

1495-1499	Synthesis of A 2′-O-(Carbomoylmethyl)Ribonucleoside H-Phosphonate Building Block and A Model Dinucleotide	Stefan Milton; Raunak Esther Yeheskiely; Roger Strömberg
1501-1504	Evaluating Coupling Procedures for Synthesis of Lna-Peptide Conjugates	Peter Steunenberg; Hans Leijonmarck; Mathias G. Svahn; C. I. Edvard Smith; Roger Strömberg
1505-1508	Synthesis of A Branched Locked Nucleic Acid (LNA) Analogue	Pawan K. Sharma; Surender Kumar; Poul Nielsen
1509-1512	2′-O-Hydroxyalkoxymethylribonucleosides and their Incorporation into Oligoribonucleotides	Sergey N. Mikhailov; Georgii V. Bobkov; Kyrill V. Brilliantov; Jef Rozenski; Arthur Van Aerschot; Piet Herdewijn; Michael H. Fisher; Rudolph L. Juliano
1513-1515	Improvement of the Synthesis of Sugar Phosphonates Using Microwave Irradiations	Suzanne Peyrottes; Franck Gallier; Alain Papillaud; Jérôme Béjaud; Christian Périgaud
1517-1521	Novel Selective Biocatalytic Deacylation Studies on Key Precursors for Bicyclonucleosides	Ashok K. Prasad; Sunil K. Singh; Neerja Kalra; Nidhi Singhal; Jesper Wengel; Virinder S. Parmar
1523-1527	Mass Spectrometry Based Methods for Analysis of Nucleosides as Antiviral Drugs and Potential Tumor Biomarkers	Luigi A. Agrofoglio; Vincent Bezy; Patrick Chaimbault; Raphaël Delépée; Boutaina Rhourri; Philippe Morin
1529-1532	Two Carbocyclic Locked Nucleic Acid Analogues Give Structural Information about the Role of Hydration in A-Type Duplexes	Nanna Albæk; Michael Petersen; Poul Nielsen
1533-1538	Porphyrin-DNA: A Supramolecular Scaffold for Functional Molecules on the Nanometre Scale	Imenne Bouamaied; Leslie-Anne Fendt; Daniel Häussinger; Markus Wiesner; Sandra Thöni; Nicolas Amiot; Eugen Stulz
1539-1542	New Pseudonucleosides Containing Chiral Oxazolidin-2-Ones and Cyclosulfamides as Aglycones: Synthesis and Antiviral Evaluation	Hocine Bouleghlem; Malika Berredjem; Marc Lecouvey; Nour-Eddine Aouf
1543-1546	2′-Deoxy-4′-C-Ethynyl-2-Fluoroadenosine: A Nucleoside Reverse Transcriptase Inhibitor with Highly Potent Activity Against Wide Spectrum of HIV-1 Strains, Favorable Toxic Profiles, and Stability in Plasma	Hiroshi Ohrui; Satoru Kohgo; Hiroyuki Hayakawa; Eiichi Kodama; Masao Matsuoka; Tomohiro Nakata; Hiroaki Mitsuya
1547-1551	NMR Study of Ammonium Ion Binding to d[G₃T₄G₄]₂ and d[G₄(T₄G₄)₃] G-Quadruplexes	Peter Podbevšek; Primož Šket; Janez Plavec
1553-1558	Antiviral Activity of 3-(3,5-Dimethylbenzyl)Uracil Derivatives Against Hiv-1 and HCMV	Tokumi Maruyama; Yosuke Demizu; Shigetada Kozai; Myriam Witvrouw; Christophe Pannecouque; Jan Balzarini; Robert Snoecks; Graciella Andrei; Erik De Clercq
1559-1563	Sequence-Specific Recognition of Double-Stranded DNA by Synthetic Minor Groove Binder Conjugates. toward the Construction of Artificial Site-Specific Deoxyribonucleases	Alexandre S. Boutorine; Ludovic Halby; Philippe Simon; Loïc Perrouault; Carine Giovannangeli; Georgy V. Gursky; Anna N. Surovaya; Sergueï L. Grokhovsky; Vladimir A. Ryabinin; Alexandre N. Sinyakov
1565-1568	Design, Synthesis, and Anti-Tumor Activity of 4′-Thionucleosides as Potent and Selective Agonists at the Human A₃ Adenosine Receptor	Lak Shin Jeong; Hyuk Woo Lee; Hea Ok Kim; Ji Young Jung; Prashantha Gunaga; Sang Kook Lee; Eun-Jin Lee; Moon Woo Chun; Zhan-Guo Gao; Kenneth A. Jacobson; Hyung Ryong Moon
1569-1572	Mismatch Discrimination of Base-Modified Nucleic Acids and their Constituents: Non-Watson-Crick Base Pairing Induced by Tautomerization	Frank Seela; Xiaohua Peng; Kuiying Xu
1573-1576	Novel Fluorophores for Labeling of Nucleosides and Oligonucleotides	Shipra Singh; Ramendra K. Singh
1577-1579	Oligonucleotide Conjugate GRN163L Targeting Human Telomerase as Potential Anticancer and Antimetastatic Agent	Sergei M. Gryaznov; Shalmica Jackson; Gunnur Dikmen; Calvin Harley; Brittney-Shea Herbert; Woodring E. Wright; Jerry W. Shay
1581-1584	DNA Labelling Topologies for Monitoring DNA-Protein Complex Formation by Fluorescence Anisotropy	Matthias Bahr; Linda Valis; Hans-Achim Wagenknecht; Elmar Weinhold
1585-1588	Thiazole Orange: A Useful Probe for Fluorescence Sensing of G-Quadruplex–Ligand Interactions	D. Monchaud; C. Allain; M. -P. Teulade-Fichou

Volume 26, Issue 10-12 (2007)

1589-1593	Biophysical Stability and Enzymatic Recognition of Oxanine in Dna	Seung Pil Pack; Akihiro Doi; Mitsuru Nonogawa; Nagendra K. Kamisetty; Kamakshaiah C. Devarayapalli; Tsutomu Kodaki; Keisuke Makino
1595-1599	Synthesis and Properties of Pyrrolidine-Based Negatively Charged Dna Mimics	Vladimir A. Efimov; Valeryi N. Klykov; Oksana G. Chakhmakhcheva
1601-1604	5-Methylcytosine-Selective Osmium Oxidation	Akimitsu Okamoto
1605-1609	A Flexible Method for the Fabrication of Gold Nanostructures Using Oligonucleotide Derivatives	Ramon Eritja; Anna Aviñó; Beatriz G. de la Torre; Donald Fitzmaurice; Andrea Ongaro; Sarmiza Elena Stanca; Andrea DiSalvo; Brendan Maninng; Daniela Iacopino
1611-1613	2′-Deoxyadenosine Bearing Hydrophobic Carborane Pharmacophore	Agnieszka Olejniczak; Blażej Wojtczak; Zbigniew J. Lesnikowski
1615-1618	Highly Effective Non-Explosive Activators Based on Saccharin for the Synthesis of Oligonucleotides and Phosphoramidites	Nanda D. Sinha; Patrick Foster; Satya N. Kuchimanchi; Greg Miranda; Saied Shaikh; Dennis Michaud
1619-1624	In Vivo and in Vitro Activity And Mechanism Of Action of the Multidrug Cytarabine-L-Glycerylyl-Fluorodeoxyuridine	Irene V. Bijnsdorp; Reto A. Schwendener; Herbert Schott; Iduna Fichtner; Kees Smid; Sarah Schott; Adrie C. Laan; Godefridus J. Peters
1625-1628	2′,4′-BNA^NC: A Novel Bridged Nucleic Acid Analogue with Excellent Hybridizing and Nuclease Resistance Profiles	S. M. Abdur Rahman; Sayori Seki; Kazushige Utsuki; Satoshi Obika; Kazuyuki Miyashita; Takeshi Imanishi
1629-1633	Mass Spectrometry of Oligonucleotides	Stefan Schürch; Jan M. Tromp; Selina T. M. Monn
1635-1639	Mismatch Base Pair Detection by Fluorescence Spectral Change Upon Addition of Metal Cation—Toward Efficient Analysis of Single Nucleotide Polymorphism	Hidetaka Torigoe; Akira Ono; Tetsuo Kozasa
1641-1643	The Effect of INA [(R)-1-O-(1-Pyrenylmethyl)Glycerol] Insertions on the Structure and Biological Activity of a G-Quadruplex from a Critical Kras G-Rich Sequence	Susanna Cogoi; Manikandan Paramasivan; L. E. Xodo; Vyacheslav V. Filichev; Erik B. Pedersen
1645-1647	At Tachment of Cholesterol to Amino-LNA: Synthesis and Hybridization Properties	Torsten Bryld; Christian Lomholt
1649-1652	Solid Phase Synthesis of Nucleobase and Ribose Modified Inosine Nucleoside Analogues	Giorgia Oliviero; Jussara Amato; Stefano D'Errico; Nicola Borbone; Gennaro Piccialli; Luciano Mayol
1653-1657	Asymmetric Synthesis and Biological Activity of l-Bicyclocarba-d4T	Hyung Ryong Moon; Ah-Young Park; Kyung Ran Kim; Moon Woo Chun; Lak Shin Jeong
1659-1664	Homogeneous Fluorescence Assays for RNA Diagnosis by Pyrene-Conjugated 2′-O-Methyloligoribonucleotides	Takashi Sakamoto; Akio Kobori; Masako Shigezawa; Yasutaka Amitani; Maiko Higuchi; Akira Murakami
1665-1668	A Simple Nucleic Acid Alternative: Aminopropyl Nucleic Acids (APNAs)	Ding Zhou; Guy Schepers; Arthur Van Aerschot
1669-1672	Detection of Terminal Mismatches on DNA Duplexes in Homogeneous Assays or with Immobilized Probes	Marcel Chassignol; Yves Aubert; Victoria Roig; Ulysse Asseline

Volume 26, Issue 8-9 (2007)

869-871	Synthesis of Fluorinated Indoles as RNA Analogues	Jelena Božilović; Joachim W. Engels
873-877	Different Strategies for the Synthesis of 2′-O-Aminoethyl Adenosine Building Blocks	Dalibor Odadzic; Joachim W. Engels
879-882	A Phenanthrene Modified RNA Hairpin	Ivan Trkulja; Alfred Stutz; Robert Häner
883-887	Aldehydic Oligonucleotide: A Key Intermediate for the Preparation of Oligonucleotide Conjugates Through Oxime Bond Formation	N. Spinelli; Y. Singh; E. Defrancq; P. Dumy
889-892	Microwave-assisted Ribosylation of modified heterocyclic bases by Vorbrüggen method	Nadja V. Nikolaus; Jelena Božilović; Joachim W. Engels
893-896	Acid-Mediated Cleavage oF Oligonucleotide P3′ → N5′ Phosphoramidates Triggered by Sequence-Specific Triplex Formation	Satoshi Obika; Masaharu Tomizu; Yoshinori Negoro; Tomohisa Osaki; Ayako Orita; Yuji Ueyama; Osamu Nakagawa; Takeshi Imanishi
897-900	5′-Carbamoylphosphonyl-[6-3H]-AZT as a Tool for Studying Metabolic Transformations of the Nonradioactive Counterpart, an Inhibitor of HIV Replication	Dmitry V. Yanvarev; Elena A. Shirokova; Maria V. Astapova; Vyacheslav I. Shram; Marina K. Kukhanova; Yury S. Skoblov
901-903	DNA Containing Non-Nucleosidic Phenanthrene Building Blocks with Asymmetrical Linkers	Simon M. Langenegger; Vladimir L. Malinovskii; Daniel Wenger; Sarah Werder; Robert Häner
905-909	An Enzymatic Transglycosylation of Purine Bases	Jarkko Roivainen; Tatiana Elizarova; Seppo Lapinjoki; Igor A. Mikhailopulo; Roman S. Esipov; Anatoly I. Miroshnikov
911-915	Design, Enantiopure Synthesis, and Biological Evaluation of Novel ISO-D-2′,3′-Dideoxy-3′-Fluorothianucleoside Derivatives as a bioisostere of Lamivudine	Kyung Ran Kim; Ah-Young Park; Hyung Ryong Moon; Moon Woo Chun; Lak Shin Jeong
917-920	New Analogs of Acyclovir Substituted at the Side Chain	Zofia Jahnz-Wechmann; Jerzy Boryski; Kunisuke Izawa; Tomoyuki Onishi; Johan Neyts; Erik De Clercq
921-925	Synthesis of Anthraquinone Oligonucleotides for Triplex Stabilization	Zhengyun Zhao; Guomei Peng; Jan Michels; Keith R. Fox; Tom Brown
927-930	Clip-Phen Conjugates for the Specific Cleavage of Nucleic Acids	Alain Laurent; Michael Wright; Ali Laayoun; Bernard Meunier; Ludivine Tissot; Marguerite Pitie
931-934	OligoPrep PVA Support for Oligonucleotide Synthesis in Columns on a Scale up to 10 μ mol	Sheena Aitken; Emma Anderson
935-937	A New and Short Convergent Synthetic Strategy to Carbocyclic Nucleosides	Bastian Reichardt; Chris Meier
939-942	Oligonucleotide Charge Reversal: 2′-O-Lysylaminohexyl Modified Oligonucleotides	Johannes Winkler; Christian R. Noe
943-947	Asymmetric Synthesis of Apio Fluoroneplanocin a Analogs as Potential AdoHcy Hydrolase Inhibitor	Ah-Young Park; Hyung Ryong Moon; Kyung Ran Kim; Jin-Ah Kang; Moon Woo Chun; Lak Shin Jeong
949-952	Hairpin Mimics with Phenanthroline- and Bipyridine-Derived Linkers	Gapian Bianké; Robert Häner
953-957	Inhibition of HIV-1 Replication in Macrophages by Red Blood Cell-Mediated Delivery of a Heterodinucleotide of Lamivudine and Tenofovir	P. Franchetti; L. Cappellacci; R. Petrelli; P. Vita; M. Grifantini; L. Rossi; F. Pierigé; S. Serafini; M. Magnani; E. Balestra; C. -F. Perno

Volume 26, Issue 8-9 (2007)

959-962	A General Route to D- and L-Six-Membered Nucleoside Analogues	Annalisa Guaragna; Daniele D'Alonzo; Mauro De Nisco; Silvana Pedatella; Giovanni Palumbo
963-967	New developments in the synthesis of oligonucleotide-peptide conjugates	Cecilia Portela; José Luis Mascareñas; Fernando Albericio; Stefania Mazzini; Clara Caminal; Roger Ramos; Sandra M. Ocampo; Ramon Eritja
969-974	Kinetics of Binding of Multisubstrate Analogue Inhibitor (2-Amino-9-[2-(Phosphonomethoxy)Ethyl]-6-Sulfanylpurine) with Trimeric Purine Nucleoside Phosphorylase	Jan Antosiewicz; Beata Wielgus-Kutrowska; Maciej Długosz; Antonin Holy; Agnieszka Bzowska
975-978	Synthesis of Enantiopure Pseudo-l-Vinylcyclopropyl Nucleosides Bearing Quaternary Carbon as Potential Anti-Herpesvirus Agent	Hyung Ryong Moon; Ah-Young Park; Kyung Ran Kim; Moon Woo Chun; Lak Shin Jeong
979-983	Triplex Formation Using Oligonucleotide Clamps Carrying 8-Aminopurines	Anna Aviñó; Marta G. Grimau; Margarita Alvira; Ramon Eritja; Raimundo Gargallo; Modesto Orozco; Carlos González
985-988	Synthesis of 2′,3′-Dideoxyinosine via Radical Deoxygenation	Takayoshi Torii; Kunisuke Izawa; Dae Hyan Cho; Doo Ok Jang
989-993	Inhibitory Properties of Nucleotides with Difluoromethylenephosphonic Acid as a Phosphate Mimic versus Calf Spleen Purine Nucleoside Phosphorylase and Effect of These Analogues on the Viability of Human Blood Lymphocytes	Ljubica Glavaš-Obrovac; Mirjana Suver; Sadao Hikishima; Tsutomu Yokomatsu; Agnieszka Bzowska
995-999	Nucleolipids as Potential Organogelators	Helmut Rosemeyer; Eva-Maria Stürenberg; Piet Herdewijn
1001-1004	Asymmetric Synthesis of Novel Pseudo-d-Vinylcyclopropyl Nucleosides Bearing Quaternary Carbon as Potential Anti-Herpesvirus Agent	Ah-Young Park; Hyung Ryong Moon; Kyung Ran Kim; Moon Woo Chun; Lak Shin Jeong
1005-1009	Photoinduced Crosslinking of Double-helical DNA by Psoralen Covalently Linked to a Triple Helix-forming Oligonucleotide under Near-physiological Conditions	Hong Li; Victoria J. Broughton-Head; Keith R. Fox; Tom Brown
1011-1014	Stereoselective Synthesis of 1′-Functionalized-4′-Thionucleosides	Lak Shin Jeong; Prashantha Gunaga; Hea Ok Kim; Dilip K. Tosh; Hyuk Woo Lee; Seung Ah Choe; Hyung Ryong Moon; Zhan-Guo Gao; Kenneth A. Jacobson; Moon Woo Chun
1015-1019	O²,1^′-Anhydro-(β -D-Psicofuranosyl)Thymine and 1-(1^′,4^′-O-Anhydro-β -D-Psicofuranosyl)Thymine: The Crystal Structures Versus the ¹H NMR and AB Initio Data	Jarkko Roivainen; Igor A. Mikhailopulo; Henning Eickmeier; Hans Reuter
1021-1024	Asymmetric Synthesis of Cyclopropyl-fused 2′-C-Methylcarbanucleosides as Potential Anti-HCV Agents	Lak Shin Jeong; Jeong A. Lee; Hea Ok Kim; Dilip K. Tosh; Hyung Ryong Moon; Seung-Jin Lee; Kang Man Lee; Yhun Y. Sheen; Moon Woo Chun
1025-1028	Syntheses of Pyrimidine Acyclic Nucleoside Phosphonates as Potent Inhibitors of Thymidine Phosphorylase (PD-ECGF) from SD-Lymphoma	Karel Pomeisl; Ivan Votruba; Antonín Holý; Radek Pohl
1029-1035	Diastereoselective Synthesis of 2′,3′-Dideoxy- β-C- Glucopyranosides as Intermediates for the Synthesis of 2′,3′-Dideoxy-β-D-Glucopyranosyl-C-Nucleosides	Michael Löpfe; Jay S. Siegel
1037-1042	Studies on Thermal Stability of Human Cytidine Deaminase	S. Vincenzetti; S. Pucciarelli; P. Mariani; G. De Sanctis; V. Polzonetti; P. Natalini; A. Vita
1043-1046	The Effects of Nucleoside Analogues on Promoter Methylation of Selected Tumor Suppressor Genes in MCF-7 and MDA-MB-231 Breast Cancer Cell Lines	B. Krawczyk; K. Rudnicka; K. Fabianowska-Majewska
1047-1050	ODN-Based Drugs for Targeting of Extracellular Proteins	E. M. Bucci; M. Valente; D. Musumeci; R. Sapio; V. Anrò; G. N. Roviello; M. Moccia
1051-1055	Novel S-Ribosylhomocysteine Analogues as Potential Inhibitors of LuxS Enzyme	Stanislaw F. Wnuk; Jennifer Lalama; Jenay Robert; Craig A. Garmendia
1057-1061	A New Family of Inhibitors of *Mycobacterium Tuberculosis* Thymidine Monophosphate Kinase	C. Gasse; V. Huteau; D. Douguet; H. Munier-Lehmann; S. Pochet

Volume 26, Issue 8-9 (2007)

1063-1066	Investigation of Novel Lipid-Functionalized PNA Monomers as Potential HIV-1 Non-Nucleoside Reverse Transcriptase and/or Integrase Inhibitors	Michael G. Thomas; Giovanni Maga; Jean-François Mouscadet; Nicola M. Howarth
1067-1071	Telomere Shortening in Human HL60 Cells by Treatment with 3′-Azido-2′,3′-Dideoxynucleosides and Telomerase Inhibition by Their 5′-Triphosphates	Xiaohong Liu; Motoko Inomata; Tsukasa Ogawara; Mineo Saneyoshi; Toyofumi Yamaguchi
1073-1077	Troxacitabine Prodrugs for Pancreatic Cancer	A. D. Adema; M. Radi; J. Daft; J. Narayanasamy; E. K. Hoebe; L. E. Alexander; C. K. Chu; G. J. Peters
1079-1082	Synthesis of Novel 2′-Deoxy Type Trans-3′,4′-Bridged Nucleic Acid	Tomohisa Osaki; Satoshi Obika; Yasuki Harada; Yasunori Mitsuoka; Kensaku Sugaya; Mitsuaki Sekiguchi; Somjing Roongjang; Takeshi Imanishi
1083-1086	Furano- and Pyrrolo [2,3-D] Pyrimidine Nucleosides and Their 5′-O-Triphospates: Synthesis and Enzymatic Activity	L. A. Alexandrova; M. A. Ivanov; L. S. Victorova; M. K. Kukhanova
1087-1093	Approach to the Synthesis of Natural and Modified Oligonucleotides by the Phosphotriester Method Using O-Nucleophilic Intramolecular Catalysis	Vladimir A. Efimov; Natalia S. Molchanova; Oksana G. Chakhmakhcheva
1095-1098	Glycosylation Reaction via a Mild and Efficient One-Pot Reaction Using Doped Natural Phosphate with Iodine as Catalyst	H. B. Lazrek; D. Ouzebla; L. Baddi; J. J. Vasseur
1099-1102	The Synthesis and Properties of Tricyclic Analogues of S⁶–MethylthioguanineandO⁶-Methylguanine	Ana R. Hornillo-Araujo; Adam J. M. Burrell; Miren K. Aiertza; Takayuki Shibata; David M. Hammond; Dolorès Edmont; Harry Adams; Geoffrey P. Margison; David M. Williams
1103-1106	A Glutaric Acid Ester as Carrier System for Sustained Delivery of Lamuvidine (3TC) Dimers	H. B. Lazrek; J. J. Vasseur; Jack Secrist III; Joachim W. Engels
1107-1110	Synthesis and Anti-HSV Activity of new N₁-Acyclic C₄ and C₆-Disubstituted Pyrazolo[3,4-D]Pyrimidine Nucleosides	Omar Moukha-chafiq; Mohamed Labd Taha; Abdelmalek Mouna
1111-1114	Stereospecific Synthesis of (-)-Neplanocin F	Sergio Rodriguez Ropero; Dolorès Edmont; Christophe Mathé; Christian Périgaud
1115-1119	Effect of Cationic Comb-Type Copolymer on Quadruplex Folding of Human Telomeric DNA	Naoki Makita; Sung Won Choi; Arihiro Kano; Asako Yamayoshi; Toshihiro Akaike; Atsushi Maruyama
1121-1124	Molecular Modelling Studies on the Binding of Some Protides to the Putative Human Phosphoramidase Hint1	C. Congiatu; A. Brancale; C. McGuigan
1125-1128	Revisited 3′-Deoxy-3′-C-Methyl-β-D-Ribonucleoside Series	Mohamed Aljarah; Sarah Couturier; Gilles Gosselin; Christophe Mathé; Christian Périgaud
1129-1132	Effect of Rubidium and Cesium Ions on the Dimeric Quaduplex formed by the Oxytricha Nova Telomeric Repeat Oligonucleotide D(GGGGTTTTGGGG)	Flaminia Cesare Marincola; Ada Virno; Antonio Randazzo; Adolfo Lai
1133-1137	Structural insight into the h TERT intron 6 sequence d(GGGGTGAAAGGGG) from ¹H-NMR study	Ada Virno; Luciano Mayol; Andres Ramos; Franca Fraternali; Bruno Pagano; Antonio Randazzo
1139-1143	Molecular Modelling Studies of Four Stranded Quadruplexes Containing A 3′-3′ or 5′-5′ Inversion of Polarity Site	Ada Virno; Francesco Zaccaria; Antonella Virgilio; Veronica Esposito; Aldo Galeone; Luciano Mayol; Antonio Randazzo
1145-1149	A Mini-Library of TBA Analogues Containing 3′-3′ and 5′-5′ Inversion of Polarity Sites	V. Esposito; A. Galeone; L. Mayol; A. Randazzo; A. Virgilio; A. Virno
1151-1154	Effect of the Introduction of an A-Residue into A Quadruplex Forming Oligonucleotide Containing A 5′-5′ Polarity of Inversion Site	A. Galeone; L. Mayol; A. Randazzo; A. Virgilio; A. Virno
1155-1159	A Topological Classification of G-Quadruplex Structures	V. Esposito; A. Galeone; L. Mayol; G. Oliviero; A. Virgilio; L. Randazzo

Volume 26, Issue 8-9 (2007)

1161-1165	Synthesis and Primary Evaluation of Novel HIV-1 Inhibitors	Yazan El Safadi; Roland Marquet; Anne-Marie Aubertin; Valérie Vivet-Boudou
1167-1172	The Support-on-Support Concept for In-Situ Oligonucleotide Synthesis on Nanoparticles	H. Seliger; M. Hinz; R. Ditz; M. Koch; P. Lapido; S. Margel
1173-1176	Thermodynamic Studies on PNA and PNA/DNA Dendrimer Formation	Maria Moccia; Domenica Musumeci; Margherita Valente; Giovanni N. Roviello; Roberto Sapio; Carlo Pedone; Enrico M. Bucci
1177-1180	Photochemically Induced RNA and DNA Abasic Sites	Pascal A. Küpfer; Christian J. Leumann
1181-1184	Cyclopentane-Nucleobase Coupling in the Synthesis of Carbocyclic L-Nucleosides: is A S_N2-Reaction an Alternative to the Mitsunobu-Reaction?	S. Jessel; E. Hense; C. Meier
1185-1188	Synthesis and Properties of Oligonucleotides Containing A 7-Membered (Oxepane) Sugar Ring	David Sabatino; Masad J. Damha
1189-1193	DNA Polymerase Recognition of 2′-Deoxy-2′-Fluoroarabinonucleoside 5′-Triphosphates (2′F-Arantps)	Chang G. Peng; Masad J. Damha
1195-1198	Introduction of Chirality into PNA By Replacement of the Achiral Methylene Carbonyl Linkage to the Nucleobase	Filip Wojciechowski; Robert H. E. Hudson
1199-1202	Synthesis of A Fluorescent PNA Monomer Containing 5-((9H-Fluoren-2-YL)Ethynyl)Uracil	Filip Wojciechowski; Robert H. E. Hudson
1203-1206	Synthesis of Modified Nucleosides for Incorporation of Formyletheno and Carboxyetheno Adducts of Adenine Nucleosides into Oligonucleotides	Niangoran Koissi; Harri Lönnberg
1207-1210	In Vitro Incorporation of LNA Nucleotides	Rakesh N. Veedu; Birte Vester; Jesper Wengel

Volume 26, Issue 6-7 (2007)

ix-xiv	PROCEEDINGS OF THE XVII INTERNATIONAL ROUNDTABLE
533-537	The 6-Methoxymethyl Derivative Of Pyrrolo-Dc For Selective Fluorometric Detection Of Guanosine-Containing Sequences	Robert H. E. Hudson; Arash Ghorbani Choghamarani
539-546	Synthesis and Biological Activity of Phosphonocarboxylate DNA	Christina M. Yamada; Douglas J. Dellinger; Marvin H. Caruthers
547-554	Synthetic Use Of Epoxy-Sugar Nucleosides	Hiromichi Tanaka; Yutaka Kubota; Shingo Takeda; Kazuhiro Haraguchi
555-558	Stabilization Of Multi-Stranded Nucleic Acid Structures Using 3″-S-Phosphorothiolate Linkages	Richard Cosstick; Joanne Buckingham; John Brazier; Julie Fisher
559-562	Florobenzene as Artificial Nucleobases-Base Pairing and Stacking Interactions	Aleksandra Živkovic; Joachim W. Engels
563-566	Some Novel Aminopropyl Nucleoside Phosphonates	Ding Zhou; Irene M. Lagoja; Arthur Van Aerschot
567-571	Reactions Of Malonaldehyde And Acetaldehyde With Calf Thymus Dna: Formation Of Conjugate Adducts	Donata Pluskota-Karwatka; Agnieszka J. Pawlowicz; Leif Kronberg
573-577	Synthesis And Anti-Hiv Activity Of Cyclic Pyrimidine Phosphonomethoxy Nucleosides And Their Prodrugs: A Comparison Of Phosphonates And Corresponding Nucleosides	Richard L. Mackman; Lijun Zhang; Vidya Prasad; Constantine G. Boojamra; James Chen; Janet Douglas; Deborah Grant; Genevieve Laflamme; Hon Hui; Choung U. Kim; Jay Parrish; Antitsa D. Stoycheva; Swami Swaminathan; KeYu Wang; Tomas Cihlar
579-583	In Vitro Anti-Malarial Activity Of N⁶-Modified Purine Analogs	Kathleen Too; Daniel M. Brown; David Loakes; Emily Bongard; Livia Vivas
585-588	Rearranging The Bicyclo[3.1.0]Hexane Template Of Carbocyclic Nucleosides To Improve Binding Recognition By Kinases	Victor E. Marquez; Maria J. Comin
589-595	Hydration Regulates The Thermodynamic Stability Of Dna Structures Under Molecular Crowding Conditions	Daisuke Miyoshi; Hisae Karimata; Naoki Sugimoto
597-601	Nucleosides And Oligonucleotides With Diynyl Side Chains: The Huisgen-Sharpless Cycloaddition “Click Reaction” Performed On Dna And Their Constituents	Frank Seela; Venkata Ramana Sirivolu
603-606	An Efficient Synthesis Of 7-Functionalized 7-Deazapurine β-D- Or β-L-Ribonucleosides: Glycosylation Of Pyrrolo[2,3-D]Pyrimidines With 1-O-Acetyl-2,3,5-Tri-O-Benzoyl-D-Or L-Ribofuranose	Xiaohua Peng; Frank Seela
607-610	Fluorinated 7-Deazapurine 2′-Deoxyribonucleosides: Modification At The Nucleobase And The Sugar Moiety	Frank Seela; Kuiying Xu; Padmaja Chittepu; Xin Ming
611-614	Foldamers Derived From Nucleoside β-Amino Acids: Pna Or Dna? Can We Have Both In One Place?	Richard Threlfall; Andrew Davies; Nicola Howarth; Richard Cosstick
615-619	Synthesis Of The Bicyclo-[4.3.0]-Thymidyl-Nucleoside Via Pd(Ii)-Mediated Ring Expansion Chemistry	Andrea Stauffiger; Christian J. Leumann
621-623	Efficient Synthesis Of Thymidine Boranophosphoramidates Conjugated With Amino Acids	Shoeb I. Khan; Barbara Ramsay Shaw
625-628	Novel Non-Nucleoside Human Cytomegalovirus Inhibitors Based Upon Tsao Nucleoside Derivatives: Structure-Activity Relationships	Sonia de Castro; Graziela Andrei; Robert Snoeck; Jan Balzarini; María-José Camarasa; Sonsoles Velázquez

Volume 26, Issue 6-7 (2007)

629-634	Methylation-Dependent Fragment Separation: Novel Analysis Of 5-Methyl Cytosine By Capillary Electrophoresis Of Amplified Dna Using Pcr Incorporation Of Chemically Modified Dctp	Victoria L. Boyd; Kristina I. Moody; Achim E. Karger; Kenneth J. Livak; Gerald Zon; John W. Burns
635-640	Discovery of ANA975: An Oral Prodrug of the TLR-7 Agonist Isatoribine	Alan X. Xiang; Stephen E. Webber; Bradley M. Kerr; Erik J. Rueden; Joseph R. Lennox; Gregory J. Haley; Tingmin Wang; John S. Ng; Mark R. Herbert; David L. Clark; Virginia N. Banh; Wei Li; Simon P. Fletcher; Kevin R. Steffy; Darian M. Bartkowski; Leonid I. Kirkovsky; Lisa A. Bauman; Devron R. Averett
641-644	Aryl-Containing Esters Of Triphosphoric Acid As Substrates Of Terminal Deoxynucleotidyl Transferase	A. L. Khandazhinskaya; E. S. Matyugina; L. A. Alexandrova; E. A. Shirokova; M. K. Kukhanova; M. V. Jasko
645-649	Selective Fluorescence Detection Of 8-Oxoguanosine With 8-Oxog-Clamp	Osamu Nakagawa; Sayaka Ono; Akira Tsujimoto; Zhichun Li; Shigeki Sasaki
651-654	Impdh As A Biological Probe For Rna Antiviral Drug Discovery: Synthesis, Enzymology, Molecular Docking, And Antiviral Activity Of New Ribonucleosides With Surrogate Bases	Vasu Nair; Xiaohui Ma; Qingning Shu; Fan Zhang; Vinod Uchil; Govardhan R. Cherukupalli
655-659	The Synthesis Of Epr Differentiable Spinlabels And Their Coupling To Uridine	Olga Frolow; Bela E. Bode; Joachim W. Engels
661-664	PNA Conjugated to High-Molecular Weight Poly(Ethylene Glycol): Synthesis and Properties	Gian Maria Bonora; Sara Drioli; Maurizio Ballico; Andrea Faccini; Roberto Corradini; Susanna Cogoi; Luigi Xodo
665-668	Biologically-Validated HIV Integrase Inhibitors with Nucleobase Scaffolds: Structure, Synthesis, Chemical Biology, Molecular Modeling, and Antiviral Activity	Vasu Nair; Vinod Uchil; Guochen Chi; Iwona Dams; Arthur Cox; Byung Seo
669-674	Biophysical Properties of Quadruplexes Containing Two or Three 8-Bromodeoxyguanosine Residues	Luigi Petraccone; Ida Duro; Antonio Randazzo; Ada Virno; Luciano Mayol; Concetta Giancola
675-679	Effect of the Incorporation of 2′-Deoxy-8-(Hydroxyl)Adenosine on the Stability of Quadruplexes Formed by Modified Human Telomeric DNA	Luigi Petraccone; Ida Duro; Eva Erra; Antonio Randazzo; Ada Virno; Concetta Giancola
681-685	Synthesis of New, Base-Modified PNA Monomers	Ferenc Sipos; Gyula Sági
687-690	Isonucleosides: Design and Synthesis of New Isomeric Nucleosides with Antiviral Potential	Vasu Nair; Dorota G. Piotrowska; Maurice Okello; Jean Vadakkan
691-694	Development Of An Antitumor Adenosine Analog, 3″-Ethynyladenosine	Yoshio Endo; Tohru Obata; Makoto Nomura; Masakazu Fukushima; Yuji Yamada; Akira Matsuda; Takuma Sasaki
695-699	7,5′-O-Dibenzylinosines: Synthesis and Studies on Their Conformational Properties	Elena Casanova; Leire Aguado; María-Luisa Jimeno; Federico Gago; María-José Camarasa; María-Jesús Pérez-Pérez
701-704	Transformation of D-(-)-Ribose into a Natural Product-Like Scaffold via a Lewis Acid Catalyzed Intramolecular Hetero-Diels-Alder Reaction	Roland Messer; Cyril A. Fuhrer; Robert Häner
705-708	Synthesis of DNA-Oligonucleotides Damaged by Arylamine-Modified 2′-Deoxyguanosine	N. Böge; Z. Szombati; C. Meier
709-712	Synthesis of 3′- S-Phosphorothiolate Oligonucleotides for their Potential Use in RNA Interference	James W. Gaynor; John Brazier; Rick Cosstick
713-716	Synthesis and Antitumor Activity of Fluorocyclopentenyl-Pyrimidines	Lak Shin Jeong; Long Xuan Zhao; Won Jun Choi; Shantanu Pal; Yeon Hee Park; Sang Kook Lee; Moon Woo Chun; Young B. Lee; Chang Ho Ahn; Hyung Ryong Moon
717-719	Synthesis of N⁶-Substituted 3′-Ureidoadenosine Derivatives as Highly Potent Agonists at the Mutant A₃ Adenosine Receptor	Lak Shin Jeong; Seung Ah Choe; Ae Yil Kim; Hea Ok Kim; Zhan-Guo Gao; Kenneth A. Jacobson; Moon Woo Chun; Hyung Ryong Moon
721-724	Asymmetric Synthesis of Novel Apio Carbocyclic Nucleoside Analogues as Potential Antiviral and Antitumor Agent	Lak Shin Jeong; Jeong A. Lee; Hyung Ryong Moon; Hea Ok Kim; Kang Man Lee; Hyun Joo Lee; Moon Woo Chun

Volume 26, Issue 6-7 (2007)

725-728	Synthesis And Anti-Hcv Activity Of 2″-β-Hydroxymethylated Nucleosides	Lak Shin Jeong; Byul Nae Yoo; Hea Ok Kim; Kang Man Lee; Hyung Ryong Moon
729-732	Stereoselective Synthesis Of Homo-Apioneplanocin A As Potential Inhibitor Of S-Adenosylhomocysteine Hydrolase	Moon Woo Chun; Hyuk Woo Lee; Jin-Hee Kim; Hea Ok Kim; Kang Man Lee; Shantanu Pal; Hyung Ryong Moon; Lak Shin Jeong
733-736	Synthesis Of Novel 4′-Modified Neplanocin A Analogues And Their Inhibitory Activity Against S-Adenosyl-L-l-Homocysteine Hydrolase	Hiroki Kumamoto; Kazuki Deguchi; Nonoko Takahashi; Hiromichi Tanaka; Yukio Kitade
737-741	7-Deaza-2′-Deoxyxanthosine: Nucleobase Protection and Base Pairing of Oligonucleotides	Khalil I. Shaikh; Peter Leonard; Frank Seela
743-746	In Search of New Inhibitors of HIV-1 Replication: Synthesis and Study of 1-(2′-Deoxy-β-D-Ribofuranosyl)-1,2,4-Triazole-3-Carboxamide as a Selective Viral Mutagenic Agent	V. Vivet-Boudou; J. -C. Paillart; A. Burger; R. Marquet
747-750	Comparative Studies of Tricyclo-DNA- and LNA-Containing Oligonucleotides as Inhibitors of HIV-1 Gene Expression	Gabriela Ivanova; Andrey Arzumanov; Michael J. Gait; Sandrine Reigadas; Jean-Jacques Toulmé; Marie-Line Andreola; Damian Ittig; Christian Leumann
751-754	Perylene Diimide–Oligonucleotide Conjugates Constructed by Click Chemistry	Alexey V. Ustinov; Veronika V. Dubnyakova; Vladimir A. Korshun
755-759	Ph-Dependent Assembly of DNA-Gold Nanoparticles Based on the i-Motif	Frank Seela; Simone Budow
761-765	Thermodynamic Analysis Of Quadruplex Dna-Drug Interaction	Bruno Pagano; Carlo A. Mattia; Ada Virno; Antonio Randazzo; Luciano Mayol; Concetta Giancola
767-772	5-Arylethynyl-2′-Deoxyuridines: Energy Transfer And Snp-Detection	Mikhail V. Skorobogatyi; Maksim V. Kvach; Marina A. Zhylinskaya; Dmitry G. Yarmolinsky; Vladimir A. Korshun; Vadim V. Shmanai
773-777	Some Novel Adenosine Mimics: Synthesis and Anticancer Potential against Cervical Cancer caused by Human Papilloma Virus	Sarika Sinha; Richa Srivastava; Bhupesh Prusty; B. C. Das; Ramendra K. Singh
779-783	Study of Different Copper (I) Catalysts for the “Click Chemistry” Approach to Carbanucleosides	Julie Broggi; Nicolas Joubert; Vincent Aucagne; Thomas Zevaco; Sabine Berteina-Raboin; Steve P. Nolan; Luigi A. Agrofoglio
785-794	Synthesis And Properties Of Oligonucleotides Containing A Cholesterol Thymidine Monomer	Adeline Durand; Tom Brown
795-798	Preparation Of 2′-Hydrazino Oligonucleotides And Their Reaction With Aldehydes And 1,3-Diketones	Timofei S. Zatsepin; Tatiana S. Oretskaya; Michael J. Gait; Dmitry A. Stetsenko
799-803	Development Of The Novel Drug Releasing System Triggered By Hybridization With Target Sequence	F. Nagatsugi; Shizuka Nakayama; Shigeki Sasaki
805-808	Lack Of Interferon (IFN) Response To T7 Transcribed pppG (n)(n = 2,3)-shRNA	Takuma Gondai; Kazuya Yamaguchi; Kahoko Hashimoto; Naoko Miyano-Kurosaki; Hiroshi Takaku
809-813	Reagents For The Selective Immobilization Of Oligonucleotides On Solid Supports	Maksim V. Kvach; Igor A. Prokhorenko; Alexey V. Ustinov; Sergei V. Gontarev; Vladimir A. Korshun; Vadim V. Shmanai
815-820	Suppression Of Hepatitis C Virus Core Protein By Short Hairpin Rna Expression Vectors In The Core Protein Expression Huh-7 Cells	Hitoshi Suzuki; Hiroyasu Kaneko; Nobushige Tamai; Kunitada Shimotohno; Naoko Miyano-Kurosaki; Hiroshi Takaku
821-825	Novel Method for the Synthesis of 2′ -Phosphorylated Oligonucleotides	Darya S. Novopashina; Olesya S. Totskaya; Maria I. Meschaninova; Dmitry A. Stetsenko; Alya G. Venyaminova
827-830	Intracellular Trapping of CycloSal-Pronucleotides by Enzymatic Cleavage	H. J. Jessen; V. Tonn; C. Meier

Volume 26, Issue 6-7 (2007)

831-834	New CycloAMB-Nucleoside Phosphonate Prodrugs	U. Görbig; J. Balzarini; C. Meier
835-839	An Alternative Synthetic Method for 4′-C-Ethynylstavudine by Means of Nucleophilic Substitution of 4′-Benzoyloxythymine Nucleoside	Kazuhiro Haraguchi; Masanori Sumino; Hiromichi Tanaka
841-847	Fluorescence studies of calf spleen purine nucleoside phosphorylase (PNP) complexes with guanine and 9-deazaguanine	Katarzyna Stępniak; Biserka Žinić; Jacek Wierzchowski; Agnieszka Bzowska
849-854	Interactions of Calf Spleen Purine Nucleoside Phosphorylase with Formycin B and its Aglycone—Spectroscopic and Kinetic Studies	Jacek Wierzchowski; Beata Iwańska; Agnieszka Bzowska; David Shugar
855-859	Cloning, Expression, Purification, and Some Properties of Calf Purine Nucleoside Phosphorylase	Katarzyna Stepniak; Agnieszka Girstun; Beata Wielgus-Kutrowska; Krzysztof Staroń; Agnieszka Bzowska
861-864	5-Diacetoxymethyl-cycloSal-d4TMP—A prototype of enzymatically activated cycloSal-pronucleotides	N. Gisch; J. Balzarini; C. Meier
865-868	Rnai Activity of Sirnas Modified with 2′-Aminoalkyl-Substituted Fluorinated Nucleobases	Jens Haas; Thea Mueller-Kuller; Stefan Klein; Joachim W. Engels

Volume 26, Issue 5 (2007)

413-421	Synthesis and Antiviral Evaluation of Azt Analogues with A Spacer Arm Between Glucidic and Base Moieties. Part II	Vincent Roy; Rachida Zerrouki; Pierre Krausz; Géraldine Laumond; Anne Marie Aubertin
423-435	Novel Regioselective Hydroxyl-Alkylation of 4,5-Diphenylimidazole-2-Thione and A Competitive Intramolecular Ring Closure of the S-Hydroxyalkyl-Imidazoles to Imidazo[2,1-b]Thiazines and Thiazoles. Role of Catalyst, Microwave Irradiation, and Solid Support	E. S. H. El Ashry; N. Rashed; L. F. Awad; E. Ramadan; S. M. Abdel-Maggeed; N. Rezki
437-451	Novel Regioselective Formation of S- and N-Hydroxyl-Alkyls of 5-(3-Chlorobenzo[b]Thien-2-yl)-3-Mercapto-4H-1,2,4-Triazole and A Facile Synthesis of Triazolo-Thiazoles and Thiazolo-Triazoles. Role of Catalyst and Microwave	E. S. H. El Ashry; A. A. Kassem; H. Abdel-Hamid; F. F. Louis; Sh. A. N. Khattab; M. R. Aouad
453-457	In Vitro Selection and Characterization of Human Immunodeficiency Virus Type 1 Resistant to Zidovudine and Tenofovir	S.-S. Park; S.-K. Hong; S.-G. Lee; J.-S. Yoon; W.-C. Yoo; S.-Y. Paik
459-471	Binding and Oxidative Cleavage Studies of DNA by Mixed Ligand Co(III) and Ni(II) Complexes of Quinolo [3,2-b]Benzodiazapine and 1,10-Phenanthroline	M. C. Prabhakara; H. S. Bhojya Naik; V. Krishna; H. M. Kumaraswamy
473-497	Improved Synthesis of Trinucleotide Phosphoramidites and Generation of Randomized Oligonucleotide Libraries	Andrey Yagodkin; Alex Azhayev; Jarkko Roivainen; Maxim Antopolsky; Alexei Kayushin; Maria Korosteleva; Anatoly Miroshnikov; John Randolph; Hugh Mackie
499-519	Design, Synthesis, and Antiviral Evaluation of Some 3′-Carboxymethyl-3′-Deoxyadenosine Derivatives	Matt A. Peterson; Pucheng Ke; Houguang Shi; Carl Jones; Brenda R. McDougall; W. Edward Robinson Jr.
521-531	Synthesis and Biophysical Studies on Fluorescently Labeled Oligodeoxyribonucleotides	Shipra Singh; Pradeep Kumar; K. C. Gupta; Ramendra K. Singh

Volume 26, Issue 4 (2007)

323-334	Synthesis of Novel Alkyl Triphosphates and Their Substrate Properties Toward Terminal Deoxynucleotidyltransferase	Maxim Jasko; Anastasiya Khandazhinskaya; Ludmila Alexandrova; Elena Shirokova; Alexander Ivanov; Marina Kukhanova
335-345	Synthesis and Biological Evaluation of Some α-[6-(1′-Carbamoylalkylthio)-1 H-Pyrazolo[3,4-D]Pyrimidin-4-yl]Thioalkylcarboxamide Acyclonucleosides	Omar Moukha-Chafiq; Mohamed Labd Taha; Abdelmalek Mouna; Hassan Bihi Lazrek; Jean-Jacques Vasseur; Erik De Clercq
347-359	Novel Simple Efficient Synthetic Approach Toward 6-Substituted-2H-[1,2,4]Triazolo[3,4-b][1,3,4]Thiadiazole-3-Thiones and First Synthesis and Biological Evaluation of N-and S-β-D-Glucosides of the[1,2,4]Triazolo [3,4-b][1,3,4]Thiadiazole Ring System	Nasser S. A. M. Khalil
361-377	First Synthesis And Antimicrobial Activity Of N- and S-α-L-Arabinopyranosyl-1,2,4-Triazoles	Nasser S. A. M. Khalil
379-390	Synthesis And Antimicrobial Activity Of Some Cyclic And Acyclic Nucleosides Of Thieno[2,3-d]Pyrimidines	Nasser A. Hassan; Mohamed I. Hegab; Aymn. E. Rashad; Afaf A. Fahmy; Farouk M. E. Abdel-Megeid
391-402	Synthesis Of 2,2,3-Tris(Hydroxymethyl)Methylenecyclopropane Analogues Of Nucleosides	Shaoman Zhou; Jiri Zemlicka
403-411	Short Synthesis And Antiviral Evaluation Of c-Fluoro-Branched Cyclopropyl Nucleosides	Chang Hyun Oh; Joon Hee Hong

Volume 26, Issue 3 (2007)

223-230	New AZT Analogues Having 5′-Alkylsulfonyl Groups: Synthesis and Anti-HIV Activity	Najim A. Al-Masoudi; Yaseen A. Al-Soud; Ibrahim A. I. Ali; Thilo Schuppler; Christoph Pannecouque; Erik De Clercq
231-243	Fluoroanalogues of Anti-Cytomegalovirus Agent Cyclopropavir: Synthesis and Antiviral Activity of (E)- and (Z)-9-{[2,2-Bis(Hydroxymethyl)-3-Fluorocyclopropylidene]Methyl}-Adenines and Guanines	Shaoman Zhou; Jiri Zemlicka; Earl R. Kern; John C. Drach
245-254	Preparation of Potential Cell-Permeant Nucleoside-2′,3′-Cyclic Phosphate Precursors	Simone Battaggia; Emma E. Smith; Joseph S. Vyle
255-258	Hypoxanthine-Guanine Phosphoribosyltransferase Deficiency: Biochemical and Molecular Findings in Six Argentine Patients	L. E. Laróvere; J. P. O'Neill; M. Randall; L. D. Fairbanks; N. Guelbert; L. Czornyj; R. Dodelson de Kremer
259-269	A Novel Universal Linker for Efficient Synthesis of Phosphorothioate Oligonucleotides	Zhiwei Wang; Phil Olsen; Vasulinga T. Ravikumar
271-275	The Fluoride Cleavable 2-(Cyanoethoxy)Methyl (CEM) Group as Reversible 3′-O-Terminator for DNA Sequencing-by-Synthesis—Synthesis, Incorporation, and Cleavage	A. Földesi; A. Keller; A. Stura; S. Zigmantas; M. Kwiatkowski; D. Knapp; J. W. Engels
277-290	Selective Photo-Cross-Linking of 2′-O-Psoralen-Conjugated Oligonucleotide with Rnas Having Point Mutations	Maiko Higuchi; Asako Yamayoshi; Takasei Yamaguchi; Reiko Iwase; Tetsuji Yamaoka; Akio Kobori; Akira Murakami
291-302	Racemic Synthesis and Antiviral Evaluation of 4′(α)-Hydroxymethyl and 6′(α)-Methyl Substituted Apiosyl Nucleosides	Aihong Kim; Joon Hee Hong
303-315	Noncovalent Interaction of G-Quadruplex DNA with Acridine at Low Concentration Monitored by MALDI-TOF Mass Spectrometry	Narayana Nagesh; Abburi Krishnaiah; Vishnu Mukund Dhople; Curum S. Sundaram; Medicharla V. Jagannadham
317-322	Application of Solid-Phase Chemistry for the Synthesis of 3′-Fluoro-3′-Deoxythymidine	Hitesh Kumar Agarwal; Keykavous Parang

Volume 26, Issue 2 (2007)

129-148	Reaction of Glycidamide with 2′-Deoxyadenosine and 2′-Deoxyguanosine—Mechanism for the Amide Hydrolysis	Josefin Backman; Leif Kronberg
149-159	N,N′-Bis-(2-(cyano)ethoxycarbonyl)-2-methyl-2-thiopseudourea: A Guanylating Reagent for Synthesis of 2′-O-[2-(Guanidinium)ethyl]-Modified Oligonucleotides	Thazha P. Prakash; Ask Püschl; Muthiah Manoharan
161-180	Molecular Recognition of Adenosine Deaminase: ¹⁵N NMR Studies	Avital Laxer; Hugo E. Gottlieb; Bilha Fischer
181-188	An Alternative Advantageous Protocol for Efficient Synthesis of Phosphorothioate Oligonucleotides Utilizing Phenylacetyl Disulfide (PADS)	R. Krishna Kumar; Phil Olsen; Vasulinga T. Ravikumar
189-204	Synthesis of 3’,5’-cyclic diguanylic acid (cdiGMP) Using 1-(4-chlorophenyl)-4-ethoxypiperidin-4-yl as a Protecting Group for 2’-hydroxy Functions of Ribonucleosides	Hongbin Yan; Aimé López Aguilar
205-222	The Chemical and Biochemical Properties of Methylphosphotriester DNA and RNA in Comparison with Their Corresponding Methylphosphonates. A Dynamic Model Description	Henk M. Buck

Volume 26, Issue 1 (2007)

1-8	Chemoselective Deprotection of α-Indole and Imidazole Ribonucleosides	Tilak Chandra; Kenneth L. Brown
9-22	Electrochemical Study on Behavior of EuMo₂ Complex and Its Interaction With DNA	Zhifeng Li; Jingwan Kang; Xiaoquan Lu
23-36	AZT 5′-Cholinephosphate as an Anti-HIV Agent: The Study of Biochemical Properties and Metabolic Transformations Using Its ³²P-Labelled Counterpart	Dmitry V. Yanvarev; Elena A. Shirokova; Maria V. Astapova; Yury S. Skoblov
37-43	Synthesis of 1,2,4-Triazole C-Nucleosides from Hydrazonyl Chlorides and Nitriles	Najim A. Al-Masoudi; Yaseen A. Al-Soud; Ibrahim A. I. Ali
45-49	Unusual β-Elimination of Carbocyclic Ketonucleosides Catalyzed by Silica Gel	Xiaozhen Liu; Xin Guo; Fei Wang; Guangqing Lei; Dongdong Luo
51-64	Synthesis and Antiviral Properties of Aza-Analogues of Acyclovir	Mariola Koszytkowska-Stawińska; Katarzyna Kaleta; Wojciech Sas; Erik De Clercq
65-82	Factors Influencing Dna Expansion in the Course of Polymerase Chain Reaction	Jitka Vondrušková; Nad'a Pařízková; Jaroslav Kypr
83-97	Synthesis and Biological Activity of 5′,9-Anhydro-3-Purine-ISONucleosides as Potential Anti-Hepatitis C Virus Agents	Byoung-Kwon Chun; Peiyuan Wang; Abdalla Hassan; Jinfa Du; Phillip M. Tharnish; Eisuke Murakami; Lieven Stuyver; Michael J. Otto; Raymond F. Schinazi; Kyoichi A. Watanabe
99-110	Characterization and Functional Analysis of the Promoter for the Human Equilibrative Nucleoside Transporter Gene, hENT1	Parween Abdulla; Imogen R. Coe
111-120	Synthesis of “Reversed” Methylenecyclopropane Analogues of Antiviral Phosphonates	Chengwei Li; Jiri Zemlicka
121-127	Deamination of 2′,3′-O-Isopropylideneadenosine-5′- Carboxylic Acid Catalyzed by Adenosine Deaminase (ADA) and Adenylate Deaminase (AMPDA): Influence of Substrate Ionization on the Activity of the Enzymes	Pierangela Ciuffreda; Laura Alessandrini; Radmila Pavlovic; Enzo Santaniello

Volume 25, Issue 12 (2006)

1309-1333	A Review: Synthesis of Aryl C-Glycosides Via the Heck Coupling Reaction	Kevin W. Wellington; Steven A. Benner
1335-1344	Synthesis and DNA Binding Properties of a New Benzo[f]Imidazo[1,5b]-Isoquinoline-Butan-1,2-Diol Derivative	Youssef L. Aly; Erik B. Pedersen
1345-1362	Oxidation Chemistry of Adenosine-3′, 5′-Cyclic Monophosphate at Pyrolytic Graphite Eletrode	Rajendra N. Goyal; Anuradha Tyagi
1363-1375	A proposal for a convenient notation for P-chiral nucleotide analogues. Part 2. Dinucleoside monophosphate analogues	Michal Sobkowski; Jacek Stawinski; Adam Kraszewski
1377-1389	A proposal for a convenient notation for P-chiral nucleotide analogues. Part 3. Compounds with one nucleoside residue and nonnucleosidic derivatives	Michal Sobkowski; Jacek Stawinski; Adam Kraszewski
1391-1397	Guanosine analog in the pyrido[2,3-d]pyrimidine ring system As a potential Toll-like receptor agonist	Guangyi Jin; Christina C. N. Wu; Dennis A. Carson; Howard B. Cottam
1399-1406	Synthesis and anti-HCMV activity of novel cyclopropyl phosphonic acid nucleosides	Aihong Kim; Joon Hee Hong; Chang Hyun Oh
1407-1424	A Simple Fluorescent Biosensor for Theophylline Based on its RNA Aptamer	C. J. Rankin; E. N. Fuller; K. H. Hamor; S. A. Gabarra; T. P. Shields
1425-1436	Action of Nucleosides and Nucleotides at 7 Transmembrane-Spanning Receptors	Kenneth A. Jacobson; Stefano Costanzi; Soo-Kyung Kim; Eunjoo Roh; Bhalchandra V. Joshi; Susanna Tchilibon; Heng T. Duong; Zhan-Guo Gao
1437	Erratum

Volume 25, Issue 9-11 (2006)

971-974	Purine and Pyrimidine Metabolism: a Firm Basis for a Transformed Society	G. J. Peters; E. A. Carrey; I. Šebesta
975-980	Thymidine Phosphorylase is Noncompetitively Inhibited by 5′-O-Trityl-Inosine (KIN59) and Related Compounds	S. Liekens; J. Balzarini; A. I. Hernández; E. De Clercq; E. M. Priego; M. J. Camarasa; M. J. Pérez-Pérez
981-986	Cellular Resistance Against Troxacitabine in Human Cell Lines and Pediatric Patient Acute Myeloid Leukemia Blast Cells	A. D. Adema; L. Zuurbier; K. Floor; I. Hubeek; G. J. L. Kaspers; F. Albertoni; G. J. Peters
987-990	Alterations of Mitochondrial DNA in CEM Cells Selected for Resistance Toward DDC Toxicity	M. Bjerke; M. Franco; M. Johansson; J. Balzarini; A. Karlsson
991-996	Catabolism of Pyrimidines in Yeast: A Tool to Understand Degradation of Anticancer Drugs	G. Andersen; A. Merico; O. Björnberg; B. Andersen; K. D. Schnackerz; D. Dobritzsch; J. Piškur; C. Compagno
997-1000	Study of the Efficacy of a Pronucleotide of 2-Chloro-2′-Deoxyadenosine in Deoxycytidine Kinase-Deficient Lymphoma Cells	F. Bontemps; C. Meier; A. Delacauw; J. Balzarini; C. Galmarini; E. Van Den Neste
1001-1007	Micro-Array Analysis of Resistance for Gemcitabine Results in Increased Expression of Ribonucleotide Reductase Subunits	K. Smid; A. M. Bergman; P. P. Eijk; G. Veerman; V. W. T. Ruiz van Haperen; P. van den Ijssel; B. Ylstra; G. J. Peters
1009-1012	Inhibition of the ERK Pathway Promotes Apoptosis Induced by 2-Chloro-2′-Deoxyadenosine in the B-Cell Leukemia Cell Line Eheb	C. Smal; S. Lisart; A. Ferrant; F. Bontemps; E. Van Den Neste
1013-1017	Antitumor Effects of 3,3′,4,4′,5,5′-Hexahydroxystilbene in hl-60 Human Promyelocytic Leukemia Cells	P. Saiko; Z. Horvath; M. Murias; N. Handler; W. Jaeger; T. Erker; M. Fritzer-Szekeres; T. Szekeres
1019-1024	Resveratrol, an Ingredient of Wine, Acts Synergistically with Ara-C and Tiazofurin in HL-60 Human Promyelocytic Leukemia Cells	Z. Horvath; P. Saiko; C. Illmer; S. Madlener; T. Hoechtl; W. Bauer; T. Erker; W. Jaeger; M. Fritzer-Szekeres; T. Szekeres
1025-1028	Studies on the Methylation Status of CpG Sequences Located in Promoters of Selected Tumour Suppressor Genes in Breast Cancer Cells	K. Fabianowska-Majewska; R. Kordek; B. Krawczyk
1029-1032	Alteration of DNA Methylation Status in K562 and MCF-7 Cancer Cell Lines by Nucleoside Analogues	B. Krawczyk; K. Fabianowska-Majewska
1033-1037	No Induction of Thiopurine Methyltransferase During Thiopurine Treatment in Inflammatory Bowel Disease	M. Lindqvist; U. Hindorf; S. Almer; P. Söderkvist; M. Ström; H. Hjortswang; C. Peterson
1039-1044	Impaired Transport as a Mechanism of Resistance to Thiopurines in Human T-Lymphoblastic Leukemia Cells	A. K. Fotoohi; M. Lindqvist; C. Peterson; F. Albertioni
1045-1049	Apically Sorted P2X7 Receptors Mediate Purinergic-Induced Pore Formation Preferentially in Apical Domains of the Plasma Membrane	X. Li; G. I. Gorodeski
1051-1054	The Novel Nucleotide 4KNTP, in High Concentrations in Erythrocytes of Renal Failure Children: a Comparison with Accumulation of Other Putative Precursors in the Plasma	E. A. Carrey; E. Synesiou; H. A. Simmonds; L. D. Fairbanks
1055-1064	Uric Acid and Renal Disease	J. Stewart Cameron
1065-1069	Hypoxanthine Effect on Equilibrative and Concentrative Adenosine Transport in Human Lymphocytes. Implications in the Phatogenesis of Lesch-Nyhan Syndrome	C. Prior; R. J. Torres; J. G. Puig
1071-1075	Familial Juvenile Hyperuricaemic Nephropathy is not Such a Rare Genetic Metabolic Purine Disease in Britain	H. A. Simmonds; J. S. Cameron; D. J. Goldsmith; L. D. Fairbanks; G. Venkat Raman
1077-1082	Efficacy and Safety of Allopurinol in Patients with the Lesch-Nyhan Syndrome and Partial Hypoxanthine- Phosphoribosyltransferase Deficiency: a Follow-up Study of 18 Spanish Patients	R. J. Torres; C. Prior; J. G. Puig
1083-1085	Effect of Beer Ingestion on the Plasma Concentrations and Urinary Excretion of Purine Bases: One-Month Study	Y. Moriwaki; T. Ka; S. Takahashi; Z. Tsutsumi; T. Yamamoto

Volume 25, Issue 9-11 (2006)

1087-1091	A Turkish Case with Molybdenum Cofactor Deficiency	K. Ichida; H. Ibrahim Aydin; M. Hosoyamada; H. Serap Kalkanoglu; A. Dursun; I. Ohno; T. Coskun; A. Tokatli; T. Shibasaki; T. Hosoya
1093-1098	Genetic Analysis of the First 4 Patients with β-Ureidopropionase Deficiency	A. B. P. van Kuilenburg; R. Meinsma; B. Assman; G. F. Hoffman; T. Voit; A. Ribes; I. Lorente; R. Busch; E. Mayatepek; N. G. G. M. Abeling; R. A. Wevers; F. Rutsch; A. H. van Gennip
1099-1102	A Neonate with Recurrent Vomiting and Generalized Hypotonia Diagnosed with a Deficiency of Dihydropyrimidine Dehydrogenase	W. Brussel; A. B. P. van Kuilenburg; P. M. W. Janssens
1103-1106	A Pivotal Role for β-Aminoisobutyric Acid and Oxidative Stress in Dihydropyrimidine Dehydrogenase Deficiency?	A. B. P. van Kuilenburg; A. E. M. Stroomer; N. G. G. M. Abeling; A. H. van Gennip
1107-1112	Adenosine Kinase from Rat Liver: New Biochemical Properties	R. Leoncini; D. Vannoni; A. Santoro; S. Giglioni; R. Carli; E. Marinello
1113-1117	cAMP Phosphodiesterase Activity Evaluation in Human Carcinoma of Salivary Glands	G. Spoto; M. della Malva; C. Rubini; M. Fioroni; A. Piattelli; E. Serra; M. Di Nicola; F. Santoleri
1119-1123	Ecto-5′-Nucleotidase (eN, CD73) is Coexpressed with Metastasis Promoting Antigens in Human Melanoma Cells	R. Sadej; J. Spychala; A. C. Skladanowski
1125-1128	Stimulatory Effects of Atorvastatin on Extracellular Nucleotide Degradation in Human Endothelial Cells	L. Osman; M. Amrani; C. Isley; M. H. Yacoub; R. T. Smolenski
1129-1132	Determination of ITPase Activity in Erythrocyte Lysates Obtained for Determination of Tpmt Activity	J. Bierau; J. A. Bakker; M. Lindhout; A. H. van Gennip
1133-1139	The Neuroleptic Chlorpromazine Inhibits the Cationic and Stimulates the Anionic Phospholipid Precursor Synthesis in Human Lymphocytes	M. Staub; A. Stenger; R. Sumeg; T. Spasokoukotskaja; L. D. Fairbanks; H. A. Simmonds; G. Keszler
1141-1146	Identification of Phosphorylation Sites on Human Deoxycytidine Kinase After Overexpression in Eucaryotic Cells	C. Smal; D. Vertommen; L. Bertrand; M. H. Rider; E. Van Den Neste; F. Bontemps
1147-1151	Deoxycytidine Kinase is Reversibly Phosphorylated in Normal Human Lymphocytes	G. Keszler; T. Spasokoukotskaja; M. Sasvári-Székely; S. Eriksson; M. Staub
1153-1158	Thymidine Kinase Diversity in Bacteria	M. P. B. Sandrini; A. R. Clausen; B. Munch-Petersen; J. Piškur
1159-1163	Thymidine Kinases in Archaea	A. R. Clausen; A. Matakos; M. P. B. Sandrini; J. Piškur
1165-1169	Purification and Characterization of Wild-Type and Mutant Tk1 Type Kinases From Caenorhabditis Elegans	T. Skovgaard; B. Munch-Petersen
1171-1175	The Role of Mitochondrial dNTP Levels in Cells with Reduced TK2 Activity	C. Desler; B. Munch-Petersen; L. J. Rasmussen
1177-1180	Enhanced Activity of Deoxycytidine Kinase After Pulsed Low Dose Rate and Single Dose Gamma Irradiation	J. Sigmond; J. Haveman; N. Castro Kreder; W. J. Loves; C. van Bree; N. A. Franken; G. J. Peters
1181-1184	Effects of Intracellular Calcium Chelation and Pifithrin-α on Deoxynucleotide Metabolism in Human Lymphocytes	T. Spasokoukotskaja; Z. Csapó; S. Virga; M. Sasvári-Székely; M. Staub; G. Keszler
1185-1188	Effect of C-Terminal of Human Cytosolic Thymidine Kinase (TK1) on in Vitro Stability and Enzymatic Properties	C. Zhu; L. S. Harlow; D. Berenstein; S. Munch-Petersen; B. Munch-Petersen
1189-1192	Substrate Specificity of Three Viral Thymidine Kinases (TK): Vaccinia Virus TK, Feline Herpesvirus TK, and Canine Herpesvirus TK	N. Solaroli; M. Johansson; J. Balzarini; A. Karlsson
1193-1196	Difference in Ki67 and Thymidylate Synthase Expression in Primary Tumour Compared with Metastatic Nodes in Breast Cancer Patients	A. Calascibetta; D. Cabibi; L. Rausa; F. Aragona; E. Barresi; A. Martorana; R. Sanguedolce

Volume 25, Issue 9-11 (2006)

1197-1200	Interacting Partners of M-PMV Nucleocapsid-DUTPase	V. Németh-Pongrácz; J. Snasel; M. Rumlova; I. Pichova; B. G. Vértessy
1201-1204	Cell Cycle Dependent Regulation of Deoxycytidine Kinase, Deoxyguanosine Kinase, and Cytosolic 5′-Nucleotidase I Activity in MOLT-4 Cells	A. Fyrberg; S. Mirzaee; K. Lotfi
1205-1209	Pharmacokinetic Modelling of [2-¹³C]Uracil Metabolism in Normal and DPD-Deficient Dogs	M. Inada; Y. Hirao; T. Koga; M. Itose; J. Kunizaki; T. Shimizu; H. Sato
1211-1214	Activity of Pyrimidine Degradation Enzymes in Normal Tissues	A. B. P. van Kuilenburg; H. van Lenthe; A. H. van Gennip
1215-1219	Evaluation of Uridine Metabolism in Human and Animal Spermatozoa	T. Niemeyer; C. Dietz; L. Fairbanks; I. Schroeder-Printzen; R. Henkel; M. Löeffler
1221-1224	Differences in Activities of the Enzymes Of Nucleotide Metabolism and its Implications for Cardiac Xenotransplantation	A. H. Y. Yuen; Z. Khalpey; M. Lavitrano; C. G. A. McGregor; K. K. Kalsi; M. H. Yacoub; R. T. Smolenski
1225-1232	Analysis of Deoxycytidine Accumulation in Gemcitabine Treated Patients	R. Honeywell; C. J. van Groeningen; A. C. Laan; E. Strocchi; R. Ruiter; G. Giaccone; G. J. Peters
1233-1236	Analysis of Intracellular Nucleotides by Capillary Electrophoresis–Mass Spectrometry	D. Friedecký; P. Bednář; M. Procházka; T. Adam
1237-1240	Synthesis and Mass Spectrometric Fragmentation Characteristics of Imidazole Ribosides–Analogs of Intermediates of Purine De Novo Synthetic Pathway	P. Vyskočilová; P. Hornik; D. Friedecký; P. Fryčák; K. Lemr; T. Adam
1241-1244	HPLC/Tandem Ion Trap Mass Detector Methods for Determination of Inosine Monophosphate Dehydrogenase (IMPDH) and Thiopurine Methyltransferase (TPMT)	K. Kalsi; A. M. Marinaki; M. H. Yacoub; R. T. Smolenski
1245-1249	Liquid Chromatographic/Mass Spectrometric Procedure for Measurement of NAD Catabolites in Human and Rat Plasma and Urine	E. M. Slominska; P. Adamski; M. Lipinski; J. Swierczynski; R. T. Smolenski
1251-1255	Analysis of Pyrimidine Synthesis De Novo Intermediates in Urine During Crisis of a Patient with Ornithine Transcarbamylase Deficiency	A. B. P. van Kuilenburg; B. T. van Maldegem; N. G. G. M. Abeling; F. A. Wijburg; M. Duran
1257-1260	Determination of 5-Fluorouracil in Plasma with HPLC-Tandem Mass Spectrometry	A. B. P. van Kuilenburg; H. van Lenthe; J. G. Maring; A. H. van Gennip
1261-1264	Determination of Thymidine Phosphorylase Activity in Human Blood Cells and Fibroblasts by a Nonradiochemical Assay Using Reversed-Phase High-Performance Liquid Chromatography	A. B. P. van Kuilenburg; L. Zoetekouw
1265-1270	5 ′-Amino-4-Imidazolecarboxamide Riboside Induces Apoptosis in Human Neuroblastoma Cells Via the Mitochondrial Pathway	M. Garcia-Gil; F. Bertini; R. Pesi; V. Voccoli; M. G. Tozzi; M. Camici
1271-1276	Endogenously Expressed Truncated P2X7 Receptor Lacking the C-Terminus is Preferentially Upregulated in Epithelial Cancer Cells and Fails to Mediate Ligand-Induced Pore Formation and Apoptosis	Y. H. Feng; X. Li; R. Zeng; G. I. Gorodeski
1277-1281	Purine Metabolism in B-Cell Lymphocytic Leukemia: A Microarray Approach	E. Marinello; F. Carlucci; F. Rosi; F. Floccari; D. Raspadori; A. Tabucchi
1283-1286	The Neuroprotective Adenosine-Activated Signal Transduction Pathway Involves Activation of Phospholipase C	A. Rogel; Y. Bromberg; O. Sperling; E. Zoref-Shani
1287-1290	Purine Metabolism and Clinical Status of Patients with Rheumatoid Arthritis Treated with Dipyridamole	C. M. Forrest; T. W. Stone; G. M. Mackay; L. Oxford; N. Stoy; G. Harman; L. G. Darlington
1291-1294	Purine Catabolism in Advanced Carotid Artery Plaque	C. Felici; I. Ciari; L. Terzuoli; B. Porcelli; C. Setacci; M. Giubbolini; E. Marinello
1295-1300	Familial Nephropathy Associated with Hyperuricemia in Spain: Our Experience with 3 Families Harbouring a UMOD Mutation	J. G. Puig; C. Prior; J. Martínez-Ara; R. J. Torres
1301-1304	Analysis of Excretion Fraction of Uric Acid	B. Stibůrková; E. Pospíšilová; S. Kmoch; I. Šebesta
1305-1308	An Unusual Cause of Renal Amyloidosis Secondary to Gout—the First Description of Familial Occurrence	Z. Vernerová; I. Rychlík; L. Brunerová; L. Dvořáková; A. Pavelková; I. Šebesta

Volume 25, Issue 8 (2006)

843-847	Synthesis of 2′-Amino-LNA Purine Nucleosides	Jacob Ravn; Christoph Rosenbohm; Signe M. Christensen; Troels Koch
849-860	Synthesis and Antiviral Activity of Some C₂-, C₄-, and C₆-Substituted Pyrazolo[3,4-D]Pyrimidine Acyclonucleosides with the Alkylating Chains of ACV, HBG, and ISO-DHPG	Omar Moukha-chafiq; Mohamed Labd Taha; Hassan Bihi Lazrek; Jean-Jacques Vasseur; Erik De Clercq
861-866	Boronated Thymidine Analogues for Boron Neutron Capture Therapy	B. T. S. Thirumamagal; Jayaseharan Johnsamuel; Guirec Y. Cosquer; Youngjoo Byun; Junhua Yan; Sureshbabu Narayanasamy; Werner Tjarks; Rolf F. Barth; Ashraf S. Al-Madhoun; Staffan Eriksson
867-870	Investigation of 1,3-Dipolar Cycloaddition Reactions of Unsaturated Nitrones in Ionic Liquids	M. Hornyák; Z. Kele; L. Kovács; P. Forgó; N. M. Howarth
871-878	Simple Synthesis and Anti-Hiv Activity of Novel 3′-Vinyl Branched Apiosyl Pyrimidine Nucleosides	Chang Hyun Oh; Jin Woo Kim; Joon Hee Hong
879-887	Simple Synthesis of Novel Acyclic (E)-Bromovinyl Nucleosides as Potential Antiviral Agents	Jin Woo Kim; Joon Hee Hong
889-907	Chemically Modified Short Interfering Hybrids (siHYBRIDS): Nanoimmunoliposome Delivery In Vitro and In Vivo for RNAi of HER-2	Richard I. Hogrefe; Alexandre V. Lebedev; Gerald Zon; Kathleen F. Pirollo; Antonina Rait; Qi Zhou; Wei Yu; Esther H. Chang
909-923	Trimethylguanosine Nucleoside Inhibits Cross-Linking Between Snurportin 1 and m₃G-CAPPED U1 snRNA	Diana Bahia; Anna Aviñó; Ramon Eritja; Edward Darzynkiewicz; Montserrat Bach-Elias
925-939	Synthesis of 2-Bromomethyl-3-Hydroxy-2-Hydroxymethyl-Propyl Pyrimidine and Theophylline Nucleosides Under Microwave Irradiation. Evaluation of Their Activity Against Hepatitis B Virus	E. S. H. El Ashry; N. Rashed; A. Abdel-Rahman; L. F. Awad; H. A. Rasheed
941-950	Synthesis and Antiviral Evaluation of Novel 5′-Norcarboacyclic Phosphonic Acid Nucleosides	Aihong Kim; Joon Hee Hong
951-968	Structure of the Biologically Relevant G-Quadruplex in The c-MYC Promoter	Danzhou Yang; Laurence H. Hurley
969	ERRATUM

Volume 25, Issue 7 (2006)

705-717	Synthesis of Poly d(G-C) Oligonucleotides	John P. Hachmann; Michal Lebl
719-734	A simple and efficient synthesis of puromycin, 2,2′-anhydro-pyrimidine nucleosides, cytidines and 2′,3′-anhydroadenosine from 3′,5′-O-sulfinyl Xylo-nucleosides	Ken-ichi Takatsuki; Sumito Ohgushi; Shigeo Kohmoto; Keiki Kishikawa; Makoto Yamamoto
735-745	Preparation of a Fludarabine Intermediate via Selective Alkylation of 2-Fluoroadenine	Brian E. Schulmeier; William R. Cantrell Jr.; William E. Bauta
747-764	Unique ³¹P Spectral Response to the Formation of a Specific Restriction Enzyme–DNA Complex	Cynthia M. Dupureur
765-770	Efficient Large-Scale Synthesis of 5′-O-Dimethoxytrityl-N⁴-Benzoyl-5-Methyl-2′-Deoxycytidine	Bruce S. Ross; Mingming Han; Vasulinga T. Ravikumar
771-784	The Influences of A Nitrogen Atom Position in Dinucleoside 2-,3-,4-Pyridylphosphonates on Fragmentation Patterns in Electrospray Ionization Multistage Tandem Mass Spectra	Sanhao Ji; Yong Ju; Hua Fu; Yufen Zhao; Tommy Johansson; Jacek Stawinski
785-793	Brief Communication: Stability and Catalytic Activity of Novel Circular DNAzymes	Georg Seifert; Tillmann Taube; Kriztina Paal; Hagen Graf von Einsiedel; Sven Wellmann; Günter Henze; Karl Seeger; Matthias Schroff; Burghardt Wittig
795-799	Silencing of HIV-1 Gene Expression by Sirnas in Transduced Cells	Masaaki Hayafune; Naoko Miyano-Kurosaki; Hiroshi Takaku; Wee-Sung Park
801-805	Inhibition of HCV Replication in HCV Replicon by shRNAs	Hiroyuki Hamazaki; Hitoshi Takahashi; Kunitada Shimotohno; Naoko Miyano-Kurosaki; Hiroshi Takaku
807-813	The Practical and Pedagogical Advantages of an Ambigraphic Nucleic Acid Notation	David A. Rozak
815-821	Effect of Microwave Irradiation on Phosphoramidite Couplings on Controlled Pore Glass	Peter Grünefeld; Clemens Richert
823-842	Characterization of the Aldehyde Reactive Probe Reaction with AP-Sites in DNA: Influence of AP-Lyase on Adduct Stability	Samuel E. Bennett; Joshua Kitner

Volume 25, Issue 4-6 (2006)

353-357	Introduction: A 70th Birthday Tribute to Eiko Ohtsuka	Hiroyuki Kamiya
359-367	Structural Studies of Heterochiral DNA/DNA, RNA/RNA, AND DNA/RNA Duplexes	Hidehito Urata; Hana Shimizu; Masao Akagi
369-382	Application of Microchip Electrophoresis in the Analysis of RNA Aptamer-Protein Interactions	Fumiko Nishikawa; Hidetoshi Arakawa; Satoshi Nishikawa
383-395	Solution Structure of a GAAG Tetraloop in Helix 6 of SRP RNA from Pyrococcus furiosus	Kiyoshi Okada; Mari Takahashi; Taiichi Sakamoto; Gota Kawai; Kouji Nakamura; Akio Kanai
397-416	A Novel Stable RNA Pentaloop that Interacts Specifically with A Motif Peptide of Lambda-N Protein	Junji Kawakami; Naoki Sugimoto; Hisanori Tokitoh; Yoshiatsu Tanabe
417-425	Structural Property of DNA That Migrates Faster in Gel Electrophoresis, as Deduced by CD Spectroscopy	Akimasa Matsugami; Keiko Tani; Kiyoshi Ouhashi; Seiichi Uesugi; Mitsunori Morita; Takashi Ohyama; Masato Katahira
427-437	Suppression of HIV-1 Replication by a Combination of Endonucleolytic Ribozymes (RNase P and tRNase ZL)	Masahiro Ikeda; Yuichiro Habu; Naoko Miyano-Kurosaki; Hiroshi Takaku
439-451	Recognition of Oxidized Thymine Base on the Single-Stranded DNA by Replication Protein A	Daisuke Irie; Akira Ono; Shunji Izuta
453-462	Conformational Changes of DNA by Photoirradiation of DNA-Bis(Zn^II-Cyclen)-Azobenzene Complex	Kenji Maie; Mitsunobu Nakamura; Kazushige Yamana
463-473	Segregation of Partly Melted DNA Molecules	Masahiko Shiraishi; Takao Sekiya
475-487	Synthesis and Hybridization Properties of Oligonucleotides Containing (2S,3R)-9-(2,3,4-Trihydroxybutyl)Adenine	Yoshihito Ueno; Shinji Ishihara; Yasutomo Ito; Yukio Kitade
489-501	Addition of an Extra Substrate Binding Site and Partial Destabilization of Stem Structures in HDV Ribozyme Give Rise to High Sequence-Specificity for its Target RNA	Tamaki Hori; Fei Guo; Seiichi Uesugi
503-521	Inhibition of VEGF mRNA by 2′-O,4′-C-Ethylene-Bridgednucleicacids (ENA®) Antisense Oligonucleotides and Their Influence on Off-Target Gene Expressions	Koji Morita; Koji Yamate; Shin-ichi Kurakata; Koji Abe; Kenji Watanabe; Makoto Koizumi; Takeshi Imanishi
523-538	Active Species for Ce(IV)-Induced Hydrolysis of Phosphodiester Linkage in cAMP AND DNA	Jun Sumaoka; Kenichiro Furuki; Yuki Kojima; Masahiko Shibata; Kimihiko Hirao; Naoya Takeda; Makoto Komiyama
539-551	Synthetic Nucleosides and Nucleotides. 43. Inhibition of Vertebrate Telomerases by Carbocyclic Oxetanocin G (C.OXT-G) Triphosphate Analogues and Influence of C.OXT-G Treatment on Telomere Length in Human HL60 Cells	Toyofumi Yamaguchi; Mineo Saneyoshi; Hazuki Takahashi; Sachiko Hirokawa; Rie Amano; Xiaohong Liu; Motoko Inomata; Tokumi Maruyama
553-560	Transient Expression of Drosophila melanogaster Deoxynucleoside Kinase Gene Enhances Cytotoxicity of Nucleoside Analogs	Hiroyuki Kamiya; Hiroshi Ochiai; Hideyoshi Harashima; Mana Ito; Akira Matsuda
561-582	Chemical Synthesis of Oligonucleotides Containing Damaged Bases for Biological Studies	Shigenori Iwai
583-599	Synthesis of Cyclic ADP-Carbocylcic-Xylose and its 3′′-O O -Methyl Analogue as Stable and Potent Ca²-Mobilizing Agents	Takashi Kudoh; Akira Matsuda; Satoshi Shuto; Takashi Murayama; Yasuo Ogawa
601-612	Synthesis and Duplex-Forming Property of Oligonucleotides Bearing a Novel Polyamine-Modified Intercalator at the Terminal or the Internal Position	Tomohisa Moriguchi; Hirokazu Sekiguchi; Makoto Tachibana; Kazuo Shinozuka

Volume 25, Issue 4-6 (2006)

613-624	NMR Spectroscopic Study of a DNA Duplex with Mercury-Mediated T-T Base Pairs	Yoshiyuki Tanaka; Hiroshi Yamaguchi; Shuji Oda; Yoshinori Kondo; Makoto Nomura; Chojiro Kojima; Akira Ono
625-634	Improved Industrial Syntheses of Penciclovir and Famciclovir Using N2-Acetyl-7-Benzylguanine and a Cyclic Side Chain Precursor	Takayoshi Torii; Keizo Yamashita; Mitsuhiko Kojima; Yumiko Suzuki; Toyoto Hijiya; Kunisuke Izawa
635-645	Apoptotic Effect of Ganciclovir on Primary Effusion Lymphoma Cells Infected with Kaposi's Sarcoma-Associated Herpesvirus	Masahiro Fujimuro; Hisanori Inoue; Yasuhiro Teishikata; Yuriko Ishida; Hideyoshi Yokosawa
647-654	Synthesis and Biological Properties of New Phosmidosine Analogs Having an N-Acylsulfamate Linkage	Haruhiko Taguchi; Akihiro Ohkubo; Mitsuo Sekine; Kohji Seio; Hideaki Kakeya; Hiroyuki Osada; Takuma Sasaki
655-665	Synthesis of 6-Arylthio Analogs of 2′,3′-Dideoxy-3′-Fluoroguanosine and Their Effect against Hepatitis B Virus Replication	Takayoshi Torii; Tomoyuki Onishi; Kunisuke Izawa; Tokumi Maruyama; Yosuke Demizu; Johan Neyts; Erik De Clercq
667-679	DNA-Binding Properties of the Antibody Specific for the Dewar Photoproduct of Thymidylyl-(3′′-5′′)-Thymidine	Hiroshi Morioka; Mikiko Kurihara; Hiroyuki Kobayashi; Kousuke Satou; Yasuo Komatsu; Makiyo Uchida; Eiko Ohtsuka; Takuya Torizawa; Koichi Kato; Ichio Shimada; Tsukasa Matsunaga; Osamu Nikaido
681-691	Comprehensive Search for DNA Polymerase in the Hyperthermophilic Archaeon, Pyrococcus furiosus	Sonoko Ishino; Yoshizumi Ishino
693-704	Crystal Structure of d(gcGXGAgc) with X = G: a Mutation at X is Possible to Occur in a Base-Intercalated Duplex for Multiplex Formation	Jiro Kondo; Tanashaya Ciengshin; Ella Czarina Magat Juan; Yoshiteru Sato; Kenta Mitomi; Satoru Shimizu; Akio Takénaka

Volume 25, Issue 3 (2006)

231-242	Comparison Between Properties Of 2′-O,4′-C-Ethylene-Bridged Nucleic Acid (Ena®) Phosphorothioate Oligonucleotides And N3′-P5′ Thiophosphoramidate Oligonucleotides	Makiko Horie; Koji Morita; Junko Kawakami; Osamu Ando; Makoto Koizumi; Shinya Tsutsumi
243-257	Synthesis and RT Inhibitory Activity Evaluation of New Pyrimidine-Based Seco-Nucleosides	Genaro Vargas; Iker S. Escalona; Magali Salas; Barbara Gordillo; Adolfo Sierra
259-278	Time And Concentration Dependence Of Fenton-Induced Oxidation Of dG	Carl Elovson Grey; Patrick Adlercreutz
279-287	The Photochemistry Of 5-BrdCpdC, dCp5-BrdCpdA, and dCp5-BrdCdT in Aqueous Solution	Yuan Gao; Yinsheng Wang
289-297	F-ara-AMP is a substrate of cytoplasmic 5′-nucleotidase II (cN-II): HPLC and NMR studies of enzymatic dephosphorylation	Lars P. Jordheim; Emeline Cros; Carlos M. Galmarini; Charles Dumontet; Anne-Sophie Bretonnet; Isabelle Krimm; Jean-Marc Lancelin; Marie-Claude Gagnieu
299-305	Synthesis of AZT analogues: 7-(3-azido-2hydroxypropyl)-, 7-(3-amino-2-hydroxypropyl)-, 7-(3-triazolyl-2-hydroxypropyl)theophyllines	El Sayed H. El Ashry; Adel Abdel-Rahman; Nagwa Rashed; Laila F. Awad; Hanaa A. Rasheed
307-314	An Efficient Process for Synthesis of 2′-O-methyl and 3′-O-methyl Guanosine from 2-aminoadenosine Using Diazomethane and the Catalyst Stannous Chloride	Anilkumar R. Kore; Gaurang Parmar; Srinu Reddy
315-323	Hydrolytic Stability of a Phosphate-Branched Oligonucleotide Incorporating a Ribonucleoside 3′-Phosphotriester Unit	Tuomas Lönnberg
325-335	Microwave-Assisted Organic Synthesis of 3-(D-gluco- Pentitol-1-Yl)-1H-1,2,4-Triazole	E. S. H. El Ashry; L. F. Awad; H. M. Abdel Hamid; A. I. Atta
337-340	An Industrial Process for Selective Synthesis of 7-methyl Guanosine 5′-Diphosphate: Versatile Synthon for Synthesis of mRNA Cap Analogues	Anilkumar R. Kore; Gaurang Parmar
341-350	Synthesis and antiviral evaluation of novel open-chain analogues of neplanocin A	Joon Hee Hong; So-Young Kim; Chang-Hyun Oh; Kyung Ho Yoo; Jung-Hyuck Cho Prof. Dr.
351-352	Erratum	Olga Adelfinskaya; Weidong Wu; V. Jo Davisson; Donald E. Bergstrom

Volume 25, Issue 2 (2006)

121-140	An Efficient Synthesis Of Acyclic N⁷- and N⁹-Adenine Nucleosides Via Alkylation With Secondary Carbon Electrophiles to Introduce Versatile Functional Groups At the C-1 Position of Acyclic Moiety	Pravin L. Kotian; V. Satish Kumar; Tsu-Hsing Lin; Yahya El-Kattan; Ajit Ghosh; Minwan Wu; Xiaogang Cheng; Shanta Bantia; Yarlagadda S. Babu; Pooran Chand
141-157	Synthesis of Potential Purinoceptor Antagonists: Application of P1-tBu Phosphazene Base for Alkylation of Adenine in Solution and on Solid Phase	Erki Enkvist; Gerda Raidaru; Asko Uri; Roshni Patel; Catherine Redick; José L. Boyer; Juhan Subbi; Indrek Tammiste
159-169	Application of 2-Amino-6-Vinylpurine As an Efficient Agent for Conjugation of Oligonucleotides	Monsur Ali; Fumi Nagatsugi; Shigeki Sasaki; Ryusuke Nakahara; Minoru Maeda
171-189	A method for finding optimal RNA secondary structures using a new entropy model (vsfold)	Wayne Dawson; Kazuya Fujiwara; Gota Kawai; Yasuhiro Futamura; Kenji Yamamoto
191-202	3′-Azido-3′-Deoxy-5′-O-Isonicotinoylthymidine: A Novel Antiretroviral Analog of Zidovudine. III. Solubility Studies	Silvina A. Teijeiro; Margarita C. Briñon
203-229	Synthesis, characterization, and biological properties of small branched RNA fragments containing chiral (R_p and S_p) 2′,5′-phosphorothioate linkages	Rawan Mourani; Masad J. Damha

Volume 25, Issue 1 (2006)

1-8	Simple Synthesis and Anti-HIV Activity of Novel Cyclopentene Phosphonate Nucleosides	Aihong Kim; Joon Hee Hong
9-15	Effects of a Modified Dye-Labeled Nucleotide Spacer Arm on Incorporation by Thermophilic DNA Polymerases	Christopher J. Lacenere; Neil K. Garg; Brian M. Stoltz; Stephen R. Quake
17-28	Synthesis and Antiviral Screening of Some Thieno[2,3-d]Pyrimidine Nucleosides	A. E. Rashad; M. A. Ali
29-35	Efficient Synthesis of [2-¹⁵N]Guanosine and 2′-Deoxy[2′-¹⁵N]Guanosine Derivatives Using N-(tert-Butyldimethylsilyl)[¹⁵N]Phthalimide as a ¹⁵N-Labeling Reagent	Kazuo Kamaike; Yoshihiro Kayama; Mitsuhisa Isobe; Etsuko Kawashima
37-54	New Azt Conjugates as Potent Anti-HIV Agents	Zhengqing You; Henry Joung Lee
55-60	Acyclic Pyrazolo[3,4-d]Pyrimidine Nucleoside as Potential Leishmaniostatic Agent	A. Hasan; M. Satyanarayana; A. Mishra; D. S. Bhakuni; Ram Pratap; A. Dube; P. Y. Guru
61-72	Solid-Phase Synthesis of 5′-Deoxy-5′-Amino-Clitocine Analogues	Chamakura V. N. S. Varaprasad; Qazi Habib; Haoyun An; Zhi Hong
73-87	Complexing Properties of Some Pyrimidines	Mamdouh S. Masoud; Sawsan S. Haggag; Ekram A. Khalil
89-107	Virologic and Enzymatic Studies Revealing the Mechanism of K65R- and Q151M-Associated HIV-1 Drug Resistance Towards Emtricitabine and Lamivudine	Joy Y. Feng; Florence T. Myrick; Nicolas A. Margot; Gilbert B. Mulamba; Laurence Rimsky; Katyna Borroto-Esoda; Boulbaba Selmi; Bruno Canard
109-117	Synthesis and Antiviral Evaluation of Novel 4′-Hydroxymethyl Branched Apiosyl Nucleosides	Jin Woo Kim; Joon Hee Hong
119	ERRATUM

Volume 24, Issue 10-12 (2005)

1387-1394	John A. Montgomery, March 29, 1924–May 24, 2004	Jack Secrist
1395-1415	John Montgomery's Legacy: Carbocyclic Adenosine Analogues as Sah Hydrolase Inhibitors with Broad-Spectrum Antiviral Activity	E. De Clercq
1417-1437	Design, Synthesis, and Antiviral Evaluation of Some Polyhalogenated Indole C-nucleosides	Jiong J. Chen; Yuan Wei; John D. Williams; John C. Drach; Leroy B. Townsend
1439-1447	Reaction of the 2′-Silyl and 2′-Stannyl Derivatives of 6-(Bromomethyl)Dimethylsilyl-1′,2′-Unsaturated Uridine Under Radical Conditions	Junko Ogamino; Hideaki Mizunuma; Hiroki Kumamoto; Kazuhiro Haraguchi; Hiromichi Tanaka
1449-1468	Synthetic Approaches to Nuclease-Resistant, Nonnatural Dinucleotides of Anti-Hiv Integrase Interest	Guochen Chi; Vasu Nair
1469-1484	Stereochemistry of Internucleotide Bond Formation by the H-Phosphonate Method. 1. Synthesis and ³¹P Nmr Analysis of 16 Diribonulceoside (3′-5′)-H-Phosphonates and the Corresponding Phosphorothioates	Michal Sobkowski; Jadwiga Jankowska; Adam Kraszewski; Jacek Stawinski
1485-1505	Oligonucleotides Containing Pyrazolo[3,4-d]Pyrimidines: 8-Aza-7-deazaadenines With Bulky Substituents in the 2- or 7-Position	Frank Seela; Anup M. Jawalekar; Lijuan Sun; Peter Leonard
1507-1517	Nucleoside Modification and Concerted Mutagenesis of the Human A³ Adenosine Receptor to Probe Interactions Between the 2-Position of Adenosine Analogs and Gln167 in the Second Extracellular Loop	Heng T. Duong; Zhan-Guo Gao; Kenneth A. Jacobson
1519-1530	Preference for Ribose Over Deoxyribose in Loop-Closing Base Pairs of Extra Stable Nucleic Acid Hairpins	Rami N. Hannoush; Masad J. Damha
1531-1542	Synthesis and Anti-Hcv Activity of N⁹, 5′-Cyclo-3-(β-D-Ribofuranosyl)-8-Azapurin-2-One Derivatives	Abdalla E. A. Hassan; Peiyuan Wang; Tamara McBrayer; Philip Tharnish; Lieven Stuyver; Michael J. Otto; Kyoichi A. Watanabe; Raymond F. Schinazi
1543-1568	Synthesis of 9-[1-(Substituted)-3-(phosphonomethoxy)propyl]adenine Derivatives as Possible Antiviral Agents	Minwan Wu; Yahya El-Kattan; Tsu-Hsing Lin; Ajit Ghosh; Satish Vadlakonda; Pravin L. Kotian; Yarlagadda S. Babu; Pooran Chand
1569-1585	Synthesis of 9-[1-(Substituted)-2-(Phosphonomethoxy)Ethyl]Adenine Derivatives as Possible Antiviral Agents	Minwan Wu; Yahya El-Kattan; Tsu-Hsing Lin; Ajit Ghosh; V. Satish Kumar; Pravin L. Kotian; Xiaogang Cheng; Shanta Bantia; Yarlagadda S. Babu; Pooran Chand
1587-1595	Synthesis of 9-[1-(1-Hydroxyethyl)-3-(Phosphonomethoxy)Propyl] Adenine and Prodrug as Possible Antiviral Agents	Ajit Ghosh; Yahya El-Kattan; Minwan Wu; Tsu-Hsing Lin; Satish Vadlakonda; Pravin L. Kotian; Yarlagadda S. Babu; Pooran Chand
1597-1611	Synthesis of N⁶-Substituted 9-[3-(Phosphonomethoxy)Propyl]Adenine Derivatives As Possible Antiviral Agents	Yahya El-Kattan; Tsu-Hsing Lin; Minwan Wu; V. Satish Kumar; Pravin L. Kotian; Ajit Ghosh; Xiaogang Cheng; Shanta Bantia; Yarlagadda S. Babu; Pooran Chand
1613-1626	Synthesis and Antiviral Activity of Some 2-Substituted 3-Formyl-and 3-Cyano-5,6-Dichloroindole Nucleosides	John D. Williams; John C. Drach; Leroy B. Townsend
1627-1633	Preparation of Nucleoside H-Phosphonoselenoate Monoesters Via the Phosphinate Approach	Martin Kullberg; Jacek Stawinsk
1635-1649	Synthetic Approaches to a Mononucleotide Prodrug of Cytarabine	R. Bazzanini; M. -H. Gouy; S. Peyrottes; G. Gosselin; C. Périgaud; S. Manfredini
1651-1664	2′,3′-Dideoxynucleoside 5′-β,γ-(Difluoromethylene) Triphosphates With α-P-Thio or α-P-Seleno Modifications: Synthesis and Their Inhibition of HIV-1 Reverse Transcriptase	Nicholas A. Boyle; Patrick Fagan; Jennifer L. Brooks; Marija Prhavc; John Lambert; P. Dan Cook
1665-1706	Nucleotides. LXXIV Synthesis of a-D-Arabino-oligonucleotides	Christoph Henke; Wolfgang Pfleiderer

Volume 24, Issue 10-12 (2005)

1707-1727	Synthesis and Anti-HIV Activity of β-D-3′-Azido-2′,3′-unsaturated Nucleosides and β-D-3′-Azido-3′-deoxyribofuranosylnucleosides	Srinivas Gadthula; Chung K. Chu; Raymond F. Schinazi
1729-1743	An Efficient Alternative Route To 3,6-Disubstituted-Furo[2,3-d]Pyrimidin-2-One Analogues	Zlatko Janeba; Noha Maklad; Morris J. Robins
1745-1761	The Middle to 3′ End of the Hiv-1 Vif Gene Sequence is Important for Vif Biological Activity and Could be Used for Antisense Oligonucleotide Targets	Jacob Samson Barn; Naoko Miyano-Kurosaki; Hiroshi Takaku; Kazuya Yamaguchi; Atsushi Sakamoto; Koichi Ishikawa; Naoki Yamamoto; Mubarak Osei-Kwasi; David Ofori-Adjei
1763-1774	Phosphoralaninate Pronucleotides of Pyrimidine Methylenecyclopropane Analogues of Nucleosides: Synthesis and Antiviral Activity	Amalraj Ambrose; Jiri Zemlicka; Earl R. Kern; John C. Drach; Elizabeth Gullen; Yung-Chi Cheng
1775-1788	A Novel Imidazole Nucleoside Containing a Diaminodihydro-S-triazine as a Substituent: Inhibitory Activity Against the West Nile Virus NTPase/Helicase	Ravi K. Ujjinamatada; Yankanagouda S. Agasimundin; Peng Zhang; Ramachandra S. Hosmane; Roman Schuessler; Peter Borowski; Kishna Kalicharran; Ali Fattom
1789-1800	Nucleosides and Nucleotides. 232. Synthesis of 2′-C-Methyl-4′-thiocytidine: Unexpected Anomerization of the 2′-Keto-4′-thionucleoside Precursor	Daisuke Kaga; Noriaki Minakawa; Akira Matsuda
1801-1815	Binding of G-Quadruplex-interactive Agents to Distinct G-Quadruplexes Induces Different Biological Effects in MiaPaCa Cells	Weijun Liu; Daekyu Sun; Laurence H. Hurley
1817-1830	Synthesis and Pharmacokinetic and Pharmacodynamic Evaluation of the Forodesine HCl Analog BCX-3040	Hollis S. Kezar III; J. Michael Kilpatrick; Deborah Phillips; Debbie Kellogg; Jianwen Zhang; Philip E. Morris Jr.
1831-1842	Synthesis of a Convenient Thymidine Glycol Phosphoramidite Monomer and Its Site-specific Incorporation into DNA Fragments	Didier Gasparutto; Sonia Cognet; Solveig Roussel; Jean Cadet
1843-1852	2′-MeO-RNA Containing Oligodeoxyribonucleotide Primers Can Prevent Template-independent Base Extension on Microarrays	Xiaodong Zhao
1853-1874	Synthesis and Application of Negatively Charged PNA Analogues	Vladimir A. Efimov; Oksana G. Chakhmakhcheva; Eric Wickstrom
1875-1884	Confocal-microscopy Studies of a Model Oligoribonucleotide HIV Inhibitor	Robyn M. Hyde; Keith Jensen; Jindrich Kopecek; Arthur D. Broom
1885-1894	Double-headed Acyclo C-Nucleoside Analogues. Functionalized 1,2-bis-(1,2,4-Triazol-3-yl)ethane-1,2-diol	A. H. Moustafa; R. A. Haggam; M. E. Younes; E. S. H. El Ashry
1895-1906	Synthesis and Biological Activity of 4′-Thio-L-xylofuranosyl Purine Nucleosides	Kamal N. Tiwari; Lea Messini; John A. Montgomery; John A. Secrist III
1907-1917	Suppression of Human Immunodeficiency Virus Type 1 (HIV-1) Replication by an HIV-1-dependent Double Locked Vector with the Cre/loxP System	Yuichiro Habu; Takashi Nagawa; Norihiko Matsumoto; Hiroaki Takeuchi; Naoko Miyano-Kurosaki; Hiroshi Takaku
1919-1945	Synthesis and Structural Analysis of Oxadiazole Carboxamide Deoxyribonucleoside Analogs	Olga Adelfinskaya; Weidong Wu; V. Jo Davisson; Donald E. Bergstrom
1947-1970	Solid-phase Parallel Synthesis of 4-β-D-Ribofuranosylpyrazolo[4,3-d]pyrimidine Nucleosides	Kanda S. Ramasamy; Roberto B. Amador; Qazi Habib; Frank Rong; Xiaogang Han; David Y. Li; Jingfan Huang; Zhi Hong; Haoyun An
1971-1996	Synthesis of 3-Aminoimidazo[4,5-c]pyrazole Nucleoside via the N-N Bond Formation Strategy as a [5:5] Fused Analog of Adenosine	Tun-Cheng Chien; David A. Berry; John C. Drach; Leroy B. Townsend
1997-2022	Pyrimidine and Purine Analogues, Effects on Cell Cycle Regulation and the Role of Cell Cycle Inhibitors to Enhance Their Cytotoxicity	Jennifer Sigmond; Godefridus J. Peters
2023-2027	Ribose-modified Mizoribine Analogues: Synthesis and Biological Evaluation	Palmarisa Franchetti; Michela Pasqualini; Loredana Cappellacci; Riccardo Petrelli; Patrizia Vita; Mario Grifantini; Hiremagalur N. Jayaram

Volume 24, Issue 9 (2005)

1277-1287	Synthesis of Novel α-l-Arabinopyranosides of β-Lactams with Potential Antimicrobial Activity	Nasser S. A. M. Khalil
1289-1292	Unusual Olefin Formation by PhSe-F trans-Elimination	Jinfa Du; Junxing Shi; Byoung-Kwon Chun; Ann Hobbs; Laurent Hollecker; Kyoichi A. Watanabe
1293-1299	Polysulfide Reagent in Solid-Phase Synthesis of Phosphorothioate Oligonucleotides: Greater than 99.8% Sulfurization Efficiency	Achim H. Krotz; Alice Hang; Dennis Gorman; Anthony N. Scozzari
1301-1307	A Proposal for a New Stereochemical Notation for P-Chiral Nucleotide Analogues and Related Compounds	Michal Sobkowski; Jacek Stawinski; Adam Kraszewski
1309-1323	Synthesis and Evaluation of RNA Transesterification Efficiency Using Stereospecific Serinol-Terpyridine Conjugates	William C. Putnam; James K. Bashkin
1325-1331	New and One Pot Chemoselective Synthesis of Nucleoside 5′-H-Phosphonate Diesters	Xin Guo; Peng Jiang; Hua Fu; Yuyang Jiang; Yufen Zhao
1333-1343	4-Aminometyl-3-Nitrobenzoic Acid—A Photocleavable Linker for Oligonucleotides Containing Combinatorial Libraries	Tatiana V. Abramova; Vladimir N. Silnikov
1345-1351	One-Pot Synthesis of TBMPS (bis [tert-Butyl)-1 Pyrenylmethyl-Silyl) Chloride as a Novel Fluorescent Silicon-Based Protecting Group for Protection of 5′-OH Nucleosides and Its Use as Purification Handle in Oligonucleotide Synthesis	Snehlata Tripathi; Krishna Misra; Yogesh S. Sanghvi
1353-1372	Synthesis of Some New 1,3/ or 1,4-Bis(Glucopyranosyl-1,2,4-Triazol-5-Ylthio)Propanes/ or Butanes as Potential Antimicrobial Agents	Ashraf A. Abbas; Nasser S. A. M. Khalil
1373-1385	Chemistry and Dynamics of Interaction of Nucleosides with Pentafluoropyridine	V. V. Litvak; I. Ya. Mainagashev; O. G. Bukhanets

Volume 24, Issue 8 (2005)

1147-1165	Regioselective Glycosylation: Synthesis of α-Indoline Nucleosides	Kenneth L. Brown; Tilak Chandra; Shawn Zou; Edward J. Valente
1167-1185	Zwitterionic Oligonucleotides: A Study on Binding Properties of 2′-O-Aminohexyl Modifications	Christian R. Noe; Johannes Winkler; Ernst Urban; Matthias Gilbert; Georg Haberhauer; Helmut Brunar
1187-1197	Synthesis of Phosphonate Analogues of the Antiviral Cyclopropane Nucleoside A-5021	Tomoyuki Onishi; Takaaki Sekiyama; Takashi Tsuji
1199-1208	Crystal Structure and Conformation of 8-(2-Hydroxyethylamino) and 8-(Pyrrolidin-1-yl) Adenosines	S. Belyakov; E. Alksnis; V. Muravenko; I. Turovskis; J. Popelis; E. Lukevics
1209-1214	N⁴-Hydroxycytosine Dioxolane Nucleosides and Their Activity Against Hepatitis B Virus	Jinfa Du; Laurent Hollecker; Junxing Shi; Byoung-Kwon Chun; Kyoichi A. Watanabe; Raymond F. Schinazi; Tammy Y. Nachman; Stefania Lostia; Lieven J. Stuyver; Michael J. Otto
1215-1225	Formation of Au(III)-DNA Coordinate Complex by Laser Ablation of Au Nanoparticles in Solution	Yoshihiro Takeda; Tamotsu Kondow; Fumitaka Mafuné
1227-1247	New Trends in Synthesis of Pyrazole Nucleosides as New Antimetabolites	Galal H. Elgemeie; Wafaa A. Zaghary; Kamelia M. Amin; Tamer M. Nasr
1249-1263	New Acyclonucleosides: Synthesis and Anti-HIV Activity	Amel Hadj-Bouazza; Rachida Zerrouki; Pierre Krausz; Géraldine Laumond; Anne Marie Aubertin; Yves Champavier
1265-1276	Synthesis of Novel Acyclonucleosides Analogs of Pyridothienopyrimidine as Antiviral Agents	Farag A. El-Essawy

Volume 24, Issue 5-7 (2005)

305-318	Zebularine: A Unique Molecule for an Epigenetically Based Strategy in Cancer Chemotherapy. The Magic of its Chemistry and Biology	Victor E. Marquez; Joseph J. Barchi Jr.; James A. Kelley; Kambhampati V. R. Rao; Riad Agbaria; Tsipi Ben-Kasus; Jonathan C. Cheng; Christine B. Yoo; Peter A. Jones
319-329	Synthesis of Complex Nucleoside Antibiotics	Satoshi Ichikawa; A. Matsuda
331-341	Antiviral Potential of a New Generation of Acyclic Nucleoside Phosphonates, the 6-[2-(Phosphonomethoxy)Alkoxy]-2,4-Diaminopyrimidines	Erik De Clercq; G. Andrei; J. Balzarini; P. Leyssen; L. Naesens; J. Neyts; C. Pannecouque; R. Snoeck; C. Ying; D. Hocková; A. Holý
343-347	A New Approach to the Synthesis of 4′-Carbon-Substituted Nucleosides: Development of a Highly Active Anti-HIV Agent 2′, 3′-Didehydro-3′-Deoxy-4′-Ethynylthymidine	Kazuhiro Haraguchi; Shingo Takeda; Masanori Sumino; Hiromichi Tanaka; Ginger E. Dutschman; Yung-Chi Cheng; Takao Nitanda; Masanori Baba
349-352	Ring-Closing Metathesis Reactions in Nucleic Acid Chemistry—Cyclic Dinucleotides for Targeting Secondary Nucleic Acid Structures	Poul Nielsen; Philip Børsting
353-357	Developing Synthetic Methods for Bioactive Phosphorus Compounds Using H-Phosphonate Chemistry: A Progress Report	Tommy Johansson; Johan Nilsson; Martin Kullberg; Gaston Lavén; Michal Sobkowski; Agnieszka Szymanska; Marzena Szymczak; Adam Kraszewski; Jacek Stawinski
359-366	A Nano-Circular Single-Stranded DNA as a Novel Tool for SNPs Detection	Tatsuo Ohmichi; Aki Takashima; Naoki Sugimoto
367-373	6-Substituted 5-Fluorouracil Derivatives as Transition State Analogue Inhibitors of Thymidine Phosphorylase	Thomas I. Kalman; Li Lai
375-381	Liver Targeting of Hepatitis-B Antiviral Lamivudine Using the HepDirect™ Prodrug Technology	K. Raja Reddy; Timothy J. Colby; James M. Fujitaki; Paul D. van Poelje; Mark D. Erion
383-385	Synthesis and Study of Conformationally Restricted 3′-Deoxy-3′,4′-Exo-Methylene Nucleoside Analogues	Julien Gagneron; Gilles Gosselin; Christophe Mathé
387-392	Design and Evaluation of 5′-Modified Nucleoside Analogs as Prodrugs for an E. coli Purine Nucleoside Phosphorylase Mutant	William B. Parker; Paula W. Allan; Steve E. Ealick; Eric J. Sorscher; Abdalla E. A. Hassan; A. V. Silamkoti; Anita T. Fowler; William R. Waud; John A. Secrist III
393-396	Antiviral Activity of Steric-Block Oligonucleotides Targeting the HIV-1 Trans-Activation Response and Packaging Signal Stem-Loop RNAs	Douglas Brown; Andrey A. Arzumanov; John J. Turner; Dmitry A. Stetsenko; Andrew M. L. Lever; Michael J. Gait
397-400	Synthesis and Biological Evaluation of Conformationally Restricted and Nucleobase-Modified Analogs of the Anticancer Compound 3′-C-Ethynylcytidine (ECYD)	Patrick J. Hrdlicka; Jan S. Jepsen; Jesper Wengel
401-408	Terminal Phosphate Labeled Nucleotides: Synthesis, Applications, and Linker Effect on Incorporation by DNA Polymerases	Shiv Kumar; Anup Sood; Jeffery Wegener; Patrick J. Finn; Satyam Nampalli; John R. Nelson; Anuradha Sekher; Paul Mitsis; John Macklin; Carl W. Fuller
409-414	Synthesis of Novel Peptide Nucleic Acid-Peptide Chimera for Non-Invasive Imaging of Cancer	A. Chakrabarti; M. R. Aruva; S. P. Sajankila; M. L. Thakur; Eric Wickstrom
415-418	Ring Opening Reactions: Synthesis of AICAR Analogs as Potential Antimetabolite Agents	S. Costanzi; C. Lambertucci; F. R. Portino; R. Volpini; S. Vittori; G. Cristalli
419-422	Borano-Nucleotides: New Analogues to Circumvent HIV-1 RT-Mediated Nucleoside Drug-Resistance	Karine Alvarez; Jérôme Deval; Boulbaba Selmi; Karine Barral; Joelle Boretto; Catherine Guerreiro; Laurence Mulard; Robert Sarfati; Bruno Canard
423-426	Synthesis of Novel Polydiamidopropanoate Dendrimer PNA-Peptide Chimeras for Non-Invasive Magnetic Resonance Imaging of Cancer	N. V. Amirkhanov; Eric Wickstrom
427-429	Microwave Irradiation for Accelerating the Synthesis of Acyclonucleosides of 1,2,4-Triazole	E. S. H. El Ashry; L. F. Awad; H. M. Abdel Hamid; A. I. Atta
431-434	Lentiviral-Mediated Delivery of Combined HIV-1 Decoy TAR and Vif siRNA as a Single 1RNA Molecule that Cleaves to Inhibit HIV-1 in Transduced Cells	Jacob Samson Barnor; Naoko Miyano-Kurosaki; Kazuya Yamaguchi; Yusuke Abumi; Koichi Ishikawa; Naoki Yamamoto; Hiroshi Takaku
435-441	E. coli RNase HI and the Phosphonate-DNA/RNA Hybrid: Molecular Dynamics Simulations	I. Barvík Jr.
443-446	A Bunch-Oligonucleotide Forming Stable Monomolecular Quadruplex Containing a T-TETRAD	Nicola Borbone; Giorgia Oliviero; Aldo Galeone; Gennaro Piccialli; Michela Varra; Luciano Mayol
447-450	Effects of Acrolein on the Quadruplex Forming d(TTAGGG)₄ Telomeric Repeat Sequence	Nicola Borbone; Giuliana D'Isa; Giorgia Oliviero; Gennaro Piccialli; Michela Varra; Luciano Mayol
451-454	Phosphate Shielding Under Different Conditions Results in an Enhanced DNA Duplex Stability	H. M. Buck
455-458	The Role of the Carboxamide Group in Nicotinamide Adenine Dinucleotide in Relation to Hydride Transfer: The Reduced Form of the Dinucleotide as Remedy in the Modulation of Neurotransmission	H. M. Buck
459-464	Spectroscopic and Kinetic Studies of Interactions of Calf Spleen Purine Nucleoside Phosphorylase with 8-Azaguanine, and Its 9-(2-Phosphonylmethoxyethyl) Derivative	Jacek Wierzchowski; Katarzyna Stępniak; Agnieszka Bzowska; David Shugar
465-469	Kinetic Model of Oxidation Catalyzed by Xanthine Oxidase—The Final Enzyme in Degradation of Purine Nucleosides and Nucleotides	Kinga Banach; Elżbieta Bojarska; Zygmunt Kazimierczuk; Lucyna Magnowska; Agnieszka Bzowska
471-476	Kinetic Properties of Cellulomonas sp. Purine Nucleoside Phosphorylase with Typical and Non-Typical Substrates: Implications for the Reaction Mechanism	Beata Wielgus-Kutrowska; Agnieszka Bzowska
477-479	Synthesis and Biological Evaluation of NAD Analogs as Human Pyridine Nucleotide Adenylyltransferase Inhibitors	Palmarisa Franchetti; R. Petrelli; L. Cappellacci; M. Pasqualini; P. Vita; L. Sorci; F. Mazzola; N. Raffaelli; Giulio Magni

Volume 24, Issue 5-7 (2005)

481-484	Design and Synthesis of Specific Inhibitors of the 3′-Processing Step of HIV-1 Integrase	Guochen Chi; Byung I. Seo; Vasu Nair
485-489	Naphthyl Phosphoramidate Derivatives of BVdU as Potential Anticancer Agents: Design, Synthesis and Biological Evaluation	C. Congiatu; C. McGuigan; W. G. Jiang; G. Davies; M. D. Mason
491-495	Control of DNA Conformation Using 3′-S-Phosphorothiolate-Modified Linkages	Joanne Buckingham; Ghalia Sabbagh; John Brazier; Julie Fisher; Rick Cosstick
497-501	Targeted Therapy of Respiratory Syncytial Virus by 2_5A Antisense	Hagen Cramer; James R. Okicki; Mei Kuang; Zan Xu
503-506	New Affinity Resin for Purification of Cap-Binding Proteins	Marzena Jankowska-Anyszka; Maciej Nogalski; Edward Darzynkiewicz
507-511	Deaggregation of eIF4E Induced by mRNA 5′ Cap Binding	Anna Niedzwiecka; Edward Darzynkiewicz; Ryszard Stolarski
513-518	Chemical Synthesis of the Novel Ca² Messenger NAADP	James Dowden; Richard S. Brown; Christelle Moreau; Antony Galione; Barry V. L. Potter
519-522	Novel Cyclosal Nucleotides with Reduced Inhibitory Potency Toward Human Butyrylcholinesterase	C. Ducho; S. Jessel; N. Gisch; J. Balzarini; C. Meier
523-525	Homo and Heterodimers of ddI, d4T and AZT: Influence of (5′-5′) Thiolcabonate-Carbamate Linkage on Anti-HIV Activity	M. Taourirte; H. B. Lazrek; A. Rochdi; J. J. Vasseur; J. W. Engels
527-531	3′-Modified Oligo(2′-O-Methylribonucleotides) as Improved Probes for Hybridization with RNA	D. S. Novopashina; O. S. Totskaya; A. A. Lomzov; A. G. Venyaminova
533-537	Chemical and Enzymatic Synthesis of 4′-Thio-β-d-Arabinofuranosylcytosine Monophosphate and Triphosphate	A. S. Fowler; K. N. Tiwari; S. R. Campbell; J. A. Secrist III
539-543	Synthesis and Structural Study of Quadruplex Structures Containing 2′-Deoxy-8-Methyladenosine	Antonio Randazzo; Veronica Esposito; Aldo Galeone; Michela Varra; Antonella Virgilio; Luciano Mayol
545-552	Epoxide Adducts at the Guanine Residue Within Single-Stranded DNA Chains: Reactivity and Stability Studies	Didier Gasparutto; T. Michel; T. Ramirez-Fuentes; C. Saint-Pierre; J. Cadet
553-555	Phosphoramidate Derivatives of 2′,5′-Dideoxyadenosine as Potential Inhibitors of the EDHF Phenomenon	F. Gavazza; F. Daverio; A. T. Chaytor; T. M. Griffith; C. McGuigan
557-569	Synthesis and Antitumor Activity of 5-Bromo-1-Mesyluracil	Ljubica Glavaš-Obrovac; Ivan Karner; Marina Pavlak; Marko Radačić; Jelena Kašnar-Šamprec; Biserka Žinić
571-575	Synthesis and Fluorescent Properties of the Tricyclic Analogues of Acyclovir Linked with Nitrogen Hetbrocyclic Units	Tomasz Goslinski; Piotr Januszczyk; Grazyna Wenska; Bozenna Golankiewicz; Erik De Clercq; Jan Balzarini
577-580	Synthesis of 2′-C-Methyl-4′-Thio Ribonucleosides	D. Dukhan; E. Bosc; J. Peyronnet; R. Storer; G. Gosselin
581-584	A Direct Synthesis of Pyrrolocytosine from 5-Iodocytosine	R. H. E. Hudson; A. K. Dambenieks; R. D. Viirre
585-588	A Solid Support with a Hydroxyallyl Linker, Full Parts of Which are Potentially Reusable for the Synthesis of Oligonucleotides	Mamoru Hyodo; Mari Morimura; Yoshihiro Hayakawa
589-593	Synthesis and Enzymatic Characterization of Methylene Analogs of Adenosine 5′-Tetraphosphate (p₄A)	Jacek Jemielity; Malgorzata Pietrowska-Borek; Elzbieta Starzynska; Joanna Kowalska; Ryszard Stolarski; Andrzej Guranowski; Edward Darzynkiewicz
595-600	Synthesis and Properties of mRNA Cap Analogs Containing Phosphorothioate Moiety in 5′,5′-Triphosphate Chain	Joanna Kowalska; Magdalena Lewdorowicz; Joanna Zuberek; Elzbieta Bojarska; Jacek Wojcik; Lean S. Cohen; Richard E. Davis; Janusz Stepinski; Ryszard Stolarski; Edward Darzynkiewicz; Jacek Jemielity
601-605	A Novel Approach to Solid Phase Chemical Synthesis of Oligonucleotide mRNA Cap Analogs	Jacek Jemielity; Petri Heinonen; Harri Lönnberg; Edward Darzynkiewicz
607-609	d-4′-Thioadenosine Derivatives as Highly Potent and Selective Agonists at the Human A₃ Adenosine Receptor	Hyouk Woo Lee; Dae Hong Shin; Ji Young Jung; Hea Ok Kim; Moon Woo Chun; N. Melman; Z. -G. Gao; Kenneth A. Jacobson; Lak Shin Jeong
611-613	Stereoselective Synthesis of 3-Hydroxymethyl-d-Cyclopentenone, the Versatile Intermediate for the Synthesis of Carbocyclic Nucleosides	Won Jun Choi; Hyung Ryong Moon; Hea Ok Kim; Young Mi Ko; Hye Jin Kim; Jeong A. Lee; Kang Man Lee; Mi Kyung Yun; Dae Hong Shin; Moon Woo Chun; Yhun Y. Sheen; Kilhyoun Kim; Lak Shin Jeong
615-621	Synthesis and Biochemical Properties of Novel mRNA 5′ Cap Analogs Resistant to Enzymatic Hydrolysis	Marcin Kalek; Jacek Jemielity; Ewa Grudzien; Joanna Zuberek; Elzbieta Bojarska; Lean S. Cohen; Janusz Stepinski; Ryszard Stolarski; Richard E. Davis; Robert E. Rhoads; Edward Darzynkiewicz
623-627	Microwaves Synthesis of Solid Supports for the Synthesis of 3′-Aminoalkyl Oligodeoxynucleotides	Charles Goussu; Jean-Jacques Vasseur; Hervé Bazin; François Morvan
629-633	Novel Dinucleoside 5′,5′-Triphosphate Cap Analogues. Synthesis and Affinity for Murine Translation Factor eIF4E	Janusz Stepinski; Joanna Zuberek; Jacek Jemielity; Marcin Kalek; Ryszard Stolarski; Edward Darzynkiewicz
635-638	Combination of Poly(l-Lysine)-Graft-Dextran Copolymer and 2′-O,4′-C-Methylene Bridged Nucleic Acid (2′,4′-BNA) Modification Synergistically Stabilizes Pyrimidine Motif Triplex at Neutral PH	Hidetaka Torigoe; Takuma Katayama; Satoshi Obika; Atushi Maruyama; Takeshi Imanishi
639-641	Synthesis and Biological Evaluation of N- and O-Alkylated Bicyclic Furanopyrimidines as Non-Nucleosidic Inhibitors of Human Cytomegalovirus	M. R. Kelleher; C. McGuigan; G. Andrei; R. Snoeck; E. De Clercq; J. Balzarini
643-645	The Journey Towards Elucidating the Anti-HCMV Activity of Alkylated Bicyclic Furano Pyrimidines	M. R. Kelleher; C. McGuigan; O. Bidet; A. Carangio; H. Weldon; G. Andrei; R. Snoeck; E. De Clercq; J. Balzarini

Volume 24, Issue 5-7 (2005)

647-650	Anti-Tumor Effect of Intravenous TNFα Gene Delivery Naked Plasmid DNA Using a Hydrodynamics-Based Procedure	Masayuki Kitajima; Youichi Tsuyama; Naoko Miyano-Kurosaki; Hiroshi Takaku
651-654	Synthesis and Purification of Fluorinated Benzimidazole and Benzene Nucleoside-5′-Triphosphates	A. E. Klöpffer; J. W. Engels
655-658	Synthesis and Biological Activity of Cyclic ADP-Carbocyclic-Ribose Analogs: Structure-Activity Relationship and Conformational Analysis of N-1-Carbocyclic-Ribose Moiety	Takashi Kudoh; Masayoshi Fukuoka; Satoshi Shuto; Akira Matsuda
659-661	Oxidative Transformations of Nucleoside Fluorenemethyl H-Phosphonoselenoate Diesters	Martin Kullberg; Jacek Stawinski
663-666	Accurate Mass Analysis of Phosphoramidites by Electrospray Mass Spectrometry	Z. Kupihár; Z. Timár; D. J. Dellinger; M. H. Caruthers
667-669	Synthesis of 2′-C-Methyl-β-d-Ribofuranosylimidazo[4,5-d]Pyridazine Derivatives (2-AZA-3-Deazapurine Nucleoside Analogues)	F. Leroy; D. Dukhan; M. Durka; D. Chaves; N. Bragnier; R. Storer; G. Gosselin
671-674	Synthesis of 5-Aza-7-Deazaguanine Nucleoside Derivatives as Potential Anti-Flavivirus Agents	D. Dukhan; F. Leroy; J. Peyronnet; E. Bosc; D. Chaves; M. Durka; R. Storer; P. La Colla; F. Seela; G. Gosselin
675-678	Model Synthesis of Nucleoside Boranophosphoramidate with Amino Acid for Prodrug Purpose	Ping Li; Barbara Ramsay Shaw
679-681	DNA Self-Assembling Systems: Branched Oligonucleotides as Building Blocks and Monitoring by Pyrene Excimer Band Formation	Dorthe Lindegaard; B. Ravindra Babu; Jesper Wengel
683-686	Synthesis of Carbocyclic Nucleotides as Potential Substrates for Thymidylate Kinase	O. R. Ludek; C. Meier
687-690	Engineering DNA Topology with Locked Nucleosides: A Structural Study	Melissa Maderia; Justin Wu; Ad Bax; Shilpa Shenoy; Barry O'Keefe; Victor E. Marquez; Joseph J. Barchi Jr.
691-694	Synthesis of Oligonucleotides Bearing an Arylamine Modification in the C8-Position of 2′-Deoxyguanosine	C. Meier; S. Gräsl; I. Detmer; A. Marx
695-699	Rapid Access to 2′-Branched-Carbocyclic Nucleosides and their 4′-Epimers from 2-Alkyl-Cyclopentene-1-Ones	J. -C. Meillon; L. Griffe; R. Storer; G. Gosselin
701-705	Comparative Conformational Analysis of Nucleosides by NMR, X-Ray, and Semi-Empirical (PM3 vs. AM1) Methods	Igor A. Mikhailopulo; Yuri A. Sokolov; Junlin He; Padmaja Chittepu; Helmut Rosemeyer; Frank Seela
707-708	Structure-Activity Relationship of 5′-Substituted Fluoro-Neplanocin A Analogues as Potent Inhibitors of S-Adenosylhomocysteine Hydrolase	Hyung Ryong Moon; Kang Man Lee; Hyun Joo Lee; Sang Kook Lee; Seung Bin Park; Moon Woo Chun; Lak Shin Jeong
709-711	Stereoselective Synthesis of Conformationally Rigid Apio Carbanucleosides as Potential Antiviral Agents	Hyung Ryong Moon; Kyung Ran Kim; Bum Tae Kim; Ki Jun Hwang; Moon Woo Chun; Lak Shin Jeong
713-715	Synthesis of Some 2′-Fluoro-2′-Deoxy-3′-C-Ethynyl and 3′-C-Vinyl-β-d-Lyxofuranosyl Nucleosides	O. Moukha-chafiq; K. N. Tiwari; J. A. Secrist III
717-720	Inhibitors of Inosine Monophosphate Dehydrogenase: Probes for Antiviral Drug Discovery	Sherry Story; Mukta Gupta; Eric Bonsu; Vasu Nair
721-724	Design of Highly Efficient and Selective Transfer Reaction of Nitrosyl Group to dC and d^MC Resulting in Specific Deamination	Md. Monsur Ali; Fumi Nagatsugi; Shizuka Nakayama; Md. Rowshon Alam; Takeshi Kawasaki; Shigeki Sasaki
725-728	Ring-Expanded Analogues of Natural Oxetanocin: ( ) and (-) Hydroxymethyl Isodideoxyadenosine	Byoung-Kwon Chun; Jean John Vadakkan; Vasu Nair
729-734	2′-Bis-Pyrene Modified Oligonucleotides: Sensitive Fluorescent Probes of Nucleic Acids Structure	D. S. Novopashina; D. A. Stetsenko; O. S. Totskaya; M. N. Repkova; A. G. Venyaminova
735-738	Synthesis of a New N-9 Ribityl Analogue of Cyclic Inosine Diphosphate Ribose (cIDPR) as a Mimic of Cyclic ADP Ribose (cADPR)	Giorgia Oliviero; Jussara Amato; Michela Varra; Gennaro Piccialli; Luciano Mayol
739-741	Unusual Monomolecular DNA Quadruplex Structures Using Bunch-Oligonucleotides	Giorgia Oliviero; Jussara Amato; Nicola Borbone; Aldo Galeone; Michela Varra; Gennaro Piccialli; Luciano Mayol
743-745	An Intramolecular 1,3-Dipolar Cycloaddition Reaction Towards the Synthesis of Chiral Azetidine Nucleoside Analogues: the d-gluco Case	P. Pádár; P. Forgó; Z. Kele; N. M. Howarth; L. Kovács
747-751	Mild, Efficient, Selective and "Green" Benzoylation of Nucleosides Using Benzoyl Cyanide in Ionic Liquid	Ashok K. Prasad; Vineet Kumar; Jyotirmoy Maity; Yogesh S. Sanghvi; Vasulinga T. Ravikumar; Virinder S. Parmar
753-756	Interaction of Porphyrin with G-Quadruplex Structures	Eva Erra; Luigi Petraccone; Veronica Esposito; Antonio Randazzo; Luciano Mayol; John Ladbury; Guido Barone; Concetta Giancola
757-760	Relative Stability of Quadruplexes Containing Different Number of G-Tetrads	Luigi Petraccone; Eva Erra; Ida Duro; Veronica Esposito; Antonio Randazzo; Luciano Mayol; Carlo Andrea Mattia; Guido Barone; Concetta Giancola
761-765	The Synthesis of Diene-Containing Nucleoside Phosphoramidites and Their Use in the Labeling of Oligonucleotides	Emma Anderson; Douglas Picken
767-770	NM 283, An Efficient Prodrug of the Potent Anti-HCV Agent 2′-C-Methylcytidine	C. Pierra; S. Benzaria; A. Amador; A. Moussa; S. Mathieu; R. Storer; G. Gosselin
771-775	Synthesis of Spin-Labeled RNAS for Long Range Distance Measurements by Peldor	Nelly Piton; Olav Schiemann; Yuguang Mu; Gerhard Stock; Thomas Prisner; Joachim W. Engels

Volume 24, Issue 5-7 (2005)

777-781	Large-Scale Synthesis of "Cpep" RNA Monomers and Their Application in Automated RNA Synthesis	R. T. Pon; S. Yu; T. Prabhavalkar; T. Mishra; B. Kulkarni; Y. S. Sanghvi
783-788	Effects of a 8-Oxoadenosine Incorporation on Quadruplex Structures: Thermal Stabilities and Structural Studies	Veronica Esposito; Antonio Randazzo; Antonella Virgilio; Luca Cozzuto; Luciano Mayol
789-794	Molecular Modeling Studies of a Parallel Stranded Quadruplexes Containing a 8-Bromoadenosine	Veronica Esposito; Antonio Randazzo; Luigi Petraccone; Concetta Giancola; Eva Erra; Antonella Virgilio; Luciano Mayol
795-800	Structural Studies on LNA Quadruplexes	Antonio Randazzo; Veronica Esposito; Oliver Ohlenschläger; Ramadurai Ramachandran; Antonella Virgilio; Luciano Mayol
801-804	Synthesis of Novel Piperidinyl Linker Based Energy Transfer Terminators and Their Potential Use in DNA Sequencing	T. Sudhakar Rao; Satyam Nampalli; Weihong Zhang; Haiguang Xiao; Shiv Kumar
805-808	Synthesis of Racemic and Enantiomeric 3-Pyrrolidinyl Derivatives of Purine and Pyrimidine Nucleobases	Petr Kocalka; Radek Pohl; Dominik Rejman; Ivan Rosenberg
809-813	bis(tBuSATE) Phosphotriester Prodrugs of 8-Azaguanosine and 6-Methylpurine Riboside; bis(POM) Phosphotriester Prodrugs of 2′-Deoxy-4′-Thioadenosine and Its Corresponding 9α Anomer	J. D. Rose; W. B. Parker; J. A. Secrist III
815-818	Kilo-Scale Synthesis Process for 2′-O-(2-Methoxyethyl)-Pyrimidine Derivatives	Bruce S. Ross; Quanlai Song; Mingming Han
819-822	Transprotection of Silyl Ethers of Nucleosides in FeCl₃ Based Ionic Liquids	Jitendra R. Harjani; Susheel J. Nara; Manikrao M. Salunkhe; Yogesh S. Sanghvi
823-827	Expansion of Triplex Recognition Codes by the Use of Novel Bicyclic Nucleoside Derivatives (WNA)	Yosuke Taniguchi; Ayako Nakamura; Yusuke Senko; Keiichi Kodama; Fumi Nagatsugi; Shigeki Sasaki
829-837	CDK Inhibitory Nucleoside Analogs Prevent Transcription from Viral Genomes	L. M. Schang; E. Coccaro; J. J. Lacasse
839-841	7-Deazapurin-2,6-Diamine and 7-Deazaguanine: Synthesis and Property of 7-Substituted Nucleosides and Oligonucleotides	Frank Seela; Xiaohua Peng; Xin Ming
843-846	Gold DNA-Conjugates: Ion Specific Self-Assembly of Gold Nanoparticles via the dG-Quartet	Frank Seela; Anup M. Jawalekar; Lifeng Chi; Dingyong Zhong; Harald Fuchs
847-850	6-Azapyrimidine and 7-Deazapurine 2′-Deoxy-2′-Fluoroarabinonucleosides: Synthesis, Conformation and Properties of Oligonucleotides	Frank Seela; Padmaja Chittepu; Yang He; Junlin He; Kuiying Xu
851-854	Propynyl Groups in Duplex, Hairpin and Triplex DNA: 7-Deazapurines and 9-Deazapurines	Frank Seela; Khalil I. Shaikh; Simone Budow; Anup M. Jawalekar
855-858	Novel DNA Nanoparticles and Networks	Frank Seela; Anup M. Jawalekar; Venkata R. Sirivolu; Helmut Rosemeyer; Yang He; Peter Leonard
859-863	l-Nucleosides Containing Modified Nucleobases	Frank Seela; W. Lin; Z. Kazimierczuk; H. Rosemeyer; V. Glaçon; X. Peng; Y. He; X. Ming; M. Andrzejewska; A. Gorska; X. Zhang; H. Eickmeier; P. La Colla
865-868	Parallel and Antiparallel DNA: Fluorescence Quenching of Ethidium Bromide by 7-Deazapurines	Hong Li; Frank Seela
869-873	7-Substituted 8-Aza-7-Deazapurines and 2,8-Diaza-7-Deaza-Purines: Synthesis of Nucleosides and Oligonucleotides	Wenqing Lin; Kuiying Xu; Frank Seela
875-879	Synthesis and in vitro Anti-HCV Activity of β-d- and l-2′-Deoxy-2′-Fluororibonucleosides	Junxing Shi; Jinfa Du; Tianwei; Krzysztof W. Pankiewicz; Steven E. Patterson; Abdalla E. A. Hassan; Phillip M. Tharnish; Tamara R. McBrayer; Stefania Lostia; Lieven J. Stuyver; Kyoichi A. Watanabe; Chung K. Chu; Raymond F. Schinazi; Michael J. Otto
881-885	Synthesis and Biological Activity of 2-Fluoro Adenine and 6-Methyl Purine Nucleoside Analogs as Prodrugs for Suicide Gene Therapy of Cancer	A. V. Silamkoti; P. W. Allan; A. E. A. Hassan; A. T. Fowler; E. J. Sorscher; W. B. Parker; J. A. Secrist III
887-890	Aryl Nucleoside H-Phosphonates as a Tool for Investigation of Stereospecificity During Coupling	Michal Sobkowski; Jadwiga Jankowska; Jacek Stawinski; Adam Kraszewski
891-896	Recent Highlights on Photolithic Oligonucleotide Array In Situ Synthesis	Klaus-Peter Stengele; Jochen Bühler; Sigrid Bühler; Evgueni Kvassiouk; Roland Green; Tamara Prykota; Wolfgang Pfleiderer
897-899	A Solid Supported Reagent for Internucleoside H-Phosphonate Linkage Formation	Nikhil Mohe; Petri Heinonen; Yogesh S. Sanghvi; Roger Strömberg
901-905	Studies in Oligonucleotide-Based Artificial Nuclease Systems. Intramolecular Copper (II) Complex Formation in an Oligonucleotide bis-Phenanthroline Conjugate	Dmitri A. Ossipov; Roger Strömberg
907-910	A Study of H-Bonding of 3- and 5-Substituted 6-Aminouracils in Duplex and Triplex Structures	E. Szájli; G. Paragi; L. Kovács
911-914	Synthesis and Biological Activity of 2′-Deoxy-4′-Thio-Pyrazolo[3,4-d]Pyrimidine Nucleosides	K. N. Tiwari; A. S. Fowler; J. A. Secrist III
915-917	Novel Strategy for Single Nucleotide Polymorphism (SNP) Genotyping by Heteroduplex Analysis: Specific Stabilization of TT Mismatch Base Pair by Mercury (II) Cation and CC Mismatch Base Pair by Silver (I) Cation	Hidetaka Torigoe; Kouji Kawahashi; Ayako Takamori; Akira Ono
919-922	Oxidation of Biotin During Oligonucleotide Synthesis	Krishna Upadhya; Iqbal K. Khattak; Bashar Mullah
923-926	Synthesis and Evaluation of Anti-HSV Activity of New 5-Alkynyl-2′-Deoxyuridines	A. A. Pchelintseva; M. V. Skorobogatyj; A. L. Petrunina; V. L. Andronova; G. A. Galegov; I. V. Astakhova; A. V. Ustinov; A. D. Malakhov; Vladimir A. Korshun

Volume 24, Issue 5-7 (2005)

927-929	A New Protecting Group for the 5′-Hydroxyl Group Having O–S Single Bond Oxidatively Cleavable Under Mild Conditions	Eri Utagawa; Kohji Seio; Mitsuo Sekine
931-934	Perylene Attached to DNA Through Stiff or Flexible Linker: Duplex Stability and Fret	Mikhail V. Skorobogatyj; Anna A. Pchelintseva; Alexei V. Ustinov; Vladimir A. Korshun; Andrei D. Malakhov
935-938	2-Substituted 5′-N-Methylcarboxamidoadenosine (MECA) Derivatives as A₃ Adenosine Receptor Ligands	S. Vittori; R. Volpini; C. Lambertucci; S. Taffi; K. N. Klotz; G. Cristalli
939-942	"Lock-in" Modified CycloSal Nucleotides—The Second Generation of CycloSal Prodrugs	D. Vukadinović; N. P. H. Böge; J. Balzarini; C. Meier
943-946	Incorporation of Ribonucleoside 5′-(α-P-Borano)Triphosphates Into a 20-MER RNA by T7 RNA Polymerase	Jing Wan; Barbara Ramsay Shaw
947-950	Synthesis of 5-(1-Propynyl)-2′-Deoxyuridine 5′-(Alpha-P-Borano)Triphosphate and Kinetic Characterization as a Substrate for MMLV Reverse Transcriptase	Joy Xin Wang; Barbara Ramsay Shaw
951-955	The Effect of a Single Boranophosphate Substitution with Defined Configuration on the Thermal Stabiltiy and Conformation of a DNA Duplex	Joy Xin Wang; Dmitri S. Sergueev; Barbara Ramsay Shaw
957-960	Synthesis of N ³,5′-Cyclo-4-(β-d-Ribofuranosyl)-vic-Triazolo[4,5-b]Pyridin-5-One and Its 3′-Deoxysugar Analogue as Potential Anti-Hepatitis C Virus Agents	Peiyuan Wang; Laurent Hollecker; Krzysztof W. Pankiewicz; Steven E. Patterson; Tony Whitaker; Tamara R. McBrayer; Phillip M. Tharnish; Lieven J. Stuyver; Raymond F. Schinazi; Michael J. Otto; Kyoichi A. Watanabe
961-964	Synthesis and Anti-Hepatitis C Virus Activity of Nucleoside Derivatives of N ³,5′-Anhydro-4-(β-d-Ribofuranosyl)-8-Azapurin-2-Ones	Abdalla E. A. Hassan; Peiyuan Wang; Tamara R. McBrayer; Phillip M. Tharnish; Lieven J. Stuyver; Raymond F. Schinazi; Michael J. Otto; Kyoichi A. Watanabe
965-969	Synthesis and Characterization of DNA Duplexes Containing an N³T-Ethyl-N³T Interstrand Crosslink in Opposite Orientations	Christopher J. Wilds; Anne M. Noronha; Sebastien Robidoux; Paul S. Miller
971-974	Antigene Property of PNA Conjugated to the Nuclear Localization Signal Peptide	Susanna Cogoi; Andrea Codognotto; Valentina Rapozzi; Luigi E. Xodo
975-977	Synthesis of 3′-Deoxy-3′-C-Hydroxymethyl Analogues of Tiazofurin and Ribavirin	Moon Woo Chun; Myong Jung Kim; Ji Hye Shin; Lak Shin Jeong
979-981	Synthesis of Homo-N-Nucleoside with 1,2,4-Triazole-3-Carboxamide	Moon Woo Chun; Jin Hee Kim; Myong Jung Kim; Bo Ram Kim; Lak Shin Jeong
983-987	Affinity of (α-P-Borano)-NTP Analogs to Rabbit Muscle Pyruvate Kinase	Mikhail I. Dobrikov; Barbara Ramsay Shaw
989-992	A Novel Amino-ON CPG-Support for the Synthesis of 3′-Aminoalkylated Oligonucleotides	Michael Leuck; Rubina Giare; Nicole Zien; Matthias Paul; Andreas Wolter
993-998	Enzymatic Resolution and Base Pairing Properties of d - and l -Cyclohexenyl Nucleic Acids (CeNA)	Ping Gu; Guy Schepers; Carsten Griebel; Jef Rozenski; Hans-Joachim Gais; Piet Herdewijn; Arthur Van Aerschot
999-1008	Photolabeling Probes of Ribavirin and Eicar	Qiongyou Wu; Fanqi Qu; Jinqiao Wan; Yi Xia; Ling Peng
1009-1013	Silyl Protecting Groups for Oligonucleotide Synthesis Removed by A ZnBr₂ Treatment	Fernando Ferreira; François Morvan
1015-1018	Synthesis of Conformationally Restricted Nucleic Acid Fragments Using Ring-Closing Alkene and Enyne Metathesis Reactions	Signe I. Steffansen; Mikkel S. Christensen; Philip Børsting; Poul Nielsen
1019-1021	Promotion of Pyrimidine Motif Triplex Formation by Morpholino Modification of Triplex-Forming Oligonucleotide: Kinetic and Thermodynamic Studies	Hidetaka Torigoe; Kouji Kawahashi; Yuusuke Tamura
1023-1027	RNA Recognition by Fluor-Aromatic Substituted	A. Živković; J. W. Engels
1029-1032	PROSIT, an Online Service to Calculate Pseudorotational Parameters of Nucleosides and Nucleotides	Guangyu Sun; Johannes H. Voigt; Victor E. Marquez; Marc C. Nicklaus
1033-1036	A Cautionary Note on the Use of the ³¹P NMR Spectroscopy in Stereochemical Correlation Analysis	Michal Sobkowski; Jadwiga Jankowska; Jacek Stawinski; Adam Kraszewski
1037-1041	Significant Improvement of Quality for Long Oligonucleotides by Using Controlled Pore Glass with Large Pores	Igor A. Kozlov; Minh Dang; Ken Sikes; Theofilos Kotseroglou; David L. Barker; Chanfeng Zhao
1043-1046	Functionalization of Pyrimidine and Purine Nucleosides at C4 and C6: C-Nucleophilic Substitution of Their C4- and C6-(1,2,4-Triazol-1-yl) Derivatives	Victor Timoshchuk
1047-1049	Synthesis of 5-Ethynyl-2′-Deoxyuridine-5′-Boranomono Phosphate as a Potential Thymidylate Synthase Inhibitor	Shoeb I. Khan; Mikhail I. Dobrikov; Barbara Ramsay Shaw
1051-1054	Synthetic Study of 3′-α-Fluoro-2′,3′-Dideoxyguanosine	Takayoshi Torii; Tomoyuki Onishi; Shigehisa Tanji; Kunisuke Izawa
1055-1058	Presence of 2′,5′-Linkages in a Homopyrimidine DNA Oligonucleotide Promotes Stable Triplex Formation Under Physiological Conditions	Satoshi Obika; Akiko Hiroto; Osamu Nakagawa; Takeshi Imanishi
1059-1061	A Convenient Method for the Synthesis of Oligonucleotide-Cationic Peptide Conjugates	G. Ferenc; Z. Kupihár; Z. Kele; L. Kovács
1063-1067	A New Approach to Oligonucleotide N3′→P5′ Phosphoramidate Building Blocks	Daria Zielinska; Krisztina Pongracz; Sergei Gryaznov

Volume 24, Issue 5-7 (2005)

1069-1074	Oligonucleotides as Coding Molecules in an Anti-Counterfeiting System	C. Wolfrum; A. Josten
1075-1079	Studies on the Attachment of DNA to Silica-Coated Nanoparticles Through a Diels-Alder Reaction	M. Proupin-Perez; R. Cosstick; L. M. Liz-Marzan; V. Salgueiriño-Maceira; M. Brust
1081-1083	Chemical Synthesis of Oligonucleotides Containing (M 4) Guanine	Ruoling Guo; Qinguo Zheng
1085-1091	Tumor-Targeting Peptide-PNA-Peptide Chimeras for Imaging Overexpressed Oncogene mRNAs	X. Tian; M. R. Aruva; H. R. Wolfe; W. Qin; E. R. Sauter; M. L. Thakur; S. A. Waldman; E. Wickstrom
1093-1095	Natural Phosphate Doped with KI in HMDS: A Mild and Efficient Reagent for Alkylation and Glycosylation of Nucleobases	H. B. Lazrek; M. Taourirte; A. Rochdi; N. Redwane; D. Ouzebla; L. Baddi; S. Sebti; J. J. Vasseur
1097-1100	Synthesis and Properties of a Novel Bridged Nucleic Acid Analogue, 5′-Amino-3′,5′-BNA	Mitsuaki Sekiguchi; Satoshi Obika; Roongjang Somjing; Takeshi Imanishi
1101-1104	Synthesis of a 2′-Amino-α-l-LNA-T Phosphoramidite	Patrick J. Hrdlicka; T. Santhosh Kumar; Jesper Wengel
1105-1109	Modified Binary Hammerhead Ribozymes with High Catalytic Activity	M. Vorobjeva; E. Gusseva; M. Repkova; N. Kovalev; M. Zenkova; A. Venyaminova; V. Vlassov
1111-1114	4,5-Bis(Ethoxycarbonyl)-[1,3]Dioxolan-2-yl as a New Orthoester-Type Protecting Group for the 2′-Hydroxyl Function in the Chemical Synthesis of RNA	Boleslaw Karwowski; K. Seio; M. Sekine
1115-1117	Stereoselective Synthesis of Novel Thioiso Dideoxy Nucleosides with Exocyclic Methylene as Potential Antiviral Agents	Prashantha Gunaga; Hea Ok Kim; Hyun Ji Kim; Moon Woo Chun; Lak Shin Jeong
1119-1121	Synthesis of 3′-Ureidoadenosine Analogues and their Binding Affinity to the A₃ Adenosine Receptor	Moon Woo Chun; Hyouk Woo Lee; Ae Yil Kim; Myong Jung Kim; Hea Ok Kim; Zhan-Guo Gao; Kenneth A. Jacobson; Lak Shin Jeong
1123-1126	Synthesis and Properties of PNA Oligomers Containing Orotic Acid Derivatives	R. H. E. Hudson; F. Wojciechowski
1127-1130	Efficient Chemo-Enzymatic Syntheses of Pharmaceutically Useful Unnatural 2′-Deoxynucleosides	Hironori Komatsu; Tadashi Araki
1131-1134	Novel Way of Capping mRNA Trimer and Studies of Its Interaction with Human Nuclear Cap-Binding Complex	Remigiusz Worch; Janusz Stepinski; Anna Niedzwiecka; Marzena Jankowska-Anyszka; Catherine Mazza; Stephen Cusack; Ryszard Stolarski; Edward Darzynkiewicz
1135-1138	Large-Scale Synthesis of 5′-O-Pixyl Protected 2′-Deoxynucleosides Useful for Oligonucleotide Synthesis	Robert T. Day; Dean Williams; Priscilla Soriano; Yogesh S. Sanghvi
1139-1146	Contributors

Volume 24, Issue 4 (2005)

233-242	Sequence Analysis of the 5′-Flanking Regions of Human Dihydropyrimidine Dehydrogenase Gene: Identification of a New Polymorphism Related with Effects of 5-Fluorouracil	Takako Hasegawa; Hye-sook Kim; Masakazu Fukushima; Yusuke Wataya
243-246	New Short Route to Unsaturated Fluoroketonucleosides: Case of 5-Fluoro-1-(6-O-Acetyl-3,4-Di-Deoxy-3-Fluoro-β-d-Glycero-Hex-3-Eno-Pyranos-2-Ulosyl) Uracil	Marie-José Egron; Dimitri Komiotis; Ismet Dorange; Jean Herscovici; Abraham P. Ollapally; Kostas Antonakis
247-257	¹³C-³¹P Couplings in the Study of Conformational Properties of Some Diastereomeric Nucleoside-3′-Thiophosphate Derivatives	Eszter Gács-Baitz; Gyula Sági; Mária Kajtár-Peredy
259-262	The Effect of N-Methyl-2-Pyridone-5-Carboxamide—A Nicotinamide Catabolite on Poly ADP-Rybosylation and Oxidative Stress Injury in Endothelial Cells	E. M. Slominska; R. T. Smolenski; F. Osborne; J. Swierczynski; M. H. Yacoub
263-266	Purine Metabolism in Pigs and Humans and Its Implications for Xenotransplantation	R. T. Smolenski; Z. Khalpey; A. Yuen; H. Dziewit; E. M. Slominska; T. Borkowski; M. Zdunek; Z. Kochan; J. Karbowska; M. Lavitrano; M. H. Yacoub
267-270	Prevention of Adriamycin Induced Heart Failure by an Increase in Endogenous Adenosine Production	A. H. Y. Yuen; M. Boscoe; R. Lango; K. Suzuki; E. M. Slominska; M. H. Yacoub; R. T. Smolenski
271-274	Exposure to Human Blood Inactivates Swine Endothelial Ecto-5′-Nucleotidase	Z. Khalpey; K. Kalsi; A. Yuen; J. Karbowska; Z. Kochan; E. M. Slominska; M. Forni; M. Bacci; M. Macherini; P. Batten; M. Lavitrano; M. H. Yacoub; R. T. Smolenski
275-277	Association of Improved Cardiac Function in Donors with C34T Mutation of the AMP Deaminase 1 Gene	A. H. Y. Yuen; M. H. Yacoub; E. J. Birks; K. K. Kalsi; P. H. Johnson; R. T. Smolenski
279-282	Lidoflazine Combined with Nucleotide Precursors Increases ATP Content and Adenosine Production in Cardiomyocytes	K. K. Kalsi; R. T. Smolenski; M. H. Yacoub
283-285	Expression of Human Ecto 5′ Nucleotidase in Pig Endothelial Cells and Its Implication for Adenosine Production and Xenotransplantation	F. N. Osborne; K. Kalsi; C. Lawson; M. Lavitrano; M. H. Yacoub; M. L. Rose; R. T. Smolenski
287-288	AMPD1 C34T Mutation Selectively Affects AMP-Deaminase Activity in the Human Heart	K. K. Kalsi; A. H. Y. Yuen; P. H. Johnson; E. J. Birks; M. H. Yacoub; R. T. Smolenski
289-301	New Dinucleoside Analogues via Cross-Coupling Metathesis	Vincent Roy; Rachida Zerrouki; Pierre Krausz
303	Errata

Volume 24, Issue 3 (2005)

161-172	Synthesis and Biological Activity of Some Unsaturated 6-Azauracil Acyclonucleosides	Youssef Kabbaj; Hassan Bihi Lazrek; Jean Louis Barascut; Jean Louis Imbach
173-178	A One-Pot Synthesis of 1-α- And 1-β-D-Arabinofuranosyl-2-Nitroimidazoles: Synthons to the Markers of Tumor Hypoxia	Ebrahim Naimi; Piyush Kumar; Alexander J. B. McEwan; Leonard I. Wiebe
179-189	Synthesis of 5′-Triphosphate Mimics (P3Ms) of 3′-Azido-3′,5′-Dideoxythymidine and 3′,5′-Dideoxy-5′-Difluoromethylenethymidine as HIV-1 Reverse Transcriptase Inhibitors	Vivek K. Rajwanshi; Marija Prhavc; Patrick Fagan; Jennifer L. Brooks; Tiffany Hurd; P. Dan Cook; Guangyi Wang
191-198	Finding Keywords for Intergenic and Gene Regions for Human Genome	Y. H. Qiao; J. L. Liu; C. G. Zhang; Yanjun Zeng
199-209	A Neural Network for Predicting the Stability of DNA/DNA Duplexes	Xiaohong Liu; Lixin; Changmei Cheng; Yong Wang; Hiromi Miyajima; Yufen Zhao
211-226	A Novel Versatile Phosphoramidite Building Block for the Synthesis of 5′- and 3′-Hydrazide Modified Oligonucleotides	Sergey I. Antsypovich; Günter von Kiedrowski
227-232	Inhibitory Mechanisms of 1-(3-C-Ethynyl-β-d-ribo-Pentofuranosyl)Uracil (EUrd) on RNA Synthesis	Tatsushi Yokogawa; Tomoharu Naito; Hiroshi Kanda; Satoshi Takatori; Kiyoko Takenaka; Takuma Sasaki; Akira Matsuda; Masakazu Fukushima; Hye-Sook Kim; Yusuke Wataya

Volume 24, Issue 2 (2005)

73-83	Synthesis of (±)-4′-Ethynyl and 4′-Cyano Carbocyclic Analogues of Stavudine (d4T)	Hiroki Kumamoto; Kazuhiro Haraguchi; Hiromichi Tanaka; Keisuke Kato; Takao Nitanda; Masanori Baba; Ginger E. Dutschman; Yung-Chi Cheng
85-110	Synthesis of Two 8-[(Anthraquinone-2-yl)-Linked]-2′-Deoxyadenosine 3′-Benzyl Hydrogen Phosphates for Studies of Photoinduced Hole Transport in DNA	Reham A. I. Abou-Elkhair; Thomas L. Netzel
111-120	Synthesis of Some Novel N-Ribosyl-1,2,4-Triazin-6(1H)-/Ones or Thiones as Potential Antibacterial and Antifungal Chemotherapeutics	Nasser S. A. M. Khalil
121-133	Novel Approach to Nucleoside-5′-(1-Hydroxymethylene-1,1-Bisphosphonates): Synthesis of New AZT Analogues	Evelyne Migianu; Maëlle Monteil; Pascale Even; Marc Lecouvey
135-145	Synthesis and Biological Evaluation of 2′,3′-Didehydro-2′,3′-Dideoxy-9-Deazaguanosine, a Monophosphate Prodrug and Two Analogues, 2′,3′-Dideoxy-9-Deazaguanosine and 2′,3′-Didehydro-2′,3′-Dideoxy-9-Deazainosine	Mao-Chin Liu; Mei-Zhen Luo; Diane E. Mozdziesz; Ginger E. Dutschman; Elizabeth A. Gullen; Yung-Chi Cheng; Alan C. Sartorelli
147-152	Co-Transfection of Messenger RNA and siRNA as a Method to Study the Efficiency of siRNA	Thorsten Mutzke; Gudrun Schubkegel; Regina Teufel; Thomas Ketterer; Jochen Probst; Birgit Scheel; Jean-Philippe Carralot; Kamran Ghoreschi; Christina Weigert; Steve Pascolo
153-160	Concise Synthesis and Antiviral Activity of Novel Unsaturated Acyclic Pyrimidine Nucleosides	Chang-Hyun Oh; Tae-Rim Baek; Joon Hee Hong

Volume 24, Issue 1 (2005)

1-14	Perfluoroarylazide Derivatives of 2′-O-Modified Oligoribonucleotides: Efficient Reagents for RNA Photomodification	D. S. Novopashina; R. N. Kulikov; M. A. Kuznetsova; A. G. Venyaminova; M. A. Zenkova; V. V. Vlassov
15-35	Synthesis and DNA Topoisomerase-II Inhibitory Activity of Unnatural Nucleosides	Ram Chandra Mishra; Namrata Dwivedi; Iti Bansal; Jitendra Kumar Saxena; Rama Pati Tripathi
37-43	Acyclic Nucleosides Bearing a Furanyl Scaffold	Vasu Nair; Sanjib Bera
45-62	Synthesis and Biological Evaluation of 2- and 7-Substituted 9-Deazaadenosine Analogues	Mao-Chin Liu; Mei-Zhen Luo; Diane E. Mozdziesz; Alan C. Sartorelli
63-72	Synthesis and Anti-HCMV Activity of Novel 2′,3′,4′-Trimethyl Branched Carbocyclic Nucleosides	Aihong Kim; Joon Hee Hong

Volume 23, Issue 12 (2004)

i-ii	List of Contributors
1815-1824	Synthesis and Antiviral Properties of Arabino and Ribonucleosides of 1,3-Dideazaadenine, 4-Nitro-1, 3-dideazaadenine and Diketopiperazine	Sarika Sinha; Richa Srivastava; Erik De Clercq; Ramendra K. Singh
1825-1832	First Synthesis of Double Headed 1,3,4-Oxadiazino[6,5-b]indole Acyclo C-Nucleosides	Adel Z. Nasr
1833-1847	The Chemical and Biochemical Properties of Methylphosphotriester DNA	Henk M. Buck
1849-1864	Effective Anomerisation of 2′-Deoxyadenosine Derivatives During Disaccharide Nucleoside Synthesis	Irina V. Gulyaeva; Kari Neuvonen; Harri Lönnberg; Andrei A. Rodionov; Elena V. Shcheveleva; Georgii V. Bobkov; Ekaterina V. Efimtseva; Sergey N. Mikhailov
1865-1874	Phosphorylation of Isocarbostyril- and Difluorophenyl-Nucleoside Thymidine Mimics by the Human Deoxynucleoside Kinases	Ashraf Said Al-Madhoun; Staffan Eriksson; Zhi-Xian Wang; Ebrahim Naimi; Edward E. Knaus; Leonard I. Wiebe
1875-1887	Synthesis of (-)-DAPD	Marcos L. Sznaidman; Jinfa Du; Amir Pesyan; Darryl G. Cleary; Kevin P. Hurley; Frank Waligora; Merrick R. Almond
1889-1910	Synthesis of Some Novel 6-Benzyl(or Substituted Benzyl)-2-β-d-Glucopyranosyl-1,2,4-Triazolo[4,3-b][1,2,4]Triazines as Potential Antimicrobial Chemotherapeutics	Nasser S. A. M. Khalil; Abdel Kader Mansour; Mohga M. Eid
1911-1927	The Solution Synthesis of Antisense Oligonucleotide-Peptide Conjugates Directly Linked via Phosphoramide Bond by Using a Fragment Coupling Approach	Nataliya V. Sumbatyan; Vassili A. Mandrugin; Alain Deroussent; Jean-Rémi Bertrand; Zsuzsa Majer; Claude Malvy; Galina A. Korshunova; Miklos Hollosi; Marina B. Gottikh
1929-1937	Phosphoramidate Protides of Carbocyclic 2′,3′-Dideoxy-2′,3′-Didehydro-7-Deazaadenosine with Potent Activity Against HIV and HBV	Kristjan S. Gudmundsson; Zhicheng Wang; Susan M. Daluge; Lance C. Johnson; Richard Hazen; Lynn D. Condreay; Christopher McGuigan

Volume 23, Issue 11 (2004)

1683-1705	Nucleosidyl-O-Methylphosphonates: A Pool of Monomers for Modified Oligonucleotides	Dominik Rejman; Milena Masojídková; Ivan Rosenberg
1707-1721	Synthesis, ¹⁸F-Radiolabelling and Biological Evaluations of C-6 Alkylated Pyrimidine Nucleoside Analogues	Silvana Raić-Malić; Anass Johayem; Simon M. Ametamey; Sanja Batinac; Erik De Clercq; Gerd Folkers; Leonardo Scapozza
1723-1738	Efficient Pyrimidine N-1-Alkylation via Activation of Electron Rich Olefins with Oxoammonium Salts: Synthesis of Methoxy TEMPO Substituted Pyrimidine Nucleoside Analogs	Kevin M. Church; Liesel M. Holloway; Ryan C. Matley; Robert J. Brower III
1739-1749	Thiosugar Nucleosides. Synthesis and Biological Activity of 1,3,4-Thiadiazole, Thiazoline and Thiourea Derivatives of 5-Thio-d-Glucose	Najim A. Al-Masoudi; Yaseen A. Al-Soud; Wasfi A. Al-Masoudi
1751-1765	Side-Chain Conformational Restriction in Template-Competitive Inhibitors of E. coliDNA Polymerase I Klenow Fragment: Synthesis, Structural Characterization and Inhibition Activity	Michael B. Doughty; Karam Aboudehen; Garland Anderson; Ke Li; Bob Moore II; Tina Poolson
1767-1777	Synthesis of Oligoribonucleotides Containing 4-Thiouridine Using the Convertible Nucleoside Approach and the 1-(2-Fluorophenyl)-4-Methoxypiperidin-4-yl Group	Anna Aviñó; Ramon Güimil García; Ramon Eritja
1779-1795	Crystal Structure and Conformation of 5-Fluorouridine: Conformational Preferences for 5-Fluorinated Pyranosides	Sunil Dutta Soni; Thamarapu Srikrishnan
1797-1811	Synthesis, In Vitro Anticancer Evaluation, and Interference with Cell Cycle Progression of N-Phosphoamino Acid Esters of Zidovudine and Stavudine	Y. W. Wu; Q. Xiao; Y. Y. Jiang; H. Fu; Y. Ju; Y. F. Zhao
1813-1814	List of Contributors

Volume 23, Issue 10 (2004)

1565-1581	Synthesis and Biological Evaluation of Novel 1′-Branched and Spironucleoside Analogues	Chryssostomos Chatgilialoglu; Carla Ferreri; Thanasis Gimisis; Marinella Roberti; Jan Balzarini; Erik De Clercq
1583-1594	7-Deaza-2′-Deoxyadenosine-5′-Triphosphate as an Alternative Nucleotide for the Pyrosequencing Technology	Jonas Eriksson; Baback Gharizadeh; Nader Nourizad; Pål Nyrén
1595-1607	An Antisense Oligodeoxynucleotide-Doxorubicin Conjugate: Preparation and Its Reversal Multidrug Resistance of Human Carcinoma Cell Line In Vitro	Yuhong Ren; Dongzhi Wei; Jianwen Liu; Wu Su
1609-1623	Thiosugars. XII. Synthesis of New 3′-O-Substituted 2′,5′-Anhydro-2′-thio-α-d-pentofuranosyl Nucleoside Analogues	Jürgen Voss; Jörn Wirsching; Oliver Schulze; Gunadi Adiwidjaja; Anja Giesler; Jan Balzarini; Erik De Clercq
1625-1637	Synthesis and Antiviral Evaluation of D4T Analogues with a Spacer Arm Between Glucidic and Base Moieties	Vincent Roy; Rachida Zerrouki; Pierre Krausz; Sylvie Schmidt; Anne Marie Aubertin
1639-1656	Interaction of 2-Chloro-N¹⁰-Substituted Phenoxazine with DNA and Effect on DNA Melting	K. H. Chandramouli; K. N. Thimmaiah; Arun Chandrashekar; Cletus J.M. D'Souza
1657-1666	Chemoselective Oxime and Thiazolidine Bond Formation: A Versatile and Efficient Route to the Preparation of 3′-Peptide-Oligonucleotide Conjugates	Mathilde Villien; Eric Defrancq; Pascal Dumy
1667-1680	Chemical Route to the Capped RNAs	I. I. Koukhareva; A. V. Lebedev
1681-1682	List of Contributors

Volume 23, Issue 8-9 (2004)

1077-1079	Purine and Pyrimidine Metabolism: New Challenges	G. J. Peters; A. B. P. van Kuilenburg; R. A. de Abreu
1081-1082	Dedication to Francoise Roch-Ramel	H. A. Simmonds
1083-1088	Antimetabolites in the Treatment of Arthritis: Current Status of the Use of Antimetabolites	B. A. C. Dijkmans; G. Jansen
1089-1100	Two Inhibitors of DNA-Synthesis Lead to Inhibition of Cytokine Production via a Different Mechanism	S. de Lathouder; A. H. Gerards; B. A. C. Dijkmans; L. A. Aarden
1101-1106	Modification of Cytokine Milieu by A_2A Adenosine Receptor Signaling–Possible Application for Inflammatory Diseases	M. Koshiba; Y. Nakamachi; H. Kosaka; T. Nakazawa; G. Tsuji; S. Kumagai
1107-1110	Purine Modulation of Cytokine Release During Diuretic Therapy of Rheumatoid Arthritis	C. M. Forrest; G. Harman; R. B. McMillan; C. Rana; S. Shaw; T. W. Stone; N. Stoy; L. G. Darlington
1111-1116	Febuxostat (TMX-67), a Novel, Non-Purine, Selective Inhibitor of Xanthine Oxidase, Is Safe and Decreases Serum Urate in Healthy Volunteers	M. A. Becker; J. Kisicki; R. Khosravan; J. Wu; D. Mulford; B. Hunt; P. MacDonald; N. Joseph-Ridge
1117-1118	PK/PD and Safety of a Single Dose of TMX-67 (Febuxostat) in Subjects with Mild and Moderate Renal Impairment	S. Hoshide; Y. Takahashi; T. Ishikawa; J. Kubo; M. Tsuchimoto; K. Komoriya; I. Ohno; T. Hosoya
1119-1122	Pharmacokinetics and Pharmacodynamics of Febuxostat (TMX-67), a Non-Purine Selective Inhibitor of Xanthine Oxidase/Xanthine Dehydrogenase (NPSIXO) in Patients with Gout and/or Hyperuricemia	K. Komoriya; S. Hoshide; K. Takeda; H. Kobayashi; J. Kubo; M. Tsuchimoto; T. Nakachi; H. Yamanaka; N. Kamatani
1123-1125	Pharmacokinetics/Pharmacodynamics of Y-700, A Novel Xanthine Oxidase Inhibitor, in Rats and Man	I. Yamada; A. Fukunari; T. Osajima; M. Kamezawa; H. Mori; J. Iwane
1127-1129	Detection of Prothrombin and Osteopontin in a Renal Stone Found in a Hyperuricemic Patient Using 2D-PAGE and LC-MS Analysis	K. Kaneko; T. Yamanobe; K. Nakagomi; K. Mawatari; M. Onoda; S. Fujimori
1131-1134	EPR Spin Trapping of a Radical Intermediate in the Urate Oxidase Reaction	E. Busi; L. Terzuoli; R. Basosi; B. Porcelli; E. Marinello
1135-1139	An Unusual Pyridine Nucleotide Accumulating in Erythrocytes: Its Identity, and Positive Correlation with Degree of Renal Failure	E. A. Carrey; R. T. Smolenski; S. M. Edbury; A. Laurence; A. M. Marinaki; J. A. Duley; L. M. Zhu; D. J. A. Goldsmith; H. A. Simmonds
1141-1145	Identification of Two Novel Mutations in Adenine Phosphoribosyltransferase Gene in Patients with 2,8-Dihydroxyadenine Urolithiasis	Atsuo Taniguchi; Sanae Tsuchida; Shin-Ichi Kuno; Masayuki Mita; Tastuya Machida; Naomasa Ioritani; Chihiro Terai; Hisashi Yamanaka; Naoyuki Kamatani
1147-1152	Medical Diagnosis, Management and Treatment of Lesch Nyhan Disease	Gillian McCarthy
1153-1160	The Spectrum of Mutations Causing HPRT Deficiency: An Update	H. A. Jinnah; J. C. Harris; W. L. Nyhan; J. P. O'Neill
1161-1164	The Motor Disorder of Classic Lesch-Nyhan Disease	Jasper E. Visser; James C. Harris; Gabor Barabas; Gary E. Eddey; H. A. Jinnah
1165-1168	Clinical and Biochemical Manifestations and Molecular Characterization of the Mutation HPRT Jerusalem	E. Zoref-Shani; Y. Bromberg; J. Hirsch; S. Feinstein; Y. Frishberg; O. Sperling
1169-1172	Mutations in the Hypoxanthine Guanine Phosphoribosyltransferase Gene (HPRT1) in Asian HPRT Deficient Families	Y. Yamada; K. Yamada; S. Sonta; N. Wakamatsu; N. Ogasawara

Volume 23, Issue 8-9 (2004)

1173-1176	Disruption of the Hypoxanthine-Guanine Phosphoribosyl-Transferase Gene Caused by a Translocation in a Patient with Lesch-Nyhan Syndrome	Makiko Mizunuma; Yasukazu Yamada; Kenichiro Yamada; Shin-Ichi Sonta; Nobuaki Wakamatsu; Kiyoko Kaneko; Nobuaki Ogasawara; Shin Fujimori
1177-1179	Effects of Hypoxanthine on Adenosine Transport in Human Lymphocytes. Implications in the Phatogenesis of Lesch–Nyhan Syndrome	R. J. Torres; I. DeAntonio; C. Prior; J. G. Puig
1181-1183	Hypoxanthine Effects on Cyclic AMP Levels in Human Lymphocytes	R. J. Torres; I. DeAntonio; C. Prior; J. G. Puig
1185-1187	Nucleotide Degradation Products in Cerebrospinal Fluid (CSF) in Inherited and Acquired Pathologies	L. D. Fairbanks; J. C. Harris; J. A. Duley; H. A. Simmonds
1189-1191	Are Allopurinol and Metabolites Found in HPRT Deficient Erythrocytes Responsible for Increased NAD Synthesis?	V. Micheli; G. Jacomelli; S. Sestini; L. Notarantonio; B. Cerboni; L. Peruzzi; G. Pompucci
1193-1196	Adenosine Transport in HPRT Deficient Lymphocytes from Lesch-Nyhan Disease Patients	R. J. Torres; I. DeAntonio; C. Prior; J. G. Puig
1197-1199	The Pathophysiology of Hyperuricemia in Essential Hypertension: A Pilot Study	Juan G. Puig; Rosa J. Torres; Luis M. Ruilope; C. Campo; Cristina Grande; Teresa Sancho; José I. Bernardino
1201-1204	Urate Oxidation in CSF and Blood of Patients with Inflammatory Disorders of the Nervous System	B. F. Becker; S. Kastenbauer; U. Ködel; D. Kiesl; H. W. Pfister
1205-1215	Deoxyribonucleoside Kinases in Mitochondrial DNA Depletion	Ann Saada-Reisch
1217-1225	Thymidine Phosphorylase Deficiency Causes MNGIE: An Autosomal Recessive Mitochondrial Disorder	M. Hirano; R. Martí; A. Spinazzola; I. Nishino; Y. Nishigaki
1227-1229	Adenylosuccinate Lyase Deficiency: Study of Physiopathologic Mechanism(s)	V. Race; S. Marie; P. Kienlen-Campard; E. Hermans; J. N. Octave; G. Van den Berghe; M. -F. Vincent
1231-1233	Adenylosuccinate Lyase Deficiency—First British Case	A. M. Marinaki; M. Champion; M. A. Kurian; H. A. Simmonds; S. Marie; M. F. Vincent; G. van den Berghe; J. A. Duley; L. D. Fairbanks
1235-1239	Modulation of Glycogen Phosphorylase Activity Affects 5-Phosphoribosyl-1-Pyrophosphate Availability in Rat Hepatocyte Cultures	Pnina Boer; Oded Sperling
1241-1244	Cyclase and Phosphodiesterase Activity on Pre-T Lymphoid Human Cells, Treated with Dimethyl Sulfoxide (DMSO)	F. Di Pietrantonio; E. Di Matteo; M. Di Nicola; O. Trubiani; R. Di Primio; E. Serra; G. Spoto
1245-1248	Evaluation of ADA Gene Expression and Transduction Efficiency in ADA/SCID Patients Undergoing Gene Therapy	F. Carlucci; A. Tabucchi; A. Aiuti; F. Rosi; F. Floccari; R. Pagani; E. Marinello
1249-1251	Urinary Methylxanthine and Autistic Disorder: Absence of Previously Reported Correlation	C. Salerno; C. Crifò
1253-1255	Biochemical and Molecular Genetic Correlation in Adenylosuccinate Lyase Deficiency	C. Salerno; C. Crifò
1257-1259	Identification of the 5′-Nucleotidase Activity Altered in Neurological Syndromes	R. Pesi; M. Camici; V. Micheli; L. Notarantonio; G. Jacomelli; M. G. Tozzi
1261-1263	The Genetic Basis of the Interaction Between Pyrimidine 5′ Nucleotidase I Deficiency and Hemoglobin E	E. Escuredo; A. M. Marinaki; J. A. Duley; S. L. Thein; D. C. Rees
1265-1267	Elevated Erythrocyte CDP-Choline Levels Associated with β-Thalassaemia in Patients with Transfusion Independent Anaemia	A. D. Laurence; M. Layton; J. A. Duley; H. A. Simmonds

Volume 23, Issue 8-9 (2004)

1269-1274	Mitochondrial Function Dependent Proliferation Assay for the Diagnosis of Mitochondrial Disorders in Human Fibroblasts	Stephen D. Hodges; Floyd F. Snyder
1275-1279	Severe Impairment of Nucleotide Synthesis Through Inhibition of Mitochondrial Respiration	N. Gattermann; M. Dadak; G. Hofhaus; M. Wulfert; M. Berneburg; M. L. Loeffler; H. A. Simmonds
1281-1285	Dihydroorotate Dehydrogenase mRNA and Protein Expression Analysis in Normal and Drug-Resistant Cells	M. Löffler; A. Klein; M. Hayek-Ouassini; W. Knecht; L. Konrad
1287-1293	Estrogen Attenuates P2X₇-R—Mediated Apoptosis of Uterine Cervical Cells by Blocking Calcium Influx	George I. Gorodeski
1295-1299	Liver Transplant: Adenosine Metabolism and Apoptosis	F. Carlucci; E. Marinello; G. Gerunda; D. Neri; F. Rosi; F. Floccari; A. Tabucchi
1301-1303	Serum Folate and Vitamin B12 Levels in Children from Mozambique	R. Leoncini; D. Vannoni; R. Guerranti; G. Cinci; A. Tabucchi; F. Carlucci; E. Marinello; A. B. Agostinho
1305-1311	Immucillins as Antibiotics for T-Cell Proliferation and Malaria	Vern L. Schramm
1313-1320	New (1-Deaza)Purine Derivatives via Efficient C-2 Nitration of the (1-Deaza)Purine Ring	M. J. Wanner; B. Rodenko; M. Koch; G. J. Koomen
1321-1327	6-[2-Phosphonomethoxy)Alkoxy]-2,4-Diaminopyrimidines: A New Class of Acyclic Pyrimidine Nucleoside Phosphonates with Antiviral Activity	J. Balzarini; C. Pannecouque; L. Naesens; G. Andrei; R. Snoeck; E. De Clercq; D. Hocková; A. Holý
1329-1333	Antiproliferative Activity and Mechanism of Action of Fatty Acid Derivatives of Gemcitabine in Leukemia and Solid Tumor Cell Lines and in Human Xenografts	A. M. Bergman; C. M. Kuiper; P. Noordhuis; K. Smid; D. A. Voorn; E. M. Comijn; F. Myhren; M. L. Sandvold; H. R. Hendriks; Ø. Fodstad; K. Breistøl; G. J. Peters
1335-1342	Selective Increase of dATP Pools upon Activation of Deoxycytidine Kinase in Lymphocytes: Implications in Apoptosis	Gergely Keszler; Tatjana Spasokoukotskaja; Zsolt Csapo; Szula Virga; Maria Staub; Maria Sasvari-Szekely
1343-1346	Fluorescence Studies of Substrate Binding to Human Recombinant Deoxycytidine Kinase	R. S. Mani; E. V. Usova; S. Eriksson; C. E. Cass
1347-1350	Quantitative Real Time PCR of Deoxycytidine Kinase mRNA by Light Cycler PCR; in Relation to Enzyme Activity	J. Sigmond; W. J. Loves; J. R. Kroep; G. J. Peters
1351-1356	Immunocytochemical Detection of Deoxycytidine Kinase in Pediatric Malignancies in Relation to In Vitro Cytarabine Sensitivity	I. Hubeek; G. J. Peters; A. J. F. Broekhuizen; I. Talianidis; A. Y. N. Schouten van Meeteren; E. R. van Wering; B. Gibson; U. Creutzig; G. J. L. Kaspers
1357-1361	Stimulation of Deoxycytidine Kinase Results in Prolonged Maintenance of the Enzyme Activity	G. Keszler; T. Spasokoukotskaja; S. Virga; M. Sasvari-Szekely; M. Staub
1363-1365	New Evidences for a Regulation of Deoxycytidine Kinase Activity by Reversible Phosphorylation	C. Smal; L. Bertrand; E. Van Den Neste; S. Cardoen; M. Veiga-da-Cunha; S. Marie; V. Race; A. Ferrant; G. Van den Berghe; F. Bontemps
1367-1370	Upregulation of Platelet Derived Endothelial Cell Growth Factor/Thymidine Phosphorylase by Interferon Alpha	M. de Bruin; K. Smid; M. A. van der Ent; M. Fukushima; H. M. Pinedo; G. J. Peters
1371-1375	Pyrimidine Degradation Defects and Severe 5-Fluorouracil Toxicity	A. B. P. van Kuilenburg; R. Meinsma; A. H. van Gennip
1377-1379	Thymidylate Synthase Polymorphism and Microsatellite Instability: Association in Colorectal Cancer	A. Calascibetta; L. Rausa; L. Gullotti; R. Buettner; R. Sanguedolce
1381-1384	Polymorphism of the Thymidylate Synthase Gene and Thymidylate Synthase Levels in Colon Cancer Cell Lines and Different Tissues of Colorectal Cancer Patients	R. Mauritz; I. J. Beumer; S. Marsh; H. L. McLeod; K. Smid; C. J. van Groeningen; H. M. Pinedo; G. J. Peters

Volume 23, Issue 8-9 (2004)

1385-1391	The Clinical Impact of Thiopurine Methyltransferase Polymorphisms on Thiopurine Treatment	S. A. Coulthard; E. C. Matheson; A. G. Hall; L. A. Hogarth
1393-1397	Mutation in the ITPA Gene Predicts Intolerance to Azathioprine	A. M. Marinaki; J. A. Duley; M. Arenas; A. Ansari; S. Sumi; C. M. Lewis; M. Shobowale-Bakre; L. D. Fairbanks; J. Sanderson
1399-1401	Allele Frequency of Inosine Triphosphate Pyrophosphatase Gene Polymorphisms in a Japanese Population	A. M. Marinaki; S. Sumi; M. Arenas; L. Fairbanks; S. Harihara; K. Shimizu; A. Ueta; J. A. Duley
1403-1405	Genetic Determinants of the Pre- and Post-Azathioprine Therapy Thiopurine Methyltransferase Activity Phenotype	M. Arenas; J. A. Duley; A. Ansari; E. A. Shobowale-Bakre; L. Fairbanks; S. Y. Soon; J. Sanderson; A. M. Marinaki
1407-1409	GTP Concentrations are Elevated in Erythrocytes of Renal Transplant Recipients when Conventional Immunosuppression is Replaced by the Inosine Monophosphate Dehydrogenase Inhibitor Mycophenolic Acid Mofetil (MMF)	D. J. A. Goldsmith; E. A. Carrey; S. M. Edbury; A. M. Marinaki; H. A. Simmonds
1411-1415	Novel Mutations and Hot-Spots in Patients with Purine Nucleoside Phosphorylase Deficiency	Eyal Grunebaum; Junyang Zhang; Chaim M. Roifman
1417-1423	Clofarabine in Adult Acute Leukemias: Clinical Success and Pharmacokinetics	Todd Cooper; Hagop Kantarjian; William Plunkett; Varsha Gandhi
1425-1429	Effects of 2-Chloro-2′-Deoxyadenosine on the Cell Cycle in the Human Leukemia EHEB Cell Line	S. Cardoen; E. Van Den Neste; C. Smal; J. F. Rosier; A. Ferrant; G. Van den Berghe; F. Bontemps
1431-1440	Management of Hyperuricemia with Rasburicase Review	J. M. de Bont; R. Pieters
1441-1444	Selective Transport of a New Class of Purine Antimetabolites by the Protozoan Parasite Trypanosoma brucei	L. J. M. Wallace; D. Candlish; A. Hagos; K. L. Seley; H. P. de Koning
1445-1450	Regulation of Equilibrative Nucleoside Uptake by Protein Kinase Inhibitors	Min Huang; Yanhong Wang; Beverly S. Mitchell; Lee M. Graves
1451-1454	Online Fluorescent Method to Assess BCRP/ABCG2 Activity in Suspension Cells	J. H. Hooijberg; G. J. Peters; G. J. L. Kaspers; P. R. Wielinga; A. J. P. Veerman; R. Pieters; G. Jansen
1455-1457	Metabolism of Adenosine in Human Colorectal Tumour	D. Vannoni; M. C. Di Pietro; F. Rosi; A. Bernini; R. Leoncini; A. Tabucchi; F. Carlucci; F. Floccari; A. Santoro; G. Tanzini; E. Marinello
1459-1465	Cloning and Expression of Malarial Pyrimidine Enzymes	R. I. Christopherson; O. Cinquin; M. Shojaei; D. Kuehn; R. I. Menz
1467-1470	Down–Regulation of Human Deoxyuridine Triphosphate Nucleotidohydrolase (dUTPase) Using Small Interfering RNA (siRNA)	M. V. Williams; A. W. Studebaker
1471-1474	Comparison of mRNA Expression Levels Determined with TAQ–Man and Competitive Template RT–PCR	R. Mauritz; W. Schwabe; P. Haeusler; P. Noordhuis; K. Smid; H. L. McLeod; D. Behnke; C. J. van Groeningen; G. J. Peters
1475-1479	Mechanistic Studies of dUTPases	J. Kovári; T. Imre; P. Szabó; B. G. Vértessy
1481-1484	A Non-Radioactive Sensitive Assay to Measure 5-Fluorouracil Incorporation into DNA of Solid Tumors	P. Noordhuis; U. Holwerda; J. A. M. Van Laar; C. L. Van der Wilt; G. J. Peters
1485-1490	Role of Platelet Derived Endothelial Cell Growth Factor/Thymidine Phosphorylase in Fluoropyrimidine Sensitivity and Potential Role of Deoxyribose-1-Phosphate	M. de Bruin; T. van Capel; K. Smid; K. van der Born; M. Fukushima; K. Hoekman; H. M. Pinedo; G. J. Peters
1491-1494	Intracellular Thymidylate Synthase Inhibition by Trifluorothymidine in FM3A Cells	O. H. Temmink; E. M. Comijn; M. Fukushima; G. J. Peters

Volume 23, Issue 8-9 (2004)

1495-1498	5-Fluoro-2′-Deoxyuridine Has Effects on Mitochondria in CEM T-Lymphoblast Cells	S. Curbo; M. Johansson; A. Karlsson
1499-1502	Effect of Fluoropyrimidines on the Growth of Ureaplasma urealyticum	Rahma Wehelie; Staffan Eriksson; Liya Wang
1503-1506	Combinations of 5-Fluorouracil with UCN-01 or Staurosporine	J. Sigmond; E. M. Comijn; J. A. E. Kamphuis; G. J. Peters
1507-1511	Cytotoxic and Apoptotic Effects of Novel Heterodinucleoside Phosphates Consisting of 5-Fluorodeoxyuridine and Ara-C in Human Cancer Cell Lines	P. Saiko; W. Bauer; Z. Horvath; T. Hoechtl; M. Grusch; C. Illmer; S. Madlener; G. Krupitza; R. M. Mader; H. Schott; M. Fritzer-Szekeres; T. Szekeres
1513-1516	Modulation of Cytarabine Induced Cytotoxicity Using Novel Deoxynucleoside Analogs in the HL60 Cell Line	I. Hubeek; G. J. Peters; A. J. F. Broekhuizen; G. J. L. Kaspers
1517-1521	Increased Cytotoxicity of 2′,2′-Difluoro-2′-Deoxycytidine in Human Leukemic Cell-Lines After a Preincubation with Cyclopentenyl Cytosine	A. C. Verschuur; A. H. Van Gennip; R. Leen; A. B. P. Van Kuilenburg
1523-1526	Antiproliferative Activity and Mechanism of Action of Fatty Acid Derivatives of Arabinosylcytosine (ara-C) in Leukemia and Solid Tumor Cell Lines	A. M. Bergman; C. M. Kuiper; F. Myhren; M. L. Sandvold; H. R. Hendriks; G. J. Peters
1527-1529	Investigation of the Substrate Recognition of Drosophila melanogaster Nucleoside Kinase by Site Directed Mutagenesis	N. Solaroli; M. Bjerke; M. Johansson; A. Karlsson
1531-1535	Combination Chemotherapy of BCNU and Didox Acts Synergystically in 9L Glioma Cells	Zsuzsanna Horvath; Wolfgang Bauer; Thomas Hoechtl; Philipp Saiko; Monika Fritzer-Szekeres; Tarik Tihan; Thomas Szekeres
1537-1539	Comparative Immunologic and Kinetic Evaluation of AMP-Deaminase Isolated from Normal Human Liver and Hepatocellular Carcinoma (HCC)	M. Szydlowska; Z. Sledzinski; M. Krzyzanowski; G. Nagel-Starczynowska; K. Kaletha
1541-1544	Amidox, an Inhibitor of Ribonucleotide Reductase, Potentiates the Action of Ara-C in HL-60 Human Promyelocytic Leukemia Cells	W. Bauer; Z. Horvath; T. Höchtl; P. Saiko; D. Karl; M. Fritzer-Szekeres; T. Szekeres
1545-1549	Potential Role of Mycophenolate Mofetil in the Management of Neuroblastoma Patients	E. Messina; L. Barile; F. Lupi; A. Giacomello
1551-1554	Cyclic Nucleotides and Neuroblastoma Differentiation	E. Messina; F. Lupi; L. Barile; A. Giacomello
1555-1558	Cyclic Guanosine Monophosphate Role in Human Carcinoma Pathogenesis	Maurizio Di Nicola; Fiorenzo Santoleri; Stefano Soscia; Massimiliano Fioroni; Corrado Rubini; Adriano Piattelli; Giuseppe Spoto
1559-1563	Author Index to Abstracts

Volume 23, Issue 6-7 (2004)

xi-xii	Preface
825-829	Alkylation and Cleavage of a DNA Fragment with Trioligonucleotide Reagent	S. I. Oshevski
831-836	Oligonucleosome DNA Fragmentation of Caspase 3 Deficient MCF-7 Cells in Palmitate-Induced Apoptosis	D. V. Semenov; P. A. Aronov; E. V. Kuligina; M. O. Potapenko; V. A. Richter
837-842	Ribonucleic Acids of Human Milk	Elena V. Kuligina; Dmitry V. Semenov; Olesya N. Shevyrina; Vladimir A. Richter
843-847	Expression of the MDR1 and MRP Genes in Patients with Lymphoma with Primary Bone Marrow Involvement	A. N. Zenkov; N. V. Scvortsova; E. L. Chernolovskaya; T. I. Pospelova; V. V. Vlassov
849-853	Oxidative DNA Cleavage by Free and Oligonucleotide-Conjugated O-Bromobenzoic Acid in the Presence of Copper(II) Ions	O. A. Koval; S. B. Oleinikova; V. V. Litvak; V. V. Vlassov; E. L. Chernolovskaya
855-859	Investigation of Tumor-Derived Extracellular DNA in Blood of Cancer Patients by Methylation-Specific PCR	Elena Y. Rykova; Tatyana E. Skvortsova; Pavel P. Laktionov; Svetlana N. Tamkovich; Olga E. Bryzgunova; Andrey V. Starikov; Nina P. Kuznetsova; Sergei A. Kolomiets; Natalia V. Sevostianova; Valentin V. Vlassov
861-866	Silencing of MDR 1 Gene in Cancer Cells by siRNA	E. B. Logashenko; A. V. Vladimirova; M. N. Repkova; A. G. Venyaminova; E. L. Chernolovskaya; V. V. Vlassov
867-872	Silencing of c-myc Expression in Tumor Cells by siRNA	T. O. Kabilova; E. L. Chernolovskaya; A. V. Vladimirova; V. V. Vlassov
873-877	Simple and Rapid Procedure Suitable for Quantitative Isolation of Low and High Molecular Weight Extracellular Nucleic Acids	Svetlana N. Tamkovich; Pavel P. Laktionov; Elena Yu. Rykova; Valentin V. Vlassov
879-883	Extracellular Circulating Nucleic Acids in Human Plasma in Health and Disease	Pavel P. Laktionov; Svetlana N. Tamkovich; Elena Yu. Rykova; Olga E. Bryzgunova; Andrey V. Starikov; Nina P. Kuznetsova; Sergey V. Sumarokov; Sergey A. Kolomiets; Natalya V. Sevostianova; Valentin V. Vlassov
885-890	Ribonuclease Activity of the Peptides with Alternating Arginine and Leucine Residues Conjugated to Tetrathymidilate	N. L. Mironova; Y. I. Boutorine; D. V. Pyshnyi; E. M. Ivanova; M. A. Zenkova; V. V. Vlassov
891-893	In Vitro Selection of Single-Stranded DNA Aptamers that Bind Human Pro-Urokinase	Natalia A. Skrypina; Larissa P. Savochkina; Robert Sh. Beabealashvilli
895-906	Hybridization of Antisense Oligonucleotides with α-Sarcin Loop Region of Escherichia coli 23S rRNA	Vladislav A. Petyuk; Roman N. Serikov; Valentin V. Vlassov; Marina A. Zenkova
907-913	The Role of Hydrophobic Interactions in Catalysis of RNA Cleavage by 1,4-Diazabicyclo[2.2.2]-Octane Based Artificial Ribonucleases	I. Kuznetsova; F. Tuzikov; N. Tuzikova; N. Tamkovich; M. Zenkova; V. Vlassov
915-920	Molecular Design of Artificial Ribonucleases Using Electrostatic Interaction	Ekaterina A. Burakova; Vladimir N. Silnikov
921-925	Photoanalogues of the Initiation Substrates of the RNA Polymerase II, 5-Azido-2-Nitrobenzoyl Derivatives of the ATP γ-Amidophosphate: The Possible Photoinduced Degradation of the Functional Group to an N-Arylhydroxylamine	T. V. Popova; V. S. Mal'shakova; P. V. Alekseyev; N. V. Kudryashova; M. M. Shakirov; L. L. Savinkova; I. A. Drachkova; T. S. Godovikova
927-930	Release of Nucleic Acids by Eukaryotic Cells in Tissue Culture	Evgeniy S. Morozkin; Pavel P. Laktionov; Elena Y. Rykova; Olga E. Bryzgunova; Valentin V. Vlassov
931-934	Preparation of DNA Chips Using Polyamine-Oligonucleotide Conjugates	Asya Levina; Elena Mikhaleva; Valentina Zarytova

Volume 23, Issue 6-7 (2004)

935-942	Properties of Antigenomic Hepatitis Delta Virus Ribozyme Cis- and Trans- Analogs	L. Savochkina; V. Alekseenkova; T. Belyanko; M. Lukin; R. Beabealashvilli
943-951	Binding Features of BCL2-Targeted Oligodeoxynucleotides with K562 Cells	A. M. Timofeev; T. V. Borovkova; T. V. Akhlynina; N. M. Nydenova; N. I. Grineva
953-968	Oligonucleotide—Minor Groove Binder 1:2 Conjugates: Side by Side Parallel Minor Groove Binder Motif in Stabilization of DNA Duplex	Vladimir A. Ryabinin; Alexandre S. Boutorine; Claude Hélène; Alexey Yu. Denisov; Dmitrii V. Pyshnyi; Alexandre N. Sinyakov
969-975	New Photoreactive Oligoribonucleotide Conjugates: Hybridization and Modification Assays	M. Repkova; M. Meshchaninova; A. Venyaminova
977-981	Ribonuclease Activity of Cationic Structures Conjugated to Lipophilic Groups	N. Koval'ov; I. Kuznetsova; E. Burakova; V. Sil'nikov; M. Zenkova; V. Vlassov
983-987	Thermodynamics of Interaction of Phthalocyanine-Oligonucleotide Conjugates with Single- and Double-Stranded DNA	A. A. Chernonosov; N. A. Kuznetsov; V. V. Koval; D. V. Pyshnyi; N. M. Derkacheva; E. A. Lukyanets; O. S. Fedorova
989-992	Toward the Development of Metal-Free Synthetic Nucleases: Cleavage of a Model Substrates by 1,4-Diazabicyclo[2.2.2]Octane Derivatives	Lyudmila S. Koroleva; Vladimir N. Silnikov
993-998	Synthesis of Monomers Bearing at the 2′-Position Cyanomethoxycarbonyl Group for Phosphoramidite Oligonucleotide Synthesis	Svetlana V. Vasilyeva; Tatyana V. Abramova; Vladimir N. Silnikov
999-1001	Assay of Random RNA Oligomerisation in Buffers with High Concentrations of Divalent Metal Ions	Alexander Vlassov
1003-1007	Characteristics of Lipids Imbalance in Patients with Tick-Borne Encephalitis	N. V. Garmashova; F. V. Tuzikov; N. A. Tuzikova; O. B. Tyshkevich; B. M. Doronin; V. N. Buneva; G. A. Nevinsky
1009-1013	Strong Changes in Lipoproteins and Autoantibodies of Blood Serum of the Tundra Nency Population as a Result of Environmental Radiation on the Territory they Inhabit	E. S. Korovkina; F. V. Tuzikov; N. A. Tuzikova; L. P. Osipova; V. N. Buneva; G. A. Nevinsky
1015-1022	Binding Properties of the Conjugates of Oligo(2′-O-Methylribonucleotides) with Minor Groove Binders Targeted to Double Stranded DNA	D. S. Novopashina; A. N. Sinyakov; V. A. Ryabinin; A. G. Venyaminova; L. Perrouault; E. Brunet; C. Giovannangeli; A. S. Boutorine
1023-1030	A New Approach to Revealing Point Mutations in DNA Analyzed by Colorimetric Detection	Marsel Kabilov; Dmitrii Pyshnyi; Grigorii Dymshits; Valentina Zarytova; Evgenia Ivanova
1031-1035	Two-Component 10–23 DNA Enzymes	A. A. Fokina; M. A. Kuznetsova; M. N. Repkova; A. G. Venyaminova
1037-1042	Binary Hammerhead Ribozymes with High Cleavage Activity	M. Kuznetsova; D. Novopashina; M. Repkova; A. Venyaminova; V. Vlassov
1043-1046	Lactoferrin Interacts with Nucleotides	S. E. Babina; G. A. Nevinsky
1047-1051	Efficient Cleavage of DS DNA by Bleomycin Conjugated via Hexaethylene Glycol Linker to Triplex-Forming Oligonucleotides	Pavel Vorobjev; Olessia Tchaika; Valentina Zarytova
1053-1056	Comparison of Enzymatic Properties of DNA-Abzymes and Human DNAses	A. G. Baranovskii; E. S. Odintsova; V. N. Buneva; B. M. Doronin; G. A. Nevinsky
1057-1064	The Influence of Nearest Neighbours on the Efficiency of Coaxial Stacking at Contiguous Stacking Hybridization of Oligodeoxyribonucleotides	Dmitrii V. Pyshnyi; Eugenia M. Ivanova
1065-1071	The Influence of the Non-Nucleotide Insert on the Hybridization Properties of Oligonucleotides	Inna A. Pyshnaya; Dmitrii V. Pyshnyi; Alexander A. Lomzov; Valentina F. Zarytova; Eugenia M. Ivanova
1073-1075	List of Contributors

Volume 23, Issue 5 (2004)

v-vi	List of Contributors
735-748	Synthesis and Antiviral Activities of New Pyrazolo[4,3-c]quinolin-3-ones and Their Ribonucleoside Derivatives	Mara R. P. de Oliveira; Thatyana R. Alves; Angelo C. Pinto; Helena de S. Pereira; Luiz R. Leão-Ferreira; Nissin Moussatché; Izabel Christina de P. P. Frugulhetti; Vitor F. Ferreira; Maria Cecília B. V. de Souza
749-754	Glycosylation Reaction of Unprotected Sugars with Hydroxyalkylthymine	Rachida Zerrouki; Luc Billard; Robert Granet; Pierre Krausz
755-765	Improved Allelic Differentiation Using Sequence-Specific Oligonucleotide Hybridization Incorporating an Additional Base-Analogue Mismatch	David Burgner; Mauro D'Amato; Dominic P. Kwiatkowski; David Loakes
767-775	Solution Stability and Degradation Pathway of Deoxyribonucleoside Phosphoramidites in Acetonitrile	Achim H. Krotz; Claus Rentel; Dennis Gorman; Phil Olsen; Hans J. Gaus; James V. McArdle; Anthony N. Scozzari
777-787	Enzymatic and Hybridization Properties of Oligonucleotide Analogs Containing Novel Phosphoramidate Internucleotide Linkages	Ahmed M. Awad; Michal Sobkowski; Hartmut Seliger
789-803	Oligonucleotide–Minor Groove Binder Conjugates and Their Complexes with Complementary DNA: Effect of Conjugate Structural Factors on the Thermal Stability of Duplexes	Vladimir A. Ryabinin; Alexandre S. Boutorine; Claude Hélène; Dmitrii V. Pyshnyi; Alexandre N. Sinyakov
805-812	Synthesis and Antiviral Evaluation of Some Novel Tricyclic Pyrazolo[3,4-b]indole Nucleosides	John D. Williams; John C. Drach; Leroy B. Townsend
813-822	Synthesis and Antiviral Activity of Novel 2′,4′-Doubly Branched Carbocyclic Nucleosides	Aihong Kim; Joon Hee Hong
823	Erratum

Volume 23, Issue 4 (2004)

v-vi	List of Contributors
647-654	Synthesis and Anti-HIV Activity of 4′-Cyano-2′,3′-didehydro-3′-deoxythymidine	Kazuhiro Haraguchi; Yoshiharu Itoh; Shingo Takeda; Yosuke Honma; Hiromichi Tanaka; Takao Nitanda; Masanori Baba; Ginger E. Dutschman; Yung-Chi Cheng
655-669	The Synthesis of [(β-d-Ribofuranosyloxy)-methyl]nucleosides	Hari Babu Mereyala; Sreeman Kumar Mamidyala
671-690	Design, Efficient Synthesis, and Anti-HIV Activity of 4′-C-Cyano- and 4′-C-Ethynyl-2′-deoxy Purine Nucleosides	Satoru Kohgo; Kohei Yamada; Kenji Kitano; Yuko Iwai; Shinji Sakata; Noriyuki Ashida; Hiroyuki Hayakawa; Daisuke Nameki; Eiichi Kodama; Masao Matsuoka; Hiroaki Mitsuya; Hiroshi Ohrui
691-700	Analysis of Local Convergence in NMR Structure Calculation for RNA by a Classification System for Nucleic Acid Structure (CSNA)	Tatsuhiko Someya; Taiichi Sakamoto; Akitsugu Takasu; Gota Kawai
701-714	Chemoenzymatic Syntheses of Homo- and Heterodimers of AZT and d4T, and Evaluation of Their Anti-HIV Activity	M. Taourirte; L. Ait Mohamed; A. Rochdi; J. -J. Vasseur; S. Fernández; M. Ferrero; V. Gotor; C. Pannecouque; E. De Clercq; H. B. Lazrek
715-724	Synthesis and Biological Evaluation of Novel Apio Nucleosides with Thiazole-4-carboxamide and 1,2,4-Triazole-3-carboxamide	Myong Jung Kim; Lak Shin Jeong; Joong Hyup Kim; Ji Hye Shin; Soon Yong Chung; Sang Kook Lee; Moon Woo Chun
725-734	The Determination of Deoxyribonucleic Acids with Triadimenol Based on the Enhancement of Resonance Light Scattering	Nianqin Jie; Shicong Hou; Fengpei Du; Chunrong Zhang; Guoxin Qin

Volume 23, Issue 3 (2004)

v-vi	List of Contributors
531-544	A Versatile Synthesis of Dihydropyrimidinone C-Nucleosides	Ram Chandra Mishra; Diksha Katiyar; Neetu Tewari; Rama Pati Tripathi
545-554	An Unusual “Senseless” 2′,5′-Oligoribonucleotide With Potent Anti-Hiv Activity	Tarek Aboul-Fadl; Vijai K. Agrawal; Robert W. Buckheit Jr.; Arthur D. Broom
555-565	Molecular Modeling of the Binding of 5-Substituted 2′-Deoxyuridine Substrates to Thymidine Kinase of Herpes Simplex Virus Type-1	Douglas G. Harris; Jianyin Shao; Benjamin D. Morrow; S. Scott Zimmerman
567-580	Reaction of Sugars with 2-Hydrazinopyridine, Precursors for Seco C-Nucleosides of 1,2,4-Triazolo[4,3-a]pyridine	E. S. H. El Ashry; M. M. Abdul-Ghani
581-598	Determination of ATP Impurity in Adenine Dinucleotides	Luminita H. Pojoga; Maricela L. Haghiac; Jana E. Moose; Richard H. Hilderman
599-611	Acyclonucleoside Iron Chelators of 1-(2-Hydroxyethoxy)methyl-2-alkyl-3-hydroxy-4-pyridinones: Potential Oral Iron Chelation Therapeutics	Gang Liu; Ping Men; Gerry H. Kenner; Scott C. Miller; Fred W. Bruenger
613-624	QSAR Analysis for ADA upon Interaction with a Series of Adenine Derivatives as Inhibitors	A. A. Moosavi-Movahedi; S. Safarian; G. H. Hakimelahi; G. Ataei; D. Ajloo; S. Panjehpour; S. Riahi; M. F. Mousavi; S. Mardanyan; N. Soltani; A. Khalafi-Nezhad; H. Sharghi; H. Moghadamnia; A. A. Saboury
625-635	Stereoselective Synthesis of Novel 4′-Branched and Bicyclo[3.1.0]hexane-Templated Nucleoside	Joon Hee Hong
637-646	Bis-Ketol Nucleoside Triesters as Prodrugs of the Antiviral Nucleoside Triphosphate Analogues of 3′-Deoxythymidine and 3′-Deoxy-2′,3′-didehydrothymidine	Kim C. Calvo; Xiaohong Wang; Gerald F. Koser

Volume 23, Issue 1-2 (2004)

xi-xiii	List of Contributors
1-5	Synthesis and Antiviral Evaluation of Some 3′-Fluoro Bicyclic Nucleoside Analogues	Christopher McGuigan; Antonella Carangio; Robert Snoeck; Graciela Andrei; Erik De Clercq; Jan Balzarini
7-29	Synthesis and Antiviral Activity of Novel Fluorinated 2′,3′-Dideoxynucleosides	Piyush Kumar; Kazue Ohkura; Jan Balzarini; Erik De Clercq; Koh-ichi Seki; Leonard I. Wiebe
31-39	An Improved Total Synthesis of Triciribine: A Tricyclic Nucleoside with Antineoplastic and Antiviral Properties	Anthony R. Porcari; Leroy B. Townsend
41-50	Tandem Mass Spectrometry for Structure Assignments of Wye Nucleosides from Transfer RNA	Shaolian Zhou; Devarasetty Sitaramaiah; Steven C. Pomerantz; Pamela F. Crain; James A. McCloskey
51-66	Nucleosides. LXV. Synthesis of New Pteridine–N₈–Nucleosides	Stefan Matysiak; Bernhard Waldscheck; Wolfgang Pfleiderer
67-76	1-Deaza-5′-noraisteromycin	Xueqiang Yin; Stewart W. Schneller
77-88	How a Modification (8-Aza-3-deaza-2′-deoxyguanosine) Influences the Quadruplex Structure of Hotoda's 6-Mer TGGGAG with 5′- and 3′-End Modifications	Suzana Jakša; Bogdan Kralj; Christophe Pannecouque; Jan Balzarini; Erik De Clercq; Jože Kobe
89-115	Second Generation of cycloSal-Pronucleotides with Esterase-Cleavable Sites: The ”Lock-In”-Concept	Chris Meier; Manuel F.H. Ruppel; Dalibor Vukadinović; Jan Balzarini
117-126	Rearrangement Reactions of 1,N²-Isopropenoguanine Cyclonucleosides	Tomasz Zandecki; Jerzy Boryski
127-136	An Efficient Route to Novel 4,5-Di- and 2,4,5-Tri Substituted Imidazoles from Imidazo[1,5-a]-1,3,5-triazine (5,8-Diaza-7,9-dideazapurine) Derivatives	Bozenna Golankiewicz; Piotr Januszczyk; Joanna Zeidler; Mariusz Popenda
137-147	Functionalization of Guanosine and 2′-Deoxyguanosine at C6: A Modified Appel Process and S_NAr Displacement of Imidazole	Zlatko Janeba; Xiaoyu Lin; Morris J. Robins
149-160	Biologically Active Antisense Phosphorothioate Oligodeoxyribonucleotides: Synthesis, Characterization, and Studies of 3′-Terminal Phosphorothioate Monoester Analogues	Vasulinga T. Ravikumar; Walt F. Lima; Kent Van Sooy; Brett Turney
161-170	Synthesis and Biological Activity of 5-Fluorotubercidin	Xiaojing Wang; Punit P. Seth; Ray Ranken; Eric E. Swayze; Michael T. Migawa
171-181	Improved and Reliable Synthesis of 3′-Azido-2′,3′-dideoxyguanosine Derivatives	Victor A. Timoshchuk; Richard I. Hogrefe; Morteza M. Vaghefi
183-193	A New Approach for the Synthesis of Novel 5-Substituted Isodeoxyuridine Analogs	Sven Guenther; Vasu Nair
195-205	Synthesis of Uridine 5′-[2-S-Pyridyl-3-thio-α-d-galactopyranosyl Diphosphate]: Precursors of UDP-Thiogal Sugar Nucleotide Donor Substrate for β-1,4-Galactosyltransferase	Jordan Elhalabi; Kevin G. Rice
207-225	Intercalating Nucleic Acids: The Influence of Linker Length and Intercalator Type on Their Duplex Stabilities	Ulf B. Christensen; Michael Wamberg; Farag A. G. El-Essawy; Abd El-Hamid Ismail; Christina B. Nielsen; Vyacheslav V. Filichev; Carsten H. Jessen; Michael Petersen; Erik B. Pedersen
227-237	Regioselective Synthesis of Indazole N¹- and N²-(β-d-Ribonucleosides)	Frank Seela; Xiaohua Peng
239-253	Synthesis of Tunicaminyluracil Derivatives	Satoshi Ichikawa; Akira Matsuda
255-262	New Sequential-Assignment Routes of Nucleic Acid NMR Signals Using a [5′-¹³C]-Labeled DNA Dodecamer	Etsuko Kawashima; Takeshi Sekine; Kaoru Umabe; Kazuo Kamaike; Toshimi Mizukoshi; Nobuhisa Shimba; Ei-ichiro Suzuki; Chojiro Kojima
263-271	Inhibitors of Adenosine Deaminase: Continued Studies of Structure-Activity Relationships in Analogues of Coformycin	Ayub Reayi; Ramachandra S. Hosmane
273-280	Use of Both Direct and Indirect ¹³C Tags for Probing Nitrogen Interactions in Hairpin Ribozyme Models by ¹⁵N NMR	Anthony J. Shallop; Barbara L. Gaffney; Roger A. Jones
281-289	The Interaction of Per-O-Acetylated Acyclic 1-(1-Butylindol-3-yl)-1-deoxy-ketoses with Silylated Uracil	S. N. Lavrenov; N. P. Solovyeva; M. I. Reznikova; O. S. Anisimova; M. N. Preobrazhenskaya

Volume 23, Issue 1-2 (2004)

291-306	Tissue Disposition of 5-o-Carboranyluracil—A Novel Agent for the Boron Neutron Capture Therapy of Prostate Cancer	Raymond F. Schinazi; Selwyn J. Hurwitz; Irina Liberman; Yuliya Glazkova; Nicolas S. Mourier; Jeffrey Olson; Thomas Keane
307-316	Synthesis of 4-Formyl-4-imidazolin-2-one Nucleosides, Isomers of Uridine and 2′-Deoxyuridine	Xiang-Jun Jiang; Thomas I. Kalman
317-337	Synthesis of Azole Nucleoside 5′-Monophosphate Mimics (P1Ms) and Their Inhibitory Properties of IMP Dehydrogenases	Guangyi Wang; Kandasamy Sakthivel; Vasanthakumar Rajappan; Thomas W. Bruice; Kathleen Tucker; Patrick Fagan; Jennifer L. Brooks; Tiffany Hurd; Janet M. Leeds; P. Dan Cook
339-346	Effect of Imino Group of a Linker Arm at the C5 Position of a Pyrimidine Nucleoside on the Thermal Stabilities of DNA/DNA and DNA/RNA Duplexes	Hiroaki Ozaki; Masayuki Mine; Kazuo Shinozuka; Hiroaki Sawai
347-359	Nucleosides. IX. Synthesis of Purine N³,5′-Cyclonucleosides and N³,5′-Cyclo-2′,3′-seconucleosides via Mitsunobu Reaction as TIBO-like Derivatives	Grace Shiahuy Chen; Chien-Shu Chen; Tun-Cheng Chien; Jun-Yen Yeh; Chia-Chi Kuo; Rahul Subhash Talekar; Ji-Wang Chern
xv-xxiii	Introduction
361-373	Uridine Recognition Motifs of Human Equilibrative Nucleoside Transporters 1 and 2 Produced in Saccharomyces cerevisiae	Mark F. Vickers; Jing Zhang; Frank Visser; Tracey Tackaberry; Morris J. Robins; Lars P. C. Nielsen; Ireneusz Nowak; Stephen A. Baldwin; James D. Young; Carol E. Cass
375-383	Anti-cowpox Virus Activities of Certain Adenosine Analogs, Arabinofuranosyl Nucleosides, and 2′-Fluoro-arabinofuranosyl Nucleosides	Donald F. Smee; Robert W. Sidwell
385-399	Synthesis and Evaluation of a Novel Synthetic Phosphocholine Lipid-AZT Conjugate That Double-Targets Wild-Type and Drug Resistant Variants of HIV	Louis S. Kucera; Susan L. Morris-Natschke; Khalid S. Ishaq; Jan Hes; Nathan Iyer; Phillip A. Furman; Ronald A. Fleming
401-410	Enhanced DNA-Directed Effects of FdUMP[10] Compared to 5FU	William H. Gmeiner; Eric Trump; Cui Wei
411-438	Synthesis of 2′-Substituted MMI Linked Nucleosidic Dimers: An Optimization Study in Search of High Affinity Oligonucleotides for Use in Antisense Constructs	Didier Peoc'h; Eric E. Swayze; Balkrishen Bhat; Yogesh S. Sanghvi
439-455	Synthesis of D-Altritol Nucleosides with a 3′-O-Tert-Butyldimethylsilyl Protecting Group	Michael Abramov; Arnaud Marchand; Agnes Calleja-Marchand; Piet Herdewijn
457-470	Nucleoside Analogues Exerting Antiviral Activity Through a Non-nucleoside Mechanism	Erik De Clercq
471-481	A_2B Adenosine Receptor Agonists: Synthesis and Biological Evaluation of 2-Phenylhydroxypropynyl Adenosine and NECA Derivatives	S. Vittori; S. Costanzi; C. Lambertucci; F. R. Portino; S. Taffi; R. Volpini; K.-N. Klotz; G. Cristalli
483-493	Monitoring the Intracellular Metabolism of Nucleoside Phosphoramidate Pronucleotides by ³¹P NMR	Jisook Kim; Daniel P. Drontle; Carston R. Wagner
495-499	Synthesis of Nucleoside Libraries on Solid Support. I. N²,N⁶-Disubstituted Diaminopurine Nucleosides	Esmir Gunic; Roberto Amador; Frank Rong; Jeffrey W. Abt; Haoyun An; Zhi Hong; Jean-Luc Girardet
501-507	Synthesis of Nucleoside Libraries on Solid Support. II. 2,6,8-Trisubstituted Purine Nucleosides Using 8-Bromoguanosine as Precursor	Yung-hyo Koh; Michael B. Landesman; Roberto Amador; Frank Rong; Haoyun An; Zhi Hong; Jean-Luc Girardet
509-520	Oligonucleotide Conjugates of Nile Red	Igor A. Prokhorenko; Natalia N. Dioubankova; Vladimir A. Korshun
521-530	Conformational Flexibility in a Triazole Nucleoside Derivative: 4-Cyano-5-cyanomethyl-1-(2,3,5-tri-O-acetyl-β-d-ribofuranosyl)-1,2,3-triazole	Ivan Leban; Marjan Ješelnik; Joachim Sieler; Jože Kobe

Volume 22, Issue 12 (2003)

v-vi	List of Contributors
ix-x	Introduction
2077-2091	Synthesis and Conformational Analysis of a Locked Analogue of Carbovir Built on a Bicyclo[3.1.0]-hex-2-enyl Template	Yongseok Choi; Guangyu Sun; Clifford George; Marc C. Nicklaus; James A. Kelley; Victor E. Marquez
2093-2104	Studies Towards the Large Scale Chemical Synthesis of the Precursors of Ribonucleosides-3′,4′,5′,5″-²H₄ and -2′,3′,4′,5′,5″-²H₅	András Földesi; Jyoti Chattopadhyaya
2105-2119	Efficacy of Methylenecyclopropane Analogs of Nucleosides Against Herpesvirus Replication In Vitro	Nicole L. Kushner; Stephanie L. Williams; Caroll B. Hartline; Emma A. Harden; Deborah J. Bidanset; Xinchao Chen; Jiri Zemlicka; Earl R. Kern
2133-2144	Design and Synthesis of a Series of Chlorinated 3-Deazaadenine Analogues	Katherine L. Seley; Peter I. O'Daniel; Samer Salim
2145-2160	Synthesis of Base Substituted 2-Hydroxy-3-(purin-9-yl)-propanoic Acids and 4-(Purin-9-yl)-3-butenoic Acids	Petra Doláková; Milena Masojídková; Antonín Holý
2161-2170	Synthesis and Anti-cancer Activity of Some Novel 5-Azacytosine Nucleosides	Kamal N. Tiwari; Loredana Cappellacci; John A. Montgomery; John A. Secrist III
2171-2193	Synthesis and Antiviral Activity of 2-Substituted Analogs of Triciribine	Anthony R. Porcari; Roger G. Ptak; Katherine Z. Borysko; Julie M. Breitenbach; John C. Drach; Leroy B. Townsend
2195-2202	Synthesis and Studies of 3′-C-Trifluoromethyl-β-D-ribonucleosides Bearing the Five Naturally Occurring Nucleic Acid Bases	Frédéric Jeannot; Gilles Gosselin; Christophe Mathé
2203-2215	Author Index to Volume 22
2217-2231	Subject Index to Volume 22

Volume 22, Issue 11 (2003)

v-vi	List of Contributors
1985-1993	Synthesis of 3′-Deoxy-3′-[4-(pyrimidin-1-yl)methyl-1,2,3-triazol-1-yl]thymidine via 1,3-Dipolar Cycloaddition	M. Tourirte; T. Oulih; H. B. Lazrek; J. L. Barascut; J. L. Imbach; N. A. Almasoudi
1995-2001	5′-Nor Carbocyclic Ribavirin	Meral Tuncbilek; Stewart W. Schneller
2003-2011	Novel Chiral Phosphoramidite Monomers from (R)- and (S)-1,3-Butanediol: Synthesis of Modified Oligonucleotides and Binding Affinity Studies	Su Jeong Kim; Byeang Hyean Kim
2013-2026	Synthesis and Biological Evaluation of Some 5-Nitro- and 5-Amino Derivatives of 2′-Deoxycytidine, 2′,3′-Dideoxyuridine, and 2′,3′-Dideoxycytidine	Evelina Colacino; Giovanni Sindona; Gilles Gosselin; Christophe Mathé
2027-2038	Synthesis and Anti-HBV Activity of Thiouracils Linked via S and N-1 to the 5-Position of Methyl β-D-Ribofuranoside	Adel A. -H. Abdel-Rahman; Ahmed E. -S. Abdel-Megied; Adel E. -S. Goda; Ibrahim F. Zeid; El Sayed H. El Ashry
2039-2048	Synthesis of 2-(3′-Azido- and 3′-Amino-3′-deoxy-β-D-ribofuranosyl)thiazole-4-carboxamide	Cheng Wu Liang; Myong Jung Kim; Lak Shin Jeong; Moon Woo Chun
2049-2060	Synthesis, Anti-HIV, and Cytotoxic Activity of New AZT Conjugates of Steroid Acids	Zhengqing You; A. Moshin Mian; Ram P. Agarwal; Henry Joung Lee
2061-2076	A New Approach to the Synthesis of Benzothiazole, Benzoxazole, and Pyridine Nucleosides as Potential Antitumor Agents	Ahmed I. Khodair; Najim A. Al-Masoudi; Jean-Pierre Gesson

Volume 22, Issue 10 (2003)

v-vi	List of Contributors
1859-1866	Study on the Interaction Between Nucleic Acids and Acetamiprid	Nianqin Jie; Shicong Hou; Fengpei Du; Linrui Huang; Guibin Jiang; Suqin Lv
1867-1897	Thiosugars. X. Novel Nucleoside Analogues Derived from 4-Thio-L-lyxofuranose	Jörn Wirsching; Jürgen Voss; Anja Giesler; Jürgen Kopf; Gunadi Adiwidjaja; Jan Balzarini; Erik De Clercq
1899-1905	Convenient Synthesis of 2′-Deoxy-2-fluoroadenosine from 2-Fluoroadenine	Song Ye; Martha M. Rezende; Wei-Ping Deng; Kenneth L. Kirk
1907-1917	Design and Synthesis of Acyclic Nucleoside Analogs with Chlorinated Imidazo[1,2-a]pyridine Bases	John D. Williams; Alaa E. Mourad; John C. Drach; Leroy B. Townsend
1919-1925	A Short, Efficient Synthesis of 2′-Deoxypseudoisocytidine Based on Heck-Chemistry	Alain Mayer; Christian J. Leumann
1927-1938	Enhancement and Inhibition by 2′-O-Hydroxyethyl Residues of Gene Targeting Mediated by Triple Helix Forming Oligonucleotides	Mrinalkanti Kundu; Fumi Nagatsugi; Alokes Majumdar; Paul S. Miller; Michael M. Seidman
1939-1952	Synthesis, Protonation Behavior, Conformational Analysis, and Regioselective Enzymatic Acylation of the Novel Diamino Analogue of (E)-5-(2-Bromovinyl)-2′-deoxyuridine (BVDU)	Iván Lavandera; Susana Fernández; Miguel Ferrero; Erik De Clercq; Vicente Gotor
1953-1961	Phosphoramidate Protides of 2′,3′-Dideoxy-3′-fluoroadenosine and Related Nucleosides with Potent Activity Against HIV and HBV	Kristjan S. Gudmundsson; Susan M. Daluge; Lance C. Johnson; Robert Jansen; Richard Hazen; Lynn D. Condreay; Christopher McGuigan
1963-1983	PNA-DNA Chimeras Containing 5-Alkynyl-pyrimidine PNA Units. Synthesis, Binding Properties, and Enzymatic Stability	Zoltán Bajor; Gyula Sági; Zsuzsanna Tegyey; Ferenc Kraicsovits

Volume 22, Issue 9 (2003)

v-vi	List of Contributors
1737-1746	A Convenient Method for the Synthesis of 2-(β-D-Glycopyranosylthio) Pyridines	Adel M. E. Attia; Ashraf A. El-Shehawy
1747-1755	Open-Chain Carbocyclic Analogs of Adenosine with Dihalovinyl Unit as Potential Inhibitors of S-Adenosyl-L-homocysteine Hydrolase	Elzbieta Lewandowska; Jennifer Lalama; Chong-Sheng Yuan; Stanislaw F. Wnuk
1757-1780	Characterization and Elucidation of Coordination Requirements of Adenine Nucleotides Complexes with Fe(II) Ions	Yael Richter; Bilha Fischer
1781-1788	Novel Synthesis of 4′C-Aryl-Branched Acyclic Nucleoside Using [3,3]-Sigmatropic Rearrangement	Gun Ha Baik; Bong Young Chung; Chang-Hyun Oh; Jung-Hyuck Cho; Ok Hyun Ko; Joon Hee Hong
1789-1803	3′-Azido-3′-deoxy-5′-O-isonicotinoylthymidine: A Novel Antiretroviral Analog of Zidovudine. II. Stability in Aqueous Media and Experimental and Theoretical Ionization Constants	Silvina A. Teijeiro; Mónica A. Raviolo; Marisa I. Motura; Margarita C. Briñón
1805-1823	Synthesis of Some New 2-α-L-Arabinopyranosyl-1,2,4-triazines as Potential Antitumor Chemotherapeutics	Abdel Kader Mansour; Mohga M. Eid; Nasser S. A. M. Khalil
1825-1833	Synthesis of Some N-Galactosides of 3-Aryl-5-benzyl (or Substituted Benzyl)-1,2,4-triazin-6(1H)-/ones or Thiones of Expected Biological Activity	Abdel Kader Mansour; Mohga M. Eid; Nasser S. A. M. Khalil
1835-1855	Permanganate Oxidation Reactions of DNA: Perspective in Biological Studies	Chinh T. Bui; Kylee Rees; Richard G. H. Cotton
1857-1858	Erratum

Volume 22, Issue 5-8 (2003)

489-505	Oligonucleotides and Derivatives as Gene-Specific Control Agents	Jian-Sheng Sun; Claude Hélène
507-517	An Industrial Process for Synthesizing Lodenosine (FddA)	Kunisuke Izawa; Satoshi Takamatsu; Satoshi Katayama; Naoko Hirose; Shigetaka Kozai; Tokumi Maruyama
519-534	Ribonucleotide Reductases: Radical Chemistry and Inhibition at the Active Site	Morris J. Robins
535-546	Inhibition of Transcription by bisPNA-Peptide Conjugates	Xin Zhao; Kunihiro Kaihatsu; David R. Corey
547-557	Recent Advances in the Synthesis of Conformationally Locked Nucleosides and Their Success in Probing the Critical Question of Conformational Preferences by Their Biological Targets	Yongseok Choi; Hyung R. Moon; Yuichi Yoshimura; Victor E. Marquez
559-571	Structures of Non-canonical Tandem Base Pairs in RNA Helices: Review	Hans A. Heus; Cornelis W. Hilbers
573-576	Pyrazolo[3,4-d]pyrimidine Nucleic Acids: Adjustment of the dA-dT to the dG-dC Base Pair Stability	J. He; G. Becher; S. Budow; F. Seela
577-581	Oligonucleotide N3′ → P5′ Thio-phosphoramidate Telomerase Template Antagonists as Potential Anticancer Agents	Sergei Gryaznov; Akira Asai; Yuko Oshima; Yoshihiro Yamamoto; Krisztina Pongracz; Ronald Pruzan; Ellen Wunder; Mieczyslaw Piatyszek; Shihong Li; Allison Chin; Calvin Harley; Shiro Akinaga; Yoshinori Yamashita
583-587	MDPSCL₂: A New Protecting Group for Chemoselective Synthesis of 2′-O-Alkylated Guanosines	Suetying Chow; Ke Wen; Yogesh S. Sanghvi; Emmanuel A. Theodorakis
589-592	Synthesis and Biological Evaluation of Halo-neplanocin A as Novel Mechanism-Based Inhibitors of S-Adenosylhomocysteine Hydrolase	Lak Shin Jeong; Hyung Ryong Moon; Jae Gyu Park; Dae Hong Shin; Won Jun Choi; Kang Man Lee; Hea Ok Kim; Moon Woo Chun; Hee-Doo Kim; Joong Hyup Kim
593-599	Phosphono Peptide Nucleic Acids with a Constrained Hydroxyproline-Based Backbone	Vladimir A. Efimov; Valeryi N. Klykov; Oksana G. Chakhmakhcheva
601-604	LNA and α-L-LNA: Towards Therapeutic Applications	Jesper Wengel; Birte Vester; Lars Bo Lundberg; Stephen Douthwaite; Mads D. Sørensen; B. Ravindra Babu; Michael J. Gait; Andrey Arzumanov; Michael Petersen; Jakob T. Nielsen
605-609	Synthesis and Biological Evaluation of β-D-Pentofuranonucleoside Derivatives of 2-Azidoadenine and 6-Azidopurines	Christophe Mathé; Thierry Lioux; Gilles Gosselin
611-615	2′-Fluoro-4′-thio-2′,3′-unsaturated Nucleosides: Anti-HIV Activity, Resistance Profile, and Molecular Modeling Studies	Youhoon Chong; Hyunah Choo; Raymond F. Schinazi; Chung K. Chu
617-621	Developing Synthetic Methods for Bioactive Phosphorus Compounds Using H-Phosphonate Chemistry: A Progress Report	Martin Bollmark; Tommy Johansson; Martin Kullberg; Johan Nilsson; Jacek Stawinski; Jacek Cieslak; Jadwiga Jankowska; Michal Sobkowski; Marzena Szymczak; Malgorzata Wenska; Adam Kraszewski
623-627	Preparation and Properties of a New Type of Acyclic, Achiral Nucleoside Analogue	Thomas Boesen; Daniel Sejer Pedersen; Jacob Jensen; Michael T. Munck; Brian M. Nielsen; Asger B. Petersen; Ulla Henriksen; Britta M. Dahl; Otto Dahl
629-633	A Short, Novel, and Cheaper Procedure for Oligonucleotide Synthesis Using Automated Solid Phase Synthesizer	Quanlai Song; Zhiwei Wang; Yogesh S. Sanghvi
635-639	Convenient Synthesis of Oligodeoxynucleotides Containing 2′-Deoxy-6-thioinosine	Christine Beuck; Elmar Weinhold
641-644	A Role for Oligonucleotide-Based RNA-Knock Down Technologies in Functional Genomics	Gabriele Dorn; Jonathan Hall; Dieter Hüsken; Jörg Lange; Pierre Martin; Francois Natt; William L. Wishart; Jan Weiler
645-648	Properties of Triple Helices Formed by Oligonucleotides Containing 8-Aminopurines	A. Aviñó; M. Frieden; J. C. Morales; B. G. de la Torre; R. Güimil-García; M. Orozco; C. González; R. Eritja
649-652	Labeling During Cleavage of Nucleic Acids for Their Detection on DNA Chips	A. Laayoun; I. Sothier; L. Menou; E. Bernal-Méndez; M. Kotera; C. Bourget; E. Trévisiol; J. Lhomme; A. Troesch
653-658	Structural Basis for Topoisomerase I Inhibition by Nucleoside Analogs	William H. Gmeiner; Shuyuan Yu; Richard T. Pon; Philippe Pourquier; Yves Pommier
659-661	Synthesis of (Z)-(1-Fluoro-2-hydroxymethyl-cyclopropylmethyl)purines	Ju-Hyun Park; Young Rang Lee; Moon Woo Chun; Lak Shin Jeong; Chong-Kyo Lee; Hee-Doo Kim
663-666	Cyclic Uridine Diphosphate Glucose: A New Pyrimidine Analog of Cyclic ADP Ribose	Marco Cipolletta; Marcella de Champdoré; Lorenzo De Napoli; Giovanni Di Fabio; Anna Messere; Daniela Montesarchio; Gennaro Piccialli
667-669	A New Approach for Syntheses of 2′,3′-Dideoxy- 2′,3′-dehydronucleosides Using 2,2-Difluoro- 1,3-dimethylimidazolidine (DFI) as a Dehydrating Reagent	Hideki Umetani; Hiroshi Sonoda; Hironori Komatsu
671-673	Synthesis of New Pseudonucleosides Containing Chiral Cyclosulfamides as Agycone	Malika Berredjem; Nour-Eddine Aouf
675-677	Synthesis of Thymine Derivatives of 4-Hydroxyvaline	Achamma Abraham; Nicola M. Howarth
679-681	Doped Natural Phosphate: A New and Environmentally Friendly Catalyst in Nucleoside Synthesis	A. Rochdi; M. Taourirte; N. Redwane; S. Sebti; J. W. Engels; H. B. Lazrek
683-685	Synthesis of Carbocyclic Analogues of Thymidine	O. R. Ludek; C. Meier
687-689	The Regiospecific One-Pot Phosphorylation of Either the 5′- or 2′-Hydroxyl in 3′-Deoxycytidines Without Protection: Critical Role of the Base	Peter D. Howes; Martin J. Slater; Katrina Wareing
691-694	Synthesis of Novel mRNA 5′ Cap-Analogues: Dinucleoside P¹, P³-Tri-, P¹, P⁴-Tetra-, and P¹, P⁵-Pentaphosphates	Jacek Jemielity; Janusz Stepinski; Magdalena Jaremko; Dorota Haber; Ryszard Stolarski; Robert E. Rhoads; Edward Darzynkiewicz
695-697	New Solid Supports Linking Nucleoside Scaffolds	Marcella de Champdoré; Lorenzo De Napoli; Giovanni Di Fabio; Anna Messere; Daniela Montesarchio; Gennaro Piccialli
699-701	One-Pot Synthesis of an AZT Boranophosphate Conjugated with Tyrosine: A Potential Prodrug Candidate	Ping Li; Barbara Ramsay Shaw
703-705	Development of a Nucleoside Analog UV Light Sensor	Shiyue Fang; Yousheng Guan; Ernest R. Blatchley III; Lian-Shin Lin; Cheng Yue Shen; Donald E. Bergstrom
707-709	4′-C-Methyl-β-D-ribofuranosyl Purine and Pyrimidine Nucleosides Revisited	J. -F. Griffon; D. Dukhan; C. Pierra; S. Benzaria; A. G. Loi; P. La Colla; J. -P. Sommadossi; G. Gosselin
711-713	A Facile Synthetic Method for 3′-α-Fluoro- 2′,3′-dideoxyadenosine	Satoshi Takamatsu; Satoshi Katayama; Masaki Naito; Keizo Yamashita; Takashi Ineyama; Kunisuke Izawa
715-717	A Zero-Length Diazirine Photoactive Nucleoside	M. Taranenko; M. Mtchedlidze; N. Sumbatyan; G. Korshunova
719-721	Synthesis and Biological Evaluation of Pyrimidine Nucleosides Fused with 3′,4′-Tetrahydrofuran Ring	Moon Woo Chun; Myong Jung Kim; Hea Ok Kim; Hyung Ryong Moon; Hee-Doo Kim; Joong Hyup Kim; Lak Shin Jeong
723-725	Bi- and Tricyclic Nucleoside Derivatives Restricted in S-Type Conformations and Obtained by RCM-Reactions	Nanna Albæk; Jacob Ravn; Morten Freitag; Helena Thomasen; Nanna K. Christensen; Michael Petersen; Poul Nielsen

Volume 22, Issue 5-8 (2003)

727-729	Synthetic Studies on Guanofosfocin: Glycosylation of 8-Oxo-purine Nucleosides via Mitsunobu Reaction	Hideyuki Sugimura; Akiyoshi Koizumi; Wataru Kiyohara
731-733	A New Type of Acyclic, Achiral Nucleoside Analogue. How Does It Simulate Nucleosides?	Asger B. Petersen; Thomas Boesen; Otto Dahl
735-737	Rearrangement Reactions of Guanosine Cyclonucleosides and Their Analogs	Jerzy Boryski; Tomasz Zandecki
739-742	Diastereo- and Enantioselective Synthesis of 1′-C-Branched N, O-Nucleosides	M. G. Saita; U. Chiacchio; D. Iannazzo; A. Corsaro; P. Merino; A. Piperno; T. Previtera; A. Rescifina; G. Romeo; R. Romeo
743-745	Reactivity Models of 1-N-Vinyluracil and Synthesis of a New Class of Potential Antiviral Agents by the Use of 1,3-Dipolar Cycloaddition Reactions	E. Colacino; G. De Luca; A. Liguori; A. Napoli; C. Siciliano; G. Sindona
747-749	Selective Metalation of 6-Methylpurines: Synthesis of 6-Fluoromethylpurines and Related Nucleosides	Abdalla E. A. Hassan; William B. Parker; Paula W. Allan; John A. Montgomery; John A. Secrist III
751-753	Chemo-enzymatic Synthesis of 3-Deoxy-β-D-ribofuranosyl Purines and Study of Their Biological Properties	Vladimir N. Barai; Anatoli I. Zinchenko; Ludmilla A. Eroshevskaya; Elena V. Zhernosek; Jan Balzarini; Erik De Clercq; Igor A. Mikhailopulo
755-758	Efficient Synthesis of 8-Thiosubstituted Guanine Derivatives as Potential Tools for Biochemical and Biological Studies	Martins Ikaunieks; Marina Madre
759-761	Synthesis of Carbocyclic Analogues of MECA and NECA 1,2-Disubstituted as Potential Adenosine Receptor Agonists	P. Besada; M. J. González-Moa; C. Terán; M. Teijeira; L. Santana
763-765	4-Thiofuranoid Glycals: Versatile Synthons for Stereoselective Synthesis of 4′-Thionucleosides	Kazuhiro Haraguchi; Haruhiko Takahashi; Hiromichi Tanaka
767-769	Stannylation Approach to the Synthesis of 2′- and 3′-Substituted Analogues of 2′,3′-Didehydro-2′,3′-dideoxynucleosides	Hiroki Kumamoto; Sayoko Onuma; Hiromichi Tanaka
771-773	Practical Synthesis of D-Cyclopent-2-enone, the Key Intermediate of Carbocyclic Nucleosides	Y. H. Jin; C. K. Chu
775-777	Covalent Analogues of Nucleobase-Pairs	Michal Hocek; Dalimil Dvořák; Martina Havelková
779-781	Introduction of a Benzyl Group onto the 2′-OH of 6-Chloropurine 3′-O-Benzoylriboside	Shigetada Kozai; Tomoyo Fuzikawa; Keisuke Harumoto; Tokumi Maruyama
783-785	Stereocontrolled Synthesis of Diene and Enyne Sugar-Modified Nucleosides and Their Interaction with S-Adenosyl-L-homocysteine Hydrolase	Stanislaw F. Wnuk; Pablo R. Sacasa; Leigh N. Crain; Elzbieta Lewandowska; Jinsong Zhang; Ronald T. Borchardt
787-789	Purine Derivatives of 1,2-Disubstituted Cyclohexane Analogues of Nucleosides	C. Terán; L. Santana; E. Uriarte; D. Viña; E. De Clercq
791-795	Study of Different Substituted Cyclic and Acyclic Benzylpronucleotides of d4T Relative to Their Hydrolytic Stability and Antiviral Activity	U. Muus; E. De Clercq; J. Balzarini; L. Naesens; C. Meier
797-799	Stereochemical Analysis of Diastereomeric 1,3-bis(Adenosine-5′-O-phosphorothioyl)glycerols	Alina Owczarek; Renata Kaczmarek; Barbara Mikołajczyk; Ewa Wasilewska; Dariusz Korczyński; Janina Baraniak; Maria Koziołkiewicz; Wojciech J. Stec; Charles Brenner
801-804	Design of Mycobacterium tuberculosis Thymidine Monophosphate Kinase Inhibitors	H. Munier-Lehmann; S. Pochet; L. Dugue; O. Dutruel; G. Labesse; D. Douget
805-807	5′-O-Ester Prodrugs of Potent and Selective Anti-HIV Agent—2′,3′-Dideoxy-3′-fluoro-2-thiothymidine (S²FLT): Synthesis and Anti-HIV Activity	A. Miazga; N. E. Poopeiko; A. Piasek; M. A. Siweckar; T. Kulikowski
809-812	2-Phenylhydroxypropynyladenosine Derivatives as High Potent Agonists at A_2B Adenosine Receptor Subtype	C. Lambertucci; R. Volpini; S. Costanzi; S. Taffi; S. Vittori; G. Cristalli
813-815	Synthesis and Biological Activity of 2-Aminopurine Methylenecyclopropane Analogues of Nucleosides	Ruifang Wang; Xinchao Chen; John C. Drach; Earl R. Kern; Jiri Zemlicka
817-819	Synthesis of Unusual Bicyclic Nucleosides Bearing an Unsaturated Side-Chain, as Potential Inhibitors of Varicella-Zoster Virus (VZV)	O. Bidet; C. McGuigan; G. Andrei; R. Snoeck; E. De Clercq; J. Balzarini
821-823	Novel Nucleotide Analogues as Potential Substrates for TMPK, a Key Enzyme in the Metabolism of AZT	H. C. Müller; C. Meier; J. Balzarini; J. Reinstein
825-827	d4TMP Delivery from 7-Substituted cycloSal-d4TMPs	C. Meier; J. T. Renze; J. Balzarini; E. De Clercq
829-831	Synthesis of New Homo and Heterodimers of 2′,3′-Dideoxyinosine (ddi) Using Ester Linkages	L. Ait Mohamed; M. Taourirte; A. Rochdi; H. B. Lazrek; J. J. Vasseur; J. W. Engels; C. Pannecouque; E. De Clercq
833-836	Synthesis and Antiviral Activity Assay of Novel (E)-3′,5′-Diamino-5-(2-bromovinyl)-2′,3′,5′-trideoxyuridine	Iván Lavandera; Susana Fernández; Miguel Ferrero; Erik De Clercq; Vicente Gotor
837-839	Optimization of Antiviral Prodrug Properties Using Combinatorial Methods	Yulia V. Berezovskaya; Mikhail V. Chudinov; Alexander M. Yurkevich
841-843	Non-inhibition of Acetylcholinesterase by cyclosal Nucleotides	C. Ducho; J. Balzarini; C. Meier
845-847	Synthesis and Biological Evaluation of a Series of New Cyclohexenyl Nucleosides	Ping Gu; Jordi Morral; Jing Wang; Jef Rozenski; Roger Busson; Arthur Van Aerschot; Erik De Clercq; Piet Herdewijn
849-851	Synthesis and Antiviral Evaluation of Ribavirin Congeners Containing a Hexitol Moiety	A. Van Aerschot; G. Schepers; R. Busson; J. Neyts; E. De Clercq; P. Herdewijn
853-855	Dinucleoside Monophosphates Containing AZT and 1-Methyladenosine or 7-Methylguanosine	Boris S. Ermolinsky; Ekaterina V. Efimtseva; Cyrill S. Alexeev; Sergey N. Mikhailov; Jan Balzarini; Erik De Clercq
857-859	2′-Deoxy-2′-C-trifluoromethyl β-D-Ribonucleoside Analogues: Synthesis and Antiviral Evaluations	Frédéric Jeannot; Gilles Gosselin; Christophe Mathé
861-863	Synthesis and Antiviral Evaluation of β-D- and β-L-Pentofuranonucleoside Derivatives Bearing 5-Trifluoromethylcytosine as the Base	Arnaud Marchand; Christophe Mathé; Gilles Gosselin
865-868	Dinucleoside Polyphosphate NAD Analogs as Potential NMN Adenylyltransferase Inhibitors. Synthesis and Biological Evaluation	P. Franchetti; L. Cappellacci; M. Pasqualini; M. Grifantini; T. Lorenzi; N. Raffaelli; G. Magni
869-872	A New Tiazofurin Pronucleotide: Synthesis and Biological Evaluation of CycloSaligenyl-Tiazofurin Monophosphate	L. Cappellacci; G. Barboni; P. Franchetti; C. Martini; H. N. Jayaram; M. Grifantini
873-875	Synthesis of Certain Heterodimers Expected as HIV-1 Reverse Transcriptase Inhibitors	D. Ladurée; E. Sugeac; C. Fossey; S. Schmidt; G. Laumond; A. M. Aubertin
877-881	Deaza- and Deoxyadenosine Derivatives: Synthesis and Inhibition of Animal Viruses as Human Infection Models	Sauro Vittori; Daniela Salvatori; Rosaria Volpini; Silvia Vincenzetti; Alberto Vita; Sara Taffi; Stefano Costanzi; Catia Lambertucci; Gloria Cristalli
883-885	Thionucleotides as Inhibitors of Ribonucleotide Reductase	B. Roy; S. Chambert; M. Lepoivre; J. -L. Décout
887-889	Synthesis of 4′-C-Ethynyl and 4′-C-Cyano Purine Nucleosides from Natural Nucleosides and Their Anti-HIV Activity	Satoru Kohgo; Kohei Yamada; Kenji Kitano; Shinji Sakata; Hiroyuki Hayakawa; Daisuke Nameki; Eiichi Kodama; Masao Matsuoka; Hiroaki Mitsuya; Hiroshi Ohrui

Volume 22, Issue 5-8 (2003)

891-894	Synthesis and Antiviral Evaluation of 2′,3′-Dideoxy-2′-fluoro-3′-C-hydroxymethyl-β-D-arabinofuranosyl Pyrimidine Nucleosides	Abdalla E. A. Hassan; Balakrina S. Pai; Stefania Lostia; Lieven Stuyver; Michael J. Otto; Raymond F. Schinazi; Kyoichi A. Watanabe
895-897	Investigations of Nucleoside H-Phosphonamidate in the Design of Nucleotide Prodrug	D. Egron; J. -L. Imbach; G. Gosselin; A. -M. Aubertin; C. Périgaud
899-901	Mononucleoside SATE Glucosyl Phosphorothiolates as a New Series of Pronucleotides	A. Jochum; N. Schlienger; G. Gosselin; J. -L. Imbach; A. -M. Aubertin; C. Périgaud
903-905	SATE (Aryl) Phosphotriester Series. I. Synthesis and Biological Evaluation	S. Peyrottes; G. Gosselin; A. -M. Aubertin; C. Périgaud
907-909	SATE (Aryl) Phosphotriester Series. II. Stability Studies and Physicochemical Parameters	G. Coussot; I. Lefebvre; D. Dimalta; S. Peyrottes; A. Pompon; G. Gosselin; C. Périgaud
911-914	Synthesis and Fluorescent Properties of 6-(4-Biphenylyl)-3,9-dihydro-9-oxo-5H-imidazo[1,2-A]purine Analogues of Acyclovir and Ganciclovir	Tomasz Goslinski; Grazyna Wenska; Bozenna Golankiewicz; Jan Balzarini; Erik De Clercq
915-917	Synthesis of 5-Azacytidine Nucleosides with Rigid Sugar Moiety as Potential Antitumor Agents	Moon Woo Chun; Myong Jung Kim; Hea Ok Kim; Hee-Doo Kim; Joong Hyup Kim; Hyung Ryong Moon; Lak Shin Jeong
919-921	Synthesis of Halogenated 9-(Dihydroxycyclopent-4′-enyl) Adenines and Their Inhibitory Activities Against S-Adenosylhomocysteine Hydrolase	Lak Shin Jeong; Jae Gyu Park; Won Jun Choi; Hyung Ryong Moon; Kang Man Lee; Hea Ok Kim; Hee-Doo Kim; Moon Woo Chun; Hea-Young Park; Kilhyoun Kim; Yhun Y. Sheen
923-925	Design and Synthesis of A₃ Adenosine Receptor Ligands, 3′-Fluoro Analogues of Cl-IB-MECA	Hea Ok Kim; Moo Hong Lim; Jae Gyu Park; Hyung Ryong Moon; Kenneth A. Jacobson; Hee-Doo Kim; Moon Woo Chun; Lak Shin Jeong
927-930	Design and Synthesis of A₃ Adenosine Receptor Ligands, 2′-Fluoro Analogues of Cl-IB-MECA	Hea Ok Kim; Jae Gyu Park; Hyung Ryong Moon; Prashantha Gunaga; Moo Hong Lim; Moon Woo Chun; Kenneth A. Jacobson; Hee-Doo Kim; Lak Shin Jeong
931-933	Bicyclic Nucleoside Inhibitors of Varicella-Zoster Virus: 5′-Chloro and 3′-Chloro Derivatives	G. Luoni; C. McGuigan; G. Andrei; R. Snoeck; E. De Clercq; J. Balzarini
935-937	Bicyclic Nucleoside Inhibitors of Varicella-Zoster Virus: Synthesis and Biological Evaluation of 2′,3′-Dideoxy- 3′-fluoro and 2′-Deoxy-xylo Derivatives	A. Carangio; C. McGuigan; G. Andrei; R. Snoeck; E. De Clercq; J. Balzarini
939-941	Synthesis of AZA Analogues of TSAO	Albert Nguyen Van Nhien; Cyrille Tomassi; Christophe Len; José Luis Marco-Contelles; Denis Postel
943-945	Synthesis, Stability, and Biological Evaluation of 1,3-Dihydrobenzo[c]furan Analogue of d4T and Its SATE Pronucleotide	Christophe Len; Abdelmajid Selouane; Denis Postel; Pierre Villa; Anne-Marie Aubertin; David Egron; Gilles Gosselin; Christian Périgaud
947-949	N-3 Substituted TSAO Derivatives as a Probe to Explore the Dimeric Interface of HIV-1 Reverse Transcriptase	María-Cruz Bonache; Cristina Chamorro; Sonsoles Velázquez; Erik De Clercq; Jan Balzarini; María-José Camarasa; Ana San-Félix
951-953	Towards New Thymidine Phosphorylase/PD-ECGF Inhibitors Based on the Transition State of the Enzyme Reaction	E. M. Priego; J. Mendieta; F. Gago; J. Balzarini; E. De Clercq; M. J. Camarasa; M. J. Pérez-Pérez
955-957	Synthesis of [1′-Fluoro-2′,2′-bis-(hydroxymethyl)-cyclopropylmethyl]purines as Antiviral Agents	Ju-Hyun Park; Myung-Hee Choi; Lak Shin Jeong; Moon Woo Chun; Hee-Doo Kim
959-961	Unusual Lability of 5′-O-tert-Butyldimethylsilyl Group On 4″-Acyl TSAO Derivatives	Sonia de Castro; María-Jesús Pérez-Pérez; Esther Lobatón; Erik De Clercq; Jan Balzarini; María-José Camarasa; Sonsoles Velázquez
963-966	Phosphorodiamides as Prodrugs for Antiviral Nucleosides	Alexander V. Shipitsyn; Natalya F. Zakirova; Evgeny F. Belanov; Tatyana R. Pronyaeva; Nina V. Fedyuk; Marina K. Kukhanova; Andrey G. Pokrovsky
967-972	Synthesis and Biological Evaluation of Some Acyclic 4,6-Disubstituted 1H-Pyrazolo[3,4-d]pyrimidine Nucleosides	O. Moukha-chafiq; M. L. Taha; A. Mouma; H. B. Lazrek; J. J. Vasseur; E. De Clercq
973-976	Thiated Analogues of 2′,3′-Dideoxy-3′-fluorothymidine and Their Phosphorylated and Phosphonylated Derivatives: Synthesis, Interaction with HIV Reverse Transcriptase, and In Vitro Anti-HIV Activity	A. Miazga; K. Felczak; M. Bretner; M. A. Siwecka; A. Piasek; T. Kulikowski
977-979	Synthesis and Antimalarial Activity of Novel N⁶-Substituted Adenosine Derivatives	P. H. Heidler; C. Herforth; A. Link
981-985	New Lipophilic Derivatives of AZT and d4T 5′-Phosphonates	Elena A. Shirokova; Maxim V. Jasko; Anastasiya L. Khandazhinskaya; Dmitry V. Yanvarev; Yury S. Skoblov; Tatyana R. Pronayeva; Nina V. Fedyuk; Andrey G. Pokrovsky; Marina K. Kukhanova
987-989	Urinary Modified Nucleosides as Tumor Markers	E. Dudley; F. Lemiere; W. Van Dongen; E. Esmans; A. M. M. El-Sharkawi; D. E. Games; A. G. Brenton; R. P. Newton
991-994	In Vitro Study of Resistance-Associated Genotypic Mutations to Nucleoside Analogs	N. Gashnikova; O. Plyasunova; Y. Kiseleva; N. Fedyuk; A. Pokrovsky
995-997	Metabolic and Pharmacological Characteristics of the Bicyclic Nucleoside Analogues (BCNAs) as Highly Selective Inhibitors of Varicella-Zoster Virus (VZV)	R. Sienaert; L. Naesens; A. Brancale; A. Carangio; G. Andrei; R. Snoeck; A. Van Kuilenburg; E. De Clercq; C. McGuigan; J. Balzarini
999-1001	Characterization of the Catalytic Subunit of the Human Herpesvirus 6 (HHV-6) DNA Polymerase Expressed in an In Vitro Transcription/Translation Assay	L. De Bolle; J. Balzarini; E. De Clercq; L. Naesens
1003-1006	Monoval-LdC: Efficient Prodrug of 2′-Deoxy-β-L-cytidine (L-dC), A Potent and Selective Anti-HBV Agent	S. Benzaria; C. Pierra; D. Bardiot; E. Cretton-Scott; E. G. Bridges; X. -J. Zhou; D. Standring; G. Gosselin
1007-1009	Synthesis of 2′-O-Substituted Ribonucleosides	V. Serebryany; L. Beigelman
1011-1015	Novel Base-Labile Protecting Groups for 5′-Hydroxy Function in Solid-Phase Oligonucleotide Synthesis	Kazuo Kamaike; Takashi Namiki; Etsuko Kawashima
1017-1022	Progress Towards a Submonomer Synthesis of Peptide Nucleic Acid	R. H. E. Hudson; R. D. Viirre
1023-1027	Towards a Circular *bis*-Peptide Nucleic Acid	R. H. E. Hudson; J. Tse
1029-1033	Nucleobase Modified Peptide Nucleic Acid	R. H. E. Hudson; R. D. Viirre; N. McCourt; J. Tse
1035-1038	A New Class of Spiegelmers Containing 2′-Fluoro-nucleotides	S. Helmling; E. Moyroud; W. Schroeder; I. Roehl; F. Kleinjung; S. Stark; G. Bahrenberg; C. Gillen; S. Klussmann; S. Vonhoff
1039-1040	Synthesis of an Asymmetrically Substituted AZA Crown Ether as Metal and Amino Acid Binding Site in DNA Conjugates	Stefan Vogel; Katja Rohr; Otto Dahl; Jesper Wengel
1041-1043	Nuclease Stability of LNA Oligonucleotides and LNA-DNA Chimeras	Miriam Frieden; Henrik F. Hansen; Troels Koch
1045-1048	Structural Pre-organization of Peptide Nucleic Acids	Vaijayanti A. Kumar
1049-1052	Oligomerization Aiming at Phosphonate Analogues of Oligoadenylates	Martina Pressová; Radek Liboska; Miloš Buděšínský; Šárka Králíková; Ivana Kavenová; Ivan Rosenberg
1053-1056	Ribo-, Xylo-, and Arabino-Configured Adenine-Based Nucleoside Phosphonates: Synthesis of Monomers for Solid-Phase Oligonucleotide Assembly	Ondřej Páv; Miloš Buděšínský; Ivan Rosenberg
1057-1060	Hybridization Properties of 4′-Branched Oligonucleotides	Radek Liboska; Miloš Buděšínský; Ivana Dvořáková-Kavenová; Ondřej Páv; Ivan Rosenberg

Volume 22, Issue 5-8 (2003)

1061-1064	α-Hydroxyphosphonate Oligonucleotides: A Promising DNA Type?	Šárka Králíková; Miloš Buděšínský; Ivan Rosenberg
1065-1067	Isosteric Phosphonate Pyrrolidine-Based Dinucleoside Monophosphate Analogues	Václav Vaněk; Miloš Buděšínský; Ivana Kavenová; Markéta Rinnová; Ivan Rosenberg
1069-1071	Oligonucleotides Containing an Acridine Group Covalently Bonded to the Nucleotide Flanking the 3′-3′ Phosphodiester Junction for Alternate Strand Triple Helix Formation	Bruno Catalanotti; Caterina Fattorusso; Luciano Mayol; Giorgia Oliviero; Gennaro Piccialli; Michela Varra
1073-1075	New Synthesis of 5-Carboxy-2′-deoxyuridine and Its Incorporation into Synthetic Oligonucleotides	V. Guerniou; D. Gasparutto; S. Sauvaigo; A. Favier; J. Cadet
1077-1079	Synthesis and Hybridization Properties of Oligonucleotide Analogues Containing Ornithine Backbone Modified with Nucleoalanines	N. Sumbatyan; A. Maksimenko; M. Gottikh; C. Malvy; G. Korshunova
1081-1083	Synthesis of Thymine-Modified Oligonucleotides	O. Gorchs; A. Grandas; J. Farràs
1085-1087	4-Guanidino-2-pyrimidinone Nucleobases: Synthesis and Hybridization Properties	J. Robles; A. Grandas; E. Pedroso
1089-1091	Synthesis and DNA Binding Properties of DNA-PNA Chimeras	G. Barone; L. De Napoli; G. Di Fabio; E. Erra; C. Giancola; A. Messere; D. Montesarchio; L. Petraccone; G. Piccialli
1093-1095	Deoxyribonolactone Lesion in DNA: Synthesis of Fluorinated Analogues	Caroline Crey; Pascal Dumy; Jean Lhomme; Mitsuharu Kotera
1097-1099	Triplex Formation Involving 2′-O,4′-C-Methylene Bridged Nucleic Acid (2′,4′-BNA) with 2-Pyridone Base Analogue: Efficient and Selective Recognition of C:G Interruption	Hidetaka Torigoe; Yoshiyuki Hari; Satoshi Obika; Takeshi Imanishi
1101-1104	Pyrrolidine PNA-DNA Chimeric Oligonucleotides with Extended Backbone	Vaijayanti A. Kumar; Meena
1105-1108	Piperidinyl Peptide Nucleic Acids: Synthesis and DNA-Complementation Studies	Pallavi Lonkar; Vaijayanti A. Kumar
1109-1111	Synthesis and Conformational Properties of O-β-D-Ribofuranosyl-(1″-2′)-guanosine and (Adenosine)-5″-phosphate	Ekaterina V. Efimtseva; Alexandra A. Shelkunova; Sergey N. Mikhailov; Koen Nauwelaerts; Jef Rozenski; Eveline Lescrinier; Piet Herdewijn
1113-1115	Chemical Incorporation of 1-Methyladenosine, Minor tRNA Component, into Oligonucleotides	E. V. Efimtseva; S. N. Mikhailov; J. Rozenski; R. Busson; A. Van Aerschot; P. Herdewijn
1117-1118	Oligonucleotides Containing Disaccharide Nucleosides: Synthesis, Physicochemical, and Substrate Properties	S. N. Mikhailov; E. V. Efimtseva; B. S. Ermolinsky; G. V. Bobkov; O. I. Andreeva; A. S. Golubeva; S. N. Kochetkov; A. Van Aerschot; G. Schepers; P. Herdewijn
1119-1121	Synthesis of Oligonucleotide Building Blocks of 2′-Deoxyguanosine Bearing a C8-Arylamine Modification	S. Gräsl; C. Meier
1123-1125	α-Hydroxybenzylphosphonate Modified Oligonucleotides: Synthesis, Properties, and a Novel Route via Monomer Building Blocks	Andreas Hohlfeld; Chris Meier
1127-1129	Determination of the Absolute P-Configuration of a Phthalidyl-Phosphonate Thymidine-Thymidine Dimer	W. Fendrich; C. Meier
1131-1133	Improved Synthesis of 2′-Amino-LNA	Signe M. Christensen; Christoph Rosenbohm; Mads Sørensen; Lotte-Emilie Larsen; Jesper Wengel; Troels Koch
1135-1137	Synthesis of an Oligonucleotide Analogue of Ethenoadenosine	Niangoran Koissi; Harri Lönnberg
1139-1141	Conformationally Restricted Dinucleotides: Tandem Ring-Closing Metathesis and Hydrogenation Approach	Philip Børsting; Poul Nielsen
1143-1145	α-LNA (α-D-Configured Locked Nucleic Acid)	Nanna K. Christensen; Michael Petersen; Birte Vester; Poul Nielsen
1147-1149	xylo-Configured Oligonucleotides (XNA, Xylo Nucleic Acids): Synthesis and Hybridization Studies	Nicolai E. Poopeiko; Britta M. Dahl; Jesper Wengel
1151-1153	RNase H Activation by Stereoregular Boranophosphate Oligonucleotide	Xin Wang; Mikhail Dobrikov; Dmitri Sergueev; Barbara Ramsay Shaw
1155-1157	Synthesis of a Base-Protected α-L-LNA Guanine Nucleoside	Gilles Gaubert; Jesper Wengel
1159-1161	Synthesis and Hybridization Properties of Oligodeoxynucleotides Containing 3′-Deoxy-3′-C-methyleneuridine	Dorthe Lindegaard; Jesper Wengel
1163-1165	Synthesis of a Base-Protected xylo-LNA Adenine Nucleoside	Torsten Bryld; Jesper Wengel
1167-1170	Synthesis of Modified RNA-Oligonucleotides for Structural Investigations	A. �ivković; J. W. Engels
1171-1173	Synthesis of Dinucleoside Boranophosphates by a Boranophosphotriester Approach	Takeshi Wada; Mamoru Shimizu; Natsuhisa Oka; Kazuhiko Saigo
1175-1178	Synthesis and Binding Properties of a Homopyrimidine 2′,5′-Linked Xylose Nucleic Acid (2′,5′-XNA)	Kazim A. Agha; Masad J. Damha
1179-1182	Conjugates of Oligo(2′-O-Methylribonucleotides) with Minor Groove Binders as New Sequence-Specific Agents Recognizing Both Grooves of Double-Stranded DNA	D. Novopashina; A. Sinyakov; V. Ryabinin; A. Venyaminova; A. Boutorine
1183-1185	Towards a DNA-Like Duplex Without Hydrogen Bonds	Gérald Mathis; Rolf Schütz; Jürg Hunziker
1187-1189	Pyrrolidino-DNA	Adrian Häberli; Alain Mayer; Christian J. Leumann
1191-1194	Fluorinated Peptide Nucleic Acid	Marcel Hollenstein; Daniel Gautschi; Christian J. Leumann
1195-1197	Transition Metal Ligands as Novel DNA-Base Substitutes	Christine Brotschi; Christian J. Leumann
1199-1201	New Nucleoside Analogues for the Recognition of Pyrimidine-Purine Inversion Sites	Sabrina Buchini; Christian J. Leumann
1203-1206	Synthetic Studies Towards a Novel, Chemical Stable, Abasic Site Analogue of DNA	Caroline Hirtz; Christian J. Leumann
1207-1210	Synthesis of a Cyclopentane Amide DNA Analogue and Its Base Pairing Properties	Dae-Ro Ahn; Markus Mosimann; Christian J. Leumann
1211-1213	Olefinic Peptide Nucleic Acid (OPA)	Daniel Gautschi; Christian J. Leumann
1215-1217	Synthesis, Biophysical, and Biochemical Properties of PNA-DNA Chimeras	Zoltán Bajor; Gyula Sági; Zsuzsanna Tegyey; László Ötvös

Volume 22, Issue 5-8 (2003)

1219-1221	Synthesis of Modified DNAs Bearing Two Different Fluorescent Probes and Its Application to Fluorescence Resonance Energy Transfer	Hiroaki Ozaki; Hiroshi Kobari; Kazuki Takagi; Hiroaki Sawai
1223-1225	Synthesis and Properties of Oligonucleotides Involving a Perylene Unit Linked to a 2′-Deoxyribose Residue	Yves Aubert; Ulysse Asseline
1227-1229	Methylated Hexitol Nucleic Acids, Towards Congeners with Improved Antisense Potential	A. Van Aerschot; A. Marchand; G. Schepers; W. Van den Eynde; J. Rozenski; R. Busson; P. Herdewijn
1231-1234	Oligonucleotides Incorporating 7-(Aminoalkyn-1-yl)-7-deaza-2′-deoxyguanosines: Duplex Stability and Phosphodiester Hydrolysis by Exonucleases	H. Rosemeyer; N. Ramzaeva; E. -M. Becker; E. Feiling; F. Seela
1235-1237	Oligonucleotides Incorporating N⁷-(2′-Deoxy-β-d-erythro-pentofuranosyl)isoguanine	P. Leonard; R. Kröschel; F. Seela
1239-1241	Synthesis and Properties of Halogenated 7-Deaza-2′-deoxyxanthosine and Protected Derivatives for Oligonucleotide Synthesis	F. Seela; K. Shaikh; T. Wiglenda
1243-1245	Synthesis of Oligonucleotide Prodrugs Bearing N-Acetyl Nucleobases	J. -C. Brès; J. -L. Imbach; F. Morvan
1247-1249	Preparation of 6-Thioguanosine Phosphoramidite for Oligoribonucleotide Synthesis	Yang Wang; Eric Lattmann; Qinguo Zheng
1251-1254	Synthesis and Physicochemical Properties of 2′-Deoxy- 2′,2″-difluoro-β-D-ribofuranosyl and 2′-Deoxy-2′,2″- difluoro-α-D-ribofuranosyl Oligonucleotides	Ekaterina Viazovkina; Maria M. Mangos; Masad J. Damha
1255-1257	Synthesis of Oligonucleotide-Peptide PEG-Conjugated: The EGG (Oligonucleotide)-Chicken (Peptide) Dilemma?	Gian Maria Bonora; Maurizio Ballico; Pietro Campaner; Sara Drioli; Ilaria Adamo
1259-1262	The Synthesis of 2′-O-Methyl G-Clamp Containing Oligonucleotides and Their Inhibition of the HIV-1 Tat-TAR Interaction	Stephen C. Holmes; Michael J. Gait
1263-1265	Imidazolethyl-Phosphoramidate α-Oligonucleotides	T. Michel; L. Mouls; F. Debart; J. -J. Vasseur
1267-1272	Stabilization of DNA Double and Triple Helices by Conjugation of Minor Groove Binders to Oligonucleotides	A. S. Boutorine; V. A. Ryabinin; D. S. Novopashina; A. G. Venyaminova; C. Hélène; A. S. Sinyakov
1273-1275	New Standards in LNA Synthesis	Henrik F. Hansen; Otto Olsen; Troels Koch
1277-1280	Synthesis and Studies of Modified Oligonucleotides- Directed Triple Helix Formation at the Purine-Pyrimidine Interrupted Site	Mohamed Jazouli; Dominique Guianvarc'h; Khalid Bougrin; Mohamed Soufiaoui; Pierre Vierling; Rachid Benhida
1281-1284	Synthesis and Triplex Binding Properties of Oligonucleotides Containing a Novel Nucleobase	Florence Lecubin; Michel Devys; Jean Louis Fourrey; Jian-Sheng Sun; Rachid Benhida
1285-1288	Synthesis of trans-L/D-2-(Tert-butoxycarbonyl- aminomethyl)-4-(thymin-1-yl) Pyrrolidin-1-yl Acetic Acid	Vaijayanti A. Kumar; Meena
1289-1291	Stabilization of RNA Bulges by Oligonucleotides Containing 2′-Naphthylmethyl-2′-deoxytubercidine	A. Madder; R. Ehrl; R. Strömberg
1293-1296	Modified Nucleoside Triphosphates: Synthesis and Applications for RNA In Vitro Selection	Th. Schoetzau; J. Langner; E. Moyroud; I. Röhl; S. Klussmann; S. Vonhoff
1297-1299	A Novel and Convenient Method for the Synthesis of Free 5′-Thiol Modified Oligonucleotides	Z. Kupihár; G. Kovács; Z. Kele; Z. Darula; L. Kovács
1301-1303	Synthesis and MS Analysis of Thiazolium and Pyridinium Derivatives of Peptide Nucleic Acids (PNAs) and Peptides	G. Kovács; P. Pádár; Z. Kupihár; Z. Kele; P. Forgó; L. Kovács
1305-1307	Synthesis of 1,4-Anhydro-2-deoxy-D-ribitol Derivatives from Thymidine	V. Serebryany; L. Beigelman
1309-1311	Synthesis and Analysis of Nucleosides Bearing Pyrrolepolyamide Binding to DNA	Etsuko Kawashima; Daisuke Itoh; Kazuo Kamaike; Yusuke Terui; Tairo Oshima
1313-1315	Synthesis of 2′-Spiro Ribo- and Arabinonucleosides	B. Ravindra Babu; Lise Keinicke; Jesper Wengel
1317-1319	Aryl-β-C-LNA Monomers as Universal Hybridization Probes[1], [2]	B. Ravindra Babu; Jesper Wengel
1321-1325	Commercial-Scale Synthesis of Protected 2′-Deoxycytidine and Cytidine Nucleosides	Kikkeri J. Divakar; Chitra M. Sawant; Y. A. Mulla; Deepak V. Zemse; Sakina M. Sitabkhan; Bruce S. Ross; Yogesh S. Sanghvi
1327-1330	Process Development for the Synthesis of 5′-O-(4,4′-Dimethoxytrityl)-N²-isobutyryl-2′-O-(2-methoxyethyl)-guanosine—A Potential Precursor for the Second Generation Antisense Oligonucleotides: An Improved Process for the Preparation of 2′-O-Alkyl-2,6-diaminopurine Riboside	Shabbir Ali S. Taj; P. Gurumurthy; R. Suresh; S. Narayanan; S. Suman Meenakshi; Yogesh S. Sanghvi
1331-1333	A Novel PNA-Monomer for Recognition of Thymine in Triple-Helix Structures	Anne Goldbech Olsen; Otto Dahl; Peter E. Nielsen
1335-1338	Synthesis and Properties of Oligonucleotide Chimeras Containing 5′-Amino-2′-deoxy-2′-fluoroarabinonucleosides	Ekaterina Viazovkina; Kyung-Lyum Min; Annie Galarneau; Masad J. Damha
1339-1342	A New Synthesis of 9-(2-Deoxy-2-fluoro-β-D-arabinofuranosyl)guanine (araF-G)	Mohamed I. Elzagheid; Ekaterina Viazovkina; Masad J. Damha
1343-1346	Synthesis of 2′,3′-Dideoxy-2′-fluoro-3′-thioarabinothymidine and Its 3′-Phosphoramidite Derivative	Mohamed I. Elzagheid; Anna Lisa Tedeschi; Masad J. Damha
1347-1350	The Effect of Universal Fluorinated Nucleobases on the Catalytic Activity of Ribozymes	A. E. Klöpffer; J. W. Engels
1351-1353	α-cycloPNA: 1-Aminocylopentane-1-carboxylic Acid-Derived Peptide Nucleic Acid	Nicola M. Howarth; Laurence P. G. Wakelin; David M. Walker
1355-1357	Oxidation of Guanine Nucleosides to 4-Amidinocarbamoyl- 5-hydroxyimidazoles by Dimethyldioxirane	R. Jeremy; H. Davies; Clarke Stevenson; Shiv Kumar; Jason Lyle; Lisa Cosby; John F. Malone; Derek R. Boyd; Narain D. Sharma; Ann P. Hunter; Bridget K. Stein
1359-1361	DNA Conjugates as Novel Functional Oligonucleotides	Takanori Kubo; Kinuko Yokoyama; Ryoji Ueki; Mayuka Yano; Yosuke Anno; Kotomi Sasaki; Hideki Ohba; Masayuki Fujii
1363-1365	Conformationally Restricted Chiral Peptide Nucleic Acids Derived from Azetidines	Lajos Kovács; Miklós Hornyák; Nicola M. Howarth
1367-1369	Control of Intracellular Delivery of Oligonucleotides by Conjugation with Signal Peptides	Mayuka Yano; Takanori Kubo; Kinuko Yokoyama; Ryoji Ueki; Kotomi Sasaki; Yosuke Anno; Hideki Ohba; Masayuki Fujii
1371-1373	Aryldiazomethane Derivatives as Reagents for Site Specific Labeling of Nucleic Acids at Phosphate	Cécile Bourget; Emmanuelle Trévisiol; Jean Lhomme; Mitsuharu Kotera; Christelle Tora; Eloy Bernal-Mendez; Ali Laayoun
1375-1378	1,2-Diol and Hydrazide Phosphoramidites for Solid-Phase Synthesis and Chemoselective Ligation of 2′-Modified Oligonucleotides	Eugeny M. Zubin; Dmitry A. Stetsenko; Tatiana S. Oretskaya; Michael J. Gait
1379-1382	Total Stepwise Solid-Phase Peptide-Oligonucleotide Conjugate Synthesis on Macroporous Polystyrene	Dmitry A. Stetsenko; Andrey D. Malakhov; Michael J. Gait

Volume 22, Issue 5-8 (2003)

1383-1385	Synthesis of 2′-Modified Oligonucleotides Containing Aldehyde or Ethylenediamine Groups	T. S. Zatsepin; E. A. Romanova; D. A. Stetsenko; M. J. Gait; T. S. Oretskaya
1387-1389	Studies on the Stability of Dinucleoside H-Phosphonates	P. Heinonen; A. Winqvist; Y. Sanghvi; R. Strömberg
1391-1393	The Cleavage of the Triphosphate Bridge of a Model for the 5′-cap mRNA Promoted by Dinuclear Bicyclic Complexes with Metal Ions	Qi Wang; Satu Mikkola; Harri Lönnberg
1395-1398	More Efficient Photolithographic Synthesis of DNA-Chips by Photosensitization	D. Wöll; S. Walbert; K. -P. Stengele; R. Green; T. Albert; W. Pfleiderer; U. E. Steiner
1399-1401	Nanoparticles and DNA Probes Based on DNA-Fluorophore Conjugates	M. A. Abdalla; J. Bayer; J. Rädler; K. Müllen
1403-1406	Novel Photocleavable Universal Support for Oligonucleotide Synthesis	Emma Anderson; Tom Brown; Douglas Picken
1407-1409	Stability, Vigor, and Inherent Versatility of Novel Amino Linker and Spacer Phosphoramidites	A. M. Morocho; V. N. Karamyshev; N. N. Polushin
1411-1413	Diastereocontrolled Synthesis of Phosphorothioate DNA via an Oxazaphospholidine Approach Using a Novel Class of Activators, Dialkyl(cyanomethyl)ammonium Salts	Natsuhisa Oka; Takeshi Wada; Kazuhiko Saigo
1415-1419	Understanding High Diastereomeric Discrimination in Formation of Oligoribonucleotide Phosphorothioate Linkages: The First Study of pKa-Dependent Activation in Solid-Supported Coupling of 2′-O-Substituted Ribonucleoside Phosphoramidites	Vasulinga T. Ravikumar; Douglas L. Cole
1421-1425	Synthesis of High Quality Phosphorothioate Oligonucleotides as Antisense Drugs. Use of I-Linker in the Elimination of 3′-Terminal Phosphorothioate Monoesters	Vasulinga T. Ravikumar; R. Krishna Kumar; Daniel C. Capaldi; Douglas L. Cole
1427-1429	Highly Efficient Synthesis of Peptide- and Carbohydrate-Oligonucleotide Conjugates Using Chemoselective Oxime and Thiazolidine Formation	D. Forget; D. Boturyn; O. Renaudet; E. Defrancq; P. Dumy
1431-1433	Reaction Mechanism for the Diastereocontrolled Synthesis of Phosphorothioate DNA by the Oxazaphospholidine Approach	Takeshi Wada; Natsuhisa Oka; Kazuhiko Saigo
1435-1437	Convenient Solid-Phase Method of Introduction of Sulfhydryl Groups into Oligodeoxyribonucleotides via 2′-O-Carbamate Linkage	S. I. Antsypovitch; S. Yu. Andreev; T. S. Oretskaya
1439-1441	Novel Biotin Phosphoramidites with Super-long Tethering Arms	A. M. Morocho; V. N. Karamyshev; O. V. Shcherbinina; A. G. Malykh; N. N. Polushin
1443-1445	Synthesis of Novel Tyrosinyl FRET Cassettes, Terminators, and Their Potential Use in DNA Sequencing	T. Sudhakar Rao; Weihong Zhang; Haiguang Xiao; Parke Flick; Shiv Kumar; Satyam Nampalli
1447-1449	Novel Synthesis of 2′-O Modified Oligonucleotides by Solid Phase Fragment Condensation	Kotomi Sasaki; Takanori Kubo; Ryoji Ueki; Mayuka Yano; Yosuke Anno; Hideki Ohba; Masayuki Fujii
1451-1453	Synthesis of DNA Conjugates by Solid Phase Fragment Condensation	Yosuke Anno; Takanori Kubo; Ryoji Ueki; Mayuka Yano; Kotomi Sasaki; Hideki Ohba; Masayuki Fujii
1455-1457	Direct Regioselective Enzymatic Acylation of Nucleosides: Building-Blocks for the Solution Phase Synthesis of Oligonucleotides	Javier García; Susana Fernández; Miguel Ferrero; Yogesh S. Sanghvi; Vicente Gotor
1459-1461	Studies Towards Synthesis of Dinucleoside Arylphosphonates with Metal Complexing Properties	Tommy Johansson; Jacek Stawinski
1463-1465	9-Fluorenemethyl H-Phosphonoselenoate—A Versatile Reagent for Transferring an H-Phosphonoselenoate Group	Martin Kullberg; Jacek Stawinski
1467-1469	Chemoselectivity in Oxidative Coupling of Bifunctional Nucleophiles with Dinucleoside H-Phosphonate and Dinucleoside H-Phosphonothioate Diesters	Johan Nilsson; Adam Kraszewski; Jacek Stawinski
1471-1474	Negatively Charged, Dye Labeled-Dideoxynucleotides for “Direct-Load” DNA Sequencing	Satyam Nampalli; Patrick J. Finn; Lei Sun; Haiguang Xiao; John R. Nelson; Gregory Grossmann; Parke K. Flick; Carl W. Fuller; Shiv Kumar
1475-1477	Design, Synthesis, and In Vitro Evaluation of APIO Analogue of Neplanocin A	Hyung Ryong Moon; Sung Hee Kwon; Jeong Ah Lee; Byul Nae Yoo; Hea Ok Kim; Moon Woo Chun; Hee-Doo Kim; Joong Hyup Kim; Lak Shin Jeong
1479-1482	A New Concept for DNA-Arrays	Kerstin Jahn-Hofmann; Nancy Holzhey; Thomas Ellinger; Joachim W. Engels
1483-1485	Molecular Recognition of Quadruplex DNA by Quinacridine Derivatives	M. -P. Teulade-Fichou; C. Hounsou; L. Guittat; J. -L. Mergny; P. Alberti; C. Carrasco; C. Bailly; J. -M. Lehn; W. D. Wilson
1487-1489	Photoadduct Leading to Crosslinking in Ru^II-Derivatized Oligonucleotides	O. Lentzen; J. -F. Constant; E. Defrancq; C. Moucheron; P. Dumy; A. Kirsch-De Mesmaeker
1491-1493	Properties of Conjugate DNA Enzymes	Takanori Kubo; Ryoji Ueki; Yosuke Anno; Mayuka Yano; Kotomi Sasaki; Hideki Ohba; Masayuki Fujii
1495-1497	Novel Method for the Covalent Immobilization of Oligonucleotides via Diels-Alder Bioconjugation	Hallie A. Latham-Timmons; Andreas Wolter; J. Shawn Roach; Rubina Giare; Michael Leuck
1499-1503	Fluorescent 2-Pyrimidinone Nucleoside in Parallel-Stranded DNA	D. N. Kaluzhny; S. N. Mikhailov; E. V. Efimtseva; O. F. Borisova; V. L. Florentiev; A. K. Shchyolkina; T. M. Jovin
1505-1507	Cross-Linking of Escherichia coli Formamidopyrymidine-DNA Glycosylase to DNA Duplexes Containing Photoactivatable Phenyl(Trifluoromethyl)diazirine Groups	M. V. Taranenko; N. V. Sumbatyan; M. T. Mtchedlidze; S. A. Kuznetsova
1509-1512	Oligoribonucleotides with Functionalized Nucleobases as New Modifiers of Biopolymers	M. Repkova; M. Meshchaninova; D. Pyshnyi; A. Venyaminova
1513-1516	Evaluation of Capillary HPLC/Mass Spectrometry as an Alternative Analysis Method for Gel Electrophoresis of Oligonucleotides	Jef Rozenski; Karen Vastmans; Arthur Van Aerschot; Piet Herdewijn
1517-1519	Structural Studies on DNA Triple Helix Formed by Intronic GAA Triplet Repeat Expansion in Friedreich's Ataxia	Aklank Jain; Faizan Ahmad; Moganty R. Rajeswari
1521-1523	Catalytic DNA and RNA for Targeting MDR1 mRNA	M. Kuznetsova; A. Fokina; M. Lukin; M. Repkova; A. Venyaminova; V. Vlassov
1525-1529	Ability of Adenosine-2′(3′)-deoxy-3′(2′)-triphosphates and Related Analogues to Replace ATP as Phosphate Donor for all Human and Drosphila melanogaster Deoxyribonucleoside Kinases	Krzysztof Krawiec; Borys Kierdaszuk; Elena N. Kalinichenko; Elena B. Rubinova; Igor A. Mikhailopulo; Staffan Eriksson; Birgitte Munch-Petersen; David Shugar
1531-1533	5′-O-Fluorosulfonylbenzoyl Esters of Purine Nucleosides as Potential Inhibitors of NTPase/Helicase and Polymerase of Flaviviridae Viruses	M. Bretner; S. Schalinski; P. Borowski; T. Kulikowski
1535-1538	Intersubunit Interactions in Human Cytidine Deaminase	S. Vincenzetti; S. Costanzi; G. Cristalli; P. Mariani; B. Quadrini; N. Cammertoni; A. Vita
1539-1543	Human Cytidine Deaminase: Understanding the Catalytic Mechanism	S. Costanzi; S. Vincenzetti; A. Vita; C. Lambertucci; S. Taffi; R. Volpini; S. Vittori; G. Cristalli
1545-1548	Nicotinamide Adenine Dinucleotide a Unique Compound for Theoretical and Synthetic Model Studies: Chirality as Source for High Stereospecificity	H. M. Buck
1549-1552	The Biochemical Significance of Parallel DNA Duplexes	H. M. Buck

Volume 22, Issue 5-8 (2003)

1553-1556	Partial Molar Volumes of mRNA 5′ Cap Analogues	Jedrzej Szymanski; Janusz Stepinski; Jaroslaw Poznanski; Edward Darzynkiewicz; Wojciech Zielenkiewicz; Ryszard Stolarski
1557-1561	Thermodynamics of 7-Methylguanosine Cation Stacking with Tryptophan upon mRNA 5′ Cap Binding to Translation Factor eIF4E	Anna Niedzwiecka; Janusz Stepinski; Lajos Balaspiri; Edward Darzynkiewicz; Ryszard Stolarski
1563-1565	Recognition of Cyclonucleoside Lesions by the Lactococcus lactis FPG Protein	Evelyne Muller; Didier Gasparutto; Bertrand Castaing; Alain Favier; Jean Cadet
1567-1570	Interactions of Potent Multisubstrate Analogue Inhibitors with Purine Nucleoside Phosphorylase from Calf Spleen—Kinetic and Spectrofluorimetric Studies	Monika Iwanow; Lucyna Magnowska; Tsutomu Yokomatsu; Shiroshi Shibuya; Agnieszka Bzowska
1571-1573	Triplex Formation Involving 2′-O,4′-C-Methylene Bridged Nucleic Acid (2′,4′-BNA) with 1-Is oquinolone Base Analogue: Efficient and Selective Recognition of C:G Interruption	Hidetaka Torigoe; Yoshiyuki Hari; Satoshi Obika; Takeshi Imanishi
1575-1577	Inhibition of Vertebrate Telomerases by the Triphosphate Derivatives of Some Biologically Active Nucleosides	Toyofumi Yamaguchi; Hazuki Takahashi; Hiroshi Jinmei; Yuko Takayama; Mineo Saneyoshi
1579-1581	Genosnip: SNP Genotyping by MALDI-TOF MS Using Photocleavable Oligonucleotides	T. Wenzel; T. Elssner; K. Fahr; J. Bimmler; S. Richter; I. Thomas; M. Kostrzewa
1583-1586	MALDI-TOF Mass Spectrometry as a Powerful Tool to Study Enzymatic Processing of DNA Lesions Inserted into Oligonucleotides	D. Gasparutto; C. Saint-Pierre; M. Jaquinod; A. Favier; J. Cadet
1587-1589	New Reagent for Protein-DNA Contacts Footprinting	O. A. Koval; S. B. Oleinikova; E. L. Chernolovskaya; V. V. Litvak; V. V. Vlassov
1591-1594	Effect of Putrescine and PEG on a Structural Transition of DNA G-Quadruplex	Daisuke Miyoshi; Akihiro Nakao; Naoki Sugimoto
1595-1598	Synthesis and Energy Transfer Efficiency of FRET Terminators Derived from Different Linkers	Shiv Kumar; Satyam Nampalli; Patrick J. Finn; T. Sudhakar Rao; Chung-Yuan Chen; Parke K. Flick; Carl W. Fuller
1599-1602	Branchpoint Sugar Stereochemistry Determines the Hydrolytic Susceptibility of Branched RNA Fragments by the Yeast Debranching Enzyme (YDBR)	Sandra Carriero; Maria M. Mangos; Kazim A. Agha; Anne M. Noronha; Masad J. Damha
1603-1605	Suppression of Exonucleolytic Degradation of Double-Stranded DNA and Inhibition of Exonuclease III by PNA	A. Slaitas; C. Ander; Z. Földes-Papp; R. Rigler; E. Yeheskiely
1607-1609	Antisense Knockdown of PKC-α Using LNA-Oligos	Jens Bo Hansen; Majken Westergaard; Charlotte Albaek Thrue; Birgit Giwercman; Henrik Oerum
1611-1613	Covalent Coupling of a PIM-1 Oncogene Targeted PNA with an Antennapedia Derived Peptide	J. -R. Bertrand; N. Sumbatyan; C. Malvy
1615-1618	Inhibition of Gene Expression by Peptide Nucleic Acids in Cultured Cells	Susanna Cogoi; Valentina Rapozzi; Luigi E. Xodo
1619-1621	2′-O,4′-C-Ethylene-Bridged Nucleic Acid (ENA^TM) for Effective Antisense Formation	Koji Morita; Koji Yamate; Shin-ichi Kurakata; Kenji Watanabe; Takeshi Imanishi; Makoto Koizumi
1623-1625	Synthesis and Antitumor Activity of N-Sulfonyl Derivatives of Nucleobases and Sulfonamido Nucleoside Derivatives	B. Žinić; I. Krizmanić; Lj. Glavaš-Obrovac; I. Karner; M. Žinić
1627-1629	Novel Short Oligonucleotide Conjugates as Inhibitors of Human Telomerase	Krisztina Pongracz; Shihong Li; Brittney-Shea Herbert; Ronald Pruzan; Ellen Wunder; Allison Chin; Mieczyslaw Piatyszek; Jerry Shay; Sergei M. Gryaznov
1631-1634	Specific Inhibition of Hepatitis C Viral Gene Expression by Non-polar (Phenylalkyl)phosphonates	S. Amberg; A. Tamke; W. H. Caselmann; J. W. Engels
1635-1637	Endcaps for Stabilizing Short DNA Duplexes	Pei-Sze Ng; Maneesh R. Pingle; Ganesan Balasundarum; Alan Friedman; Xiaolin Zu; Donald E. Bergstrom
1639-1645	Diastereomeric Process Control in the Synthesis of 2′-O-(2-Methoxyethyl) Oligoribonucleotide Phosphorothioates as Antisense Drugs	Vasulinga T. Ravikumar; Douglas L. Cole
1647-1649	Universal Labeling Chemistry for Nucleic Acid Detection on DNA-Arrays	E. Bernal-Méndez; C. Tora; I. Sothier; M. Kotera; A. Troesch; A. Laayoun
1651-1655	Incorporation of (α-P-Borano)-2′,3′-dideoxycytidine 5′-Triphosphate into DNA by Drug-Resistant MMLV Reverse Transcriptase and Taq DNA Polymerase	Mikhail I. Dobrikov; Zinaida A. Sergueeva; Barbara Ramsay Shaw
1657-1659	Synthesis of 2′-Deuterio and 3′-Deuterio Cytidine 5′-Diphosphate	Jessica Sandbrink; Roger Strömberg
1661-1664	Determination of RNA Tertiary Structure by Electron Paramagnetic Resonance Spectroscopy (EPR)	Nelly Piton; Joachim W. Engels
1665-1667	Synthesis and Recognition by DNA Polymerases of a Reactive Nucleoside for DNA Diversification	S. Pochet; L. Dugué; H. Strobel
1669-1672	Conformationally Restricted 2-Substituted Wyosine Derivatives. ¹H, ¹³C, and ¹⁵N NMR Study	Daniel Baranowski; Bozenna Golankiewicz; Janez Plavec
1673-1675	³¹P NMR Studies on the Putative Chemoselective Activation of Nucleoside-3′-thiophosphate-O-esters	Gyula Sági; Zoltán Bajor; Roland Mizda; Gyöngyi Kenesi
1677-1680	¹H-NMR Study of the Quadruplex [d(TGGGT)]₄ Containing a Modified Thymine	Luigi Petraccone; Eva Erra; Lucia Nasti; Aldo Galeone; Antonio Randazzo; Veronica Esposito; Luciano Mayol; Guido Barone; Concetta Giancola
1681-1684	PNA-DNA Chimeras Forming Quadruplex Structures	Veronica Esposito; Aldo Galeone; Luciano Mayol; Anna Messere; Gennaro Piccialli; Antonio Randazzo
1685-1686	Synthesis of 2-Deoxy-β-D-ribose 1-Phosphate, NMR Comparison and Its Enzymatic Activity for Structural Elucidation of Synthetic α-Isomer	Hironori Komatsu; Ichirou Ikeda
1687-1690	Structure of 2′,5′-Linked Tetraribonucleotide Loops: A Novel RNA Motif	Rami N. Hannoush; Alexei Yu. Denisov; Kalle Gehring; Masad J. Damha
1691-1693	Structural Characterization of LNA and α-L-LNA Hybridized to RNA	Michael Petersen; Jakob T. Nielsen; Kent Bondensgaard; Jesper Wengel; Jens Peter Jacobsen
1695-1698	Interactions of Trimeric Purine Nucleoside Phosphorylases with Ground State Analogues—Calorimetric and Fluorimetric Studies	Beata Wielgus-Kutrowska; Joachim Frank; Antonin Holý; Gertraud Koellner; Agnieszka Bzowska
1699-1702	Crystal Structure of Calf Spleen Purine Nucleoside Phosphorylase in a Complex with Multisubstrate Analogue Inhibitor with 2,6-Diaminopurine Aglycone	Gertraud Koellner; Albrecht Stroh; Grzegorz Raszewski; Antonin Holý; Agnieszka Bzowska
1703-1706	Binding Studies of Eukaryotic Initiation Factor eIF4E with Novel mRNA Dinucleotide Cap Analogues	Joanna Zuberek; Jacek Jemielity; Janusz Stepinski; Magdalena Lewdorowicz; Anna Niedzwiecka; Dorota Haber; Ryszard Stolarski; Robert E. Rhoads; Edward Darzynkiewicz
1707-1710	Influence of the Length of the Phosphate Chain in mRNA 5′ Cap Analogues on Their Interaction with Eukaryotic Initiation Factor 4E	Joanna Zuberek; Jacek Jemielity; Anna Niedzwiecka; Janusz Stepinski; Aleksandra Wyslouch-Cieszynska; Ryszard Stolarski; Edward Darzynkiewicz
1711-1714	Interaction Between Yeast Eukaryotic Initiation Factor eIF4E and mRNA 5′ Cap Analogues Differs from That for Murine eIF4E	Katarzyna Kiraga-Motoszko; Janusz Stepinski; Anna Niedzwiecka; Jacek Jemielity; Malgorzata Wszelaka-Rylik; Ryszard Stolarski; Wojciech Zielenkiewicz; Edward Darzynkiewicz
1715-1719	Cell Surface Oligonucleotide-Binding Proteins of Human Squamous Carcinoma A431 Cells	P. P. Laktionov; B. P. Chelobanov; M. V. Kharkova; E. Yu. Rykova; D. V. Pyshnyi; I. A. Pyshnaya; K. Marcus; H. E. Meyer; V. V. Vlassov

Volume 22, Issue 5-8 (2003)

1721-1723	Geniom® Technology—The Benchtop Array Facility	R. Güimil; M. Beier; M. Scheffler; H. Rebscher; J. Funk; A. Wixmerten; M. Baum; C. Hermann; H. Tahedl; E. Moschel; F. Obermeier; I. Sommer; D. Büchner; R. Viehweger; J. Burgmaier; C. F. Stähler; M. Müller; P. F. Stähler
1725-1727	Resistance of Human Cytomegalovirus to D- and L-Ribosyl Benzimidazoles as a Tool to Identify Potential Targets for Antiviral Drugs	Gloria Komazin; Roger G. Ptak; Brian T. Emmer; Leroy B. Townsend; John C. Drach
1729-1731	Linear Polyethylenimine as a Tool for Comparative Studies of Antisense and Short Double-Stranded RNA Oligonucleotides	Jean-Charles Bologna; Gabriele Dorn; Francois Natt; Jan Weiler
1733-1736	The Use of Triisopropylsilyl-oxymethyl (TOM) in the Synthesis of Anti-telomerase 2-5A Antisense Compound RBI 011	Hagen Cramer; Rachele Rhea; Jim Okicki; Karen Yirava; Robert Silverman

Volume 22, Issue 4 (2003)

359-371	Synthesis and Properties of Phosphorylated 3′-O-β-D-Ribofuranosyl-2′-deoxythymidine	Ekaterina V. Efimtseva; Alexandra A. Shelkunova; Sergey N. Mikhailov; Koen Nauwelaerts; Jef Rozenski; Eveline Lescrinier; Piet Herdewijn
373-389	Synthesis, Structural Studies, and Biological Evaluation of Some Purine Substituted 1-Aminocyclopropane-1-carboxylic Acids and 1-Amino-1-hydroxymethylcyclopropanes	Zoran Džolić; Vedran Krištafor; Mario Cetina; Ante Nagl; Antonija Hergold-Brundić; Draginja Mrvoš-Sermek; Thomas Burgemeister; Mira Grdiša; Neda Slade; Krešimir Pavelić; Jan Balzarini; Erik De Clercq; Mladen Mintas
391-404	C-5 Modified Nucleosides: Direct Insertion of Alkynyl-Thio Functionality in Pyrimidines	Heike A. Held; Abhijit Roychowdhury; Steven A. Benner
405-417	The Analogue of Thymidine Triphosphate Containing a Methylene Group in Place of the 5′ Oxygen Can Serve as a Substrate for Reverse Transcriptase	M. A. Bell; G. R. Gough; P. T. Gilham
419-435	Synthesis of Triazole Nucleoside Derivatives	Zicheng Li; Shuhua Chen; Ning Jiang; Gang Cui
437-451	Synthesis of Carbocyclic 1-[4-(Hydroxymethyl)cyclopent-2-enyl]-1,2,4-triazole-3-carboxamide and Its Derivatives	Gwang-il An; Hakjune Rhee
453-460	2-Methyl-5-tert-butylthiophenol—An Odorless Deprotecting Reagent Useful in Synthesis of Oligonucleotides and Their Analogs	R. Krishna Kumar; Douglas L. Cole; Vasulinga T. Ravikumar
461-468	Solid Phase Synthesis of Phosphorothioate Oligonucleotides Utilizing Diethyldithiocarbonate Disulfide (DDD) as an Efficient Sulfur Transfer Reagent	Zacharia S. Cheruvallath; R. Krishna Kumar; Claus Rentel; Douglas L. Cole; Vasulinga T. Ravikumar
469-487	6-(Levulinyloxymethyl)-3-methoxy-2-nitrobenzoyl and 2-(Levulinyloxymethyl)-5-methoxy-4-nitrobenzoyl Groups as Novel Base-Labile Groups for 5′-Hydroxy Protection in Solid-Phase Oligonucleotide Synthesis	Kazuo Kamaike; Takashi Namiki; Etsuko Kawashima

Volume 22, Issue 3 (2003)

239-247	Cyclopropyl and Related Analogs of the Anti-HIV Compound, Isodideoxyadenosine	Vasu Nair; Travis Mickle; Sanjib Bera
249-263	Structural Properties of the Neutral and Monoanionic Forms of Xanthosine, Highly Relevant to Their Substrate Properties with Various Enzyme Systems	Jarosław Poznanski; Borys Kierdaszuk; David Shugar
265-274	Synthesis of (Z)-(2,3-bis-Hydroxymethyl)methylenecyclopropane Analogues of Purine Nucleosides	Xinchao Chen; Shintaro Matsumi; Hiroaki Mitsuya; Jiri Zemlicka
275-282	Introduction of the α-P-Borano-Group into Deoxynucleoside Triphosphates Increases Their Selectivity to HIV-1 Reverse Transcriptase Relative to DNA Polymerases	Mikhail I. Dobrikov; Kristen M. Grady; Barbara Ramsay Shaw
283-297	Conformational Properties of Nucleotide-Based Template-Competitive HIV-1 Reverse Transcriptase Inhibitors: Analysis of Enzyme Binding Modes	Weiying Lin; Ke Li; Bob M. Moore II; Michael B. Doughty
299-307	Synthesis of N-Substituted 1-Amino-2,3-dihydro-1H-imidazole-2-thione-N-nucleosides and S-Glycosylated Derivatives	Iman A. Al-Masoudi; Ahmed I. Khodair; Yaseen A. Al-Soud; Najim A. Al-Masoudi
309-317	Stacking Conformation of 9-[ω-(Thymin-1-yl)alkyl]adenine in Aqueous Solution	Toshio Itahara
319-328	Synthesis and Antiherpetic Activity of Acyclovir Phosphonates	Inna L. Karpenko; Maxim V. Jasko; Valeriya L. Andronova; Alexander V. Ivanov; Marina K. Kukhanova; Georgy A. Galegov; Yury S. Skoblov
329-347	Study on Reactivity and Protection of the α-Hydroxyphosphonate Moiety in 5′-Nucleotide Analogues: Formation of the 3′-O-P-C(OH)-C4′ Internucleotide Linkage	Šárka Králíková; Milena Masojídková; Miloš Buděšínský; Ivan Rosenberg
349-357	Synthesis of Double Headed Imidazoline Acyclo C-Nucleosides: 1,4-bis[1-Amino-5-oxo-4-Substituted-(Imidazolin-2-yl)]galacto-tetritols	Adel Z. Nasr

Volume 22, Issue 2 (2003)

109-114	Building Blocks for Polyamide Nucleic Acids: Facile Synthesis Using Potassium Fluoride Doped Natural Phosphate as Basic Catalyst	A. Alahiane; M. Taourirte; A. Rochdi; N. Redwane; S. Sebti; J. W. Engels; H. B. Lazrek
115-127	Synthesis and Biological Activities of 2-Functionalized Purine Nucleosides	Vasu Nair; Bindu Bera; Earl R. Kern
129-134	Synthesis of Antisense Oligonucleotides with Minimum Depurination	Achim H. Krotz; Douglas L. Cole; Vasulinga T. Ravikumar
135-144	Synthesis and Biological Activity of 2-Aminopurine Methylenecyclopropane Analogues of Nucleosides	Ruifang Wang; Xinchao Chen; John C. Drach; Earl R. Kern; Jiri Zemlicka
145-151	A New Method for the Synthesis of 2′-O-Benzyladenosine Using Mitsunobu Reaction	Shigetada Kozai; Tomoyo Fuzikawa; Keisuke Harumoto; Tokumi Maruyama
153-173	Striking Ability of Adenosine-2′(3′)-deoxy-3′(2′)-triphosphates and Related Analogues to Replace ATP as Phosphate Donor for All Four Human, and the Drosophila Melanogaster, Deoxyribonucleoside Kinases	Krzysztof Krawiec; Borys Kierdaszuk; Elena N. Kalinichenko; Elena B. Rubinova; Igor A. Mikhailopulo; Staffan Eriksson; Birgitte Munch-Petersen; David Shugar
175-192	Hydrodynamic and Spectroscopic Studies of Substrate Binding to Human Recombinant Deoxycytidine Kinase	Rajam S. Mani; Elena V. Usova; Staffan Eriksson; Carol E. Cass
193-202	Convenient Synthesis of 8-Amino-2′-deoxyadenosine	Miriam Frieden; Anna Aviñó; Ramon Eritja
203-221	Structural Polymorphism of Telomeric DNA Regulated by pH and Divalent Cation	Daisuke Miyoshi; Shizuka Matsumura; Wei Li; Naoki Sugimoto
223-238	Synthesis, Conformation, and Antiviral Activity of 5-Methoxymethyl-2′-deoxycytidine Analogs	Wajdi M. Zoghaib; Shajan Mannala; V. Sagar Gupta; Guy Tourigny; R. Stephen Reid

Volume 22, Issue 1 (2003)

1-12	Side Reactions in the H-Phosphonate Approach to Oligonucleotide Synthesis: A Kinetic Investigation on Bisacylphosphite Formation and 5′-O-Acylation	Susannah Sigurdsson; Roger Strömberg
13-19	Microwave-Assisted Synthesis of O′-Adamantylated Uracil-Derived Nucleosides	Agata Górska; Mariola Andrzejewska; Jarosław Kamiński; Zygmunt Kazimierczuk
21-44	Selective Synthesis and Reactions of 6-Substituted- 2-β-galactosyl-1,2,4-triazines of Potential Anticancer Activity	Abdel Kader Mansour; Mohga M. Eid; Nasser S. A. M. Khalil
45-62	Conformational Studies of Novel Antiretroviral Analogs of Zidovudine	María T. Baumgartner; Marisa I. Motura; Rubén H. Contreras; Adriana B. Pierini; Margarita C. Briñón
63-69	Synthesis of Serine/Alanine Conjugated 3′,5′-TpT	Zhi-Hui Qin; Chang-Xue Lin; Yong Ju; Yu-Fen Zhao
71-84	Synthesis of a Novel Aldehyde: 4-O-Methyl-5-formylmethyl- 2′-deoxyuridine	Chung-Shan Yu; Franz Oberdorfer
85-98	Fluorescent 7- and 8-Methyl Etheno Derivatives of Adenosine and 6-Amino-9-ethylpurine: Syntheses and Fluorescence Properties	Piritta Virta; Toni Holmström; Tony Munter; Thomas Nyholm; Leif Kronberg; Rainer Sjöholm
99-107	Nucleic Acid Component Analogues: Synthesis of 2′-Deoxynucleosides from 5-Substituted-4- Hydroxy-6(1H)-Pyrimidinones	Ahmed F. Khattab; Ahmed E.-S. Abdel Megied; Erik B. Pedersen

Volume 21, Issue 11-12 (2002)

737-751	THE SYNTHESIS OF ANTI-FIXED 3-METHYL-3- DEAZA-2′-DEOXYADENOSINE AND OTHER 3H-IMIDAZO[4,5-c]PYRIDINE ANALOGS	Rostem J. Irani; John SantaLucia Jr.
753-764	AFFINITY MODIFICATION OF EcoRII DNA METHYLTRANSFERASE BY THE DIALDEHYDE-SUBSTITUTED DNA DUPLEXES: MAPPING THE ENZYME REGION THAT INTERACTS WITH DNA	Oksana M. Gritsenko; Elizaveta V. Koudan; Sergey N. Mikhailov; Boris S. Ermolinsky; Arthur Van Aerschot; Piet Herdewijn; Elizaveta S. Gromova
765-774	SYNTHESIS of 2′-DEOXY-2′-FLUOROGUANYL-(3′,5′)-GUANOSINE	Tokumi Maruyama; Shigetada Kozai; Kazuo Nakamura; Masachika Irie
775-784	TARGETING OF A701G NUCLEOTIDE AT THE HUMAN ATP1A1 LOCUS USING A RNA/DNA CHIMERA	Tiziana Cervelli; Grazia Lombardi; Lorenzo Citti; Alvaro Galli; Maria Teresa Locci; Giuseppe Rainaldi
785-801	A COMPARISON OF THE PROPERTIES AND THE SOLUTION STRUCTURE FOR RNA AND DNA QUADRUPLEXES WHICH CONTAIN TWO GGAGG SEQUENCES JOINED WITH A TETRANUCLEOTIDE LINKER	Hui Liu; Atsushi Kugimiya; Tokuhiro Sakurai; Masato Katahira; Seiichi Uesugi
803-812	PROCEDURE FOR SELECTING STARTING CONFORMATIONS FOR ENERGY MINIMIZATION OF NUCLEOSIDES AND NUCLEOTIDES	Douglas G. Harris; Jianyin Shao; Jonathan M. Anderson; Douglas P. Marx; S. Scott Zimmerman
813-823	KINETIC AND MOLECULAR MODELING OF NUCLEOSIDE AND NUCLEOTIDE INHIBITION OF MALATE DEHYDROGENASE	Douglas G. Harris; Douglas P. Marx; S. Scott Zimmerman; Ronald W. McCune
825-835	SYNTHESIS AND ANTIVIRAL EVALUATION OF ISATIN RIBONUCLEOSIDES	Mara R. P. deOliveira; José C. Torres; Simon J. Garden; Carla Veronica B. dos Santos; Thatyana Rocha Alves; Angelo C. Pinto; Helena de S. Pereira; Luiz Roberto Leão Ferreira; Nissin Moussatché; Izabel Christina de P. P. Frugulhetti; Vitor F. Ferreira; Maria Cecília B. V. de Souza
837-847	A NEW CLASS OF BIHETEROCYCLIC THIOGLYCOSIDES FROM PYRIDINE-2-(1H)-THIONES	Galal H. Elgemeie; Mona A. Ahmed
849-861	CONVENIENT SYNTHESIS OF FLUORINATED NUCLEOSIDES WITH PERFLUOROALKANESULFONYL FLUORIDES	Satoshi Takamatsu; Satoshi Katayama; Naoko Hirose; Etienne De Cock; Geert Schelkens; Marc Demillequand; Jozef Brepoels; Kunisuke Izawa
863-882	SYNTHESIS, STRUCTURE, AND CONFORMATION OF ANTI-TUMOR AGENTS IN THE SOLID AND SOLUTION STATES: HYDROXYL DERIVATIVES OF FTORAFUR	David M. Stokes; Brajeswar Paul; James L. Alderfer; Robert M. Wollman; Thamarapu Srikrishnan
883-889	APPLICATION OF MITSUNOBU REACTION TO SOLID-PHASE PEPTIDE NUCLEIC ACID (PNA) MONOMER SYNTHESIS	Bogdan Falkiewicz
891-901	SYNTHESIS OF NOVEL 8-SUBSTITUTED CARBOCYCLIC ANALOGS OF 2′,3′-DIDEOXYADENOSINE WITH ACTIVITY AGAINST HEPATITIS B VIRUS	Kristjan S. Gudmundsson; Susan M. Daluge; Lynn D. Condreay; Lance C. Johnson

Volume 21, Issue 10 (2002)

619-635	A NEW CLASS OF ACYCLIC NUCLEOSIDE PHOSPHONATES: SYNTHESIS AND BIOLOGICAL ACTIVITY OF 9-{[(PHOSPHONOMETHYL)AZIRIDIN-1-YL]METHYL}GUANINE (PMAMG) AND ANALOGUES	Ghassan Abu Sheikha; Paolo La Colla; Anna Giulia Loi
637-649	DAUNOMYCIN BINDING TO DEOXYPOLYNUCLEOTIDES WITH ALTERNATING SEQUENCES: COMPLETE THERMODYNAMIC PROFILES OF HETEROGENEOUS BINDING SITES	Dongchul Suh; Yu-Kyoung Oh; Man-Wook Hur; Byungchan Ahn; Jonathan B. Chaires
651-664	INCORPORATION OF 8-HISTAMINYL-DEOXYADENOSINE [8-(2-(4-IMIDAZOLYL)ETHYLAMINO)-2′-DEOXYRIBOADENOSINE] INTO OLIGODEOXYRIBONUCLEOTIDES BY SOLID PHASE PHOSPHORAMIDITE COUPLING	Leonard Lermer; John Hobbs; David M. Perrin
665-680	SYNTHESIS AND BIOLOGICAL EVALUATION OF ENDOCYCLIC 2′,3′-DIDEHYDRO- 2′,3′-DIDEOXYMETHANOCARBA ADENOSINE	Danaè R. Quirk Dorr; Robert Vince
681-694	SYNTHESIS OF 5-(PYRIDINYL AND PYRIDINIUMYL)-2′-DEOXYURIDINE NUCLEOSIDES: REVERSIBLE ELECTRON TRAPS FOR DNA	Samir T. Gaballah; Thomas L. Netzel
695-708	INHIBITION OF SOME HEPATIC GLYCOSIDASES BY THE DISECO NUCLEOSIDE, 4-AMINO-3-(D-GLUCOPENTITOL-1-YL)- 5-MERCAPTO-1,2,4-TRIAZOLE AND ITS 3-METHYL ANALOG	Mahmoud Balbaa; Hamdi Mansour; Hany El-Sawy; El-Sayed H. El-Ashry
709-721	SYNTHESIS AND ANTI-HCMV ACTIVITY OF NOVEL ACYCLIC NUCLEOSIDES	Jae Young Lee; Chang Hyun Oh; Ok Hyun Ko; Joon Hee Hong
723-735	REACTION OF N³-BENZOYL-3′,5′-O-(DI-TERT-BUTYLSILANEDIYL)URIDINE WITH HINDERED ELECTROPHILES: INTERMOLECULAR N³ To 2′-O PROTECTING GROUP TRANSFER	Lei Zhu; Osvaldo dos Santos; Nadrian C. Seeman; James W. Canary

Volume 21, Issue 8-9 (2002)

505-533	SYNTHESIS AND ANTI-HIV ACTIVITY OF [D4U]-[TROVIRDINE ANALOGUE] AND [D4T]-[TROVIRDINE ANALOGUE] HETERODIMERS AS INHIBITORS OF HIV-1 REVERSE TRANSCRIPTASE	D. Gavriliu; C. Fossey; A. Ciurea; Z. Delbederi; E. Sugeac; D. Ladurée; S. Schmidt; G. Laumond; A. M. Aubertin
535-545	INTERACTION OF DISTAMYCIN A AND NETROPSIN WITH QUADRUPLEX AND DUPLEX STRUCTURES: A COMPARATIVE ¹H-NMR STUDY	Antonio Randazzo; Aldo Galeone; Veronica Esposito; Michela Varra; Luciano Mayol
547-560	SYNTHESIS OF 5-(2,2′-BIPYRIDINYL AND 2,2′-BIPYRIDINEDIIUMYL)-2′-DEOXYURIDINE NUCLEOSIDES: PRECURSORS TO METALLO-DNA CONJUGATES	Samir T. Gaballah; Charles E. Kerr; Bruce E. Eaton; Thomas L. Netzel
561-580	TWO EFFICIENT POLYMERIC CHEMICAL PLATFORMS FOR OLIGONUCLEOTIDE MICROARRAY PREPARATION	Clarissa Consolandi; Bianca Castiglioni; Roberta Bordoni; Elena Busti; Cristina Battaglia; Luigi Rossi Bernardi; Gianluca De Bellis
581-598	SYNTHESES OF NOVEL SUBSTITUTED-BORANOPHOSPHATE NUCLEOSIDES	Kamesh Vyakaranam; Geeta Rana; Bernard F. Spielvogel; John A. Maguire; Narayan S. Hosmane
599-617	SYNTHESIS AND HYBRIDIZATION PROPERTIES OF RNA CONTAINING 8-CHLOROADENOSINE	Lisa S. Chen; Terry L. Sheppard

Volume 21, Issue 6-7 (2002)

411-416	A DIRECT ROUTE TO 2-(β-D-RIBOFURANOSYLTHIO)PYRIDINE GLYCOSIDES	Galal H. Elgemeie; Abdel-Fatah Z. Heikel; Mona A. Ahmed
417-426	CHEMICAL STABILITY OF 2′-DEOXY-5-METHYLISOCYTIDINE DURING OLIGODEOXYNUCLEOTIDE SYNTHESIS AND DEPROTECTION	Chenxia Wang; Jialiang Jiang; Thomas R. Battersby
427-433	FORMATION OF 2′-DEOXY-2-NITROADENOSINES BY REACTION OF 2′-DEOXYADENOSINES WITH COPPER(II) NITRATE/ACETIC ANHYDRIDE	Toyo Kaiya; Haruko Tanaka; Kohfuku Kohda
435-447	REGIOSELECTIVE 1-ALKYLATION OF 2′-DEOXYGUANOSINE	Yanhe Huang; Francis Johnson
449-462	ANALYSIS OF RELATIVE POSITIONS OF RIBONUCLEOTIDE BASES IN A CRYSTAL STRUCTURE OF RIBOSOME	Akitsugu Takasu; Kimitsuna Watanabe; Gota Kawai
463-467	SYNTHESIS AND CHARACTERIZATION OF ADENOSINE ADDUCTS OF ARYLAMINES	N. V. Anil Kumar; K. Mantelingu; K. S. Rangappa
469-475	SYNTHESIS OF 1-(2-NAPHTHYLSULFONYL)PYRAZOLE-C-GLYCOSIDES	Abd El-Hamid Ismail; Abdel Aleem Hassan Abdel Aleem; Hamed Abdel Bary; Samy El-Assaly
477-493	NUCLEIC ACID COMPONENTS AND THEIR ANALOGUES: A NOVEL AND EFFICIENT METHOD FOR THE SYNTHESIS OF A NEW CLASS OF BIPYRIDYL AND BIHETEROCYCLIC-NITRO GEN THIOGLYCOSIDES FROM PYRIDINE-2(1H)-THIONES	Galal H. Elgemeie; Mervat M. El-Enany; Mohamed M. Ismail; Eman K. Ahmed
495-503	CONSEQUENCES OF POLYMORPHISM OF 5′-GMP.Na₂ IN THE VIBRATIONAL SPECTRA OF METAL COMPLEXES AND ISOTOPIC DERIVATIVES	M. de la Fuente; R. Navarro; A. Hernanz

Volume 21, Issue 4-5 (2002)

275-286	SULFOXIDE-METAL EXCHANGE FOR THE SYNTHESIS OF THE 2′-TRIBUTYLSTANNYL DERIVATIVE OF 2′,3′-DIDEHYDRO-2′,3′-DIDEOXYURIDINE (d4U): A GENERAL ENTRY TO 2′-CARBON-SUBSTITUTED ANALOGUES OF d4U	Hiroki Kumamoto; Sayoko Onuma; Kumiko Tsuchiya; Yuko Egusa; Hiromichi Tanaka; Tsuyoshi Satoh
287-325	PYRIMIDINETHIONE NUCLEOSIDES AND THEIR DEAZA ANALOGUES	Galal H. Elgemeie; Eman A. Kamal
327-334	UNSATURATED FLUOROKETONUCLEOSIDES AS ANTICANCER AGENTS: THE SYNTHESIS AND BIOLOGICAL ACTIVITY OF 5-FLUORO-1-(3,4-DI-DEOXY-3-FLUORO-6-O-TRITYL-β-D-GLYCERO-HEX-3-ENO-PYRANOS-2-ULOSYL) URACIL	M. J. Egron; B. I. Dorange; K. Antonakis; J. Herscovici; A. P. Ollapally
335-360	SYNTHESIS OF THIAAZAHETEROCYCLE NUCLEOSIDE ANALOGUES	A. Ané; G. Prestat; M. Thiam; S. Josse; M. Pipelier; J. P. Pradère; D. Dubreuil
361-375	NEW GLYCOSYL-(CARBOXAMIDE)-1,2,3-TRIAZOLE-N-NUCLEOSIDES: SYNTHESIS AND ANTITUMOR ACTIVITY	Najim A. Al-Masoudi; Yaseen A. Al-Soud
377-383	SYNTHESIS OF 1-(2-HYDROXY-3-METHOXYPROPYL)URACILS AND THEIR ACTIVITY AGAINST L1210 AND MACROPHAGE RAW 264.7 CELLS	Alicja Copik; Jerzy Suwinski; Krzysztof Walczak; Joanna Bronikowska; Zenon Czuba; Wojciech Król
385-392	SYNTHESIS AND CHARACTERIZATION OF NUCLEOSIDE DERIVATIVES, N-(BENZOYL)-N-(DEOXYGUANOSIN-8-YL)-4-AMINOBIPHENYL AND N-(2′-DEOXYGUANOSIN-8-YL)-4-AMINOBIPHENYL VIA α-PHENYL-N-(4-BIPHENYL)NITRONE	H. Mallesha; K. R. Ravi Kumar; K. S. Rangappa
393-400	MICROWAVE ASSISTED HIGH YIELDING PREPARATION OF N-PROTECTED 2′-DEOXYRIBONUCLEOSIDES USEFUL FOR OLIGONUCLEOTIDE SYNTHESIS	N. S. Rao; P. Kumar; V. K. Chauhan; B. S. Garg; K. C. Gupta
401-409	REACTION Of GLYCOSYL ISOTHIOCYNATES WITH 3-INDOLYLAMINOMETHYL-KETONE HYDROCHLORIDE	Mohamed A. Saleh

Volume 21, Issue 3 (2002)

191-206	SYNTHESIS AND IN VITRO CYTOTOXIC AND ANTIVIRAL ACTIVITIES OF 1-(2,5,6-TRIDEOXY-6-HALOGENOHEPT-5-ENOFURANURONONITRILE)THYMINE AND DERIVATIVES	Jean M. J. Tronchet; Frederic Chalard; Elisabeth Rivara-Minten; Michel Seman; Erik De Clercq; Jan Balzarini; Pierre Dilda
207-216	SYNTHESIS AND BIOLOGICAL EVALUATION OF S-GLYCOSYLATED PYRIDINES	Adel M. E. Attia
217-230	3′-AZIDO-3′-DEOXY-5′-O-ISONICOTINOYLTHYMIDINE, A NEW PRODRUG OF ZIDOVUDINE. SYNTHESIS, SOLID STATE CHARACTERIZATION AND ANTI HIV-1 ACTIVITY	Marisa I. Motura; Guillermo N. Moroni; Silvina A. Teijeiro; Horacio Salomón; Margarita C. Briñón
231-241	SYNTHESIS AND IN VITRO ANTIBACTERIAL ACTIVITY OF NOVEL 5′-O-ANALOG DERIVATIVES OF ZIDOVUDINE AS POTENTIAL PRODRUGS	Guillermo N. Moroni; Patricia M. Bogdanov; Margarita C. Briñón
243-255	SYNTHESIS, ANTIVIRAL AND CYTOSTATIC ACTIVITIES, OF CARBOCYCLIC NUCLEOSIDES INCORPORATING A MODIFIED CYCLOPENTANE RING. IV. ADENOSINE AND URIDINE ANALOGUES	M. Isabel Nieto; Olga Caamaño; Franco Fernández; María Gómez; Jan Balzarini; Erik De Clercq
257-274	SYNTHESIS AND BIOLOGICAL EVALUATION OF ISONUCLEOSIDES DERIVED FROM METHYL 3,5-ANHYDRO-2-O-(2-FLUOROBENZYL)-d-XYLOFURANOSIDES	Jörn Wirsching; Oliver Schulze; Jürgen Voss; Anja Giesler; Jürgen Kopf; Gunadi Adiwidjaja; Jan Balzarini; Erik De Clercq

Volume 21, Issue 2 (2002)

111-123	SYNTHESIS AND HYBRIDIZATION STUDIES OF A 5-AMINOPENTANOIC ACID NUCLEOBASE (APN) DIMER	Susan F. Donaldson; Stephen C. Bergmeier; Jennifer V. Hines; Melinda S. Gerdeman
125-137	STRUCTURAL TRANSITIONS IN POLYCYTIDYLIC ACID: PROTON BUFFER CAPACITY DATA	Margarita I. Zarudnaya; Svitlana P. Samijlenko; Andriy L. Potyahaylo; Dmytro M. Hovorun
139-154	EFFECT OF 5-FU SUBSTITUTION AND MUTATION ON Sm PROTEIN BINDING TO HUMAN U4 snRNA	Wei Cui; William H. Gmeiner
155-163	NEW SYNTHESIS OF L-FMAU FROM L-ARABINOSE	Marcos L. Sznaidman; Merrick R. Almond; Amir Pesyan
165-176	SYNTHESIS AND BIOLOGICAL EVALUATION OF SOME ACYCLIC α-(1H-PYRAZOLO[3,4-d]PYRIMIDIN-4-YL)THIOALKYLAMIDE NUCLEOSIDES	O. Moukha-chafiq; M. L. Taha; H. B. Lazrek; J. J. Vasseur; E. De Clercq
177-190	P-CHIRAL OLIGONUCLEOTIDES. 2D ROESY NMR ASSIGNMENT OF ABSOLUTE CONFIGURATION AT PHOSPHORUS AND CONFORMATIONAL ANALYSIS OF 5′-O-MONOMETHOXYTRITYL-(2′-O-DEOXYRIBONUCLEOSIDE) 3′-O-[O-(4-NITROPHENYL)]METHANEPHOSPHONATES	Stefan Jankowski; Agnieszka B. Olejniczak; Zbigniew J. Lesnikowski

Volume 21, Issue 1 (2002)

1-13	NEW METHOD FOR THE PREPARATION OF 3′- AND 2′-O-PHOSPHORAMIDITES OF 2′- AND 3′-DIFLUOROMETHYLURIDINE DERIVATIVES	Pawel J. Serafinowski; Catherine A. Brown
15-21	Glucopyranosides Derived From 6-Aryl-5-Cyano-2-(Methylthio)Pyrimidin-4(3H)Ones	Ibrahim M. Abdou; Adel M. Attia; Lucjan Strekowski
23-43	SYNTHESIS OF NOVEL HYDROXYMETHYL SUBSTITUTED ANALOGUES RELATED TO CARBOVIR AND NEPLANOCIN A	Henrik Franzyk; Søren Rosendal Jensen; Carl Erik Olsen; Jon Holbech Rasmussena
45-54	“SENSELESS” ANTIVIRAL POLYRIBONUCLEOTIDES: POLY (1-PROPARGYLINOSINIC ACID)	Robyn M. Hyde; Robert W. Buckheit Jr.; Arthur D. Broom
55-64	DIFFICULTIES IN THE DEPROTECTION OF 1,2-KETALS IN NUCLEOSIDES CONTAINING ALKYLIDENCARBAZOYL GROUPS	Julia Magdalena; Susana Fernández; Miguel Ferrero; Vicente Gotor
65-72	A FACILE SYNTHESIS OF CIS-4-AMINO-2-CYCLOPENTENE-1-METHANOL, A KEY INTERMEDIATE FOR THE SYNTHESIS OF CARBOCYCLIC NUCLEOSIDES	Gwang-il An; Hakjune Rhee
73-78	Microwave Induced Synthesis of Ribonucleosides on Solid Support	Mariola Andrzejewska; Jarosław Kamiński; Zygmunt Kazimierczuk
79-82	SYNTHESIS AND ENZYMATIC CHARACTERIZATION OF P₁-THIO-P₂-OXO TRIDEOXYNUCLEOSIDE DIPHOSPHATES HAVING AZT, FdU, OR dT AT THE 3′-POSITION	László Ötvös; Zoltán Bajor; Ferenc Kraicsovits; Gyula Sági; Zsuzsanna Tegyey
93-106	SYNTHESIS AND ANTIVIRAL EVALUATION OF SOME NEW GLYCOSYLTHIOUREAS CONTAINING A QUINAZOLINONE NUCLEUS	Mohamed A. Saleh; Mohamed F. Adbel-Megged; Mohamed A. Abdo; Abdel-Basset M. Shokr

Volume 20, Issue 12 (2001)

1903-1913	PREPARATION OF BASE-DEUTERATED 2′-DEOXYADENOSINE NUCLEOSIDES AND THEIR SITE-SPECIFIC INCORPORATION INTO DNA	Panadda Chirakul; Justin R. Litzer; Snorri Th. Sigurdsson
1915-1925	SYNTHESIS OF CARBOCYCLIC OROTIDINE ANALOGS AS POTENTIAL OROTIDINE DECARBOXYLASE INHIBITORS	Gyu Y. Song; Fardos N. M. Naguib; Mahmoud H. el Kouni; Chung K. Chu
1927-1939	SYNTHESIS AND ANTI-HIV ACTIVITY OF THYMIDINE ANALOGUES BEARING A 4′-CYANOVINYL GROUP AND SOME DERIVATIVES THEREOF	Jean M. J. Tronchet; Imre Kovacs; Pierre Dilda; Michel Seman; Graciela Andrei; Robert Snoeck; Erik De Clercq; Jan Balzarini
1941-1948	SYNTHESIS OF CYCLOBUTANE ANALOGUES OF THE ANTIVIRAL CYCLOPROPANE NUCLEOSIDE A-5021	Tomoyuki Onishi; Takashi Tsuji
1949-1960	SYNTHESIS AND ANTI-HIV ACTIVITY OF NEW MODIFIED 1,2,3-TRIAZOLE ACYCLONUCLEOSIDES	H. B. Lazrek; M. Taourirte; T. Oulih; J. L. Barascut; J. L. Imbach; C. Pannecouque; M. Witrouw; E. De Clercq
1961-1973	REGIOSELECTIVE SYNTHESIS OF 1,3,5-¹³C₃ AND 2,4-¹³C₂-LABELED 2-DEOXYRIBONOLACTONES	Paul J. Hatala; James Kallmerten; Philip N. Borer
1975-2000	SYNTHESIS OF HALOGEN-SUBSTITUTED 3-DEAZAADENOSINE AND 3-DEAZAGUANOSINE ANALOGUES AS POTENTIAL ANTITUMOR/ANTIVIRAL AGENTS	Mao-Chin Liu; Mei-Zhen Luo; Diane E. Mozdziesz; Tai-Shun Lin†; Ginger E. Dutschman; Elizabeth A. Gullen; Yung-Chi Cheng; Alan C. Sartorelli

Volume 20, Issue 10-11 (2001)

1751-1760	TT DINUCLEOTIDES CONTAINING AN ISOXAZOLINE MOIETY: SYNTHESIS AND BINDING AFFINITY STUDY	Jong Rock Kong; Sang Kook Kim; Byung Jo Moon; Su Jeong Kim; Byeang Hyean Kim
1761-1774	CONDENSATION OF TRIFORMYLMETHANE WITH GUANOSINE	Niangoran Koissi; Kari Neuvonen; Tony Munter; Leif Kronberg; Harri Lönnberg
1775-1781	PREPARATION OF 1-(3-C-(PROPA-1,2-DIENYL)-D-RIBO-PENTOFURANOSYL)URACIL, AN ALLENIC NUCLEOSIDE	Jérôme Dauvergne; Alain Burger; Jean-François Biellmann
1783-1796	CONFORMATIONAL RIGIDITY INTRODUCED BY 2′,5′-PHOSPHODIESTER LINKS IN DNA	Anil Kumar; Debasis Dass; M. Atreyi; M. V. R. Rao; S. B. Katti
1797-1810	SYNTHESIS AND BIOLOGICAL ACTIVITY OF 4-SUBSTITUTED 1-[1-(2-HYDROXYETHOXY)- METHYL-1,2,3-TRIAZOL-(4 & 5)-YLMETHYL]-1H-PYRAZOLO[3,4-d]PYRIMIDINES	O. Moukha-Chafiq; M. L. Taha; H. B. Lazrek; C. Pannecouque; M. Witvrouw; E. De Clercq; J. L. Barascut; J. L. Imbach
1811-1821	SYNTHESIS AND BIOLOGICAL EVALUATION OF SOME 4-SUBSTITUTED 1-[1-(4-HYDROXYBUTYL)-1,2,3-TRIAZOL-(4 & 5)-YLMETHYL]-1H-PYRAZOLO-[3,4-d]PYRIMIDINES	O. Moukha-Chafiq; M. L. Taha; H. B. Lazrek; J. J. Vasseur; C. Pannecouque; M. Witvrouw; E. De Clercq
1823-1830	SYNTHESIS OF CARBOCYCLIC ANALOGS OF 2′,3′-DIDEOXYSANGIVAMYCIN, 2′,3′-DIDEOXYTOYOCAMYCIN, AND 2′,3′-DIDEOXYTRICIRIBINE	Kristjan S. Gudmundsson; Zhicheng Wang; Susan M. Daluge; Paul L. Feldman
1831-1841	SYNTHESIS OF 5-METHYLAMINO-2′-DEOXYURIDINE DERIVATIVES	Bruno Catalanotti; Aldo Galeone; Luciano Mayol; Giorgia Oliviero; Daniela Rigano; Michela Varra
1843-1849	THE SYNTHESIS OF DITHYMIDINE BORANOPHOSPHATE BY THE OXATHIAPHOSPHOLANE APPROACH	Andrzej Okruszek; Agnieszka Sierzchała; Katarzyna Żmudzka; Wojciech J. Stec
1851-1858	SITE SPECIFIC INCORPORATION OF 6-AZAURIDINE INTO THE GENOMIC HDV RIBOZYME ACTIVE SITE	Adegboyega K. Oyelere; Scott A. Strobel
1859-1870	5′-BIS-PYRENYLATED OLIGONUCLEOTIDES DISPLAY ENHANCED EXCIMER FLUORESCENCE UPON HYBRIDIZATION WITH DNA AND RNA	E. Kostenko; M. Dobrikov; N. Komarova; D. Pyshniy; V. Vlassov; M. Zenkova
1871-1879	EFFICIENT ASSESSMENT OF MODIFIED NUCLEOSIDE STABILITY UNDER CONDITIONS OF AUTOMATED OLIGONUCLEOTIDE SYNTHESIS: CHARACTERIZATION OF THE OXIDATION AND OXIDATIVE DESULFURIZATION OF 2-THIOURIDINE	E. Sochacka
1881-1889	O-GLYCOSIDES OF N-HYDROXYINDOLES[1]	S. N. Lavrenov; A. M. Korolev; M. N. Preobrazhenskaya
1891-1902	SYNTHESIS AND ANTIVIRAL EVALUATION OF N-GLYCOSIDES DERIVED FROM 6-AMINO-3-ARYL-2-METHYL-4-(3H)-QUINAZOLINONES	Mohamed A. Saleh; Youssef A. Abbas; Fouad Eabdel-Hai; Shaban A. Youssef

Volume 20, Issue 9 (2001)

1615-1623	SYNTHESIS AND STEREOCHEMICAL CHARACTERIZATION OF DIASTEREOMERIC NUCLEOSIDE-PHOSPHOROTHIOSELENOATES BY NMR METHODS	Mária Kajtár-Peredy; István Tömösközi; Eszter Gács-Baitz
1647-1654	A NOVEL AFFINITY CHROMATOGRAPHY METHOD FOR THE CO-PURIFICATION OF DEOXYCYTIDINE KINASE AND CYTIDINE DEAMINASE	Hiroyuki Uchida; Hidetaka Morinaga; Takashi Misaki; Takamichi Miyazaki; Takayuki Uwajima; Tohru Obata; Yoshio Endo; Akira Matsuda; Takuma Sasaki
1655-1670	SYNTHESIS OF 5-ALKENYLATED D4T ANALOGUES VIA THE Pd-CATALYZED CROSS-COUPLING REACTION	A. Ciurea; C. Fossey; S. Benzaria; D. Gavriliu; Z. Delbederi; B. Lelong; D. Ladurée; A. M. Aubertin; A. Kirn
1671-1682	SYNTHESIS AND STRUCTURE DETERMINATION OF SOME OXADIAZOLE-2-THIONE AND TRIAZOLE-3-THIONE GALACTOSIDES	Roshan Ahmad; Rashid Iqbal; Humaira Akhtar; Zia-ul-Haq; Helmut Duddeck; Lech Stefaniak†; Jerzy Sitkowski
1683-1690	NOVEL REVERSION REACTION OF D-ARABINO-HEXOSE PHENYLOSOTRIAZOLE. A USEFUL MODEL IN NATURAL GLYCOSIDE AND POLYSACCHARIDE ANALYSIS	Hammed H. A. M. Hassan; Amel H. F. El-Husseiny
1691-1704	SYNTHESIS OF CERTAIN 2′-DEOXYURIDINE DERIVATIVES CONTAINING SUBSTITUTED PHENOXY GROUPS ATTACHED TO C-5′; EVALUATION AS POTENTIAL dUTP ANALOGUES	Jonathan H. Marriott; G. Wynne Aherne; Anthea Hardcastle; Michael Jarman
1705-1721	SYNTHESIS AND BINDING AFFINITY OF A CHIRAL PNA ANALOGUE	Ying Li; Tao Jin; Keliang Liu
1723-1734	SYNTHESIS OF SELENIUM-DERIVATIZED NUCLEOSIDES AND OLIGONUCLEOTIDES FOR X-RAY CRYSTALLOGRAPHY	Nicolas Carrasco; Dov Ginsburg; Quan Du; Zhen Huang
1735-1750	SYNTHESIS OF 2-THIOHYDANTOINS AND THEIR S-GLUCOSYLATED DERIVATIVES AS POTENTIAL ANTIVIRAL AND ANTITUMOR AGENTS	Ahmed I. Khodair

Volume 20, Issue 8 (2001)

1439-1447	SYNTHESIS AND BIOLOGICAL ACTIVITIES OF (Z) AND (E) α-ETHENYL ACYCLONUCLEOSIDES	N. Redwane; H. B. Lazrek; J. L. Barascut; J. L. Imbach; J. Balzarini; M. Witvrouw; E. De Clercq
1449-1461	SYNTHESIS OF A NEW 5′-O-TRIPHOSPHATE ANALOG OF 5-METHYL 2′-O-DEOXYCYTIDINE. PRELIMINARY IN VITRO LABELING FOR NON-RADIOACTIVE DETECTION OF DNA	Ch. Rodríguez-Tanty; R. Pérez; J. Miranda; H. Vélez-Castro; A. Rosado; A. Macías; V. Vidal-Alles; M. J. Araña; N. Pérez Souto; D. Higginson-Clarke; A. M. Riverón
1463-1471	CONVENIENT METHOD FOR THE PREPARATION OF 2′-DEOXYRIBOSYLUREA BY THYMIDINE OXIDATION AND NMR STUDY OF BOTH ANOMERS	Igor Dubey; Genevi�ve Pratviel; Anne Robert; Bernard Meunier
1473-1483	HIGHLY EFFICIENT RANDOM MUTAGENESIS IN TRANSCRIPTION-REVERSE-TRANSCRIPTION CYCLES BY A HYDROGEN BOND AMBIVALENT NUCLEOSIDE 5′-TRIPHOSPHATE ANALOGUE: POTENTIAL CANDIDATES FOR A SELECTIVE ANTI-RETROVIRAL THERAPY	K. Moriyama; C. Otsuka; D. Loakes; K. Negishi
1485-1495	NMR STUDIES AND SEMI-EMPIRICAL ENERGY CALCULATIONS FOR CYCLIC ADP-RIBOSE	Trevor J. Rutherford; John Wilkie; Chinh Q. Vu; Klaus D. Schnackerz; Myron K. Jacobson; David Gani
1497-1522	2′-C-ALKOXY AND 2′-C-ARYLOXY DERIVATIVES OF N-(2-PHOSPHONOMETHOXYETHYL)-PURINES AND -PYRIMIDINES: SYNTHESIS AND BIOLOGICAL ACTIVITY	Dominik Rejman; Milena Masojídková; Eric De Clercq; Ivan Rosenberg
1523-1531	A NEW METHOD FOR THE SYNTHESIS OF N²-ALKYLGUANOSINES USING MITSUNOBU REACTION AS A KEY STEP	Shigetada Kozai; Aya Yorikane; Tokumi Maruyama
1555-1569	SYNTHESIS OF 4-ACYL-1H-1,2,3-TRIAZOLIC NUCLEOSIDES	Anna C. Cunha; Letícia O. R. Pereira; Rodrigo O. P. de Souza; Maria Cecília B. V. de Souza; Vitor F. Ferreira
1571-1582	COMPARISON OF THE ANTIVIRAL ACTIVITY OF HYDROPHOBIC AMINO ACID PHOSPHORAMIDATE MONOESTERS OF 2′, 3′-DIDEOXYADENOSINE (DDA) AND 3′-AZIDO-3′-DEOXYTHYMIDINE (AZT)	Shu-ling Chang; George Griesgraber; Carston R. Wagner
1583-1598	SYNTHESIS AND BIOLOGICAL ACTIVITY OF 4′-C-HYDROXYMETHYL-2′-FLUORO- D-ARABINOFURANOSYLPURINE NUCLEOSIDES	Anita T. Shortnacy-Fowler; Kamal N. Tiwari; John A. Montgomery; John A. Secrist III
1599-1614	ACYCLIC NUCLEOSIDE/NUCLEOTIDE ANALOGUES WITH AN IMIDAZOLE RING SKELETON	Huan-Ming Chen; Ramachandra S. Hosmane

Volume 20, Issue 4-7 (2001)

271-285	ACYCLIC/CARBOCYCLIC GUANOSINE ANALOGUES AS ANTI-HERPESVIRUS AGENTS	E. De Clercq; G. Andrei; R. Snoeck; L. De Bolle; L. Naesens; B. Degrève; J. Balzarini; Y. Zhang; D. Schols; P. Leyssen; C. Ying; J. Neyts
287-296	NOVEL ARYL SUBSTITUTED BICYCLIC FURO NUCLEOSIDES AS EXTREMELY POTENT AND SELECTIVE ANTI-VZV AGENTS	Christopher McGuigan; Hubert Barucki; Antonella Carangio; Sally Blewett; Sheila Srinivasan; Graciela Andrei; Robert Snoeck; Erik De Clercq; Jan Balzarini
297-306	ACTIVATION OF ANTI-REVERSE TRANSCRIPTASE NUCLEOTIDE ANALOGS BY NUCLEOSIDE DIPHOSPHATE KINASE: IMPROVEMENT BY α-BORANOPHOSPHATE SUBSTITUTION	Benoit Schneider; Philippe Meyer; Simon Sarfati; Laurence Mulard; Catherine Guerreiro; Joëlle Boretto; Joël Janin; Michel Véron; Dominique Deville-Bonne; Bruno Canard
307-314	SYNTHESIS, HYDROLYSIS AND ANTI-EBV ACTIVITY OF A SERIES OF 3′-MODIFIED cycloSal-BVDUMP PRONUCLEOTIDES	C. Meier; A. Lomp; A. Meerbach; P. Wutzler
315-321	DESIGN OF NEW MONONUCLEOTIDE PRODRUGS: ARYL (SATE) PHOSPHOTRIESTER DERIVATIVES	S. Peyrottes; N. Schlienger; T. Beltran; I. Lefebvre; A. Pompon; G. Gosselin; A. -M. Aubertin; J. -L. Imbach; C. Périgaud
323-328	SYNTHESIS AND ANTICANCER ACTIVITY OF 4-AMINO-5-OXO-8-(β-D-XYLOFURANOSYL) PYRIDO[2,3-d]PYRIMIDINE	Zbigniew Pietrzkowski; Jean-Luc Girardet; Cathey Esler; Guangyi Wang
329-332	SYNTHESIS AND ANTIVIRAL ACTIVITY OF METHYLENEDIFLUOROCYCLOPROPANE ANALOGUES OF NUCLEOSIDES	R. Wang; M. B. Ksebati; J. C. Drach; J. Zemlicka
333-341	RIBOSE MODIFIED NUCLEOSIDES AND NUCLEOTIDES AS LIGANDS FOR PURINE RECEPTORS	K. A. Jacobson; R. G. Ravi; E. Nandanan; H. S. Kim; S. Moro; Y. C. Kim; K. Lee; D. Barak; V. E. Marquez; X. D. Ji
343-360	2-SUBSTITUTED PI SYSTEM DERIVATIVES OF ADENOSINE THAT ARE CORONARY VASODILATORS ACTING VIA THE A_2A ADENOSINE RECEPTOR	J. Zablocki; V. Palle; B. Blackburn; E. Elzein; G. Nudelman; S. Gothe; Z. Gao; Z. Li; S. Meyer; L. Belardinelli
361-367	FLUORESCENCE RESONANCE ENERGY TRANSFER DYE NUCLEOTIDE TERMINATORS: A NEW SYNTHETIC APPROACH FOR HIGH-THROUGHOUT DNA SEQUENCING	Satyam Nampalli; Mahesh Khot; John R. Nelson; Parke K. Flick; Carl W. Fuller; Shiv Kumar
369-374	DESIGN OF MULTIDYE SYSTEMS FOR FRET-BASED APPLICATIONS	Mikhail S. Shchepinov; Vladimir A. Korshun
375-381	ANALYSIS OF ANTI-HIV NUCLEOSIDE INHIBITORS BY CAPILLARY ELECTROPHORESIS-ELECTROSPRAY IONIZATION MASS SPECTROMETRY	L. A. Agrofoglio; X. Cahours; T. T. Tran; H. Dessans; C. Kieda; P. Morin
383-384	THE CONFORMATIONAL SPACE OF NASCENT PEPTIDE-ACCEPTING 3′-AMINOACYL RIBONUCLEOS(T)IDES: ¹H NMR DATA AND AB INITIO CALCULATIONS OF PUROMYCIN AND SOME SYNTHETIC ANALOGS	Nhat Quang Nguyen Trung; Peter Strazewski; Martin Olsson; Måns Ehrenberg
385-388	UNDERSTANDING THE MODE OF ACTION OF L-NUCLEOSIDES AS ANTIVIRAL AGENTS: A MOLECULAR MODELING APPROACH	Kyeong Lee; Youhoon Chong; Chung K. Chu
389-396	LNA (LOCKED NUCLEIC ACID) AND THE DIASTEREOISOMERIC α-L-LNA: CONFORMATIONAL TUNING AND HIGH-AFFINITY RECOGNITION OF DNA/RNA TARGETS	Jesper Wengel; Michael Petersen; Kathrine E. Nielsen; Gitte A. Jensen; Anders E. Håkansson; Ravindra Kumar; Mads D. Sørensen; Vivek K. Rajwanshi; Torsten Bryld; Jens Peter Jacobsen
397-399	THE ROLE OF ANTISENSE OLIGONUCLEOTIDES IN THE WAVE OF GENOMIC INFORMATION	Brenda F. Baker
401-410	TELOMERASE INHIBITORS – OLIGONUCLEOTIDE PHOSPHORAMIDATES AS POTENTIAL THERAPEUTIC AGENTS	S. Gryaznov; K. Pongracz; T. Matray; R. Schultz; R. Pruzan; J. Aimi; A. Chin; C. Harley; B. Shea-Herbert; J. Shay; Y. Oshima; A. Asai; Y. Yamashita
411-417	DNA TRIPLE-HELIX FORMATION AT PYRIMIDINE-PURINE INVERSION SITES	Serge P. Parel; Judith Marfurt; Christian J. Leumann
419-428	PNA-RELATED OLIGONUCLEOTIDE MIMICS AND THEIR EVALUATION FOR NUCLEIC ACID HYBRIDIZATION STUDIES AND ANALYSIS	V. Efimov; M. Choob; A. Buryakova; D. Phelan; O. Chakhmakhcheva
429-440	PROPERTIES OF ARABINONUCLEIC ACIDS (ANA & 20′F-ANA): IMPLICATIONS FOR THE DESIGN OF ANTISENSE THERAPEUTICS THAT INVOKE RNASE H CLEAVAGE OF RNA	M. J. Damha; A. M. Noronha; C. J. Wilds; J. -F. Trempe; A. Denisov; R. T. Pon; K. Gehring
441-449	RNA AND N3′ → P5′ KISSING APTAMERS TARGETED TO THE TRANS-ACTIVATION RESPONSIVE (TAR) RNA OF THE HUMAN IMMUNODEFICIENCY VIRUS-1	Fabien Darfeuille; Christian Cazenave; Sergei Gryaznov; Frédéric Ducongé; Carmelo Di Primo; Jean-Jacques Toulmé
451-459	INHIBITION OF (CYTOSINE C5)-METHYLTRANSFERASE BY OLIGONUCLEOTIDES CONTAINING FLEXIBLE (CYCLOPENTANE) AND CONFORMATIONALLY CONSTRAINED (BICYCLO[3.1.0]HEXANE) ABASIC SITES	Victor E. Marquez; Peiyuan Wang; Marc C. Nicklaus; Martin Maier; Muthiah Manoharan; Judith K. Christman; Nilesh K. Banavali; Alexander D. Mackerell Jr.
461-470	INTRACELLULAR Ca²-MOBILIZING ADENINE NUCLEOTIDES. SYNTHESIS AND BIOLOGICAL ACTIVITY OF CYCLIC ADP-CARBOCYCLIC-RIBOSE AND C-GLYCOSIDIC ANALOG OF ADENOPHOSTIN A	Satoshi Shuto; Masayoshi Fukuoka; Hiroshi Abe; Akira Matsuda
471-480	OLIGONUCLEOTIDE ANALOGUE INTERFERENCE WITH THE HIV-1 TAT PROTEIN-TAR RNA INTERACTION	Andrey Arzumanov; Andrew P. Walsh; Xiaohai Liu; Vivek K. Rajwanshi; Jesper Wengel; Michael J. Gait
481-486	6-OXOCYTIDINE CONTAINING OLIGONUCLEOTIDES INHIBIT THE HIV-1 INTEGRASE IN VITRO	P. Brodin; M. Pinskaya; U. Parsch; J. Bischerour; H. Leh; E. Romanova; J. W. Engels; M. Gottikh; J. F. Mouscadet
487-492	ZIDOVUDINE (AZT) RESISTANCE IN H9 CELLS DUE TO DECREASED TK EXPRESSION IS ASSOCIATED WITH HYPERMETHYLATION OF TK GENE	B. Gröschel; G. Höver; H. W. Doerr; J. Cinatl Jr.
493-499	STRUCTURAL, DYNAMIC, AND ENZYMATIC PROPERTIES OF MIXED α/β-OLIGONUCLEOTIDES CONTAINING POLARITY REVERSALS	M. W. Germann; J. M. Aramini; B. W. Kalisch; J. H. van de Sande
501-506	ANALOGS OF GUANINE NUCLEOSIDE TRIPHOSPHATES FOR SEQUENCING APPLICATIONS	Mark G. McDougall; Lei Sun; Inna Livshin; Louis P. Hosta; Bernard F. McArdle; Sui-Bi Samols; Carl W. Fuller; Shiv Kumar
507-514	2′-MODIFIED OLIGONUCLEOTIDES FROM METHOXYOXALAMIDO AND SUCCINIMIDO PRECURSORS: SYNTHESIS, PROPERTIES, AND APPLICATIONS	N. Polushin; A. Malykh; O. Malykh; M. Zenkova; N. Chumakova; V. Vlassov; S. Kozyavkin
515-523	ENHANCED INHIBITION OF HIV-1 REPLICATION IN MACROPHAGES BY ANTISENSE OLIGONUCLEOTIDES, RIBOZYMES AND ACYCLIC NUCLEOSIDE PHOSPHONATE ANALOGS DELIVERED IN pH-SENSITIVE LIPOSOMES	N. Düzgünes; S. Simões; V. Slepushkin; E. Pretzer; J. J. Rossi; E. De Clercq; V. P. Antao; M. L. Collins; M. C. Pedroso de Lima
525-531	PHOTOLITHOGRAPHIC SYNTHESIS OF HIGH-DENSITY OLIGONUCLEOTIDE PROBE ARRAYS	Anthony D. Barone; Jody E. Beecher; Paul A. Bury; Chuan Chen; Tina Doede; Jacqueline A. Fidanza; Glenn H. McGall
533-538	HIGH CAPACITY SUBSTRATES AS A PLATFORM FOR A DNA PROBE ARRAY GENOTYPING ASSAY	Jacqueline Fidanza; Marc Glazer; Daniel Mutnick; Glenn McGall; Curt Frank
539-550	SYNTHESIS OF PEPTIDE-OLIGONUCLEOTIDE PHOSPHOROTHIOATE CONJUGATES BY CONVERGENT OR STEPWISE SOLID-PHASE STRATEGIES	Maxim Antopolsky; Alex Azhayev
551-558	NOVEL CLASS OF DNA BINDING MOTIFS BASED ON BISTETRAHYDROFURAN AND BISFURAN SKELETON WITH LONG ALKYL CHAINS	Shigeki Sasaki; Takayuki Shibata; Hidemine Torigoe; Yosinori Shibata; Minoru Maeda
559-566	COVALENT MODIFICATION AND SURFACE IMMOBILIZATION OF NUCLEIC ACIDS VIA THE DIELS-ALDER BIOCONJUGATION METHOD	Gregory M. Husar; Dominick J. Anziano; Michael Leuck; David P. Sebesta
567-576	A CASE STUDY: OLIGONUCLEOTIDE PURIFICATION FROM GRAM TO HUNDRED GRAM SCALE	Ranjit R. Deshmukh; Kjell-Ove Eriksson; Peter Moore; Douglas L. Cole; Yogesh S. Sanghvi
577-585	8-AZA-7-DEAZAADENINE AND 7-DEAZAGUANINE: SYNTHESIS AND PROPERTIES OF NUCLEOSIDES AND OLIGONUCLEOTIDES WITH NUCLEOBASES LINKED AT POSITION-8	F. Seela; H. Debelak
587-596	SYNTHESIS OF NEW CLASSES OF BORON-CONTAINING NUCLEOTIDES	Jinlai Lin; Barbara Ramsay Shaw
597-607	ANTI-HBV SPECIFIC β-L-2′-DEOXYNUCLEOSIDES	Martin L. Bryant; Edward G. Bridges; Laurent Placidi; Abdesslem Faraj; Anna-Giulia Loi; Claire Pierra; David Dukhan; Gilles Gosselin; Jean-Louis Imbach; Brenda Hernandez; Amy Juodawlkis; Bud Tennant; Brent Korba; Paul Cote; Erika Cretton-Scott; Raymond F. Schinazi; Jean-Pierre Sommadossi

Volume 20, Issue 4-7 (2001)

609-619	1-(3-C-ETHYNYL-β-D-RIBO-PENTOFURANOSYL)CYTOSINE (ECYD, TAS-106)1: ANTITUMOR EFFECT AND MECHANISM OF ACTION	Atsushi Azuma; Akira Matsuda; Takuma Sasaki; Masakazu Fukushima
621-628	PRACTICAL SYNTHESIS, SEPARATION, AND STEREOCHEMICAL ASSIGNMENT OF THE PMPA PRO-DRUG GS-7340	H. Chapman; M. Kernan; E. Prisbe; J. Rohloff; M. Sparacino; T. Terhorst; R. Yu
629-634	AN ASSAY SYSTEM TO DETECT THE SELECTIVE ADVANTAGE OF ANTI-HIV RIBOZYME EXPRESSING CD4 T-LYMPHOCYTES	Stefan A. Klein; Christian Klebba; Joachim W. Engels
635-639	TENOFOVIR (PMPA) IS LESS SUSCEPTIBLE TO PYROPHOSPHOROLYSIS AND NUCLEOTIDE-DEPENDENT CHAIN-TERMINATOR REMOVAL THAN ZIDOVUDINE OR STAVUDINE	Lisa K. Naeger; Nicolas A. Margot; Michael D. Miller
641-648	HUMAN RENAL ORGANIC ANION TRANSPORTER 1 (hOAT1) AND ITS ROLE IN THE NEPHROTOXICITY OF ANTIVIRAL NUCLEOTIDE ANALOGS	Tomas Cihlar; Edmund S. Ho; Deborah C. Lin; Andrew S. Mulato
649-652	SYNTHESIS AND ANTIPROLIFERATIVE ACTIVITY OF SOME 4′-C-HYDROXYMETHYL-α- AND -β-D-ARABINO-PENTOFURANOSYL PYRIMIDINE NUCLEOSIDES	Jean-François Griffon; John A. Montgomery; John A. Secrist III
653-656	SYNTHESIS AND IN VITRO EVALUATION OF NOVEL ANTI-VARICELLA-ZOSTER VIRUS (VZV) NUCLEOSIDES	Antonella Carangio; Christopher McGuigan; D. Cahard; Graciela Andrei; Robert Snoeck; Erik De Clercq; Jan Balzarini
657-660	STRUCTURE-ACTIVITY RELATIONSHIPS OF APIO NUCLEOSIDES AS POTENTIAL ANTIVIRAL AGENTS	Lak Shin Jeong; Hyung Ryong Moon; Jun Hee Hong; Su Jeong Yoo; Won Jun Choi; Hea Ok Kim; Hee Sung Ahn; Hye Woo Baek; Moon Woo Chun; Hee-Doo Kim; Jeongmin Kim; Jong-Ryoo Choi
661-664	SYNTHESIS OF CARBOCYCLIC PHOSPHONONUCLEOSIDES	B. Legeret; Z. Sarakauskaite; F. Pradaux; Y. Saito; S. Tumkevicius; L. A. Agrofoglio
665-668	SYNTHESIS AND ANTIVIRAL ACTIVITY OF D- AND L-2′-AZIDO-2′,3′-DIDEOXY-4′-THIOPYRIMIDINE AND PURINE NUCLEOSIDES	Lak Shin Jeong; Yun Ha Kim; Hea Ok Kim; Su Jeong Yoo; Yong Hee Park; Sook Hee Yeon; Moon Woo Chun; Hee-Doo Kim
669-672	DNA SEQUENCE RECOGNITION BY NFκB p50 HOMODIMER: STRICT AND OBSCURE RECOGNITION SITES IN THE BINDING SEQUENCE	Atsushi Kittaka; Hiroaki Takayama; Masaaki Kurihara; Chikafumi Horii; Hiromichi Tanaka; Tadashi Miyasaka; Jun-ichiro Inoue
673-676	FOUR COLOR FRET DYE NUCLEOTIDE TERMINATORS FOR DNA SEQUENCING	T. Sudhakar Rao; Satyam Nampalli; Kate Lavrenov; Weihong Zhang; Haiguang Xiao; John Nelson; Shiv Kumar
677-679	DESIGN AND SYNTHESIS OF NOVEL FLUOROCYCLOPROPANOID NUCLEOSIDES	Young Rang Lee; Ju-Hyun Park; Raok Jeon; Lak Shin Jeong; Moon Woo Chun; Hee-Doo Kim
681-684	NOVEL NUCLEOSIDES WITH VINYL FLUORIDE OR VINYL BROMIDE MOIETY AS OPEN-CHAIN ANALOGS OF NEPLANOCIN A	Myung-Hee Choi; Chong-Kyo Lee; Lak Shin Jeong; Moon Woo Chun; Hee-Doo Kim
685-688	MECHANISM OF INACTIVATION OF S-ADENOSYL-L-HOMOCYSTEINE HYDROLASE BY 5′-DEOXY-5′-S-ALLENYLTHIOADENOSINE AND 5′-DEOXY-5′-S-PROPYNYLTHIOADENOSINE	G. Guillerm; D. Guillerm; C. Witkowski-Vandenplas
689-693	INACTIVATION OF S-ADENOSYL-L-HOMOCYSTEINE HYDROLASE WITH FLUORINATED ANALOGS OF 2′- AND 3′-DEOXY-5′-METHYLTHIOADENOSINE	D. Guillerm; G. Guillerm; C. Witkowski-Vandenplas
695-698	SYNTHESIS AND BIOLOGICAL EVALUATION OF BORONATED NUCLEOSIDES FOR BORON NEUTRON CAPTURE THERAPY (BNCT) OF CANCER	W. Tjarks; J. Wang; S. Chandra; W. Ji; J. Zhuo; A. J. Lunato; C. Boyer; Q. Li; E. V. Usova; S. Eriksson; G. H. Morrison; G. Y. Cosquer
699-702	SYNTHESIS OF NOVEL 3′-DEOXY-3′-C-HYDROXYMETHYL NUCLEOSIDES WITH CONFORMATIONALLY RIGID SUGAR MOIETY AS POTENTIAL ANTIVIRAL AGENTS	Moon Woo Chun; Myung Jung Kim; Un Hee Jo; Joong Hyup Kim; Hee-Doo Kim; Lak Shin Jeong

Volume 20, Issue 4-7 (2001)

703-706	SYNTHESIS OF NOVEL D- AND L-3′-DEOXY-3′-C-HYDROXYMETHYL NUCLEOSIDE WITH EXOCYCLIC METHYLENE AS POTENTIAL RIBONUCLEOTIDE REDUCTASE INHIBITOR	Moon Woo Chun; Myung Jung Kim; Un Hee Jo; Joong Hyup Kim; Hee-Doo Kim; Lak Shin Jeong
707-710	“SECOND GENERATION” OF TSAO COMPOUNDS DIRECTED AGAINST HIV-1 TSAO-RESISTANT STRAINS	E. Lobatón; S. Velázquez; M. J. Pérez-Pérez; M. L. Jimeno; A. San-Félix; E. De Clercq; J. Balzarini; M. J. Camarasa
711-714	4″-H-TSAO-T, A NOVEL PROTOTYPE IN THE HIV-1 SPECIFIC TSAO FAMILY	E. Lobatón; S. Velázquez; A. San-Félix; E. De Clercq; J. Balzarini; M. J. Camarasa
715-718	A NEW CLASS OF ANTI-HIV-1 OLIGONUCLEOTIDE TARGETED TO THE POLYPURINE TRACT OF VIRAL RNA	Takashi Hiratou; Naoko Miyano-Kurosaki; Hiroshi Gushima; Hiroshi Takaku
719-722	EFFECTIVE SUPPRESSION OF HIV-1 GENE EXPRESSION BY A MAMMALIAN tRNA 3′ PROCESSING ENDORIBONUCLEASE AND EXTERNAL GUIDE SEQUENCE OLIGOZYMES	Michiko Kitano; Jaco S. Barnor; Naoko Miyano-Kurosaki; Yumihiko Endo; Masakazu Yukita; Hiroaki Takeuchi; Yutaka Tamura; Kazuyuki Takai; Masayuki Nashimoto; Hiroshi Takaku
723-726	INHIBITION OF HIV-1 REPLICATION BY THE CRE-LOXP HAMMERHEAD RIBOZYME	Yuichiro Habu; Naoko Miyano-Kurosaki; Hiroaki Takeuchi; Norihiko Matsumoto; Yutaka Tamura; Hiroshi Takaku
727-730	(D)- AND (L)-CYCLOHEXENYL-G, A NEW CLASS OF ANTIVIRAL AGENTS: SYNTHESIS, CONFORMATIONAL ANALYSIS, MOLECULAR MODELING, AND BIOLOGICAL ACTIVITY	J. Wang; M. Froeyen; C. Hendrix; C. Andrei; R. Snoeck; E. Lescrinier; E. De Clercq; P. Herdewijn
731-733	SYNTHESIS AND BIOLOGICAL EVALUATION OF PYRIDIN-2-ONE NUCLEOSIDES	Caroline M. Huntley; Ann S. Cotterill; Jean-Yves Maillard; Jan Balzarini; Claire Simons
735-738	ISONUCLEOSIDES INCORPORATING UNIVERSAL BASES	Vasu Nair; David S. Sosnouski; Qingming Zhu
739-742	A NEW PROCEDURE FOR THE PHOSPHORYLATION OF NUCLEOSIDES: APPLICATION TO THE DISCOVERY OF INHIBITORS OF HIV INTEGRASE	Vasu Nair; Michael Taktakishvili
743-746	SYNTHESIS AND BIOLOGICAL ACTIVITY OF 4′-THIO-L-XYLOFURANOSYL NUCLEOSIDES	Kamal N. Tiwari; Lea Messini; John A. Montgomery; John A. Secrist III
747-750	SYNTHESIS AND BIOLOGICAL ACTIVITY OF 4′-C-HYDROXYMETHYL-2′-FLUORO-D-ARABINOFURANOSYLPURINE NUCLEOSIDES	A. T. Shortnacy-Fowler; K. N. Tiwari; J. A. Montgomery; J. A. Secrist III
751-754	SYNTHESIS AND STUDY OF A NEW SERIES OF PHOSPHORAMIDATE DERIVATIVES AS MONONUCLEOTIDE PRODRUGS	David Egron; Christian Périgaud; Gilles Gosselin; Anne-Marie Aubertin; Jean-Louis Imbach
755-758	SYNTHESIS AND ANTIVIRAL EVALUATION OF 3′-C-TRIFLUOROMETHYL NUCLEOSIDE DERIVATIVES BEARING ADENINE AS THE BASE	Frédéric Jeannot; Christophe Mathé; Gilles Gosselin
759-762	SYNTHESIS OF 5-CHLORO-1-(2,3-DIDEOXY-3-FLUORO-β-D-GLYCERO-HEX-2-ENOPYRANOSE-4-ULOSYL)URACIL AS POTENTIAL ANTICANCER/ANTIVIRAL AGENT	Abdul R. Khan; Kimberly X. Mulligan; Abraham P. Ollapally
763-766	BICYCLIC NUCLEOSIDE INHIBITORS OF VARICELLA-ZOSTER VIRUS (VZV): EFFECT OF TERMINAL UNSATURATION IN THE SIDE-CHAIN	Sheila Srinivasan; Christopher McGuigan; Graciela Andrei; Robert Snoeck; Erik De Clercq; Jan Balzarini
767-769	ANTI-HIV ACTIVITY OF NOVEL PHOSPHONATE DERIVATIVES OF AZT, d4T, AND ddA	A. G. Pokrovsky; T. R. Pronayeva; N. V. Fedyuk; E. A. Shirokova; A. L. Khandazhinskaya; N. B. Tarusova; I. L. Karpenko; A. A. Krayevsky
771-774	COUPLING OF 2,6-DISUBSTITUTED PURINES TO RIBOSE-MODIFIED SUGARS	S. Vittori; S. Costanzi; C. Lambertucci; R. Volpini; G. Cristalli
775-779	SYNTHETIC PROCEDURE FOR THE PREPARATION OF NOVEL POTENT AND SELECTIVE A₃ ADENOSINE RECEPTOR RADIOLIGANDS	R. Volpini; S. Costanzi; C. Lambertucci; S. Vittori; G. Cristalli
781-784	INCREASED RNA AFFINITY OF HNA ANALOGUES BY INTRODUCING ALKOXY SUBSTITUENTS AT THE C-1 OR C-3 POSITION	A. Van Aerschot; M. Meldgaard; F. Volders; G. Schepers; J. Rozenski; P. Herdewijn
785-788	CYCLOHEXENE NUCLEIC ACIDS (CeNA) FORM STABLE DUPLEXES WITH RNA AND INDUCE RNASE H ACTIVITY	J. Wang; B. Verbeure; I. Luyten; M. Froeyen; C. Hendrix; H. Rosemeyer; F. Seela; A. Van Aerschot; P. Herdewijn
789-795	SYNTHESIS OF OLIGONUCLEOSIDE BORANOPHOSPHATES VIA AN H-PHOSPHONATE METHOD WITHOUT NUCLEOBASE PROTECTION	Dmitri S. Sergueev; Zinaida A. Sergueeva; Barbara Ramsay Shaw
797-799	α-OLIGONUCLEOTIDES WITH ANIONIC PHOSPHODIESTER AND CATIONIC PHOSPHORAMIDATE LINKAGES ENHANCED STABILITY OF DNA TRIPLE HELIX	F. Ehrenmann; J. -J. Vasseur; F. Debart

Volume 20, Issue 4-7 (2001)

801-804	A NEW “NATIVE LIGATION” PROCEDURE FOR PEPTIDE-OLIGONUCLEOTIDE CONJUGATION	Dmitry A. Stetsenko; Michael J. Gait
805-808	POLYIMIDAZOLE CONJUGATED OLIGONUCLEOTIDES REACH THE NUCLEUS OF HELA CELLS	François Morvan; C. Castex; E. Vivès; Jean-Louis Imbach
809-813	RECOGNITION OF DNA BY STRAND INVASION WITH OLIGONUCLEOTIDE-SPERMINE CONJUGATES	Pierre F. Potier; Jean-Paul Behr
815-818	STACKING AND STABILITY OF RNA DUPLEXES CONTAINING FLUOROBENZENE AND FLUOROBENZIMIDAZOLE NUCLEOSIDES	Jörg Parsch; Joachim W. Engels
819-823	OLIGONUCLEOTIDES WITH ISOPOLAR PHOSPHONATE INTERNUCLEOTIDE LINKAGE: A NEW PERSPECTIVE FOR ANTISENSE COMPOUNDS?	D. Rejman; J. Snášel; R. Liboska; Z. Točík; O. Pačes; Š. Králíková; M. Rinnová; P. Koiš; I. Rosenberg
825-828	SYNTHESIS AND EVALUATION OF α-LNA	Nanna K. Christensen; Jakob K. Dalskov; Paul Nielsen
829-832	ANTISENSE PROPERTIES OF 2′-O-DIMETHYLAMINOOXYETHYL (2′-O-DMAOE) OLIGONUCLEOTIDES	Thazha P. Prakash; Andrew M. Kawasaki; Joseph F. Johnston; Mark J. Graham; Thomas P. Condon; Muthiah Manoharan
833-835	RAPID RNA CLEAVAGE USING AN ANTISENSE SYSTEM WITH TWO TERPYRIDINE · Cu(II) COMPLEXES	Hideo Inoue; Takako Furukawa; Takashi Tamura; Akihiro Kamada; Eiko Ohtsuka
837-840	UNNATURAL ENANTIOMERS OF 5-AZACYTIDINE ANALOGUES: SYNTHESES AND ENZYMATIC PROPERTIES	G. Gaubert; G. Gosselin; S. Eriksson; A. Vita; G. Maury
841-846	A CODE RELATING SEQUENCE TO STRUCTURE IN NUCLEIC ACIDS	Mieczysław Remin
847-850	INTERACTION OF LNA OLIGONUCLEOTIDES WITH MDR1 PROMOTER	E. L. Chernolovskaya; A. A. Koshkin; V. V. Vlassov
851-854	Cu²-DEPENDENT DNA-CLEAVING ACTIVITY OF ARENES	O. A. Koval; E. L. Chernolovskaya; V. V. Litvak; V. V. Vlassov
855-858	SIMULTANEOUS HPLC ANALYSIS OF HYDROPHOBIC PRODRUGS AND THEIR HYDROPHILIC METABOLITES IN BIOLOGICAL MEDIA WITHOUT SAMPLE PREPARATION. APPLICATION TO THE BIOTRANSFORMATION STUDIES OF PRONUCLEOTIDES DERIVED FROM 5-FLUOROURACIL	G. Coussot; I. Lefebvre-Tournier; L. Hollecker; G. Gosselin; J. -L. Imbach; A. Pompon
859-862	INTERACTION OF OLIGONUCLEOTIDES WITH CELLULAR PROTEINS	P. Laktionov; B. Chelobanov; E. Rykova; V. Vlassov
863-867	GLYCERALDEHYDE-3-PHOSPHATE DEHYDROGENASE IS RESPONSIBLE FOR INTRANUCLEAR LOCALIZATION OF SOME OLIGONUCLEOTIDES	V. Tomasi; P. P. Laktionov; A. V. Bryksin; N. V. Volod'ko; C. Griffoni; E. Y. Rykova; E. Spisni; R. Kraft; V. V. Vlassov
869-871	5-PROPYNYLPYRIMIDINE NUCLEOSIDE DERIVATIVES: RATIONALLY DESIGNED MECHANISM-BASED INACTIVATORS OF THYMIDYLATE SYNTHASE	Thomas I. Kalman; Zhe Nie; Ashwini Kamat
873-877	INHIBITION OF IN VITRO PRE-mRNA SPLICING IN S. CEREVISIAE BY BRANCHED OLIGONUCLEOTIDES	S. Carriero; R. S. Braich; R. H. E. Hudson; D. Anglin; J. D. Friesen; M. J. Damha
879-882	SYNTHESIS OF 3′-THIOAMIDO-MODIFIED 3′-DEOXYTHYMIDINE-5′-TRIPHOSPHATES AND THEIR USE AS CHAIN TERMINATORS IN SANGER-DNA SEQUENCING	K. Schwarzer; C. Wojczewski; J. W. Engels
883-887	NOVEL PROPARGYLAMINE-LINKED NUCLEOSIDES FOR HIGH THROUGHPUT SNP GENOTYPING BY MALDI-TOF MS	Thomas Wenzel; Thomas Fröhlich; Kathrin Strassburger; Susann Richter; Jacqueline Bimmler; Constance Franke; Isabell Thomas; Markus Kostrzewa
889-891	LIPOPLEX-MEDIATED STABLE GENE TRANSFER INTO HeLa CELLS	Moganavelli Singh; Sharda Balram; Mario Ariatti
893-894	ROLLING CIRCLE AMPLIFICATION FOR SCORING SINGLE NUCLEOTIDE POLYMORPHISMS	A. Rösler; L. Bailey; S. Jones; J. Briggs; S. Cuss; I. Horsey; M. Kenrick; S. Kingsmore; L. Kent; J. Pickering; T. Knott; E. Shipstone; G. Scozzafava
895-899	THE USE OF (OLIGONUCLEOTIDE-MALEIC ANHYDRIDE COPOLYMER) CONJUGATES IN NUCLEIC ACID DIAGNOSTIC ASSAYS: EFFECT OF THE NUMBER OF OLIGONUCLEOTIDES PER POLYMER ON TEST SENSITIVITY IMPROVEMENT	C. Minard-Basquin; C. Chaix; C. Pichot

Volume 20, Issue 4-7 (2001)

901-902	SECO C-NUCLEOSIDE ANALOGS OF THE 1,2,4-TRIAZOLE	El Sayed H. El Ashry; Laila F. Awad
903-907	2′-O-MODIFIED OLIGORIBONUCLEOTIDES WITH TERMINAL 3′-3′-INTERNUCLEOTIDE LINKAGE AND THEIR DERIVATIVES	D. Novopashina; M. Kuznetsova; A. Venyaminova
909-914	DESIGN AND SIMPLE ROUTES OF SYNTHESIS OF OLIGONUCLEOTIDE CONJUGATES FOR STUDIES OF DNA TRIPLE HELIX FORMATION	G. N. Grimm; A. S. Boutorine; P. Lincoln; C. Hélène
915-919	SITE-DIRECTED ALKYLATION TO CYTIDINE WITHIN DUPLEX BY THE OLIGONUCLEOTIDES CONTAINING FUNCTIONAL NUCLEOBASES	Fumi Nagatsugi; Takeshi Kawasaki; Natsuko Tokuda; Minoru Maeda; Shigeki Sasaki
921-925	SYNTHESIS OF SOME 2′- AND 3′-FLUOROALKYL SUBSTITUTED NUCLEOSIDES AND OLIGONUCLEOTIDES	Pawel J. Serafinowski; Catherine A. Brown; Colin L. Barnes
927-929	SYNTHESIS AND PHOTOCHEMICAL BEHAVIOUR OF A T-T DIMER CONTAINING AN AMIDE LINKAGE	Martial Thomas; Pascale Clivio; Dominique Guillaume; Jean-Louis Fourrey
931-934	BENZYL-FUNCTIONALIZED cycloSal-d4T MONOPHOSPHATES	J. Renze; M. Plath; C. Ducho; J. Balzarini; E. De Clercq; C. Meier
935-936	SYNTHESIS OF N²-ALKYLGUANOSINE USING MITSUNOBU REACTION AS A KEY STEP	Tokumi Maruyama; Aya Yorikane; Shigetada Kozai
937-940	EFFICIENT SYNTHESIS OF D-[1′-¹³C]-RIBONUCLEOSIDES FOR INCORPORATION INTO OLIGO-RNA	Y. Saito; A. Nyilas; L. A. Agrofoglio
941-945	BORANE-AMINE COMPLEXES - VERSATILE REAGENTS IN THE CHEMISTRY OF NUCLEIC ACIDS AND THEIR ANALOGS	Zinaida A. Sergueeva; Dmitri S. Sergueev; Barbara Ramsay Shaw
947-950	PRO-OLIGONUCLEOTIDE SYNTHESIS USING ALLYL AND ALLYLOXYCARBONYL PROTECTIONS: DIRECT MALDI-TOF MS ANALYSIS ON SOLID SUPPORT	N. Spinelli; J. -J. Vasseur; Y. Hayakawa; J. -L. Imbach
951-954	STEP-BY-STEP CONTROL BY MALDI-TOF MS OF AN OLIGONUCLEOTIDE SYNTHESIS ON STANDARD CPG SOLID-SUPPORT	A. Meyer; F. Debart; J. -L. Imbach; J. -J. Vasseur
955-958	SYNTHESIS OF SOME ACYCLONUCLEOSIDES α-(PYRAZOLO[3,4-d]PYRIMIDIN-4-YLTHIO)-ALKYLAMIDES	M. L. Taha; O. Moukha-Chafiq; H. B. Lazrek; J. J. Vasseur; J. L. Imbach
959-962	SYNTHESIS OF NEW HOMO AND HETERODINUCLEOSIDES CONTAINING THE 2′,3′-DIDEOXYNUCLEOSIDES AZT AND D4T	M. Taourirte; H. B. Lazrek; J. J. Vasseur; M. Ferrero; S. Fernandez; V. Gotor
963-966	DIRECT MALDI-TOF MS ANALYSIS OF OLIGONUCLEOTIDES ON SOLID SUPPORT THROUGH A PHOTOLABILE LINKER	A. Meyer; N. Spinelli; J. -C. Brès; C. Dell'Aquila; F. Morvan; I. Lefebvre; B. Rayner; J. -L. Imbach; J. -J. Vasseur
967-971	5-(PHENYLTHIOMETHYL)-2′-DEOXYURIDINE AS AN EFFICIENT PHOTOREACTIVE PRECURSOR TO GENERATE SINGLE AND MULTIPLE LESIONS WITHIN DNA FRAGMENTS	Sophie Bellon; Didier Gasparutto; Anthony Romieu; Jean Cadet
973-976	THE MOX/SUC PRECURSOR STRATEGIES: ROBUST WAYS TO CONSTRUCT FUNCTIONALIZED OLIGONUCLEOTIDES	N. Polushin
977-979	RECOMBINANT BACTERIAL CELLS AS EFFICIENT BIOCATALYSTS FOR THE PRODUCTION OF NUCLEOSIDES	E. Spoldi; D. Ghisotti; S. Calì; M. Grisa; G. Orsini; G. Tonon; G. Zuffi
981-983	METHYL 5-O-BENZOYL-2,3-OXAZOLE-D-RIBOFURANOSIDE: A USEFUL INTERMEDIATE FOR THE SYNTHESIS OF CONFORMATIONALLY RESTRAINED NUCLEOSIDES	José Molina; Hannah L. Maslen; Claire Simons
985-989	MULTIPLE OLIGONUCLEOTIDE SYNTHESIS IN TANDEM ON SOLID-PHASE SUPPORTS FOR SMALL AND LARGE SCALE SYNTHESIS	R. T. Pon; S. Yu; Y. S. Sanghvi
991-994	STUDIES OF A CHEMICALLY MODIFIED OLIGODEOXYNUCLEOTIDE CONTAINING A 5-ATOM AMIDE BACKBONE WHICH EXHIBITS IMPROVED BINDING TO RNA	Christopher J. Wilds; George Minasov; François Natt; Peter von Matt; Karl-Heinz Altmann; Martin Egli
995-997	CHIMERIC RNA WITH MODIFIED BACKBONES: ALTERNATING METHYLENE(METHYLIMINO) LINKED PHOSPHODIESTER BACKBONE OLIGONUCLEOTIDES WITH 2′-OH AND 2′-OMe GROUPS	Marija Prhavc; Balkrishen Bhat; George Just; P. Dan Cook; Muthiah Manoharan
999-1002	SYNTHESIS AND STRUCTURAL STUDY OF PYRIMIDYL CARBOCYCLIC ANALOGUES OF NUCLEOSIDES BASED ON CYCLOPENTENE RINGS	C. Terán; M. J. González Moa; R. Mosquera; L. Santana

Volume 20, Issue 4-7 (2001)

1003-1006	SYNTHESIS OF 6-FORMYLURIDINE 5′-MONOPHOSPHATE: 6-FORMYL-UMP	Michael P. Groziak
1007-1010	EFFICIENT SYNTHESIS OF OLIGONUCLEOTIDE-PEPTIDE CONJUGATES ON LARGE SCALE	Svetlana O. Doronina; Andrei P. Guzaev; Muthiah Manoharan
1011-1014	A NOVEL PROTECTING STRATEGY FOR INTERNUCLEOSIDIC PHOSPHATE AND PHOSPHOROTHIOATE GROUPS	Andrei P. Guzaev; Muthiah Manoharan
1015-1018	SYNTHESIS OF CHIMERIC OLIGONUCLEOTIDES CONTAINING INTERNUCLEOSIDIC PHOSPHODIESTER AND S–PIVALOYLTHIOETHYL PHOSPHOTRIESTER RESIDUES	Andrei P. Guzaev; Balkrishen Bhat; Guity Balow; Muthiah Manoharan
1019-1023	SYNTHESIS AND PROPERTIES OF NOVEL TRIPHOSPHATE ANALOGUES: RIBONUCLEOSIDE AND DEOXYRIBONUCLEOSIDE (α-P-BORANO, α-P-THIO)TRIPHOSPHATES	Jinlai Lin; Kenneth W. Porter; Barbara Ramsay Shaw
1025-1028	ANTIVIRAL ACTIVITY OF TENOFOVIR (PMPA) AGAINST NUCLEOSIDE-RESISTANT CLINICAL HIV SAMPLES	Michael D. Miller; Nicolas A. Margot; Kurt Hertogs; Brendan Larder; Veronica Miller
1029-1032	SYNTHESIS AND ANTIVIRAL EVALUATION OF C-4-HYDRAZIDE DERIVATIVES OF 2′,3′-DIDEOXYCYTIDINE	Valérie Boudou-Vivet; Christophe Mathé; Gilles Gosselin
1033-1036	MODIFIED DINUCLEOSIDE TETRAPHOSPHONATES, NEW POTENTIAL INHIBITORS OF HIV REVERSE TRANSCRIPTASE	E. A. Shirokova; A. L. Khandazhinskaya; Yu. S. Skoblov; L. Ye. Goryunova; R. S. Beabealashvilli; A. A. Krayevsky
1037-1041	3′-DEOXYRIBOFURANOSE DERIVATIVES OF 1-DEAZA AND 3-DEAZA-ADENOSINE AND THEIR ACTIVITY AS ADENOSINE DEAMINASE INHIBITORS	S. Costanzi; C. Lambertucci; R. Volpini; S. Vittori; G. Lupidi; G. Cristalli
1043-1045	POTENT IN VITRO ANTICANCER ACTIVITIES OF RING-EXPANDED (“FAT”) NUCLEOSIDES CONTAINING THE IMIDAZO[4,5-E][1,3]DIAZEPINE RING SYSTEM	Juliana K. Gill; Lijuan Wang; Maria Bretner; Rachel Newman; Natasha Kyprianou; Ramachandra S. Hosmane
1047-1048	N-PHENYLIMIDAZOLIUM TRIFLATE AS A HIGHLY EFFECTIVE PROMOTER FOR THE INTERRIBONUCLEOTIDE-BOND FORMATION VIA THE PHOSPHORAMIDITE METHOD	Rie Kawai; Jun-ichiro Sugimoto; Masanori Kataoka; Yoshihiro Hayakawa
1049-1051	SYNTHESIS AND STUDY OF THE FLUORESCEIN CONJUGATE OF THE NUCLEOTIDE dPTP	W. J. Cummins; A. L. Hamilton; C. L. Smith; M. S. J. Briggs
1053-1057	SYNTHESIS AND IN VITRO ANTIVIRAL ACTIVITY EVALUATION OF 9-(2-AZIDO-2,3-DIDEOXY-β-D-THREO-PENTOFURANOSYL)ADENINE DERIVATIVES	Satoshi Takamatsu; Kunisuke Izawa; Tokumi Maruyama; Satoshi Katayama; Naoko Hirose; Erik De Clercq
1059-1062	SYNTHESIS AND ANTIVIRAL ACTIVITY OF NOVEL EXOMETHYLENE CYCLOPROPYL NUCLEOSIDES	Bo Gil Choi; Eun Yee Kwak; Joon Hee Hong; Chong Kyo Lee
1063-1066	BICYCLIC FURO PYRIMIDINE NUCLEOSIDES WITH ARYLOXYPHENYL AND HALOPHENYL SUBSTITUTED SIDE CHAINS AS POTENT AND SELECTIVE VARICELLA-ZOSTER VIRUS INHIBITORS	Sally Blewett; Christopher McGuigan; Hubert Barucki; Graciela Andrei; Robert Snoeck; Erik De Clercq; Jan Balzarini
1067-1078	THE DESIGN AND SYNTHESIS OF PURINE INHIBITORS OF CDK2. III	P. W. Shum; N. P. Peet; P. M. Weintraub; T. B. Le; Z. Zhao; F. Barbone; B. Cashman; J. Tsay; S. Dwyer; P. C. Loos; E. A. Powers; K. Kropp; P. S. Wright; A. Bitonti; J. Dumont; D. R. Borcherding
1079-1083	CHEMICAL CROSS-LINKING OF PEPTIDES DERIVED FROM RECA WITH SINGLE-STRANDED OLIGONUCLEOTIDES CONTAINING 5-FORMYL-2′-DEOXYURIDINE	Toru Sugiyama; Atsushi Kittaka; Hiroaki Takayama; Mitsugu Tomioka; Yoshiteru Ida; Reiko Kuroda
1085-1090	PURIFICATION OF PMPA AMIDATE PRODRUGS BY SMB CHROMATOGRAPHY AND X-RAY CRYSTALLOGRAPHY OF THE DIASTEREOMERICALLY PURE GS-7340	H. Chapman; M. Kernan; J. Rohloff; M. Sparacino; T. Terhorst
1091-1098	METABOLISM OF GS-7340, A NOVEL PHENYL MONOPHOSPHORAMIDATE INTRACELLULAR PRODRUG OF PMPA, IN BLOOD	Eugene J. Eisenberg; Gong-Xin He; William A. Lee
1099-1102	AN EFFICIENT PROCESS FOR THE SYNTHESIS OF CYCLIC HPMPC	Michael S. Louie; Harlan Chapman

Volume 20, Issue 4-7 (2001)

1103-1106	SYNTHESIS OF 8-AMINO AND 8-SUBSTITUTED AMINO DERIVATIVES OF ACYCLIC PURINE NUCLEOSIDE AND NUCLEOTIDE ANALOGS. ALKYLATION OF 8-SUBSTITUTED PURINE BASES	Z. Janeba; A. Holý
1107-1111	MESSENGER RNA ISOLATION USING NOVEL PNA ANALOGUES	D. Phelan; K. Hondorp; M. Choob; V. Efimov; J. Fernandez
1113-1115	SYNTHESIS OF MODIFIED NUCLEOSIDE 5′-TRIPHOSPHATES FOR IN VITRO SELECTION OF CATALYTIC NUCLEIC ACIDS [1]	Jasenka Matulic-Adamic; Andrew T. Daniher; Alexander Karpeisky; Peter Haeberli; David Sweedler; Leonid Beigelman
1117-1121	LIN-BENZOARISTEROMYCIN	Vasanthakumar P. Rajappan; Stewart W. Schneller
1123-1125	SYNTHESIS AND IN VITRO ACTIVITY OF D- AND L-ENANTIOMERS OF 5-(TRIFLUOROMETHYL)URACIL NUCLEOSIDE DERIVATIVES	Raul Salvetti; Massimo Pregnolato; Annalisa Verri; Federico Focher; Silvio Spadari; Arnaud Marchand; Christophe Mathé; Gilles Gosselin
1127-1128	NEW CARBOCYCLIC NUCLEOSIDES DERIVED FROM INDAN	F. Abad; F. Álvarez; F. Fernández; X. García-Mera; J. E. Rodríguez-Borges
1129-1131	MODIFIED CYCLOBUTANE CARBONUCLEOSIDES: SYNTHESIS AND EVALUATION OF THEIR ANTIVIRAL ACTIVITY	F. Fernández; A. R. Hergueta; C. López; E. De Clercq; J. Balzarini
1133-1135	A CYCLOBUTANE CARBONUCLEOSIDE WITH MARKED SELECTIVITY AGAINST TK AND TK^- VARICELLA ZOSTER VIRUS	C. López; C. Balo; J. M. Blanco; F. Fernández; E. De Clercq; J. Balzarini
1137-1139	SYNTHESIS AND EVALUATION OF ANTIVIRAL ACTIVITY OF HIGHER HOMOLOGUES OF XYLO-CARBOCYCLIC NUCLEOSIDES	O. Caamaño; M. J. Figueira; F. Fernández; M. D. García; M. I. Nieto; E. de Clercq; J. Balzarini
1141-1145	NOVEL NUCLEOSIDE TRIPHOSPHATE ANALOGS FOR THE ENZYMATIC LABELING OF NUCLEIC ACIDS	A. D. Barone; C. Chen; G. H. McGall; K. Rafii; Philip R. Buzby; James J. Dimeo
1147-1152	6-AZACYTIDINE - COMPOUND WITH WIDE SPECTRUM OF ANTIVIRAL ACTIVITY	I. Alexeeva; N. Dyachenko; L. Nosach; V. Zhovnovataya; S. Rybalko; R. Lozitskaya; A. Fedchuk; V. Lozitsky; T. Gridina; A. Shalamay; L. Palchikovskaja; O. Povnitsa
1153-1157	SYNTHESIS AND ADENOSINE RECEPTOR AFFINITY AND POTENCY OF 8-ALKYNYL DERIVATIVES OF ADENOSINE	C. Lambertucci; S. Costanzi; S. Vittori; R. Volpini; G. Cristalli
1159-1163	KINETICS STUDY OF THE BIOTRANSFORMATION OF AN OLIGONUCLEOTIDE PRODRUG IN CELLS EXTRACT BY MATRIX-ASSISTED LASER DESORPTION/IONIZATION TIME-OF-FLIGHT MASS SPECTROMETRY	François Morvan; Jean-Charles Brès; Isabelle Lefebvre; Jean-Jacques Vasseur; Alain Pompon; Jean-Louis Imbach
1165-1168	CELLULAR UPTAKE AND INTRACELLULAR QUANTIFICATION OF FLUORESCENT LABELED T₂₀ ME-SATE PROOLIGONUCLEOTIDES	François Morvan; J. C. Bologna; E. Vivès; Jean-Louis Imbach
1169-1172	KINETICALLY SELECTIVE BINDING OF SINGLE STRANDED RNA OVER DNA BY A PYRROLIDINE-AMIDE OLIGONUCLEOTIDE MIMIC (POM)	David T. Hickman; Paul M. King; Jonathan M. Slater; Matthew A. Cooper; Jason Micklefield
1173-1176	SYNTHESIS AND BIOPHYSICAL STUDIES OF OLIGONUCLEOTIDES CONTAINING HYDROXAMATE LINKAGES	Kanda S. Ramasamy; Vesna Stoisavljevic; Johnson Y. N. Lau
1177-1179	LABELING DURING CLEAVAGE (LDC), A NEW LABELING APPROACH FOR RNA	V. Monnot; C. Tora; S. Lopez; L. Menou; A. Laayoun
1181-1185	NEW APPROACHES TOWARDS FLUORESCENCE LABELLING OF MESSENGER RNA TRANSCRIPTS	Arlette Garnier; Dieter Hüsken; Jan Weiler
1187-1191	ENGINEERING PREFERENCES OF HAIRPIN PNA BINDING TO COMPLEMENTARY DNA: EFFECT OF N7G IN aeg/aep PNA BACKBONE	V. A. Kumar; M. D'Costa; K. N. Ganesh
1193-1196	SYNTHESIS AND EVALUATION OF PROLYL CARBAMATE NUCLEIC ACIDS (PrCNA)	Meena; V. A. Kumar; K. N. Ganesh
1197-1200	CONSTRAINED FLEXIBILITY IN PNA: DNA BINDING STUDIES WITH BRIDGED AMINOPROPYLGLYCYL PNA	P. S. Lonkar; V. A. Kumar; K. N. Ganesh

Volume 20, Issue 4-7 (2001)

1201-1204	EXTRA STABLE 2′,5′-LINKED RNA LOOPS	Rami N. Hannoush; Masad J. Damha
1205-1209	EFFECT OF SUBSTITUTING ARABINONUCLEOSIDES FOR DEOXYNUCLEOTIDES IN THE DNA PRIMING STRAND ON THE POLYMERASE ACTION OF HIV-1 RT	Anne M. Noronha; Dominique Arion; Michael A. Parniak; Masad J. Damha
1211-1217	MOLECULAR MODELLING OF 2′-OH MEDIATED HYDROGEN BONDING IN RIBONUCLEOS(T)IDES BY NMR CONSTRAINED AM1 AND MMX CALCULATIONS	Parag Acharya; Irina Velikian; Sandipta Acharya; Jyoti Chattopadhyaya
1219-1223	DO THE 16 MER, 5′-GUGGUCUGAUGAGGCC-3′ AND THE 25 MER, 5′-GGCCGAAACUCGUAAGAGUCACCAC-3′, FORM A HAMMERHEAD RIBOZYME STRUCTURE IN PHYSIOLOGICAL CONDITIONS? AN NMR AND UV THERMODYNAMIC STUDY	Edouard Zamaratski; Anna Trifonova; Parag Acharya; Johan Isaksson; Tatiana Maltseva; Jyoti Chattopadhayaya
1225-1228	THE NMR CONFORMATION STUDY OF THE COMPLEXES OF DEOXYCYTIDINE KINASE (dCK) AND 2′-DEOXYCYTIDINE/2′-DEOXYADENOSINE	T. Maltseva; E. Usova; S. Eriksson; J. Milecki; A. Földesi; J. Chattopadhayaya
1229-1233	AN ENERGETIC CORRELATION OF AB INITIO AND NMR STUDIES OF THE 3′-GAUCHE EFFECT IN 3′-SUBSTITUTED THYMIDINES	Parag Acharya; Christophe Thibaudeau; Jyoti Chattopadhyaya
1235-1238	PROMOTION OF TRIPLEX FORMATION BY 2′-O,4′-C-METHYLENE BRIDGED NUCLEIC ACID (2′,4′-BNA) MODIFICATION: THERMODYNAMIC AND KINETIC STUDIES	Hidetaka Torigoe; Satoshi Obika; Takeshi Imanishi
1239-1241	A DNA-BINDING PEPTIDE FROM A PHAGE DISPLAY LIBRARY	Julian Wölcke; Elmar Weinhold
1243-1246	INHIBITION OF HUMAN TELOMERASE BY L-ENANTIOMERS OF NATURAL 2′-DEOXYRIBONUCLEOSIDE 5′-TRIPHOSPHATES	Toyofumi Yamaguchi; Rieko Yamada; Aki Tomikawa; Koichi Shudo; Motoki Saito; Fuyuki Ishikawa; Mineo Saneyoshi
1247-1250	MECHANISTIC STUDIES TO UNDERSTAND THE INHIBITION OF WILD TYPE AND MUTANT HIV-1 REVERSE TRANSCRIPTASE BY CARBOVIR-TRIPHOSPHATE	Adrian S. Ray; Karen S. Anderson
1251-1254	ACCELERATION OF NUCLEIC ACID HYBRIDIZATION ON DNA MICROARRAYS DRIVEN BY pH TUNABLE MODIFICATIONS	Peiming Zhang; Natalia Briones; Chang-Gong Liu; Charles K. Brush; Tom Powdrill; Yuri Belosludtsev; Mike Hogan
1255-1258	LABORATORY DIAGNOSIS OF RESPIRATORY DISEASES: PCR VERSUS SEROLOGY	H. Haaheim; L. Vorland; T. J. Gutteberg
1259-1262	PHOTOSENSITIZED AND CATALYTIC OXIDATION OF DNA BY METALLOPHTHALOCYANINE-OLIGONUCLEOTIDE CONJUGATES	V. V. Koval; A. A. Chernonosov; T. V. Abramova; T. M. Ivanova; O. S. Fedorova; V. M. Derkacheva; E. A. Lukyanets
1263-1266	SYNTHESIS OF 2′,3′-DIDEOXY-2′,3′-DIDEHYDRO NUCLEOSIDES VIA A SERENDIPITOUS ROUTE	Z. Guo; Y. S. Sanghvi; L. E. Brammer Jr.; T. Hudlicky
1267-1270	UNEXPECTED RESULTS AND RECOURSE IN PROCESS OPTIMIZATION OF NUCLEOSIDE 3′-O-SUCCINATES	Quanlai Song; Yogesh S. Sanghvi
1271-1274	A NEW FACILE METHOD FOR SPIN-LABELING OF OLIGONUCLEOTIDES	Thorsten Strube; Olav Schiemann; Fraser MacMillan; Thomas Prisner; Joachim W. Engels
1275-1278	PHENYLALKYL BACKBONE MODIFIED OLIGODEOXYNUCLEOTIDES, THEIR SYNTHESIS AND THE INFLUENCE OF THE ALKYL CHAIN LENGTH	Stefan Amberg; Joachim W. Engels
1279-1282	SYNTHESIS AND BASE PAIRING PROPERTIES OF 9-DEAZAPURINE N⁷-NUCLEOSIDES IN OLIGONUCLEOTIDE DUPLEXES AND TRIPLEXES	P. Leonard; T. Wiglenda; F. Seela
1283-1286	PARALLEL DNA CONTAINING PYRAZOLO[3,4-D]PYRIMIDINE ANALOGUES OF ISOGUANINE	F. Seela; R. Kröschel; Y. He
1287-1289	BRIDGED CYCLIC OLIGORIBONUCLEOTIDES—TOWARDS MODELS FOR CODON-ANTICODON PAIRING	R. Micura; W. Pils; K. Grubmayr; M. -O. Ebert; B. Jaun
1291-1293	LARGE-SCALE MANUFACTURING OF ALL FOUR 2′-DEOXYNUCLEOSIDES VIA NOVEL STRATEGIES INCLUDING A CHEMO-ENZYMATIC PROCESS	Hironori Komatsu; Hirokazu Awano; Hiroharu Tanikawa; Kiyoshi Itou; Ichirou Ikeda
1295-1298	KINETIC STUDIES OF THE DEGRADATION OF OXYCARBONYLOXYMETHYL PRODRUG OF ADEFOVIR AND TENOFOVIR IN SOLUTION	Reza Oliyai; Lung-Chi Yuan; Terry Dahl
1299-1302	DEALKYLATION OF PHOSPHONATE ESTERS WITH CHLOROTRIMETHYLSILANE	A. J. Gutierrez; E. J. Prisbe; J. C. Rohloff

Volume 20, Issue 4-7 (2001)

1303-1307	SYNTHESES OF DNA DUPLEXES CONTAINING A C–C INTERSTRAND CROSS-LINK	Anne M. Noronha; David M. Noll; Paul S. Miller
1309-1312	SYNTHESIS AND NMR-ANALYSIS OF TRICYCLIC NUCLEOSIDES	Poul Nielsen; Michael Petersen; Jens Peter Jacobsen
1313-1316	SPECIFIC BINDING AND STABILIZATION OF DNA AND PHOSPHOROTHIOATE DNA BY AMPHIPHILIC α-HELICAL PEPTIDES	Takanori Kubo; Masayuki Fujii
1317-1320	AMPHIPHILIC β-SHEET PEPTIDES CAN BIND TO DOUBLE AND TRIPLE STRANDED DNA	Kinuko Yokoyama; Takanori Kubo; Masayuki Fujii
1321-1324	A NOVEL APPROACH FOR THE SOLID PHASE SYNTHESIS OF DNA-PEPTIDE CONJUGATES	Takanori Kubo; Krishna Dubey; Masayuki Fujii
1325-1328	SYNTHESIS OF A NOVEL NUCLEIC ACID MIMIC: P-BORANOMETHYLPHOSPHONATE	Jinlai Lin; Barbara Ramsay Shaw
1329-1331	A NEW SYNTHETIC METHODOLOGY FOR TIAZOFURIN	Kanda S. Ramasamy; Johnson Y. N. Lau
1333-1337	SYNTHETIC STUDIES TO IMPROVE THE DEUTERIUM LABELLING IN NUCLEOSIDES FOR FACILITATING STRUCTURAL STUDIES OF LARGE RNAS BY HIGH-FIELD NMR SPECTROSCOPY	Mrinal K. Kundu; Anna Trifonova; Zoltán Dinya; András Földesi; Jyoti Chattopadhyaya
1339-1341	THE SYNTHESIS OF, AND STUDIES ON, 2′-C-MODIFIED NUCLEOTIDES	Lavinia Brennan; Kevin J. Fettes; Ian A. O'Neil; Richard Cosstick
1343-1346	DESIGN AND PROPERTIES OF HEPATITIS C VIRUS ANTISENSE OLIGONUCLEOTIDES FOR LIVER SPECIFIC DRUG TARGETING	Thomas J. Lehmann; Matthias Serwe; Wolfgang H. Caselmann; Joachim W. Engels
1347-1350	NOVEL MACROCYCLES DERIVED FROM NUCLEOSIDES	Noelia Calcerrada-Muñoz; Ian O'Neil; Richard Cosstick
1351-1354	SOLID-PHASE SYNTHESIS OF OLIGODEOXYNUCLEOTIDES CONTAINING 3′-S-PHOSPHOROTHIOLATE LINKAGES	Kevin J. Fettes; Ian O'Neil; Stanley M. Roberts; Richard Cosstick
1355-1358	SYNTHESIS AND BIOLOGICAL ACTIVITIES OF CYCLIC ADP-CARBOCYCLIC-RIBOSE AND ITS ANALOGS	Masayoshi Fukuoka; Satoshi Shuto; Noriaki Minakawa; Yoshihito Ueno; Akira Matsuda
1359-1361	RESOLUTION OF RACEMIC MIXTURES OF CARBOCYCLIC ANALOGUES OF NUCLEOSIDES AND ASSIGNMENT OF THEIR ABSOLUTE CONFIGURATION	P. Besada; C. Terán; E. Quezada; J. M. Seco; E. Uriarte
1363-1365	1,2-DISUBSTITUTED CYCLOHEXANE CARBOCYCLIC ANALOGUES OF NUCLEOSIDES	D. Viña; L. Santana; E. Uriarte
1367-1370	ASYMMETRIC SYNTHESIS OF CARBOCYCLIC PYRIMIDINE NUCLEOSIDES VIA π-ALLYLPALLADIUM COMPLEX	Junxing Shi; Raymond F. Schinazi
1371-1375	THE USE AND EVALUATION OF 2 2 PHOTOADDITION IN IMMOBILIZATION OF OLIGONUCLEOTIDES ON A THREE DIMENSIONAL HYDROGEL MATRIX	R. Elghanian; Y. Xu; J. McGowen; M. Seithoff; C. G. Liu; J. Winick; N. Fuller; R. Ramakrishnan; A. Beuhler; T. Johnson; A. Mazumder; C. K. Brush
1377-1379	SYNTHESIS AND HYBRIDIZATION OF NOVEL CHIRAL PYRROLIDINE BASED PNA ANALOGUE	Andis Slaitas; Esther Yeheskiely
1381-1384	EVALUATION OF SEVERAL ECONOMICAL COMPUTATIONAL METHODS FOR GEOMETRY OPTIMISATION OF PHOSPHORUS ACID DERIVATIVES	Susannah Sigurdsson; Roger Strömberg
1385-1388	A METHOD FOR SYNTHESIS OF AN ARTIFICIAL RIBONUCLEASE	Hans Åström; Roger Strömberg
1389-1392	PREPARATION OF 3′-C-BRANCHED URIDINE ANALOGUES, SUITABLE FOR CONVERSION INTO FUNCTIONALISED 3′-C-METHYLENE DERIVATIVES	Anna Winqvist; Roger Strömberg
1393-1397	SYNTHESIS OF NEW CHIRAL PEPTIDE NUCLEIC ACID (PNA) MONOMERS	Bogdan Falkiewicz; Wojciech Wiśniowski; Aleksandra S. Kołodziejczyk; Kazimierz Wiśniewski
1399-1402	RESTRICTED ROTATION IN CHIRAL PEPTIDE NUCLEIC ACID (PNA) MONOMERS - INFLUENCE OF SUBSTITUENTS STUDIED BY MEANS OF ¹H NMR	Marta Oleszczuk; Sylwia Rodziewicz-Motowidło; Bogdan Falkiewicz
1403-1409	PREPARATION OF OLIGODEOXYNUCLEOTIDE 5′-TRIPHOSPHATES USING SOLID SUPPORT APPROACH	A. V. Lebedev; I. I. Koukhareva; T. Beck; M. M. Vaghefi
1411-1414	PHARMACOKINETICS OF SALICYLATE ESTER PRODRUGS OF CYCLIC HPMPC IN DOGS	Reza Oliyai; Murty N. Arimilli; Robert J. Jones; William A. Lee
1415-1419	LC/MS DETERMINATION OF THE INTRACELLULAR CONCENTRATION OF TWO NOVEL ARYL PHOSPHORAMIDATE PRODRUGS OF PMPA AND THEIR METABOLITES IN DOG PBMC	Theresa Lynch; Gene Eisenberg; Michael Kernan
1421-1424	PHOSPHORAMIDITES AND OLIGONUCLEOTIDES CONTAINING 7-DEAZAPURINES AND PYRIMIDINES CARRYING AMINOPROPARGYL SIDE CHAINS	F. Seela; N. Ramzaeva; P. Leonard; Y. Chen; H. Debelak; E. Feiling; R. Kröschel; M. Zulauf; T. Wenzel; T. Fröhlich; M. Kostrzewa
1425-1428	ANTISENSE OLIGONUCLEOTIDE ISIS 2922 TARGETS IE-EXPRESSION AND PREVENTS HCMV-IE-INDUCED SUPPRESSION OF TSP-1 AND TSP-2 EXPRESSION	S. Margraf; M. Bittoova; J-U. Vogel; R. Kotchekov; H. W. Doerr; J. Cinatl Jr.
1429-1432	BASE MUTATION ANALYSIS BY A FERROCENYL NAPHTHALENE DIIMIDE DERIVATIVE	Shigeori Takenaka; Hiroyoshi Miyahara; Kenichi Yamashita; Makoto Takagi; Hiroki Kondo
1433-1437	CYTARABINE TREATMENT OF HUMAN T-LYMPHOID CELLS INDUCES DECREASED HIV-1 RECEPTOR EXPRESSION AND REDUCED HIV-1 SUSCEPTIBILITY	B. Gröschel; A. Kaufmann; J. Cinatl; H. W. Doerr

Volume 20, Issue 3 (2001)

169-183	NMR SOLUTION STRUCTURE AND CONFORMATIONAL ANALYSIS OF THE CALCIUM RELEASE AGENT CYCLIC ADENOSINE 5′-DIPHOSPHATE RIBOSE (cADPR)	Steven M. Graham; Sarah C. Pope
185-196	PHOTOCHEMICAL SYNTHESIS OF NOVEL DIDEOXYNUCLEOSIDES	E. Lee-Ruff; R. Margau
197-211	AN IMPROVED SYNTHESIS OF THE DINUCLEOTIDES pdCpA AND pdCpdA	Xue-Feng Zhu; A. Ian Scott
213-227	A FACILE SYNTHESIS OF 5′-END SOLID-ANCHORED, 3′-END FREE OLIGODEOXYRIBONUCLEOTIDES VIA THE (5′ → 3′)-ELONGATED PHOSPHORAMIDITE STRATEGY	Akira Sakakura; Yoshihiro Hayakawa
243-250	THE PRODUCTION AND EVALUATION OF ANTIBODIES FOR ENZYME IMMUNOASSAY OF AZTTP	Fatima Akeb; Christophe Creminon; Jacques Grassi; Roger Guedj; Danièle Duval
251-260	SYNTHESIS AND PROPERTIES OF OLIGONUCLEOTIDES CONTAINING 8-BROMO-2′-DEOXYGUANOSINE	Carme Fàbrega; Maria J. Macías; Ramon Eritja
261-269	A NEURAL NETWORK TO PREDICT MELTING TEMPERATURE (T_m) OF RNA DUPLEX	Changmei Cheng; Lixin; Hiromi Miyajima; Piet Herdewijn

Volume 20, Issue 1-2 (2001)

1-9	PREPARATION OF OLIGODEOXYNUCLEOTIDES CONTAINING 5-(N-METHYLPIPERAZINYL) AND 5-BENZYLOXYMETHYL URACILS	Ahmed E.-S. Abdel Megied; Omar M. Ali; Thomas Kofoed; Erik B. Pedersen
59-75	EFFICIENT METHODS FOR THE SYNTHESIS OF [2-¹⁵N]GUANOSINE AND 2′-DEOXY[2-¹⁵N]GUANOSINE DERIVATIVES	Kazuo Kamaike; Kazutomo Kinoshita; Katsuyuki Niwa; Kumi Hirose; Kazuhiro Suzuki; Yoshiharu Ishido
77-91	THE CHEMICAL STABILITY OF S-(2-ACYLTHIOETHYL) AND S-ACYLOXYMETHYL PROTECTED THYMIDYLYL-3′,5′-THYMIDINE PHOSPHOROMONOTHIOLATES AND THEIR DEACYLATION PRODUCTS IN AQUEOUS SOLUTION	Päivi Poijärvi; Mikko Oivanen; Harri Lönnberg
93-101	NEW 3′-DEOXYTHYMIDINES BEARING A NUCLEOPHILIC 3′-SUBSTITUENT	Anatoly M. Belostotskii; Helen Keren-Yeshuah; Jael Lexner; Alfred Hassner
103-116	NOVEL SYNTHESIS OF seco TYPE OF ACYCLO C-NUCLEOSIDES OF 1,2,4-TRIAZOLE AND 1,2,4-TRIAZOLO[3,4-b][1,3,4]THIADIAZINE	El Sayed H. El Ashry; Laila F. Awad
117-130	SYNTHESIS AND CHARACTERIZATION OF POLYAMINE-BASED BIOMIMETIC CATALYSTS AS ARTIFICIAL RIBONUCLEASE	Kazuo Shinozuka; Yoshimitu Nakashima; Kazuhiro Shimizu; Hiroaki Sawai
131-143	BINDING OF A PORPHYRIN CONJUGATE OF HOECHST 33258 TO DNA. I. UV-VISIBLE AND MELTING STUDIES DETECT MULTIPLE BINDING MODES TO A 12-MER NONSELF-COMPLEMENTARY DUPLEX	Silvana Frau; Elena V. Bichenkova; Olga S. Fedorova; Serghei Lokhov; Kenneth T. Douglas
145-156	BINDING OF A PORPHYRIN CONJUGATE OF HOECHST 33258 TO DNA. II. NMR SPECTROSCOPIC STUDIES DETECT MULTIPLE BINDING MODES TO A 12-MER NONSELF-COMPLEMENTARY DUPLEX DNA	Silvana Frau; Elena V. Bichenkova; Gareth A. Morris; Kenneth T. Douglas
157-168	BINDING OF A DESMETALLO-PORPHYRIN CONJUGATE OF HOECHST 33258 TO DNA. III. STRONG BINDING TO SINGLE-STRAND OLIGONUCLEOTIDES	Elena V. Bichenkova; Silvana Frau; Olga S. Fedorova; Kenneth T. Douglas

Volume 19, Issue 10-12 (2000)

a-c	Editorial board page for “Nucleosides, Nucleotides & Nucleic Acids”, Volume 19, Number 10-12
xiii-xxv	Biographical Sketch
xxvii-xl	Selected Publications (1961–2000) Alexander Krayevsky
1487-1503	Studies on Reactions of Nucleoside H-Phosphonates with Bifunctional Reagents. Part VI. Reaction with Diols	Michal Sobkowski; Malgorzata Wenska; Adam Kraszewski; Jacek Stawiński
1505-1516	The Mechanism of Dna Repair by Uracil-Dna Glycosylase: Studies Using Nucleotide Analogues	Angelika Rösler; George Panayotou; David P. Hornby; Tom Barlow; Tom Brown; Laurence H. Pearl; Renos Savva; G. Michael Blackburn
1517-1530	Synthesis and Antiviral Evaluation of the β-L-Enantiomers of Some Thymine 3′-Deoxypentofuranonucleoside Derivatives	Christophe Mathé; Gilles Gosselin
1531-1541	Guanosine Analogues as Anti-Herpesvirus Agents	E. De Clercq
1543-1552	Synthesis and Properties of 2′-Deoxycytidine Triphosphate Carrying C-Myc Tag Sequence	Michael Hinz; Dirk Gottschling; Ramon Eritja; Hartmut Seliger
1553-1567	A Remarkable Stabilization of Complexes Formed by 2,6-Diaminopurine Oligonucleotide N3′→P5′ Phosphoramidates	Tracy Matray; Soya Gamsey; Krisztina Pongracz; Sergei Gryaznov
1569-1580	Transglycosylation Reactions of 6-Thioguanine Acyclonucleosides	Andrzej Manikowski; Jerzy Boryski
1581-1598	Fluorescence Properties and Base Pair Stability of Oligonucleotides Containing 8-Aza-7-deaza-2′-deoxyisoinosine or 2′-Deoxyisoinosine	Frank Seela; Georg Becher; Yaoming Chen
1599-1614	Synthesis and Incorporation of Pyrrole Carboxamide Nucleoside Triphosphates by DNA Polymerases	D. Loakes; M. J. Guo; D. M. Brown; S. A. Salisbury; C. L. Smith; I. Felix; S. Kumar; S. Nampalli
1615-1656	The Synthesis of Deuterionucleosides	András Földesi; Anna Trifonova; Mrinal K. Kundu; Jyoti Chattopadhyaya
1657-1673	Nucleophilic N¹ → N³ Rearrangement of 5′-O-Trityl-O²,3′-Cycloanhydrothymidine	Xian-Bin Yang; Konrad Misiura; Wojciech J. Stec; Marek J. Potrzebowski; Sławomir Kaźmierski; Michał Wieczorek; Wiesław R. Majzner; Grzegorz D. Bujacz
1675-1692	Cleavage of the Phosphodiester Bond of Uridylyl-(3′,5′)-8-Carboxymethylaminoadenosine by Hydronium, Hydroxide and Zinc(Ii) Ions: A Model Study Aimed at Elucidating the Potential of a Carboxylate Function as an Intramolecular Catalyst	Satu Mikkola; Mikko Oivanen; Kari Neuvonen; Suvi Piitari; Kaisa Ketomäki; Harri Lönnberg
1693-1707	Synthesis of Modified Nucleotide Building Blocks Containing Electrophilic Groups in the 2′-Position	Anna V. Kachalova; Timofei S. Zatsepin; Elena A. Romanova; Dmitry A. Stetsenko; Michael J. Gait; Tatiana S. Oretskaya
1709-1719	Antisense Phosphorothioate Oligonucleotides Targeted to the Human Chemokine Receptor CXCR4	Akiko Kusunoki; Naoko Miyano-kurosaki; Tohru Kimura; Kazuyuki Takai; Naoki Yamamoto; Hiroshi Gushima; Hiroshi Takaku
1721-1734	Anti-HIV-1 Activity by a Triple-Helix Forming Oligonucleotides Targeted to Polypurine Tract on Viral RNA	Takashi Hiratou; Satoru Tsukahara; Naoko Miyano-kurosaki; Kazuyuki Takai; Takeshi Saito; Naoki Yamamoto; Hiroshi Takaku
1735-1750	Fluorescent α-Anomeric 1,N(6)Etheno- Deoxyadenosine in DNA Duplexes. the α-εdA / dG Pair	L. Bielecki; B. Skalski; I. Zagórowska; R. E. Verrall; R. W. Adamiak

Volume 19, Issue 10-12 (2000)

1751-1764	New Phosphoramidite Reagents for the Synthesis of Oligonucleotides Containing a Cysteine Residue Useful in Peptide Conjugation	Dmitry A. Stetsenko; Michael J. Gait
1765-1777	Nucleotides LXIV[1]: Synthesis, Hybridization and Enzymatic Degradation Studies of 2′-O-Methyl-Oligoribonucleotides and 2′-O-Methyl/Deoxy Gapmers	Hagen Cramer; Wolfgang Pfleiderer
1779-1785	New Efficient Synthesis of Thymidine Cyclic 3′, 5′- Phosphorofluoridate and Its Sulfur Analogue via the Phosphoroamidite Route	Wojciech Dąbkowski; Izabela Tworowska; Jan Michalski; Friedrich Cramer
1787-1793	Synthesis of Non-Nucleoside Triphosphate Analogues, a New Type of Substrates for Terminal Deoxynucleotidyl Transferase	Andrey A. Arzumanov; Lyubov S. Victorova; Maxim V. Jasko
1795-1804	P-(Alkyl)-Nucleoside 5′-Hydrogenphosphonates as Depot Forms of Antiviral Nucleotide Analogues	A. L. Khandazhinskaya; E. A. Shirokova; I. L. Karpenko; N. F. Zakirova; N. B. Tarussova; A. A. Krayevsky
1805-1820	Probing the MvaI Methyltransferase Region that Interacts with DNA: Affinity Labeling with the Dialdehyde-Containing DNA Duplexes	O. M. Gritsenko; S. N. Mikhailov; E. V. Efimtseva; A. Van Aerschot; P. Herdewijn; E. S. Gromova
1821-1830	Synthesis and RNase L Binding and Activation of a 2-5A-(5′)-DNA-(3′)-PNA Chimera, a Novel Potential Antisense Molecule	Jeroen C. Verheijen; Ling Chen; Suzanne F. Bayly; Paul F. Torrence; Gijsbert A. van der Marel; J. H. Van Boom
1831-1846	New Pyrimidine Cyclonucleosides with Hydrogenated Aglycones: Synthesis and X-Ray Structures	Anatoly D. Shutalev; Valeriy E. Zavodnik; Galina V. Gurskaya
1847-1859	Synthesis and Properties of O-β-D-Ribofuranosyl-(1″-2′)-Adenosine-5″-O-Phosphate and Its Derivatives	Andrei A. Rodionov; Ekaterina V. Efimtseva; Sergey N. Mikhailov; Jef Rozenski; Ingrid Luyten; Piet Herdewijn
1861-1884	Oligonucleotides Containing 9-(2-Deoxy-2-Fluoro-β-D-Arabinofuranosyl)-Adenine and -Guanine: Synthesis, Hybridization and Antisense Properties	Tuula Tennilä; Elena Azhayeva; Jouko Vepsäläinen; Reino Laatikainen; Alex Azhayev; Igor A. Mikhailopulo
1885-1909	Pyrophosphoryl Derivatives of 1-(2-Deoxy-3-O-Phosphonomethyl-β-and-α-D-Erythro-Pentofuranosyl)Thymine: Synthesis and Substrate Properties Towards Some DNA Polymerases	Igor A. Mikhailopulo; Tamara I. Kulak; Olga V. Tkachenko; Svetlana L. Sentyureva; Lyubov S. Victorova; Helmut Rosemeyer; Frank Seela
1911-1929	Substituent — Directed Aralkylation and Alkylation Reactions of the Tricyclic Analogues of Acyclovir and Guanosine	Tomasz Ostrowski; Joanna Zeidler; Tomasz Goslinski; Bozenna Golankiewicz
1931-1941	A New Strategy of Discrimination of a Point Mutation by Tandem of Short Oligonucleotides	D. V. Pyshnyi; S. G. Lokhov; M. A. Podyminogin; E. M. Ivanova; V. F. Zarytova
1943-1965	Rapid Routes of Synthesis of Oligonucleotide Conjugates from Non-Protected Oligonucleotides and Ligands Possessing Different Nucleophilic or Electrophilic Functional Groups	Gunther N. Grimm; Alexandre S. Boutorine; Claude Helene
1967-1976	Large-Scale Solid-Phase Preparation of 3′-Unprotected Trinucleotide Phosphotriesters - Precursors for Synthesis of Trinucleotide Phosphoramidites	A. Kayushin; M. Korosteleva; A. Miroshnikov
1977-1991	S,X-Acetals in Nucleoside Chemistry. III¹. Synthesis of 2′-and 3′-O-Azidomethyl Derivatives of Ribonucleosides	S. G. Zavgorodny; A. E. Pechenov; V. I. Shvets; A. I. Miroshnikov
1993-2003	Synthesis Of N-Labeled Peptidyl AMP	Hidehiko Narita; Tomohisa Moriguchi; Kohji Seio; Mitsuo Sekine; Hajime Miyaguchi; Kensaku Sakamoto; Shigeyuki Yokoyama
2005-2017	Synthesis and Structure Activity Relationships of 5-Substituted - 4′-thio-β-D-Arabinofuranosylcytosines	Kamal N. Tiwari; Anita T. Shortnacy-fowler; Loredana Cappellacci; William R. Waud; William B. Parker; John A. Montgomery; John A. Secrist III
2019-2024	Inhibition of Human Immunodeficiency Virus Type-1 (HIV-1) Replication by Immunor (Im²⁸), a New Analog of Dehydroepiandrosterone	Karidia Diallo; Hugues Loemba; Maureen Oliveira; Donatien D. Mavoungoua; Mark A. Wainberg

Volume 19, Issue 9 (2000)

a	Editorial board page for “Nucleosides, Nucleotides & Nucleic Acids”, Volume 19, Number 9
1381-1396	The Synthesis of Novel 6,5- and 6,6-Membered Fused Heterocyclic Compounds Derived from Thymine	Milan Jokić; Zlatica Raza; Darinka Katalenić
1397-1411	Syntheses of 1-[(2-Hydroxyethoxy)methyl]- and 1-[(1,3-Dihydroxy-2-Propoxy)methyl]- Derivatives of 5-Substituted-2,4-difluorobenzene: Unnatural Acyclo Thymidine Mimics for Evaluation as Anticancer and Antiviral Agents	Zhi-Xian Wang; Weili Duan; Leonard I. Wiebe; Erik De Clercq; Jan Balzarini; Edward E. Knaus
1413-1425	Conformationally Locked Nucleosides. Synthesis of Oligodeoxynucleotides Containing 3′-Amino-3′-deoxy-3′-N,5′(R)-C-ethylenethymidine	Guangyi Wang; Vesna Stoisavljevic
1427-1439	Fluorescent Labelling of Oligodeoxyribonucleotides by the Oxyamino-Aldehyde Coupling Reaction	Emmanuelle Trévisiol; Annabelle Renard; Eric Defrancq; Jean Lhomme
1441-1461	Synthesis and Antiviral Activity of C-5 Substituted β-D- and β-L-D4T Analogues	Z. Delbederi; C. Fossey; G. Fontaine; S. Benzaria; D. Gavriliu; A. Ciurea; B. Lelong; D. Ladurée; A. M. Aubertin; A. Kirn
1463-1474	Europium Cryptate Labeled Deoxyuridine-Triphosphate Analog: Synthesis and Enzymatic Incorporation	B. Alpha-bazin; H. Bazin; S. Guillemer; S. Sauvaigo; G. Mathis
1475-1486	2,2′-Anhydro-4′-Thionucleosides: Precursors for 2′-Azido- and 2′-Chloro-4′-thionucleosides and for a Novel Thiolane to Thietane Rearrangement	J. Allen Miller; Ashley W. Pugh; G. Mustafa Ullah

Volume 19, Issue 8 (2000)

a-b	Editorial board page for “Nucleosides, Nucleotides & Nucleic Acids”, Volume 19, Number 8
vii-viii	Preface	Manlio Palumbo
1205-1218	Linkage of a Triple Helix-Forming Oligonucleotide to Amsacrine-4-carboxamide Derivatives Modulates the Sequence-Selectivity of Topoisomerase II-Mediated DNA Cleavage	Paola Arimondo; Christian Bailly; Alexandre Boutorine; Ulysse Asseline; Jian-Sheng Sun; ThÉRÈSe Garestier; Claude Hélène
1219-1229	[2,1-c] [1,4]Benzodiazepine (PBD)-Distamycin Hybrid Inhibits DNA Binding to Transcription Factor Sp1	P. G. Baraldi; B. Cacciarit; A. Guiotto; R. Romagnoli; G. Spalluto; A. Leoni; N. Bianchi; G. Feriotto; C. Rutigliano; C. Mischiati; Roberto Gambari
1231-1240	DNA Accessibility to Minor Groove Ligands in Core Nucleosome and Chromatosome	R. Fodera; R. Caneva; C. Canzonetta; M. Savino
1241-1248	Down-Regulation of H Tau 40 Protein Expression by Minor Groove Binders	Leonhard Kittler; Leo Wollweber
1249-1264	The Interaction of Drugs with DNA Gyrase: A Model for the Molecular Basis of Quinolone Action	Jonathan G. Heddle; Faye M. Barnard; Lois M. Wentzell; Anthony Maxwell
1265-1271	DNA Phosphodiester Bond Hydrolysis Mediated by Cu(II) and Zn(II) Complexes of 1,3,5,-Triamino-cyclohexane Derivatives	Claudia Sissi; Fabrizio Mancin; Manlio Palumbo; Paolo Scrimin; Paolo Tecilla; Umberto Tonellato
1273-1279	BCL-2 Regulation Targeting the AU-Rich Domain	Annamaria Bevilacqua; Maria Cristina Ceriani; Nicola Schiavone; Angelo Nicolin
1281-1288	PAcM-AN: Poly(N-Acryloylmorpholine)-Conjugated Antisense Oligonucleotides	G. M. Bonora; A. M. De Franco; R. Rossin; P. M. Veronese; P. Ferrutic; O. Plyasunova; P. E. Vorobjev; D. V. Pyshnyi; N. I. Komarova; V. F. Zarytova
1289-1299	Glycosylations of Inosine and Uridine Nucleoside Bases and Synthesis of the New 1-(β-D-Glucopyranosyl)-Inosine-5′, 6″-diphosphate	Antonia De Capua; Lorenzo De Napoli; Giovanni Di Fabio; Anna Messere; Daniela Montesarchio; Gennaro Piccialli
1301-1310	Oligonucleotide Labeling: Synthesis of a New Spin-Labeled 2′-Deoxyguanosine Analogue	Cesare Giordano; Francesco Pedone; Paola Fattibene; Luciano Cellai
1311-1326	Molecular Structure and Cytotoxicity of 3D-Transition Metal Complexes Capable to Form a Stable Metal-Nitrogen Bond	A. Marzotto; D. A. Clemente; A. Zampiron; M. Carrara
1327-1336	6-Hydroxy Derivative as New Desfluoroquinolone (DFQ): Synthesis and DNA-Binding Study	Oriana Tabarrini; Claudia Sissi; Arnaldo Fravolini; Manlio Palumbo
1337-1353	DNA Recognition by Quinoline Antibiotics: Use of Base-Modified DNA Molecules to Investigate Determinants of Sequence-Specific Binding of Luzopeptin	Christian Bailly; Stephen Crow; Andrew Minnock; Michael J. Waring
1355-1364	Double-Stranded Nucleic Acids in Liquid-Crystalline Dispersions as Building Blocks for Cross-Linked Supramolecular Structures	Yu. M. Yevdokimov; V. I. Salyanov; B. V. Mchedlischvili; V. A. Bykov; A. V. Belyaev; S. A. Saunin; F. Spener; M. Palumbo
1365-1379	Shape-Selective Binding of Geometrically-Constrained bis-Distamycins to a DNA Duplex and a Model Okazaki Fragment of Identical Sequence	William H. Gmeiner; Wei Cui; Sanjay Sharma; Ana Maria Soto; Luis A. Marky; J. William Lown

Volume 19, Issue 7 (2000)

a	Editorial board page for “Nucleosides, Nucleotides & Nucleic Acids”, Volume 19, Number 7
1057-1091	Synthesis and anti-HIV evaluation of new 2′,3′- dideoxy-3′-thiacytidine prodrugs	Nicolas Mourier; Michel Camplo; Giovanna Schioppacassi Della Bruna; Francesco Pellacini; Domenico Ungheri; Jean-Claude Chermann; Jean-Louis Kraus
1093-1100	Facile Synthesis of N-(1-Alkenyl) Derivatives of 2,4-Pyrimidinediones	Ulla Henriksen
1101-1109	Ribonuclease T1 Cleaves RNA After Guanosines Within Single-Stranded Gaps of Any Length	Thomas Greiner-Stöffele; Hans-Heinrich Foerster; Ulrich Hahn
1111-1122	A Facile Synthesis of cis-9-[4-(1,2-Dihydroxyethyl)-cyclopent-2-enyl]guanine and Its Derivative	Gwang-Il An; Hakjune Rhee
1123-1134	Convenient Syntheses of 6-Methylpurine and Related Nucleosides	Abdalla E. A. Hassan; Reham A. I. Abou-elkair; John A. Montgomery; John A. Secrist III
1135-1143	A One-Pot Preparation of 1-Benzyl-2′-deoxyinosine from ionized 2′-Deoxyinosine	Ki-Young Moon; Yeong Shik Kim
1145-1158	Invasion of Strongly Binding Oligonucleotides into tRNA Structure	V. Petyuk; R. Serikov; V. Tolstikov; V. Potapov; R. Giege; M. Zenkova; V. Vlassov
1159-1183	Efficient Synthesis of 2′-Deoxynucleoside 3′-C-Phosphonates: Reactivity of Geminal Hydroxyphosphonate Moiety	Śárka Králíková; Miloś Buděšínský; Milena Masojídková; Ivan Rosenberg
1185-1191	Self-Assembly and Lyomesophases Formed by Long-Chain Alkoxymethyl-Nucleobase Derivatives	W. V. Meister; S. Lindau; C. Bohley; U. Gromann; M. Madre; L. Kovalenko; G. Bischoff; R. Zhuk; S. Hoffmann
1193-1203	Method for the Synthesis of Uric Acid Derivatives	Tokumi Maruyama; Shigetada Kozai; Fumi Sasaki

Volume 19, Issue 5-6 (2000)

a-b	Editorial board page for “Nucleosides, Nucleotides & Nucleic Acids”, Volume 19, Number 5-6
845-849	Synthesis and Antiviral Activity of 3-(β-D-Ribofuranosyl)-1,2,4-oxadiazole-5-carboxamide	Ram Pratap; V. N. Yarovenko
851-866	Synthesis of N,N-Dialkylaniline-2′-deoxyuridine Conjugates for DNA-Mediated Electron Transfer Studies	E. Charles Kerr; E Bruce Eaton; L. Thomas Netzel
867-879	Synthesis of Unsaturated Carboacyclic Nucleoside Analogues via Mitsunobu Reactions	Jinfa Du; Guangyi Wang
881-889	Synthesis of [bis(Inosine-5′)]-tetraphosphate and [bis(Inosine-5′)]-pentaphosphate Analogues Bearing the Residues of Methylenediphosphonic Acid	A. V. Shipitsyn; N. B. Tarussova; E. A. Shirokova; A. A. Krayevsky
891-902	Kinetic Studies on CE(IV)-Induced Hydrolysis of Single-Stranded and Double-Stranded Oligonucleotides	Tomoyuki Igawa; Jun Sumaoka; Makoto Komiyama
903-915	Synthesis and NMR Characterization of Diastereomeric C_PSMeG Derivatives	Daisy Machytka; Gyula Sági; MÁRia Kajtár-peredy; Eszter Gács-baitz
917-933	The Chemical Synthesis of Oligoribonucleotides with Selectively Placed 2′-O-Phosphates	Ryszard Kierzek; Michelle A. Steiger; Sherry L. Spinelli; Douglas H. Turner; Eric M. Phizicky
935-940	A Convenient Synthesis of A Novel Nucleoside Analogue: 4-(δ-Diformyl-methyl)-1-(β-D-ribofuranosyl)-2-pyrimidinone	Kui Gao; Leslie E. Orgel
941-954	Studies on Epimeric D-xylo-and D-lyxo-Tetritol-yl-2-phenyl-2H-1,2,3-triazoles. Synthesis and Anomeric Configuration of 4-(α- and β-D-Threofuranosyl)-2-phenyl-2H-1,2,3-triazole C-Nucleoside Analogs	Mohammed A. E. Sallam; Farida F. Louis; John M. Cassady
955-962	Investigation of a Facile Synthetic Method for Phosphorothioate Dimer Synthons In Oligonucleotide Phosphorothioates Synthesis	Takanori Miyashita; Kohei Yamada; Kazuhiko Kondo; Kenya Mori; Kazuo Shinozuka
963-975	Inhibition of Cell Growth and Proliferation in Human Glioma Cells and Normal Human Astrocytes Induced by 8-Cl-cAMP and Tiazofurin	M. Pesic; K. Drabek; C. Esler; S. Ruzdijic; V. Pejanovic; Z. Pietrzkowski
977-994	The Nonenzymatic Hydrolysis of Oligoribonucleotides VII. Structural Elements Affecting Hydrolysis	Arkadiusz Bibillo; Marek Figlerowicz; Krzysztof Ziomek; Ryszard Kierzek
995-1003	Prooligonucleotides Exhibit Less Serum-Protein Binding Than Phosphodiester and Phosphorothioate Oligonucleotides	Guilhem Tosquellas; Anton Bryksin; Karine Alvarez; François Morvan; Jean-Jacques Vasseur; Bernard Rayner; Elena Rykova; Pavel Laktionov; Valentin Vlassov; Jean-Louis Imbach
1005-1015	Synthesis of 6-Alkyl- and Arylamino-9-(tetrahydro-2-pyranyl)purines via 6-Methylsulfonylpurine	José Daniel Figueroa Villar; Marita Almeida Motta
1017-1031	Synthesis and Antiviral Activity of C-5 Substituted Analogues of D4T Bearing Methylamino- or Methyldiamino-Linker Arms	D. Gavriliu; C. Fossey; G. Fontaine; S. Benzaria; A. Ciurea; Z. Delbederi; B. Lelong; D. Ladurée; A. M. Aubertin; A. Kirn
1033-1054	Synthesis, Mechanism and Fluorescence Properties of 8-(Aryl)-3-β-D-Ribofuranosylimidazo[2,1-i]purine 5′-Phosphate Derivatives	Bilha Fischer; Eihab Kabha; Fernand-Pierre Gendron; Adrien R. Beaudoin

Volume 19, Issue 4 (2000)

a	Editorial board page for “Nucleosides, Nucleotides & Nucleic Acids”, Volume 19, Number 4
705-722	Pyrazole Related Nucleosides 5.¹ Synthesis and Biological Activity of 2′-Deoxy- 2′, 3′-dideoxy- and Acyclo-analogues of 4-Iodo-1-β-D-ribofuranosyl-3-carboxymethyl Pyrazole (IPCAR)	Stefano Manfredini; Pier Giovanni Baraldi; Rita Bazzanini; Elisa Durini; Silvia Vertuani; Alessandra Pani; Tiziana Marceddu; Francesca Demontis; Laura Vargiu; Paolo La Colla
723-733	Nucleic Acid Components and Their Analogues: New Synthesis of Bicyclic Thiopyrimidine Nucleosides	Galal E. H. Elgemeie; Adel M. E. Attia; Sherifa S. Alkabai
735-748	Synthesis of 3′-O2-(Azaheterocycle)-Thymidines	Guillaume Prestat; Didier Dubreuil; Ané Adjou; Jean Paul Pradère; Jacques Lebreton; Michel Evers; Yvette Henin
749-756	Replacement of the Phosphodiester Bond Between U4 and G5 in the U-Turn of a Chemically Modified Hammerhead Ribozyme by an Amide Bond	Martin Dunkel; Vivian Reither
757-774	Synthesis of 3′-Trifluoromethyl Nucleosides as Potential Antiviral Agents	Pawan K. Sharma; Vasu Nair
775-794	Highly Stereoselective Synthesis and Biological Properties of Nucleoside Analogues Bearing a Spiro Inserted Oxirane Ring	Jean M. J. Tronchet; Imre Kovacs; Michel Seman; Pierre Dilda; Erik De Clercq; Jan Balzarini
795-804	Metabolism of O⁶-Propyl and N⁶-Propyl-carbovir in CEM Cells	William B. Parker; Sue C. Shaddix; Lucy M. Rose; Phuong T. Pham; Mei Hua; Robert Vince
805-813	The Synthesis of Cyclonucleotides with Fixed Glycosidic Bond Linkages as Putative Agonists for P2-Purinergic Receptors	Girolamo Tusa; Juta K. Reed
815-825	New Purine Derivatives as Efficient Preparation of Nucleoside Analogs via Alkylation	Kirill A. Lukin; Chengxi Yang; John R. Bellettini; B. A. Narayanan
827-838	Preparation, Hydrolysis and Intramolecular Transesterification of 3′-Deoxy-3′-thioinosine 3′-S-Dimethylphosphorothiolate	Mohamed I. Elzagheid; Esa Mäki; Ulla Kaukinen; Mikko Oivanen; Harri Lönnberg
839-843	Synthesis of 9-(2-Deoxy-β-D-ribofuranosyl)purine-2-thione	Harry P. Rappaport

Volume 19, Issue 3 (2000)

a	Editorial board page for “Nucleosides, Nucleotides & Nucleic Acids”, Volume 19, Number 3
515-531	Synthesis and Properties of Uniquely Modified Oligoribonucleotides: Yeast Trna^Phe Fragments with 6-Methyluridine and 5,6-Dimethyluridine at Site-Specific Positions	Elzbieta Sochacka; Grazyna Czerwinska; Richard Guenther; Robert Cain; Paul F. Agris; Andrzej Malkiewicz
533-543	Influence of Diastereomeric Ratios of Deoxyribonucleoside Phosphoramidites on the Synthesis of Phosphorothioate Oligonucleotides	Z. S. Cheruvallath; H. Sasmor; D. L. Cole; V. T. Ravikumar
545-558	Development of a Purification Procedure for the Isolation of Nucleosides from Urine Prior to Mass Spectrometric Analysis	E. Dudley; S. El-shakawi; D. E. Games; R. P. Newton
559-565	A Convenient Synthesis of 2′-Deoxy-2-fluoroadenosine; a Potential Prodrug for Suicide Gene Therapy	Abdalla E. A. Hassan; Anita T. Shortnacy-fowler; John A. Montgomery; John A. Secrist III
567-584	Synthesis and Biological Activities of New Carbaacyclonucleosides and 1′-Oxaacyclonucleosides Related to Clitocine	Corinne Bacchelli; Roger Condom; Nadia Patino; Anne-Marie Aubertin
585-591	Formation and Reactivity of 2,4-Ditriazolyl Pyrimidine C-Nucleoside Derived from Pseudouridine	Natalia Dyatkina; Alexander Khorlin; Kyoichi A. Watanabe
593-601	Synthesis of Oligodeoxyribonucleotide Bearing 2′-S-Alkyl Residue and its Effect on the Duplex Stability	Hiroaki Ozaki; Yuichi Sato; Sadaji Azuma; Hiroaki Sawai
603-618	Synthesis and Biological Evaluation of 1,3-Oxathiolane 5-Azapyrimidine, 6-Azapyrimidine, and Fluorosubstituted 3-Deazapyrimidine Nucleosides	Mao-Chin Liu; Mei-Zhen Luo; Diane E. Mozdziesz; Tai-Shun Lin; Ginger E. Dutschman; Elizabeth A. Gullen; Yung-Chi Cheng; Alan C. Sartorelli
619-628	Efficient Synthesis of Carbocyclic Nucleoside, (±)-Homocarbovir Via π-Allylpalladium Complex Formation from the Allyl N,N-Ditosylimide Substrate	Hakjune Rhee; Dong-Oh Yoon; Michael E. Jung
629-635	Stereoselective Synthesis and X-Ray Structure of 1-(4-O-Benzyl-1,5-anhydro-2,3-dideoxy-D-arabino-hex-1-enitol-3-yl)-4-methoxy-1H-pyrimidin-2-one	Hideyuki Sugimura
637-650	Syntheses, Crystal Structures, and Hydrogen Bonding Patterns of 3′-C-Methylenecarboxylic-3′-deoxythymidine and 3′-C-Methyleneamidilylic-3′-deoxythymidine	Joong Young Kim; Byeang Hyean Kim
651-690	The Latest Progress in the Synthesis of Carbocyclic Nucleosides	Xue-Feng Zhu
691-702	Cellular Pharmacology of the D- and L-Enantiomers of β-5-o-Carboranyl-2′-deoxyuridine	Selwyn J. Hurwitz; Li; Alessandra Eleuteri; Janis Wright; Josef Moravek; Raymond F. Schinazi
703	Erratum

Volume 19, Issue 1-2 (2000)

xiii-xiv	Guest Editorial	T. A. Krenitsky; G. W. Koszalka
xv-xvii	Biographical Sketch	William H. Prusoff
a-b	Editorial board page for “Nucleosides, Nucleotides & Nucleic Acids”, Volume 19, Number 1-2
1-12	The “β-Fluorine Effect” in the Non-Metal Hydride Radical Deoxygenation of Fluorine-Containing Nucleoside Xanthates	Maqbool A. Siddiqui; John S. Driscoll; Elie Abushanab; James A. Kelley; Joseph J. Barchi Jr.; Victor E. Marquez
13-29	Conformation and Local Environment of Nucleotides Bound To Hiv Type 1 Reverse Transcriptase (HIV-1 RT) in The Ground State	George R. Painter; C. Webster Andrews; Phillip A. Furman
31-37	Synthesis of (Z)- and (E)-9-[(2-Hydroxyethylidene)cyclopropyl]adenine—New Methylenecyclopropane Analogues of Adenosine and Their Substrate Activity for Adenosine Deaminase	Yao-Ling Qiu; Mohamad B. Ksebati; Jiri Zemlicka
39-68	Synthesis of 4-Substituted Imidazo[4,5-d][1,2,3]triazine (2-Azapurine)nucleosides	Steven Krawczyk; Michael T. Migawa; John C. Drach; Leroy B. Townsend
69-86	Synthesis of Amide-Linked [(3′)CH₂CO-NH(5′)] Nucleoside Analogues of Small Oligonucleotides	Morris J. Robins; Bogdan Doboszewski; Bradley L. Nilsson; Matt A. Peterson
87-100	Synthesis and Antiviral Activity of Amino Acid Carbamate Derivatives of AZT	Shu-Ling Chang; George Griesgraber; Timothy W. Abraham; Tullika Garg; Heng Song; Cheryl L. Zimmerman; Carston R. Wagner
101-123	Synthesis and Evaluation of a Series of 2′-Deoxy Analogues of The Antiviral Agent 5,6-Dichloro-2-Isopropylamino-1-(β-L-Ribofuranosyl)-1H-Benzimidazole (1263W94)	Joseph H. Chan; Stanley D. Chamberlain; Karen K. Biron; Michelle G. Davis; Robert J. Harvey; Dean W. Selleseth; Ronna E. Dornsife; Ernest H. Dark; Lloyd W. Frick; Leroy B. Townsend; John C. Drach; George W. Koszalka
125-153	Design, Synthesis, and Antiviral Evaluation of 2-Deoxy-D-Ribosides of Substituted Benzimidazoles as Potential Agents for Human Cytomegalovirus Infections	Ruiming Zou; Etsuko Kawashima; George A. Freeman; George W. Koszalka; John C. Drach; Leroy B. Townsend
155-174	Benzimidazole 2′-Isonucleosides: Design, Synthesis, and Antiviral Activity of 2-Substituted-5,6-Dichlorobenzimidazole 2′-Isonucleosides	G. A. Freeman; D. W. Selleseth; J. L. Rideout; R. J. Harvey
175-187	Nucleosides and Nucleotides. 192. Toward the Total Synthesis of Cyclic ADP-Carbocyclic-Ribose. Formation of the Intramolecular Pyrophosphate Linkage by a Conformation-Restriction Strategy in a Syn-form Using a Halogen Substitution at the 8-Position of the Adenine Ring	Yuji Sumita; Michiyo Shirato; Yoshihito Ueno; Akira Matsuda; Satoshi Shuto
189-203	Investigation of The Kinetics of Degradation of Hexopyranosylated Cytosine Nucleosides Using Liquid Chromatography	Grace N. Thoithi; Ann Van Schepdael; Roger Busson; Gerard Janssen; Arthur Van Aerschot; Piet Herdewijn; EugÈNe Roets; Jos Hoogmartens
205-217	Synthesis and Antiviral Evaluation of Unnatural β-L-Enantiomers of 3′-Fluoro- and 3′-Azido-2,3′-dideoxyguanosine Derivatives	Arnaud Marchand; Christophe Mathé; Jean-Louis Imbach; Gilles Gosselin
219-236	Synthesis of L-3′-Hydroxymethylribonucleosides	John S. Cooperwood; Vincent Boyd; Giuseppe Gumina; Chung K. Chu
237-251	Pyrrolo[2,3-d]Pyrimidine Nucleosides: Synthesis and Antitumor Activity of 7-Substituted 7-Deaza-2′-Deoxyadenosines	Frank Seela; Matthias Zulauf; Shih-Fong Chen
253-268	Synthesis and Antiviral Activities of Enantiomeric 1-[2-(Hydroxymethyl) Cyclopropyl] Methyl Nucleosides	Claire Pierra; Sureyya Olgen; Sócrates C. H. Cavalcanti; Yung-Chi Cheng; Raymond F. Schinazi; Chung K. Chu
269-273	Carbocyclic 5′-Noruridine	Vishnumurthy R. Hegde; Katherine L. Seley; Stewart W. Schneller

Volume 19, Issue 1-2 (2000)

275-282	Rapid and Selective Reduction of Amide Group by Borane-Amine Complexes in Acyl Protected Nucleosides	Zinaida A. Sergueeva; Dmitri S. Sergueev; Barbara Ramsay Shaw
283-295	Synthesis of Biomimetic Analogs of Neomycin B: Potential Inhibitors of the HIV RNA Rev Response Element	Naozumi Nishizono; Vasu Nair
297-327	An Efficient, Scalable Synthesis of the HIV Reverse Transcriptase Inhibitor Ziagen® (1592U89)	Susan M. Daluge; Michael T. Martin; Barry R. Sickles; Douglas A. Livingston
329-340	Synthesis of 4′-Thio-β-D-arabinofuranosylcytosine (4′-Thio-ara-C) and Comparison of Its Anticancer Activity with That of Ara-C	Kamal N. Tiwari; Anita T. Shortnacy-fowler; Loredana Cappellacci; William B. Parker; William R. Waud; John A. Montgomery; John A. Secrist III
341-356	Phosphorylation of Ganciclovir Phosphonate by Cellular GMP Kinase Determines the Stereoselectivity of Anti-Human Cytomegalovirus Activity	Wayne H. Miller; Lilia M. Beauchamp; Eric Meade; John E. Reardon; Karen K. Biron; Albert A. Smith; Charles A. Goss; Richard L. Miller
357-369	Rational Design of Selective Antimetabolites of DNA-Thymine Biosynthesis: 5-Propynylpyrimidine Nucleoside Derivatives	Thomas I. Kalman; Zhe Nie
371-377	Potentiation of The Anti-HIV Activity of Zalcitabine and Lamivudine by a CTP Synthase Inhibitor, 3-Deazauridine	Wen-Yi Gao; David G. Johns; Hiroaki Mitsuya
379-404	Synthesis and Biological Activity of a Novel Class of Purine Nucleoside Phosphorylase Inhibitors	Philip E. Morris Jr.; Arthur J. Elliott; Sandra P. Walton; Carl H. Williams; John A. Montgomery
405-413	Cellular Phosphorylation of 2′, 3′-Dideoxyadenosine-5′-monophosphate, a Key Intermediate in The Activation of the Antiviral Agent DDI, in Human Peripheral Blood Mononuclear Cells	Brian L. Robbins; Jack Greenhaw; Arnold Fridland
415-434	Differential Transport of Cytosine-Containing Nucleosides by Recombinant Human Concentrative Nucleoside Transporter Protein hCNT1	Kathryn A. Graham; Jackie Leithoff; Imogen R. Coe; Delores Mowles; John R. Mackey; James D. Young; Carol E. Cass
435-446	Excision of β-L- and β-D-Nucleotide Analogs From DNA by p53 Protein	Marina Kukhanova; Tsung-Wu Liu; Helene Pelicano; Yung-Chi Cheng
447-460	Preclinical Antitumor Activity of 2-Chloro-9-(2-deoxy-2-fluoro-β-D-arabinofuranosyl)adenine (C1-F-Ara-A)	William R. Waud; Steven M. Schmid; John A. Montgomery; John A. Secrist III
461-470	Early Therapy with Valaciclovir or Famciclovir Reduces But Does Not Abrogate Herpes Simplex Virus Neuronal Latency	Hugh J. Field; Alana M. Thackray
471-479	Synthesis and Antiviral Evaluation of 1-O-Hexadecylpropanediol-3-P-acyclovir: Efficacy Against HSV-1 Infection in Mice	James R. Beadle; Ganesh D. Kini; Kathy A. Aldern; Michael F. Gardner; Kristine N. Wright; Rachel J. Rybak; Earl R. Kern; Karl Y. Hostetler
481-499	In Vitro and In Vivo Metabolism and Pharmacokinetics of bis [(T-Butyl)-S-acyl-2-thioethyl]-β-L-2′,3′-dideoxy-5-fluorocytidine Monophosphate	Lee T. Martin; Erika Cretton-scott; Laurent Placidi; Abdesslem Faraj; Anna Giulia Loi; Raymond F. Schinazi; Harold M. McClure; Gilles Gosselin; Jean-Louis Imbach; Jean Pierre Sommadossi
501-513	Efficacy of Topical Acyclovir Monophosphate, Acyclovir, or Penciclovir in Orofacial HSV-1 Infections of Mice and Genital HSV-2 Infections of Guinea Pigs	Earl R. Kern; Joyce Palmer; George Szczech; George Painter; Karl Y. Hostetler

Volume 18, Issue 11-12 (1999)

In Memory of Dr. Gordon Shaw

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 18, Number 11-12
xiii-xv	Biographical Sketch
2345-2356	Analogs of AICA- and IsoAICA Ribosides and Their Methylated Base Counterparts	Raymond P. Panzica; Leroy B. Townsend
2357-2365	Improved Synthesis of 2-Deoxy-L-ribose	Weijian Zhang; Kanda S. Ramasamy; Devron R. Averett
2367-2377	Transglycosylation Reaction of 6-Thioguanosine	Andrzej Manikowski; Jerzy Boryski
2379-2395	Synthesis and Antiviral Studies of Unsaturated Analogues of Isomeric Dideoxynucleosides	Sanjib Bera; Travis Mickle; Vasu Nair
2397-2414	Synthetic Oligonucleotide Combinatorial Libraries. 3. Synthesis of Polyamevonucleosides	Przemyslaw Godzina; Katarzyna Adrych-Rozek; Wojciech T. Markiewicz
2415-2423	Intramolecular Glycosylation to Form 4-Methoxy-2,6-Dioxopyrimidine Nucleosides via O⁶,5′-Cyclonucleosides	Claire Castro; Chuan Chen; Michael E. Jung
2425-2431	A Modified Synthesis of Tiazofurin	Kanda S. Ramasamy; Devron Averett
2433-2442	Synthesis of 8-Substituted Analogues of 2′-Deoxy-2′-Fluoroadenosine	Tokumi Maruyama; Shigetada Kozai; Takako Manabe; Yuko Yazima; Yoshiko Satoh; Hiroshi Takaku
2443-2461	Certain 3,9-Dideazapurines as Inhibitors of Purine Nucleoside Phosphorylase	Jerry D. Rose; John A. Secrist III; John A. Montgomery
2463-2473	Synthesis and Biological Evaluation of 9-(β-L-Arabinofuranosyl)Adenine	Valérie Boudou; Jean-Louis Imbach; Grilles Gosselin
2475-2497	Acyclic Sugar Analogs of Triciribine: Lack of Antiviral and Antiproliferative Activity Correlate with Low Intracellular Phosphorylation	Anthony R. Porcari; Katherine Z. Borysko; Roger G. Ptak; Julie M. Breitenbach; Linda L. Wotring; John C. Drach; Leroy B. Townsend
2499-2510	Synthesis, Cytotoxic Effect and Antiviral Activity of 1-(β-D-Arabinofuranosyl)-5-Bromo-N⁴-Substitutedcytosine and 1-(β-D-Arabinofuranosyl)-5-Bromo-4-Methoxypyrimidin-2(1h)-One Derivatives	Raffaele Saladino; Maurizio Mezzetti; Enrico Mincione; Anna Teresa Palamara; Patrizia Savini; Stefano Marini
2511-2520	Synthesis of Di- And Tri-Substituted Adenosine Derivatives and Their Affinities at Human Adenosine Receptor Subtypes	R. Volpini; E. Camaioni; S. Costanzi; S. Vittori; K. -N. Klotz; G. Cristalli
2521-2532	L-Nucleoside Analogues as Potential Antimalarials That Selectively Target Plasmodium Falclparum Adenosine Deaminase	David M. Brown; Andrew G. Netting; Byoung K. Chun; Yongseok Choi; Chung K. Chu; Annette M. Gero
2533-2549	Polyester and N-Methyl Analogues of Peptide Nucleic Acids: Synthesis and Hybridization Properties	V. A. Efimov; A. A. Buryakova; M. V. Choob; O. G. Chakhmakhcheva
2551-2564	Inhibitory Potency of 5-Benzyluracil, 5-Phenylcytosine and 5-Phenylpyrimidin-2-one Nucleosides Against Uridine Phosphorylase from Mouse Leukemic L1210 Cells	Ivan Votruba; Marcela Krečmerová; Hubert Hřebabecký; Antonín Holý
2565-2580	Straightforward Synthesis of Lipophilic Thymidine Glucopyranosyl Monophosphates as Models for a Drug Delivery System Across Cellular Membranes	Emilia Belsito; Angelo Liguori; Anna Napoli; Carlo Siciliano; Giovanni Sindona

Volume 18, Issue 11-12 (1999)

In Memory of Dr. Gordon Shaw

2581-2599	Crystal and Solution Structure of 5′-O-(Guanosine-2′-O-Phosphonomethyl)Cytidine, an Isopolar Nonisosteric Phosphonate Analog Of GpC	J. Zachová; I. Císaŕová; M. Buděšíns�; R. Liboska; Z. Točík; I. Rosenberg
2601-2611	Synthesis of a Novel Pyrazolo[1, 5-C]Pyrimidine C-Nucleoside and Conformational Analysis By NMR Spectroscopy	Marija Prhavc; Janez Plavec; Joźe Kobe; Ivan Leban; Gerald Giester
2613-2630	Nucleoside Analogues with a Novel Glycone Based on the Benzo[C]Furan Core	David F. Ewing; Nour-Eddine Fahmi; Christophe Len; Grahame Mackenzie; Gino Ronco; Pierre Villa; Gordon Shaw
2631-2660	The Synthesis of Geometric Variants of Rigidly-Linked Uracil-{Spacer}-Uracil and Uracil-{Spacer}-Effector Molecules Using Block Assembly Methods	R. N. Warrener; D. N. Butler; M. Golic
2661-2676	A Pyrene Seco-Pseudonucleoside in Constructing Interaction-Sensitive Fluorescent DNA Probes	Vladimir A. Korshun; Konstantin V. Balakin; Tatyana S. Proskurina; Ilya I. Mikhalev; Andrei D. Malakhov; Yuri A. Berlin
2677-2684	Random Mutagenesis Using 2-Amino-9-(2-Deoxy-β-D-Ribofuranosyl)Purine-5′-Triphosphate and the Polymerase Chain Reaction	F. Hill; I. Felix; M. G. McDougall; S. Kumar; D. Loakes; D. M. Brown
2685-2695	5′-Tailed Octanucleotide Primers for Cycle Sequencing	D. Loakes; F. Hill; D. M. Brown; S. Ball; M. A. Reeve; P. S. Robinson
2697-2709	Incorporation of 2′-Deoxysangivamycin in DNA Duplexes: The Conversion of a Pyrrolo[2, 3-d]Pyrimidine Nitrile to a Carboxamide upon Oligonucleotide Deprotection	Frank Seela; Matthias Zulauf
2711-2719	Oligodeoxyribonucleotides with Internucleotidic or Terminal Phosphorothioate Groups: Different Pathways in the Reaction with Water-Soluble Carbodhmide	Valeri G. Metelev; Oxana A. Borisova; Nina G. Dolinnaya; Zoe A. Shabarova
2721-2744	d(GCGTAGC), an Equilibrium Between a Hairpin Structure and an Unusual Duplex	Evline Lescrinier; Shqun Sheng; Ja Schraml; Roger Busson; Piet Herdewijn
2745-2750	Oligonucleotide Conjugated to Linear and Branched High Molecular Weight Polyethylene Glycol as Substrates for RNase H	P. E. Vorobjev; V. F. Zarytova; G. M. Bonora
2751-2768	Structural Characterization of Intact Covalently Linked DNA Adducts by Electrospray Mass Spectrometry	Joeph Banoub; Stven Combden; Judith Miller-Banoub; George Sheppard; Howard Hodder
2769-2783	Introduction of 6-Formylcytidine into a Myb Binding Sequence	Atushi Kittaka; Tesuya Kuze; Miori Amano; Hiomichi Tanaka; Taashi Miyasaka; Kuihiko Hirose; Taao Yoshida; Aknori Sarai; Taashi Yasukawa; Shnsuke Ishii
2785-2818	Physico-Chemical Properties of 5′-Polyarene Tethered DNA-Conjugates, and Their Duplexes with Complementary RNA	Nitin Puri; Jyoti Chattopadhyaya
2819-2835	Stereoselective Synthesis of β-L-2′, 3′-Dideoxy-and L-2′,3′-Didehydro-2′,3′-Dideoxy Purine Nucleosides	Peiyuan Wang; Pascal J. Bolon; M. Gary Newton; Chung K. Chua

Volume 18, Issue 10 (1999)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 18, Number 10
2141-2146	Site-Specific Formation of A basic Lesions in DNA	Robert S. Coleman; Richard M. Pires
2147-2154	Tetra-Thymidine Phosphorofluoridates via Tetra-Thymidine Phosphoro-selenoates: Synthesis and Stability	Janina Baraniak; Dariusz Korczynski; Renata Kaczmarek; Wojciech J. Stec
2155-2173	Isolation and Characterization of 5-Carbamoylmethyluridine and 5-Carbamoylmethyl-2-Thiouridine from Human Urine	G. B. Chheda; H. B. Patrzyc; H. A. Tworek; S. P. Dutta
2175-2191	The Synthesis and Biological activity of a Highly Selective Adenosine A_2a. Receptor Agonist	David R. Borcherding; Nelsen L. Lentz; Philip M. Weintraub; Mark W. Dudley; Roberta Secrest; Philip R. Kastner; Norton P. Peet; Hoechst Marion Roussel
2193-2199	Sensitivity of Bacteriophage RB69 DNA Polymerase to n²-(p-n-Butylphenyl)-2′-Deoxyguanosinenucleotides	James M. Stattel; George E. Wright
2201-2217	A Spectroscopic and Thermodynamic Study of Taxol Nucleic Acid Complexes	G. Bischoff; U. Gromann; S. Lindau; W. V. Meister; S. Hoffmann
2219-2231	Synthesis of c-5′-nor-Dideoxycarbanucleosides Structurally Related to Neplanocin C	Maria J. Comin; Carlos A. Pujol; Elsa B. Damonte; Juan B. Rodriguez
2233-2252	Synthesis of 2′,3′-Dideoxy-2′-Fluoro-l-threo-Pentofuranosyl Nucleosides as Potential Antiviral Agents	Socrates C. H. Cavalcanti; Yuejun Xiang; M. Gary Newton; Raymond F. Schinazi; Yung-Chi Cheng; Chung K. Chu
2253-2263	Synthesis and Antiviral Activity of Carbocyclic Nucleosides Incorporating a Modified Cyclopentane Ring. Part 3: Adenosine and Uridine Analogues	M. Isabel Nieto; J. Manuel Blanco; Olga Caamaño; Franco Fernández; Xerardo Garcia-mera; Carmen Lopez; Jan Balzarini; Erik De Clercq
2265-2283	Selective Synthesis and Structure of 6-Arylvinyl-2- and 4-Glucosyl-1,2,4-triazines of Expected Interesting Biological Activity	Abdel Kader Mansour; Yehia A. Ibrahim; Nasser S. A. M. Khalil
2285-2300	Synthesis of New Nucleoside Analogues Comprising a Geminal Difluorocyclopropane Moiety as Potential Antiviral/Antitumor Agents	Yao-Ling Qiu; Jiri Zemlicka
2301-2306	Synthesis of Some Pyridine Ribosides and Their Biological Activity	Adel M. Attla; Hanaa A. Mansour; Ahmed A. Almehdi; Mohammed M. Abbasi
2307-2315	Synthesis and Biological Activity of Modified Thiopyrimidine Nucleosides	Adel M. Attia; Morsala A. Sallam; Ahmed A. Almehdi; Mohammed M. Abbasi
2317-2325	Synthesis and Anti-Retroviral Activity of O,O′-BIS(3′-Azido-2′,3′-Dideoxythymidin-5′-yl) Phosphoramidate Derivatives	Inger Kers; Jacek Stawiński; Jean-Luc Girardet; Jean-Louis Imbach; Christian Perigaud; Gilles Gosselin; Anne-Marie Aubertin
2327-2333	Utilization Of Tetrabutylammonium Triphenyldifluorosilicate (TBAT) In The Synthesis of 6-Fluoropurine Nucleosides	Vadim Gurvich; Hye-Young Kim; Richard P. Hodge; Constance M. Harris; Thomas M. Harris
2335-2343	Synthesis of N-Glycosylated Pyridiines as New Antimetabolite Agents	Badria A. Hussain; Adel M. Attia; Galal E. H. Elgemeie

Volume 18, Issue 9 (1999)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 18, Number 9
1911-1928	Synthesis of Chiral Carbocyclic Ribonucleotides	Vincent D. Antle; Carol A. Caperelli
1929-1933	Base Modified Oligodeoxynucleotides. II. Increase of Stability to Nucleases by 5-Alkyl-, 5-(1-Alkenyl)-, and 5-(1-Alkynyl)-pyrimidines	L. Ötvös; J. Sági; Gy. Sági; A. Szemz
1935-1944	Identification of a Good C-MYC Antisense Oligodeoxynucleotide Target Site and the Inactivity at This Site of Novel NCH Triplet-Targeting Ribozymes	Richard V. Giles; David G. Spiller; Richard E. Clark; David M. Tidd
1945-1960	Application of Oligonucleoside Methylphosphonates in the Studies on Phosphodiester Hydrolysis by Serratia Endonuclease	Tushar Kumar Srivastava; Peter Friedhoff; Alfred Pingoud; S. B. Katti
1961-1976	Homologues of Isomeric Dideoxynucleosides as Potential Antiviral Agents: Synthesis of Isodideoxy-Nucleosides with a Furanethanol Sugar Moiety	Xiaoping Zheng; Vasu Nair
1977-1984	Asymmetric Synthesis of 4′-Methyl-2′,3′-dideoxynucleosides	Frederick A. Luzzio; Alexander V. Mayorov; Michael E. Menes; William L. Champion Jr.
1985-1994	Synthesis and Antiviral Activity of 1,5-and 1,3-Dialkyl-1,2,4-triazole C-Nucleosides Derived from 1-(Chloroalkyl)-1-aza-2-azoniaallene Salts	Yaseen A. Al-soud; Wasfi A. Al-masoudi; Rajab Abu El-halawa; Najim Al-masoudi
1995-2016	Synthesis of Iodoaminoimidazole Arabinoside (IAIA): A Potential Reductive Metabolite of the Spect Imaging Agent, Iodoazomycin Arabinoside (IAZA)	Herbert C. Lee; Piyush Kumar; Leonard I. Wiebe; Robert McDonald; John R. Mercer; Kazue Ohkura; Koh-Ichi Seki
2017-2030	Evaluation of Oligonucleotides Containing Two Novel 2′-O-Methyl Modified Nucleotide Monomers: A 3′-C-Allyl and a 2′-O-3′-C-Linked Bicyclic Derivative	Henrik M. Pfundheller; Alexei A. Koshkin; Carl Erik Olsen; Jesper Wengel
2031-2042	Synthesis and Nuclease Stability of Dinucleotides Containing an Anti- conformationally Constrained Acyclic Thymidine	Ling-Yih Hsu; Kuo-Tsao Yang
2043-2049	Nucleosides. II. Synthesis and Properties of 3,4-Diaryl-4,5-dihydro-1-(β-D-ribofuranosyl)-1,2,4-triazole-5-thiones	Mosselhi A. N. Mosselhi
2051-2069	Evaluation of Different Types of End-Capping Modifications on the Stability of Oligonucleotides Toward 3′- and 5′-Exonucleases	Daniela Pandolfi; Francesca Rauzi; Massimo L. Capobianco
2071-2091	Physico-chemical and Biological Properties of Antisense Phosphodiester Oligonucleotides with Various Secondary Structures	Andrei V. Maksimenko; Marina B. Gottikh; Valerie Helin; Zoe A. Shabarova; Claude Malvy
2093-2108	Hydrolytic Reactions of 3′-Deoxy-3′-thioinosylyl-(3′→ >5′)-uridine; An RNA Dinucleotide Containing a 3′-S-Phosphorothiolate Linkage	Mohamed I. Elzagheid; Mikko Oivanen; Karel D. Klika; Bryan C. N. M. Jones; Richard Cosstick; Harri Lönnberg
2109-2120	A Simple and Efficient Procedure for the Synthesis of an Alendronate- Oligonucleotide Conjugate via a Carbamate Linker	M. Lecouvey; C. Dufau; El D. Manouni; Y. Leroux
2121-2126	Palladium-Catalyzed Animation of 6-Chloropurine. Synthesis of N⁶-Substituted Adenosine Analogues	Judith Barends; Johannes van der Linden; Floris Van Delft; Gerrit-Jan Koomen
2127-2139	Regioselective N¹-Alkylation of Guanosine Derivatives Protected at N² by an N,N-Dialkyl Amidine Group	Stéphane P. Vincent; Charles Mioskowski; Luc Lebean

Volume 18, Issue 8 (1999)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 18, Number 8
1751-1769	Synthesis and Triplex Forming Properties of Pyrimidine Derivative Containing Extended Functionality	Diego A. Gianolio; Larry W. McLaughlin
1771-1787	Improved Methods for the Preparation of 2′-Deoxyribonucleoside and Ribonucleoside 3′-Phosphoramidites with Allylic Protectors	Sophie B. Heidenhain; Yoshihiro Hayakawa
1789-1802	Increased Cytotoxicity and Decreased In Vivo Toxicity of FdUMP[10] Relative to 5-FU	Jinqian Liu; Alan Skradis; Carol Kolar; Jeff Kolath; James Anderson; Terrence Lawson; James Talmadge; William H. Gmeiner
1803-1807	Synthesis of Dimer Phosphoramidite Synthons for Oligodeoxyribonucleotide Phosphorothioates Using Diethyldithiocarbonate disulfide as an Efficient Sulfurizing Reagent	Alessandra Eleuteri; Zacharia S. Cheruvallath; Daniel C. Capaldi; Douglas Cole Vasulinga; T. Ravikumar
1809-1824	A Phosphate Bound Universal Linker for DNA Synthesis	Matthew H. Lyttle; Daren J. Dick; Derek Hudson; Ronald M. Cook
1825-1843	Cytidinium H-Phosphonate Monohydrate, bis 2′-Deoxycytidinium H-Phosphonate and 2′-Deoxycytromium H-Phosphonate -Structures and Properties	Maria D. Bratek-Wiewiórowska; Maciej Wiewiórowski; Magdalena Alejska; Agnieszka Olszewska; Krzysztof Woźniak
1845-1861	Synthesis and Biophysical Studies of Modified Oligonucleotides Containing Acyclic Amino Alcohol Nucleoside Analogs	Kanda S. Ramasamy; Vesna Stoisavljevic
1863-1877	Evaluation of the Kinetics of Hydrolysis of Diamino Analogues of 2′- Or 3′-Deoxyadenosine and of 9-(2-Deoxy-β-D-threo-Pentofuranosyl)adenine or 9-(3-Dexoy-β-D-threo-Pentofuranosyl)adenine By Liquid Chromatography	G. Thoithi; A. Van Schepdaer; C. Vinckier; P. Herdewijn; E. Roets; J. Hoogmartens
1879-1882	Efficient Synthesis of Deoxyribonucleoside Phosphoramidites by Eliminating the Use of Additional Activator	Alessandra Eleuteri; Daniel C. Capaldi; Douglas Cole Vasulinga; T. Ravikumar
1883-1903	Substrate/Inhibitor Properties of Human Deoxycytidine Kinase (dCK) and Thymidine Kinases (Tk1 And Tk2) Towards the Sugar Moiety of Nucleosides, Including O′-Alkyl Analogues	Borys Kierdaszuk; Krzysztof Krawiec; Zygmunt Kazimierczuk; Ulla Jacobsson; Nils G. Johansson; Birgitte Munch-petersen; Staffan Eriksson; David Shugar
1905-1910	The Synthesis of Carbocyclic 5′-Nor Thymidine and an Isomer as Oligonucleotide Monomers	Vishnumurthy R. Hegde; Katherine L. Seley; Xing Chen; Stewart W. Schneller

Volume 18, Issue 6-7 (1999)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 18, Number 6-7
xxxix-xl	Preface	Gilles Gosselin
1141-1162	Making Drugs Out of Oligonucleotides: A Brief Review and Perspective	P. Dan Cook
1163-1168	Synthesis of Artificially Bent Oligonucleotides by Incorporation of Conformationally Rigid 5′-Cyclouridylic Acid Derivatives	Mitsuo Sekine; Osamu Kurasawa; Kohji Seio; Koh-Ichiroh Shohda; Takeshi Wada
1169-1174	Triarylmethyl Substituted 4,5-Dicyanoimidazoles as Activators for Rp-Diastereoselective Synthesis of TpN Dinucleoside Methylphosphonates	Peter Schell; Wolfgang H. G. Laux; Joachim W. Engels
1175-1180	A New Approach to the Synthesis of Linear and Cyclic Oligoribonucleotides	Colin B. Reese; Quanlai Song
1181-1182	Progress in the Synthesis of Cyclic Deoxyribo- and Oligoribonucleotides	M. Frieden; A. Grandas; E. Pedroso
1183-1185	Reversed(5′-3′)Oligonucleotide Synthesis on Oxalyl-CPG Support	J. Bogan; L. Ignatovich; E. Stankevic
1187-1189	Stability of Phosphorothioate Oligonucleotides in Aqueous Ammonia in Presence of Stainless Steel	Brett J. Turney; Zacharia S. Cheruvallath; Mark Andrade; Douglas L. Cole; Vasulinga T. Ravikumar
1191-1194	Diastereomeric Process Control in the Synthesis of Oligodeoxyribonucleotide Phosphorothioates	Zacharia S. Cheruvallath; Tadeusz K. Wyrzykiewicz; Douglas L. Cole; Vasulinga T. Ravikumar
1195-1197	Use of Phenylacetyl Disulfide (PADS) in the Synthesis of Oligodeoxyribonucleotide Phosphorothioates	Zacharia S. Cheruvallath; Patrick D. Wheeler; Douglas L. Cole; Vasulinga T. Ravikumar
1199-1201	A New Protecting Group Strategy for Amino Groups in Oligonucleotide Chemistry: CEOC Group	Muthiah Manoharan; Thazha P. Prakash; Isabelle Barber-peoc'h; Balkrishen Bhat; Guillermo Vasquez; Bruce S. Ross; P. Dan Cook
1203-1204	A New, Efficient Exocyclic Amine Protection Scheme for 2-Aminoadenosine and Derivatives for Incorporation into Oligonucleotides	Bruce S. Ross; Robert H. Springer; Ramesh Bharadwaj; Alice M. Symons; Muthiah Manoharan
1205-1206	An Improved Deprotection Procedure of Amine-Containing Oligonucleotides from Acrylonitrile Modification	Chu-An Chang; Thomas Horn
1207-1209	Dimethoxytrityl Removal in Organic Medium: Efficient Oligonucleotide Synthesis Without Chlorinated Solvents	Achim H. Krotz; Douglas L. Cole; Vasulinga T. Ravikumar
1211-1213	Oligodeoxyribonucleotide Phosphorothioates: Substantial Reduction of (N-1)-Mer Content Through the Use of Blockmer Phosphoramidite Synthons	Alessandra Eleuteri; Zacharia S. Cheruvallath; Daniel C. Capaldi; Achim H. Krotz; Douglas L. Cole; Vasulinga T. Ravikumar
1215-1217	Synthesis of Deoxyribonucleoside Phosphorodithioate Dimers by a Triester Method	Daniel C. Capaldi; Douglas L. Cole; Vasulinga T. Ravikumar
1219-1220	The 9-Fluorenylmethoxycarbonyl (Fmoc) Group and Its Use in Oligonucleotide Synthesis	H. Schirmeister-tichy; G. G. Alvarado; W. Pfleiderer
1221-1222	Antiviral Activity of Magnesium and Magnesium/poly r(A-U) Combinations Against two RNA Viruses	J. Jamison; J. Gilloteaux; M. R. Nassiri; C. C. Tsai; J. Summers
1223-1224	Tetraethylene Glycol-Derived Spacer for Oligonucleotide Synthesis	Sigmund Gunzenhauser; Ewa Biala; Peter Strazewski
1225-1226	A New H-Phosphonate Approach Using N-Unprotected Monomers and Phosphonium Condensing Reagents	Takeshi Wada; Yuichi Sato; Fumio Honda; Shun-Ichi Kawahara; Akira Mochizuki; Mitsuo Sekine
1227-1229	An Improved Method for the Preparation of 4-Cyano-2-butenyl-deoxyribonucleosidephosphoramidites	G. Duckworth; J. Ackroyd
1231-1234	A Biotin Phosphoramidite Reagent for the Automated Synthesis of 5′-Biotinylated Oligonucleotides	Zhengyun Zhao; John Ackroyd
1235-1236	A Simple Solid-Phase Based Purification Procedure for Oligodeoxynucleotides	Thomas Horn; Mickey S. Urdea
1237-1238	Reusable Solid-Phase Supports for Oligonucleotide Synthesis Using Hydroquinone-O,O'-diacetic Acid (“Q-Linker”)	R. T. Pon; S. Yu; Z. Guo; X. Yang; Y. S. Sanghvi
1239-1240	Synthesis of Mixed Ribo/Deoxyribopolynucleotides by Mutant T7 RNA Polymerase	V. L. Tunitskaya; S. O. Gudima; D. A. Kostyuk; S. N. Kochetkov
1241-1242	Chemoselective Synthesis of Dithymidine Phosphorothioate in Solution Using O-Protected Thiophosphate Monomers	Thomas Boesen; Jan Kehler; Otto Dahl
1243-1244	A Mild Method for the Preparation of Nucleoside Phosphorofluoridate and Phosphorofluoridothioate Diesters	Martin Bollmark; Jacek Stawinski
1245-1246	New Methods for Multiple Modifications of a Phosphorus Centre. Their Relevance to Nucleotide and Oligonucleotide Analogues Synthesis	Inger Kers; Jacek Cieslak; Jadwiga Jankowska; Adam Kraszewski; Jacek Stawinski

Volume 18, Issue 6-7 (1999)

1247-1248	New Phosphitylating Reagents Containing P-F Bond and Their Application in the Synthesis of P-Fluoro Nucleosidyl Phosphates, Thiophosphates and Selenophosphates	W. Dąbkowski; I. Tworowska; E. Poniatowska; J. Michalski; F. Cramer
1249-1250	Synthesis and Properties of Some (2′-5′) Linked Dinucleoside Monophosphates Modified with 3′-Difluoromethylene Groups	C. A. Brown; C. L. Barnes; P. J. Serafinowski
1251-1252	Studies on the Phosphonate Isostere of Nucleoside 3′- and 2′-Phosphates as Precursors of the Related Oligonucleotides	Igor A. Mikhailopulo; Tamara M. Tsvetkova; Grigorii G. Sivets; Nicolai E. Poopeiko
1253-1254	Dimeric Oligonucleotide Synthons Containing 2-Deoxy-3-O-Phosphonomethyl-α-D-erythro-pentofuranosyl Nucleosides	Igor A. Mikhailopulo; Tamara I. Kulak; Olga V. Tkachenko; Svetlana L. Sentyureva; Frank Seela
1255-1256	Stereoselective 5′-Monodeuterated Ribonucleoside Phosphoramidites as Tools for Conformational Studies of RNA by the NMR Approach	M. A. Lukin; V. N. Bushuev
1257-1259	Synthesis of 5′-Ethynyl-2′-deoxynucleoside Analogues as Building Block for Antisense Oligonucleotide	Hassan B. Lazrek; Abdelalli Rochdi; Joachim W. Engels
1261-1262	Synthesis and Enzymatic Stability of Acyclic Thymidine Dimer Analogues having a Constrained Anti-Glycosidic Conformation	Ling-Yih Hsu; Kuo-Tsao Yang
1263-1264	Ethyl[2-Deoxy-5-O-(4,4′-dimethoxytrityl)-α- and β-D-erythro-Pentofuranosyl] Acetates as Versatile Intermediates in Nucleic Acid Chemistry	Jari Hovinen; Alex Azhayev; Harri Salo; Juhani Vilpo
1265-1266	Hydrolytic Reactions of an RNA Dinucleotide Containing a 3′-S-Phosphorothiolate Linkage	Mohamed Elzagheid; Mikko Oivanen; B. Colin; N. M. Jones; Richard Cosstick; Harri Lönnberg
1267-1268	Zn² Promoted Hydrolysis of RNA	Satu Mikkola; Izabela Zagorowska; Harri Lönnberg
1271-1276	Development of a Rapid Screening System to Test Antisense ODN Modifications and Carriers	Valérie Hélin; Marina Gottikh; Zohar Mishal; Frédéric Subra; Claude Malvy; Marc Lavignon
1277-1278	New Homogeneous Reverse Transcriptase and Nuclease Assays Based on Rare Earth Cryptate and Fluorescent Energy Transfer	Alpha-Bazin Béatrice; Mathis Gérard
1279-1280	Perylene-Labeled Oligonucleotide as a Probe in Homogeneous Hybridization Assay	K. V. Balakin; V. A. Korshun; D. S. Esipov; I. I. Mikhalev; Yu. A. Berlin
1281-1283	New Photolabile Protecting Groups of the 2-(2-Nitrophenyl)ethoxycarbonyl- and the 2-(2-Nitrophenyl)ethylsulfonyl-Type for the Oligonucleotide Synthesis	S. Bühler; H. Giegrich; W. Pfleiderer
1285-1287	Oligonucleotide Synthesis on Linear Reactive Polymer Grafted onto Solid Support, Medical Diagnostics Applications	C. Minard-basquin; C. Chaix; C. Pichot; B. Mandrand
1289-1291	Improved Solid Supports and Spacer/Linker Systems for the Synthesis of Spatially Addressable PNA-Libraries	S. Matysiak; N. C. Hauser; S. Würtz; J. D. Hoheisel
1293-1295	High-Density Nucleoside Analog Probe Arrays for Enhanced Hybridization	Jacqueline A. Fidanza; Glenn H. McGall
1297-1299	Detection of Nucleic Acids by Cycling Probe Technology on Magnetic Particles: High Sensitivity and Ease of Separation	Ram Bhatt; Brad Scott; Scott Whitney; Robert N. Bryan; Lynn Cloney; Alexandre Lebedev
1301-1304	New Developments in Light-Controlled Synthesis of DNA-Arrays	M. Beier; J. D. Hoheisel
1305-1307	Solid-Supported Oligonucleotide Systems for Special Biomedical Applications	Hartmut Seliger; Michael Hinz; Sigalit Gura; Boa Nitzan; Shlomo Margel
1309-1310	Peptide-and Biotin-Oligonucleotide-Pyrrole Conjugates for Electrochemical Addressing on Silicon Chip	H. Bazin; T. Livache
1311-1312	Efficient Automated Synthesis of Molecular Beacons	Bashar Mullah; Ken Livak
1313-1315	Long Range Electron Transfer in PNA/DNA Duplexes	Troels Koch; Bruce Armitage; Henrik F. Hansen; Henrik Ørum; Gary B. Schuster
1317-1318	Hole Transport Between G Bases in DNA	Eric Meggers; Bernd Giese
1319-1320	Oligonucleotides Derivatized with Luminescent and Photoreactive RU(II) Complexes: Models for Photoelectron Transfer and Photocrosslinking	J. F. Constant; E. Defrancq; J. Lhomme; N. Boutonnet; S. Content; I. Ortmans; A. Kirsch-De Mesmaeker
1321-1322	Interactions of High Affinity Anti (6-4) Photoproduct Antibody Fragments with Damaged DNA	Eiko Ohtsuka; Hiroyuki Kobayashi; Hiroshi Morioka; Kousuke Sato; Yasuo Komatsu; Osamu Nikaido; Yoshinori Satow; Ichio Shimada
1323-1324	Efficient Chemical Synthesis of Oligonucleotides Containing the 2-Deoxyribonolactone Site	Mitsuharu Kotera; Anne-Gaëlle Bourdat; Eric Defrancq; Muriel Jourdan; Julian Garcia; Christian Coulombeau; Jean Lhomme
1325-1327	Chemical Synthesis of Oligonucleotides Containing The (6-4) Photoproduct at the Thymine-Cytosine Site and Its Repair By (6-4) Photolyase	Shigenori Iwai; Toshimi Mizukoshi; Kenichi Hitomi; Takeshi Todo
1329-1330	Differences Between 4′-RNA and 4′-DNA Radicals During Anaerobic Strand Cleavage	Harald Strittmatter; Urs Schwitter; Bernd Giese
1331-1333	Synthesis and Characterization of Oligodeoxynucleotides Containing 5′,8-Cyclopurine-2′-Deoxyribonucleosides	Anthony Romieu; Didier Gasparutto; Didier Molko; Jean Cadet

Volume 18, Issue 6-7 (1999)

1335-1337	Misreading of RNA Templates Containing 8-Oxo-7,8-Dihydroguanosine Or 8-Oxo-2′-O-Methylguanosine in cDNA Synthesis by Reverse Transcriptases	Sang Kook Kim; Ji Young Kim; Shigeyuki Yokoyama; Hiroshi Takaku; Byung Jo Moon
1339-1341	Synthesis and Biological Evaluation of Modified DNA Fragments for The Study of Nucleotide Excision Repair in E. coli	Vania Monaco; Karin I. van de Wetering; Nico J. Meeuwenoord; Hans A. van den Elst; Hanneke R. Stuivenberg; Rob Visse; Janco C. van der Kaaden; Geri F. Moolenaar; Esther E. A. Verhoeven; Nora Goosen; Gijs A. van der Marel; Jacques H. van Boom
1343-1344	Spontaneous Cleavage of Single and Double Stranded 4′-DNA Radicals Under Aerobic Conditions	Adrian Dussy; Bernd Giese
1345-1347	5-Deazaflavins: New Very Efficient DNA Photosensitisers, Synthesis of Oligonucleotide Conjugates	I. Girault; J. L. Ravanat; C. Frier; M. Fontecave; J. Cadet; J. L. Décout
1349-1350	Synthesis and Characterization of Oligodeoxyribonucleotides Containing Tandem Base Damage	A. G. Bourdat; D. Gasparutto; C. D'ham; J. Cadet
1351-1353	Specific Recognition and Stabilization of an Abasic Site-Containing DNA Duplex by a Macrocyclic Bisacridine	M. P. Teulade-Fichou; J. P. Vigneron; J. M. Lehn; N. Berthet; J. Michon; J. Garcia; M. Jourdan; J. Lhomme
1355-1358	Higher Binding Affinity of Duplex Oligodeoxynucleotides Containing 1,2-Dideoxy-D-Ribose to The N6-Adenine DNA Methyltransferase M·TAQI Supports a Base Flipping Mechanism	Birgit Holz; Elmar Weinhold
1359-1360	Localization of The Initiation Site in T7 RNA Polymerase by Affinity Labeling	E. Rusakova; V. Tunitskaya; L. Memelova; B. Ermolinsky; S. Kochetkov; S. Mikhailov
1363-1364	Pyranosyl - Oligonucleotides	A. Eschenmoser
1365-1370	Lna (Locked Nucleic Acid)	Jesper Wengel; Alexei Koshkin; Sanjay K. Singh; Poul Nielsen; Michael Meldgaard; Vivek K. Rajwanshi; Ravindra Kumar; Jan Skouv; Christina B. Nielsen; Jens Peter Jacobsen; Nana Jacobsen; Carl E. Olsen
1371-1376	Properties of Oligonucleotides with Six Membered Carbohydrate Mimics and a 1,4-Relationship Between the Base Moiety and the Hydroxymethyl Group	P. Herdewijn; B. Allart; B. De Bouvere; H. De Winter; C. Hendrix; N. Hossain; G. Schepers; I. Verheggen; B. Wroblowski; A. Van Aerschot
1377-1378	Synthesis of ²H,¹³C-Labelled 2′-Deoxynucleosides and Their Site Specific Incorporation into Oligo-DNA for Structural Studies via Relaxation Time Measurements	A. Földesi; T. V. Maltseva; J. Chattopadhyaya
1379-1380	Boranophosphate Nucleic Acids - A Versatile DNA Backbone	Vladimir Rait; Dmitri Sergueev; Jack Summers; Kaizhang He; Faqing Huang; Bozenna Krzyzanowska; Barbara Ramsay Shaw
1381-1382	2′-DMAOE RNA: Emerging Oligonucleotides with Promising Antisense Properties	Thazha P. Prakash; Andrew M. Kawasaki; Guillermo Vasquez; Allister S. Fraser; Martin D. Casper; P. Dan Cook; Muthiah Manoharan
1383-1384	NMI Linkage Modification Increases Potency and Stability of H-RAS Antisense Oligonucleotides	Lex M. Cowsert; Cara T. Ohashi; Balkrishen Bhat; Didier Peoc'h; Alice M. Symons; P. Dan Cook; Muthiah Manoharan
1385-1386	Synthesis of New Pseudonucleosides Containing Sulfamylated Derivatives of Natural Amino Acids as Aglycone	Nour-Eddine Aouf; Ouassila Attoui; Abdelghani Djahoudi
1387-1388	2′-Deoxy-2′(S)-ethynyl Oligonucleotides: Synthesis and Pairing Properties	Rolf Buff; Jürg Hunziker
1389-1390	Use of [4,6-Di-¹⁴C]-5′-DMT-thymidine Phosphoramidite Reagent for the Radiolabeling of Synthetic Oligonucleotides	Andrei Guzaev; Brunel Boyode; Guity Balow; Muthiah Manoharan
1391-1392	Synthesis of Chimerical Oligonucleotides Containing Internucleosidic Phosphodiester and S-Pivaloyl Mercaptoethyl Phosphotriester Linkages	Andrei Guzaev; Guity Balow; Muthiah Manoharan
1393-1396	Phosphonate Analogues of Peptide Nucleic Acids and Related Compounds: Synthesis and Hybridization Properties	V. A. Efimov; A. A. Buryakova; M. V. Choob; O. G. Chakhmakhcheva
1397-1398	A New Strategy for DNA Inhibition with Backbone Substituted DNA Analogues	H. M. Buck
1399-1400	8-Aza-7-deazapurine DNA: Synthesis and Duplex Stability of Oligonucleotides Containing 7-Substituted Bases	F. Seela; G. Becher; M. Zulauf
1401-1402	Synthesis of Oligodeoxynucleotides Containing 4′-C-Aminoalkyl-thymidines and Their Thermal Stability and Nuclease-Resistance Properties	Yoshihito Ueno; Makiko Kanazaki; Satoshi Shuto; Akira Matsuda
1403-1404	Synthesis and Biological Properties of 2′-5′ Oligodeoxyribonucleotide, an Isomer of Biologic DNA	Ramendra K. Sing; H. Takaku
1405-1406	Improvements in the Synthesis of L-Ribonucleosides for the Preparation of Mirror-Image Oligoribonucleotides	F. Santamaria; B. Rayner
1407-1408	γ-Aminobutyric Acid as Enzymolabile Groups for the Pro-oligonucleotide Approach	N. Mignet; F. Morvan; B. Rayner; J. L. Imbach
1409-1411	Conformationally Restrained Chiral PNA Conjugates: Synthesis and DNA Complementation Studies	B. P. Gangamani; M. Decosta; V. A. Kumar; K. N. Ganesh
1413-1415	Bicyclo[3.2.1]-DNA: A DNA Analog Containing a Rigid Backbone and a Flexible Base-Pairing Region	C. Roberts; C. Epple; C. Leumann
1417-1418	Elucidation of the Hydrolytical Properties of α-Hydroxybenzylphosphonates as a New Potential Pro-Oligonucleotide Concept	R. P. Mauritz; F. S. Schmelz; C. Meier
1419-1420	Synthesis, Hybridization, and Nuclease Resistance Properties of 2′-O-Aminooxyethyl Modified Oligonucleotides	Andrew M. Kawasaki; Martin D. Casper; Thazha P. Prakash; Sheri Manalili; Henri Sasmor; Muthiah Manoharan; P. Dan Cook

Volume 18, Issue 6-7 (1999)

1421-1422	Nucleic Acid Analog Peptide Containing β-Aminoalanine Modified with Nucleobases	Masayuki Fujii; Jinsai Hidaka
1423-1424	4′-Thio-RNA: Synthesis, Base Pairing Properties and Interaction with Dimerization Initiation Site of HIV-1	David Dukhan; Florence De Valette; Roland Marquet; Bernard Ehresmann; Chantal Ehresmann; François Morvan; Jean-Louis Barascut; Jean-Louis Imbach
1425-1426	Novel Oligonucleotide Analogues Derived From Serine and 4-Hydroxyproline	V. A. Efimov; M. V. Choob; A. A. Buryakova; O. G. Chakhmakhcheva
1427-1428	Synthesis and Properties of Some Morpholino Oligonucleotide Analogues	O. Chakhmakhcheva; M. Andrianov; A. Buryakova; M. Choob; V. Efimov
1429-1431	Oligonucleotides with 2,6-Diaminopurine Base Replacing for Adenine: Synthesis and Properties	V. Boudou; K. Rothenbacher; A. Van Aerschot; P. Herdewijn
1433-1434	The Prooligonucleotide Approach: Synthesis of Mixed SATE-Phosphotriester Phosphodiester Oligonucleotides	J. C. Bologna; G. Tosquellas; F. Morvan; B. Rayner; J. L. Imbach
1435-1436	Use of Photolabile Amino-Protecting Groups in the Synthesis of Base-Sensitive DNA SATE-Phosphotriesters	Karine Alvarez; Jean-Jacques Vasseur; Jean-Louis Imbach
1437-1438	Synthesis of Spirannic Nucleosides and Their Incorporation into Oligonucleotides	A. Renard; M. Kotera; J. Lhomme
1439-1440	7-Deaza-2′-deoxyguanosines Functionalized with 7-(ω-Aminoalk-1-YNYL) Residues	N. Ramzaeva; C. Mittelbach; F. Seela
1443-1448	Studies Towards the Synthesis of Peptide-Oligonucleotide Conjugates	Suzanne Peyrottes; Béatrice Mestre; Fabienne Burlina; Michael J. Gait
1449-1454	Synthesis of Polyaminooligonucleotides and Their Combinatorial Libraries	Wojciech T. Markiewicz; Przemysław Godzina; Maria Markiewicz
1455-1456	Synthesis of Oligonucleotide Conjugates with the Aid of N-Chloroacetamidohexyl Phosphoramidite Reagent	Andrei Guzaev; Muthiah Manoharan
1457-1458	Conversion of Unprotected Amino-Link Oligonucleotides into Their Tetramethylguanidinium Derivatives	B. Greiner; E. Uhlmann
1459-1461	Interaction of Complementary Oligonucleotides with the 3′-End of Yeast tRNA^PHE	V. Petyuk; M. Zenkova; R. Giege; V. Vlassov
1463-1465	Mechanism and Specificity of RNA Cleavage by Chemical Ribonucleases	N. Beloglazova; A. Vlassov; D. Konevetc; V. Sil'nikov; M. Zenkova; R. Giege; V. Vlassov
1467-1468	Synthesis of Oligonucleotides Bearing Polyamine Groups for Recognition of DNA Sequences	Pierre Potier; Abdennaji Adib; Alexeï Kochkine; Ivan Huc; Jean-Paul Behr
1469-1470	Oligonucleotides with Reactive Dialdehyde Groups as Novel Affinity Reagents	S. N. Mikhailov; B. S. Ermolinsky; E. V. Efimtseva; M. G. Brevnov; O. M. Gritsenko; E. S. Gromova; A. Van Aerschot; P. Herdewijn
1471-1472	Synthesis of Fully Protected Nucleoside- Folic Acid Conjugated Phosphoramidites and Their Incorporation into Antisense Oligonuleotides	Balkrishen Bhat; Guity Balow; Andrei Guzaev; P. Dan Cook; Muthiah Manoharan
1473-1476	A New Fluorescent Probe for Studies of Interactions Between Hydrophobic Oligonucleotides and Cellular Membranes	C. Gosse; A. S. Boutorine; L. Jullien; C. Hélène
1477-1478	Thermodynamic Melting Studies on Oligonucleotide-Peptide Conjugates	C. Frier; J. G. Harrison; S. Balasubramanian
1479-1481	Tc-99m-Labeling of Modified RNA	Christoph S. Hilger; Michael C. Willis; Mark Wolters; Wolfgang A. Pieken
1483-1484	Synthesis and Biological Activity of 2′,5′-Oligoadenylate Trimers Containing 5′-Terminal 5′-Amino-5′-deoxy- and 5′-Amino-3′,5′-dideoxyadenosine Derivatives	Evgeny I. Kvasyuk; Igor A. Mikhailopulo; Robert J. Suhadolnik; Earl E. Henderson; Nicholas F. Muto; Kathryn T. Iacono; Joseph Homon; Wolfgang Pfleiderer
1485-1486	2-5A-PNA Complexes: A Novel Class of Antisense Compounds	J. C. Verheijen; S. F. Bayly; M. R. Player; P. F. Torrence; G. A. van der Marel; J. H. Van Boom
1487-1488	Convenient Method for the Synthesis of DNA Conjugate	Masayuki Fujii; Taro Hasegawa; Shuji Takase; Koichiro Goto
1489-1490	Synthesis of Nucleopeptide-Oligonucleotide Conjugates	Natalia V. Sumbatyan; Elena A. Artsatbanova; Olga V. Baeva; Kwang-Chul Hyun; Svetlana A. Kuznetsova; Marina B. Gottikh; Galina A. Korshunova
1491-1492	Synthesis and Characterization of Artificial Ribonucleases	N. S. Zhdan; I. L. Kuznetsova; M. A. Zenkova; A. V. Vlassov; V. N. Silnikov; R. Giege; V. V. Vlassov
1493-1494	The Stepwise Solid-Phase Synthesis Methodology is Suitable for the Preparation of a Great Variety of Nucleopeptides	V. Marchán; L. Debéthune; M. Beltrán; J. Robles; I. Travesset; G. Fábregas; E. Pedroso; A. Grandas
1495-1496	Intercalating Insert into Internucleotide Linkages as Way for Stabilization and Detection of of Short DNA Duplexes	S. V. Kochetkova; E. I. Tishchenko; E. N. Timofeev; I. L. Shchaveleva; V. L. Florentiev
1497-1499	Conception, Preparation and Biological Evaluation of One Inhibitor of the HIV-1 Tat-TAR Complex	Sandrine Pairot; Audrey Farese-Di Giorgio; Christophe Di Giorgio; Nadia Patino; Roger Condom; Roger Guedj
1501-1502	Oligonucleotides Containing a 6-Substituted Pyrimidine Base: A Design for Myb Inhibitors	Atsushi Kittaka; Tetsuya Kuze; Hiromichi Tanaka; Tadashi Miyasaka; Kunihiko Hirose; Tadao Yoshida; Akinori Sarai; Takashi Yasukawa; Shunsuke Ishii

Volume 18, Issue 6-7 (1999)

1503-1505	Site-Specific RNA Cleavage Using Terpyridine·Cu(II)-Linked 2′-O-Methyloligonucleotides	Hideo Inoue; Masaki Shimizu; Takako Furukawa; Takashi Tamura; Miwa Matsui; Eiko Ohtsuka
1507-1511	Combinatorial Library of Artificial Ribonucleases	Dieter Hüsken; Andrea Deichert; Jonathan Hall; Robert Häner
1513-1514	Synthesis of New Photocross-Linking 5-C-Base-Substituted UTP Analogs and Their Application in Highly Selective Affinity Labelling of the Tick-Borne Encephalitis Virus RNA Replicase Proteins	O. V. Morozova; D. M. Kolpashchikov; T. M. Ivanova; T. S. Godovikova
1515-1516	Synthesis of New Oligonucleotide Derivatives with Porphyrins and Phthalocyanins	T. Abramova; T. Ivanova; V. Koval; O. Fedorova
1517-1518	Visible Light Activatable Binary System of Oligonucleotide Conjugates for Nucleic Acids Modification	M. I. Dobrikov; T. I. Gainutdinov; V. V. Vlassov
1519-1520	Structural Requirements at the 15.1–16.1 Position of the Hammerhead Ribozyme	J. Ludwig; M. Blaschke; M. Dunkel; B. Beijer; K. Ross; B. S. Sproat
1521-1522	Construction of a Modified Hairpin Ribozyme for Investigations of the Structure-Function Relationship	Yasuo Komatsu; Shigeko Yamashita; Eiko Ohtsuka
1523-1525	Using Fluorescence Resonance Energy Transfer (FRET) for Measuring 2-5A Analogues Ability to Activate RNase L	Hagen Cramer; Daniel A. Geselowitz; Paul F. Torrence
1527-1529	5′-C-Tosyloxyalkylnucleosides. Models for Oligonucleotide Coupling with Nucleophiles	V. Banuls; V. Sarramegna; C. Froment; J. M. Escudier; L. Gorrichon
1531-1533	A New Approach to the Synthesis of Trinucleotide Phosphoramidites - Synthons for the Generation of Oligonucleotide/Peptide Libraries	A. Kayushin; M. Korosteleva; A. Miroshnikov; W. Kosch; D. Zubov; N. Piel; W. Weichel; U. Krenz
1535-1538	Investigations on Sarcosine and Isonipecotic Acid Containing Peptide Nucleic Acids	T. Lescrinier; C. Hendrix; P. Herdewijn
1539-1540	Characterization of Oligonucleotide Sequence Isomers in Mixtures Using HPLC/MS	Jef Rozenski; James A. McCloskey
1543-1548	Parallel-Stranded DNA Formed by New Base Pairs Related to the Isoguanine-Cytosine or Isocytosine-Guanine Motifs	Frank Seela; Changfu Wei; Alexander Melenewski; Yang He; Rita Kröschel; Elisabeth Feiling
1549-1553	New Techniques for the Rapid Characterization of Oligonucleotides by Mass Spectrometry	J. A. McCloskey; A. B. Whitehill; J. Rozenski; F. Qiu; P. F. Crain
1555-1562	Parallel-Stranded Oligonucleotides with Alternating d(A-isoG)/d(T·C) and d(A·G)/d(T·m⁵isoC) Sequences	A. K. Shchyolkina; O. F. Borisova; T. M. Jovin
1563-1564	Glycerol-Furcated Oligonucleotides: Synthesis and Aggregation	H. Rosemeyer; E. Feiling; Wolfgang Nierling; F. Seela
1565-1566	Oligonucleotides Labeled by Fluorophores at the Sugar 2′-Positions for Fluorescence Energy Transfer Study of Nucleic Acid Structure	Kazushige Yamana; Tsuneo Mitsui
1567-1569	Crystal Structure of a Left-Handed Z-DNA Hexamer, d(CG)₃, Duplex Complexed with Synthetic Polyamine Reveals Binding of a Polyamine in the Minor Groove	Ken-Ichi Tomita; Hirofumi Ohishi; Isao Nakanishi; Toshio Hakoshima; Alexander Rich
1571-1573	The Computational Studies on the Conformation-Stabilizing Factors of the Left-Handed Z-DNA	Hirofumi Ohishi; Isao Nakanishi; Ken-Ichi Tomita; Tosimasa Ishida
1575-1576	Thermodynamics of Site-Specific Variant tRNA^Ala Acceptor Stem Microhairpins	Ewa Biala; William McClain; Peter Strazewski
1577-1578	Cytarabine-Induced Destabilization and Bending of a Model Okazaki Fragment	William H. Gmeiner; Alan Skradis; Richard T. Pon; Jinqian Liu
1579-1581	Nucleoside Modifications Affect the Structure and Stability of the Anticodon of tRNA^Lys,3	Darrell R. Davis; Philippe C. Durant
1583-1585	Four-Stranded Intercalated Cytosine-Rich Molecules: Novel Insights into DNA Structure and Stability	Imre Berger; Martin Egli; Nada Spackova; Jiri Sponer; Alexander Rich
1587-1592	Formation of Triple Helices at Irregular Poly (R·Y) Sites Located in Critical Positions in the Human BCR Promoter	L. E. Xodo; E. Del Terra; B. Scaggiante; G. Manzini; F. Quadrifoglio
1593-1596	A Single Carbocyclic Nucleotide Substitution in a 12mer DNA Gives a Hoogsteen Basepaired Duplex (Till 38°C) and a Hairpin (Till 65°C). A 600 MHz NMR Spectroscopic Study	J. Isaksson; T. Maltseva; P. Agback; X. Luo; A. Kumar; E. Zamaratski; J. Chattopadhyaya
1597-1598	Synthesis of 2′-Deoxy[5′-¹³C]Ribonucleotides and HMQC-Noesy NMR Study of the Dickerson's Dodecamer with ¹³C-Labeling at the 5′ Positions	Etsuko Kawashima; Takeshi Sekine; Kaoru Umabe; Yuhki Naito; Kazuo Kamaike; Chojiro Kojima; Toshimi Mizukoshi; Ei-Ichiro Suzuki; Yoshiharu Ishido
1599-1600	The Application of “The Uppsala NMR-Window” Concept for Conformational Analysis of Large DNA & RNA by High-Field NMR Spectroscopy	A. Földesi; T. V. Maltseva; J. Chattopadhyaya
1601-1602	Crystal and Solution Structure of the Bi-Loop Motif in Cyclic Octanucleotides	N. Escaja; E. Pedroso; S. A. Salisbury; C. Gonzàlez
1603-1607	NMR Structure of an Oligonucleotide Containing A Base Pair 3-(2-Hydroxyethyl) Deoxyuridine-Adenine	Y. Boulard; L. C. Sowers; G. V. Fazakerley
1609-1613	NMR Studies of Triplex Formation - Recognition of C•G Base Pairs by New Heterocyclic Systems	Florence Lecubin; Jean Louis Fourrey; Jian-Sheng Sun; R. Benhida

Volume 18, Issue 6-7 (1999)

1615-1616	Sequence-Specific Alkylation of DNA by Duocarmycin A and Its Novel Derivatives Bearing PY/IM Polyamides	Z. F. Tao; T. Fujiwara; I. Saito; H. Sugiyama
1617-1618	DNA Recognition by Non-Natural Oligonucleotides	Svetlana O. Doronina; Stéphanie Blanalt-Feidt; Jean-Paul Behr
1619-1621	Modified Oligonucleotides with Triple-Helix Stabilization Properties	Ramon Eritja; Elisenda Ferrer; Ramón Güimil García; Modesto Orozco
1623-1624	Enhancement of Stability of Double and Triple Stranded DNA by Cationic Amphiphilic α-Helix Peptide	Masayuki Fujii; Taro Hasegawa; Takuro Niidome; Haruhiko Aoyagi
1625-1627	Oligodeoxyxylonucleotides Form Stable Triplexes with Single-Stranded DNA	M. B. Gottikh; Y. I. Alekseev; A. V. Perminov; M. D. Pinskaya; Z. A. Shabarova
1629-1630	DNA Triple Helix Formation by N-Alkylphosphoramidate α-Oligonucleosides	A. Laurent; M. Naval; F. Debart; J. J. Vasseur; B. Rayner
1631-1632	Triplex Formation of α-Oligodeoxynucleotides Containing 5-Me-α-dC(N-4-Spermine)	A. Meyer; F. Morvan; B. Rayner; J. L. Imbach
1633-1637	Use of C5-Diamino-Substituted-Pyridine in Triple Helix Forming Oligonucleotides	J. Michel; S. Moreau
1639-1640	New 3′-3′ Linkers for Alternate Strand Triplex Forming Oligonucleotides	L. De Napoli; G. Di Fabio; A. Messere; D. Montesarchio; D. Musumeci; G. Piccialli
1641-1643	Selective Recognition of Triplex and Duplex Melting in Triple-Helical Nucleic Acids by Circular Dichroism Spectroscopy	Uwe Parsch; Karlheinz Wörner; Joachim W. Engels
1645-1646	Synthesis of Oligonucleotide-Intercalator Conjugates Capable to Inhibit HIV-1 DNA Integration	M. B. Gottikh; E. M. Volkov; E. A. Romanova; T. S. Oretskaya; Z. A. Shabarova
1647-1650	Binding of Chemically-Modified Oligonucleotides to the Double-Stranded Stem of an RNA Hairpin	Karine Aupeix; Jean-Jacques Toulmé
1651-1653	Relative Effects of Graft Copolymer and Polyamines on Triplex Stabilization Under Physiological Conditions	A. Ferdous; H. Watanabe; T. Akaike; A. Maruyama
1655-1656	Poly(L-Lysine)-Graft-Dextran Copolymer Remarkably Promotes Pyrimidine-Motif Triplex Formation at Neutral Ph: Thermodynamic and Kinetic Studies	H. Torigoe; A. Ferdous; H. Watanabe; T. Akaike; A. Maruyama
1657-1658	New Nucleobase Analogs for the Extension of the Triple Helix Recognition Code	David Lengeler; Klaus Weisz
1659-1660	Experimental and Theoretical Volumes of Nucleic Acids	L. M. Rellick; W. J. Becktel
1663-1664	The Concept of ‘Minimally Modified’ Antisense Oligonucleotides for Specific Inhibition of Gene Expression	E. Uhlmann; A. Peyman
1665-1666	Enzymatic Hydrolysis and Biological Activity of Oligonucleotides Containing 5-Substituted Pyrrmidine Bases	L. Ötvös; J. Sági; Gy. Sági; A. Szemzõ; F. D. Tóth; A. Jeney
1667-1668	Translation Arrest by RNase h Incompetent Antisense Oligonucleotides	I. Robbins; J. E. Gee; G. Mitta; B. Rayner; S. Vichier-guerre; M. Leng; A. van der Laan; J. van Boom; J. S. Nelson; B. Lebleu
1669-1671	Inhibition of DNA Transcription Elongation and Unwinding by Bis-Pna	L. Bastide; G. Villani; P. Nielsen; P. E. Boehmer; B. Lebleu
1673-1676	A 38 kDa Nuclear Protein Is Involved in the Retention of an Antisense Oligonucleotide Directed Against Cytosolic Phospholipase A2	C. Griffoni; E. Spisni; M. Orlandi; S. Santi; M. Riccio; V. Tomasi
1677-1679	Specifically Designed Polymeric Nanospheres Increase Cellular Uptake of Unmodified Antisense ODNs	Luisa Tondelli; Michele Laus; Alfredo Ricca; Gennaro Citro
1681-1682	Comb-Type Copolymers for Controlled DNA Delivery	A. Maruyama; A. Ferdous; T. Ishihara; S. Asayama; J. U. Park; M. Nogawa; H. Watanabe; Y. Takei; T. Akaike
1683-1684	Synthesis and Cellular Uptake of Fluorescently Labeled Oligodeoxynucleotide Prodrugs	C. Dell'aquila; E. Vives; J. L. Imbach; B. Rayner
1685-1688	In Vitro and In Vivo Anti-influenza A Virus Activity of Antisense Oligonucleotides	Takayuki Abe; Tadashi Mizuta; Shin-Ichi Suzuki; Toshifumi Hatta; Kazuyuki Takai; Tomoyuki Yokota; Hiroshi Takaku
1689-1691	Thermodynamic Studies on Hairpin Forming Antisense-Oligodeoxynucleotides Directed Against Hepatitis C Virus RNA	Thomas J. Lehmann; Stefan Eisenhardt; Joachim W. Engels
1693-1695	Activation of Spleen Lymphocytes by Plasmid DNA	E. Rykova; P. Laktionov; V. Vlassov
1697-1699	Uptake of Oligonucleotides by Keratinocytes	P. Laktionov; J-E Dazard; J. Piette; E. Vives; E. Rykova; V. Vlassov; B. Lebleu
1701-1704	Antisense Effects of Oligonucleotides Complementary to the Hairpin of the Leishmania Mini-exon RNA	Daniel Compagno; Jean-Jacques Toulmé
1705-1708	Antisense Oligodeoxynucleotide Complementary to CXCR4 mRNA Block Replication of HIV-1 in COS Cells	Akiko Kusunoki; Akira Wada; Naoko Kurosaki; Tohru Kimura; Kazuyuki Takai; Naoki Yamamoto; Hiroshi Takaku

Volume 18, Issue 6-7 (1999)

1709-1710	The Cytotoxicity of Anti-PAI-I Oligonucleotides and Their Conjugates	Anna Kobylańska; Elżbieta Pluskota; Zofia Pawtowska; Andrzej Okruszek; Czeslaw S. Cierniewski; Wojciech J. Stec
1711-1716	Effect of Oligomer Length and Base Substitutions on the Cytotoxic Activity and Specific Nuclear Protein Recognition of GTn Oligonucleotides in the Human Leukemic CCRF-CEM Cell Line	Carla Morassutti; Barbara Dapas; Bruna Scaggiante; Gabriela Paroni; Luigi Xodo; Franco Quadrifoglio
1717-1718	Inhibition of HIV-1 Integration by Mono- & Bifunctionalized Triple Helix Forming Oligonucleotides	Priscille Brodin; Marina Gottikh; Christian Auclair; Jean-François Mouscadet
1719-1720	Protein and RNA of Human Telomerase as Targets for Modified Oligonucleotides	M. von Janta-lipinski; K. Gaertner; C. Lehmann; H. Scheer; J. Schildt; E. Matthes
1721-1722	Uptake and Intracellular Distribution of Oligonucleotides Vectorized by a PAMAM Dendrimer	Valérie Hélin; Marina Gottikh; Zohar Mishal; Frédéric Subra; Claude Malvy; Marc Lavignon
1723-1725	Biological Properties of Antisense Oligonucleotides Conjugated to Different High-Molecular Mass Poly(Ethylen Glycols)	G. M. Bonora; E. Ivanova; N. Komarova; D. Pishiniyi; P. Vorobjev; V. Zarytova; S. Zaramella; F. M. Veronese
1727-1728	Synthesis of Fluorescent Cationic Lipids for Evaluation of Cellular Pathways and Delivery Mechanisms of Antisense Oligonucleotides	Balkrishen Bhat; Normand Heber't; Eric G. Marcusson; Nicholas M. Dean; C. Frank Bennett; Muthiah Manoharan
1729-1730	Cytotoxicity and In Vivo Tolerance of FdUMP[10]: A Novel Pro-Drug of the TS Inhibitory Nucleotide FdUMP	William H. Gmeiner; Alan Skradis; Richard T. Pon; Jinqian Liu
1731-1733	In Vivo Imaging and Pharmacokinetics of Oligonucleotides	Stéphana Marzabal; S. Terrazzino; B. Kühnast; F. Dollé; J. R. Deverre; A. Jobert; C. Crouzel; L. Di Giamberardino; B. Tavitian
1737-1746	Carbohydrate Modifications in Antisense Oligonucleotide Therapy: New Kids on the Block	Muthiah Manoharan; Andrew M. Kawasaki; Thazha P. Prakash; Allister S. Fraser; Marija Prhavc; Gopal B. Inamati; Martin D. Casper; P. Dan Cook
1747-1748	Synthesis of Modified Thiopurine Nucleosides for Structural Characterization of Human Thiopurine S-Methyltransferase	Galina A. Korshunova; Eugene Y. Krynetski; Manana T. Mtchedlidze; Denis V. Agapkin; William E. Evans; Natalia F. Krynetskaia

Volume 18, Issue 4-5 (1999)

a	Editorial board page for “Nucleosides, Nucleotides & Nucleic Acids”, Volume 18, Number 4-5
xxxix-xl	Preface	Gilles Gosselin
509-519	Studies Designed to Increase the Stability and Antiviral Activity (HCMV) of the Active Benzimidazole Nucleoside, TCRB	Leroy B. Townsend; Kristjan S. Gudmundsson; Susan M. Daluge; Jiong J. Chen; Zhijian Zhu; George W. Koszalka; Leslie Boyd; Stanley D. Chamberlain; George A. Freeman; Karen K. Biron; John C. Drach
521-530	Conformationally Restricted Nucleosides. The Reaction of Adenosine Deaminase with Substrates Built on a Bicyclo[3.1.0]hexane Template	Victor E. Marquez; Pamela Russ; Randolph Alonso; Maqbool A. Siddiqui; Kye-Jung Shin; Clifford George; Marc C. Nicklaus; Fang Dai; Harry Ford Jr.
531-536	Conformationally Locked Nucleoside Analogs. Synthesis of 2′-Deoxy-2′-C, 4′-C-Bridged Bicyclic Nucleosides	Guangyi Wang; Esmir Gunic
537-540	New Classes of Fluorinated L-Nucleosides; Synthesis and Antiviral Activity	Kyeong Lee; Yongseok Choi; Joon H. Hong; Raymond F. Schinazi; Chung K. Chu
541-546	Synthesis and Testing of New Modified Nucleosides	Michael E. Jung; Christopher J. Nichols; Oliver Kretschik; Yue Xu
547-553	Mechanistic and Synthetic Aspects of the C-1′ Radicals in Modified Nucleosides	Chryssostomos Chatgilialoglu
555-556	Recent Advances in the Synthesis of 6-Vinyl-N,N-Dialkylcytosine Derivatives	Maurizio Botta; Raffaele Saladino; Luigi Stasi; Umberto Ciambecchini; Rosario Nicoletti
557-558	A Novel Approach for the Synthesis of seco C-Nucleoside Analogues	Laila F. Awad; El Sayed H. El Ashry
559-563	Simple and Stereoselective Syntheses of Nucleoside Analogues with a Benzo[c]furan Glycone Moiety	David F. Ewing; Noureddine Fahmi; Grahame Mackenzie; Alessandra Pranzo
565-567	A Convenient Approach to N-3 Alkylation of 9-Substituted Guanines	Tomasz Ostrowski; Joanna Zeidler; Tomasz Goelizski; Bozenna Golankiewicz
569-570	A New Series of Mechanism-Based Inhibitors of S-Adenosyl-L-Homocysteine Hydrolase from Beef Liver	Corinne Vandenplas; Danielle Guillerm; Georges Guillerm
571-572	Synthesis and Antiviral Activity of L-2′-Deoxy-2′-up-fluoro-4′-thionucleosides	Lak Shin Jeong; Hyung Ryong Moon; Su Jeong Yoo; Sun Nan Lee; Hee-Doo Kim; Moon Woo Chun
573-574	Synthesis and Polymerase Incorporation Properties of a Tricyclic Pyrrolopyrimidine Related to N⁶-Hydroxy-2′-deoxyadenosine	F. Hill; D. Loakes; C. L. Smith; D. M. Williams; D. M. Brown
575-576	Synthesis and Biological Evaluation of New Enantiomers of 5-O-Carboranyl Pyrimidine Nucleosides	Nicolas Mourier; Alessandra Eleuteri; Raymond F. Schinazi
577-579	Synthesis of Novel Isomeric Dideoxydidehydronucleosides	Vasu Nair; Sanjib Bera; Travis Mickle; Serge Van Calenbergh
581-583	Synthesis of Isoxazolidino Analogues of 2′,3′-Dideoxynucleosides	Evelina Colacino; Antonella Converso; Antonio De Nino; Antonella Leggio; Angelo Liguori; Loredana Maiuolo; Anna Napoli; Antonio Procopio; Carlo Siciliano; Giovanni Sindona
585-586	Lithiation-Stannylation Chemistry of Nucleosides	Hiromichi Tanaka; Hiroki Kumamoto; Satoru Shindoh; Hiroyuki Hayakawa; Keisuke Kato; Tadashi Miyasaka
587-590	Coupling of 2,6-Dichloropurine and 2,6-Dichlorodeazapurines with Ribose and Ribose Modified Sugars	S. Vittori; E. Camaioni; S. Costanzi; R. Volpini; G. Cristalli
591-592	A Novel and Enantioselective Approach to the Synthesis of Cyclohexane Carbocyclic Nucleosides Starting from (-)-Carvone	Jing Wang; Piet Herdewijn
593-594	Enantioselective Synthesis and Conformational Analysis of Cyclohexene Carbocyclic Nucleosides	Jing Wang; Piet Herdewijn
595-596	Design and Biological Evaluation of New Mechanismbased Inhibitors of S-Adenosyl-L-homocysteine Hydrolase	Stanislaw F. Wnuk; Chong-Sheng Yuan; Ronald T. Borchardt; J. Robins Morris
597-598	Methylenecyclopropane Analogues of Nucleosides: Synthesis, Absolute Configuration, and Enantioselectivity of Antiviral Effect of (R)-(-)- and (S)-( )-Synadenol	Y-L. Qiu; A. Hempel; N. Camerman; A. Camerman; F. Geiser; R. G. Ptak; J. M. Breitenbach; T. Kira; L. Li; E. Gullen; Y-C. Cheng; J. C. Drach; J. Zemlicka
599-600	Synthesis of 5′-Thioalkyl, Sulfoxide and Sulfone Pyrimidine Nucleosides	L. A. Agrofoglio; F. Girard; F. Fleury; S. Léonce
601-602	Stereoselective Synthesis of Carbocyclic α-L-Homonucleosides	L. A. Agrofoglio; F. Girard; C. Demaison; M-G. Lee; P. Roingeard; A. Fridland
603-604	Efficient Stereoselective Synthesis of New C-Nucleosides via Intramolecular Mitsunobu Cyclization	R. Benhida; D. Guianvarch; J-L. Fourrey; J. S. Sun
605-606	Synthesis of Non-Natural Pyrimidine Nucleosides	Stephanie Blanalt-feidt; Svetlana O. Doronina; Jean-Paul Behr
607-609	A New and Convenient Approach for the Synthesis of Ribo- and 2′-Deoxyribo-β-L-Furanonucleosides Starting From β-L-Xylofuranonucleosides	V. Boudou; G. Gosselin; J-L. Imbach

Volume 18, Issue 4-5 (1999)

611-612	Synthesis of a C-8 Modified Adenosine Analogue as a Potential Mechanistic Probe for Ribonucleotide Reductases	G. C. Magnin; J. Dauvergne; A. Burger; J-F. Biellmann
613-614	Synthesis and Biological Activity of 5-Azacytosine Nucleosides Derived from 4-Thio-2-Deoxy-L-threo-Pentofuranose and 4-Thio-2-Deoxy-D-erythro-Pentofuranose	Loredana Cappellacci; Kamal N. Tiwari; John A. Montgomery; John A. Secrist III
615-616	Synthesis and Antiviral Activities of 1,3-Oxathiolanyl Nucleosides with 5-Hydroxymethyl Substituent	Moon Woo Chun; Sung Pil Choi; Myong Jung Kim; Chol Joon Bae; Hyung Ryong Moon; Hee-Doo Kim; Lak Shin Jeong
617-618	Synthesis of L-Sangivamycin and Toyocamycin Analogues and Their Inhibitory Activities of SER/THR Protein Kinases	Moon Woo Chun; Dae Hong Shin; Sun Yong Song; Yong Hee Lee; Chul Hoon Lee; Lak Shin Jeong; Seung Ki Lee
619-620	As-Triazine Derivatives with Potential Therapeutic Action XXVII. Synthesis of 5-[Alkyl-(ethoxycarbonyl)methyl]mercapto-6-azauridines	Francisc Czobor; Carol Cristescu
621-622	Synthesis of Novel Pyrene-Bearing C-Nucleoside and Its Incorporation into Oligonucleotides	Natalia Dyatkina; Alexander Khorlin; Yuri Khrlin; Kyoichi A. Watanabe
623-624	Synthesis of O-β-D-Ribofuranosyl-(1″-2′)-adenosine-5″-O-phosphate	Andrei A. Rodionov; Ekaterina V. Efimtseva; Sergey N. Mikhailov
625-626	Synthesis of (±)-cis-3-Aminomethyl-1-indanylmethanol as a Precursor of Carbocyclic Analogues of Nucleosides	M. Escobar; F. Fernández; X. García-Mera; J. E. Rodriguez-Borges
627-632	Configuration and Conformation Studies of Nucleoside Analogues Based on the Benzo[c]furan Core	D. F. Ewing; N. Fahmi; G. Mackenzie; A. Pranzo
633-634	3′-(N-Hydroxyimino)-2′,3-dideoxynucleosides and Their Derivatives: Synthesis, Broad Spectrum Antiviral Properties and Synthetical Application for the Preparation of Other Nucleoside Analogues	I. Fedorov; E. Kazmina; M. Jasko; J. Balzarini; E. De Clercq; J-P. Sommadossi; J-L. Imbach; G. Gosselin
635-636	Synthesis, Conformation and Biological Properties of Selenonucleosides	Krzysztof Felczak; Agnieszka Miazga; Barbara Golos; Wojciech Rode; David Shugar; Tadeusz Kulikowski
637-639	Ex-Novo and Revisum Procedures for the Preparation of C-1′ Branched Nucleosides	C. Chatgilialoglu; C. Costantino; C. Ferreri; T. Gimisis; A. Romagnoli; R. Romeo
641-642	Synthesis of Novel Carbocyclic Nucleosides with a Modified Cyclopentane Ring and Evaluation of Their Antiviral Activity	Isabel Nieto; M. José Figueira; J. Manuel Blanco; Olga Caamaño; Franco Fernández; Erik De Clercq; Jan Balzarini
643-644	Stereospecific Synthesis and Antiviral Activities of β-L-2′,3′-Dideoxy-5-chloropyrimidine Nucleoside Derivatives	C. Pierra; G. Gosselin; J-P. Sommadossi; A. Faraj; E. De Clercq; J. Balzarini; J-L. Imbach
645-648	Synthesis of cis-Disubstituted Cyclobutenyl Nucleoside Analogues	M-E. Gourdel-Martin; F. Huet
649-650	Novel Types of Spin Labelled Nucleoside Analogues	J. M. J. Tronchet; M. Zsély; E. Grand; N. Laroze; M. Iznaden; M. Sollini; M. Geoffroy
651-652	A Versatile Synthesis of Enantiomerically Pure D- and L-Pyranosyl Nucleoside Analogues	Romualdo Caputo; Annalisa Guaragna; Giovanni Palumbo; Silvana Pedatella
653-654	An Economical Synthesis of Famciclovir	Toyoto Hijiya; Keizo Yamashita; Mitsuhiko Kojima; Yumiko Uchida; Satoshi Katayama; Takayoshi Torii; Hiroshi Shiragami; Kunisuke Izawa
655-656	Synthesis and Antiviral Activity of D- and L-Isodideoxy Nucleosides with Exocyclic Methylene	Lak Shin Jeong; Su Jeong Yoo; Hyung Ryong Moon; Moon Woo Chun; Chong-Kyo Lee
657-658	Synthesis of Nucleosides Having Unusual Branched Sugars as Potential Antiviral Agents	Kuniki Kato; Shosuke Yamamura
659-660	Solution Phase Combinatorial Chemistry. Purine- and Pyrimidine-Based Libraries with Antibacterial Activity via Solution Phase Simultaneous Addition of Functionalities	Andrew M. Kawasaki; Martin D. Casper; Hans J. Gaus; Rigo Herrmann; Richard H. Griffey; P. Dan Cook
661-671	Synthesis of N-Aryl Uracils and Hypoxanthines and Their Biological Properties	Tokumi Maruyama; Shigetada Kozai; Mayuko Uchida
673-674	Synthesis of Alkenyl Acyclonucleosides Derivatives of 5-Halogenouracil as Antiviral and Antitumoral Agents	A. Rochdi; M. Taourirte; N. Redwane; H. B. Lazrek; J. L. Barascut; J. L. Imbach
675-676	Novel TSAO Derivatives Modified at Positions 3′ and 4′ Of the Spiro Moiety	E. Lobatón; S. Velázquez; A. San-Félix; C. Chamorro; V. Tuñón; A. Esteban-gamboa; E. De Clercq; J. Balzarini; M. J. Camarasa; M. J. Pérez-Pérez
677-678	Triazole and Imidazole Reversed Nucleosides of L-Idose and D-Glucose	L. Vanbaelinghem; P. Martin; D. Postel; G. Goethals; D. F. Ewing; G. Mackenzie; G. Ronco; P. Villa
679-680	Structure-Activity Relationships of Tiazofurin Analogs: Synthesis and Computational Studies of 4′-Thio Derivatives of Thiophenfurin and Furanfurin	P. Franchetti; S. Marchetti; L. Cappellacci; M. Grifantini; B. M. Goldstein; D. Dukhan; J-L. Barascut; J-L. Imbach
681-682	Potential Inhibitors of HIV Integrase	Christophe Mathe; Vasu Nair
683-685	Synthesis and Biological Activity of 4′-Thio-2′-deoxy Purine Nucleosides	Lea Messini; Kamal N. Tiwari; John A. Montgomery; John A. Secrist III
687-688	Chemical and Enzymatic Synthesis and Antiviral Properties of 2′-Deoxy-2′-fluoroguanosine	Galina V. Zaitseva; Anatoli I. Zinchenko; Vladimir N. Barai; N. I. Pavlova; Evgeny I. Boreko; Igor A. Mikhailopulo
689-690	A Novel Route for the Synthesis of Fluorodeoxy Sugars and Nucleosides	Igor A. Mikhailopulo; Grigorii G. Sivets; Natalia B. Khripach

Volume 18, Issue 4-5 (1999)

691-692	Studies on Disaccharide Nucleoside Synthesis. Mechanism of the Formation of Trisaccharide Purine Nucleosides	Sergey N. Mikhailov; Andrei A. Rodionov; Ekaterina V. Efimtseva; Boris S. Ermolinsky; Marina V. Fomitcheva; Nelly Sh. Padyukova; Klaus Rothenbacher; Eveline Lescrinier; Piet Herdewijn
693-695	L-R_{ibonucleosides for} R_acemic RNA	E. Moyroud; O. Botta; P. Strazewski
697-699	A Serendipitous Synthesis of 8-Dimsyl-2′-deoxyguanosine	Satyam Nampalli; Inna Livshin; Shiv Kumar
701-702	A New Synthetic Approach Towards α- and β-LNA (Locked Nucleic Acids)	Poul Nielsen; Jesper Wengel
703-705	5-Fluoro-1-(3,4-dideoxy-3-fluoro-6-0-trityl-beta-D-glycero-hex-3-eno-pyranos-2-ulosyl (Uracil): Anticancer Agent	Abraham P. Ollapally; Ismet Bennouna-dorange; Thomas L. Whitaker Jr.
707-708	“Mixed Inhibitors” of HIV-Reverse Transcriptase: Synthesis and Antiviral Activity	R. Pontikis; R. Note; E. Dechaux; J. Guillaumel; A-M. Aubertin; D. S. Grierson; C. Monneret
709-711	Synthesis and Molecular Modeling of Novel HSV1 Uracil-DNA Glycosylase Inhibitors	M. Pregnolato; D. Ubiali; A. Verri; F. Focher; S. Spadari; H. Sun; C. Zhi; G. E. Wright
713-714	Synthesis and Inhibitory Activity Against Phosphatidylinositol 4-Kinase of Echiguanine Analogs	Yoshio Saito; Kuniki Kato; Kazuo Umezawa
715-716	Unexpected Results in the Reaction of 5′-Tosyl TSAO-m³T With Amines	C. Chamorro; S. Velázquez; M. L. Jimeno; M. J. Pérez-Pérez; E. Lobatón; V. Tuñón; A. Esteban-gamboa; F. Gago; E. De Clercq; J. Balzarini; M. J. Camarasa; A. San-Félix
717-719	Synthesis of New Fluorescent Nucleoside Analogues and Application to the Study of Human Deoxycytidine Kinase	M. Shafiee; G. Gosselin; J-L. Imbach; S. Eriksson; G. Maury
721-723	Synthesis of an Alanyl Adenosine Analog	Oliver Botta; Peter Strazewski
725-726	Nucleoside Analogues of Purine with a 1,2-Disubstituted Cyclopentene Ring	P. Besada; C. Terán; L. Santana; M. Teijeira; E. Uriarte
727-729	Synthesis of Peptide Nucleic Acid Monomers	L. Kovács; Z. Timár; B. Penke
731-732	Synthesis of Some Fully 3′ and 4′-C-Branched-Chain Sugar Nucleoside Analogues	T. Ton-That
733-734	Synthesis and Biological Evaluation of 1,2-Disubstituted Carbonucleosides of 6-Substituted Purine and 8-Azapurine	L. Santana; M. Teijeira; E. Uriarte; C. Terán; G. Andrei; R. Snoeck; J. Balzarini; E. De Clercq
735-736	Lead Optimization of N⁶-Cyclopentyl-3′-amido-3′-deoxyxylofuranosyladenines as Adenosine A₁ Receptor Antagonists	S. Van Calenbergh; A. Link; D. De Keukeleire; P. Herdewijn
737-738	Synthesis of a Nucleoside Bioconjugate System as a Potential Anti-HIV Agent	Serge Van Calenbergh; Vasu Nair
739-740	Synthesis and Receptor Affinity of Polysubstituted Adenosines	S. Vittori; E. Camaioni; S. Costanzi; R. Volpini; K-N. Klotz; G. Cristalli
741-742	Structure-Activity Relationships of Adenosine Deaminase Inhibitors	S. Vittori; E. Camaioni; S. Costanzi; R. Volpini; G. Lupidi; G. Cristalli
745-757	Gene Therapy of Cancer: Activation of Nucleoside Prodrugs with E. coli Purine Nucleoside Phosphorylase	John A. Secrist III; William B. Parker; Paula W. Allan; L. Lee Bennett Jr.; William R. Waud; Jackie W. Truss; Anita T. Fowler; John A. Montgomery; Steven E. Ealick; Alan H. Wells; G. Yancey Gillespie; V. K. Gadi; Eric J. Sorscher
759-771	Antitumor Potential of Acyclic Nucleoside Phosphonates	E. De Clercq; G. Andrei; J. Balzarini; S. Hatse; S. Liekens; L. Naesens; J. Neyts; R. Snoeck
773-778	Resistance Profiles of ( ) 2′-Deoxy-3′-oxa-4′-thiocytidine and (-) 2′-Deoxy-3′-oxa-4′-thio-5-fluorocytidine	Nathalie Richard; Horacio Salomon; Maureen Oliveira; Robert Rando; Mark A. Wainberg
779-793	Mechanism-Based Inhibition of Ribonucleotide Reductases: New Mechanistic Considerations and Promising Biological Applications	Morris J. Robins
795-805	Structural Determinants of HIV-1 Reverse Transcriptase Stereoselectivity Towards (β)-L-Deoxy- and Dideoxy-Pyrimidine Nucleoside Triphosphates: Molecular Basis for the Combination of L-Dideoxynucleoside Analogs with Non-nucleoside Inhibitors in Anti HIV Chemotherapy	G. Maga; M. Amacker; U. Hübscher; G. Gosselin; J-L. Imbach; C. Mathé; A. Faraj; J. P. Sommadossi; S. Spadari
807-810	The Enantioselectivity of the Cellular Deoxynucleoside Kinases	Jianghai Wang; Jyoti Chattopadhyaya; Staffan Eriksson
811-814	A New Antitumor Nucleoside, 1-(3-C-Ethynyl-β-_d-ribo-pentofuranosyl)-cytosine (ECyd), Is a Potent Inhibitor of RNA Synthesis	Akira Matsuda; Masakazu Fukushima; Yusuke Wataya; Takuma Sasaki
815-820	Synthetic Studies on 2′-Substituted-4′-thiocytidine Derivatives as Antineoplastic Agents	Yuichi Yoshimura; Mikari Endo; Kenji Kitano; Kohei Yamada; Shinji Sakata; Shinji Miura; Haruhiko Machida
821-827	Design and SAR Study of a Novel Class of Nucleotide Analogues as Potent Anti-HCMV Agents	N. Nguyen-ba; L. Chan; M. Quimpère; N. Turcotte; N. Lee; H. Mitchell; J. Bédard
829-830	Phosphorylation of Anti-HIV Nucleoside Analogs by Nucleoside Diphosphate Kinase	Benoit Schneider; Yingwu Xu; Olivier Sellam; Robert Sarfati; Joel Janin; Michel Véron; Dominique Deville-bonne
831-834	Distinct Inhibitory Effects of 2-Chloro-2′-deoxyadenosine and 9-β-D-Arabinosyl-2-fluoroadenine on DNA Methyltransferase in Human T-Lymphocytes	Dorota Wyczechowska; Katarzyna Ruckemann; John A. Duley; Anne H. Simmonds; Krystyna Fabianowska-majewska

Volume 18, Issue 4-5 (1999)

835-836	Investigations into Biochemical Mode of Inhibition of Guanase by Azepinomycin: Synthesis and Biochemical Screening of Several Analogues of Azepinomycin	Vasanthakumar P. Rajappan; Ramachandra S. Hosmane
837-838	Potent Anti-hepatitis B Viral Activity and Inhibition of Bacteriophage T7 RNA Polymerase by a “Fat” Nucleoside and Its 5′-Triphosphate Derivative: Synthetic, Biochemical, and Biological Studies of 4,8-Diamino-6-imino-6h-1-β-D-ribofuranosylimidazo[4,5-E][1,3]diazepine-5′-triphosphate	Maria Bretner; Dorothy Beckett; Ramachandra S. Hosmane
839-842	Enzymatic Preparation of ³²P-Labeled β-L-2′, 3′-dd-5′ ATP and Its Use as a High-Affinity, Conformation-Specific Ligand for Labeling Adenylyl Cyclases	Roger A. Johnson; Ilana Shoshani; Carmen Dessauer; Gilles Gosselin
843-844	A New Look at the Molecular Mechanism of Thymidylate Synthase and Its Interaction with Nucleotide Analogues	T. I. Kalman; D. A. Matthews
845-846	Mechanistic Similarities Between Thymidylate Synthase and IMP Dehydrogenase: A Common Strategy of Catalysis	T. I. Kalman
847-848	Mechanism of Inhibition of HIV Reverse Transcriptase by 1-(2-Deoxy-β-_d-ribofuranosyl)-4-acetylimidazolin-2-one (Imidine)	T. I. Kalman; K. Sen; X-J. Jiang
849-851	Effect of Acyclic Nucleoside Phosphonates on the HIV-1 Integrase in Vitro	G. Abu Sheika; E. Tramontano; A. G. Loi; P. Franchetti; M. Grifantini; P. La Colla
853-855	Pyrimidine Nucleotidases/Phosphotransferases from Human Erythrocyte	A. Amici; M. Emanuelli; N. Raffaelli; S. Ruggieri; G. Magni
857-860	Derivatives of L-Adenosine and L-Guanosine as Substrates for Human Deoxycytidine Kinase	G. Gaubert; G. Gosselin; J-L. Imbach; S. Eriksson; G. Maury
861-862	On The Catalytic Mechanism of Adenosylhomocysteine/Methylthioadenosine Nucleosidase From E. coli.	Brigitte Allart; Danielle Guillerm; Georges Guillerm
863-864	Reasons and Limits of Substrate Activity of Modified L-dNTP in DNA Biosynthesis	Alexander A. Krayevsky; Natalya B. Dyatkina; Dmitry G. Semizarov; Liubov S. Victorova; Elena A. Shirokova; Fritz Theil; Martin Von Janta Lipinski; Gilles Gosselin; Jean-Louis Imbach
865-866	Investigation of the Ternary Complex Formed Between Recombinant Rat Hepatoma Thymidylate Synthase, FdUMP op S⁴FdUMP and N⁵, N¹⁰-Methylenetetrahydrofolate with the Use of ¹H AND ¹⁹F NMR	W. Szeszkowski; J. Cieśla; R. Stolarski; W. Rode; T. Kulikowski
867-869	Interaction of β-L-Adenosine-5′-triphosphate (L-ATP) with Human Deoxycytidine Kinase, Human DNA Primase and T4 DNA Ligase: Does the Chance Direct Enzymatic Enantioselectivity?	A. Verri; A. Montecucco; G. Gosselin; V. Boudou; S. Spadari; J-L. Imbach; F. Focher
871-872	Binding of Substrates by Purine Nucleoside Phosphorylase (PNP) from Cellulomonas Sp. - Kinetic and Spectrofluorimetric Studies	B. Wielgus-kutrowska; J. Tebbe; J. Wierzchowski; D. Shugar; W. Saenger; G. Koellner; A. Bzowska
873-874	Synthesis of 2-Chloro-6-aryloxy- and 2-Chloro-6-alkoxyarylpurines and Their Properties in the Purine Nucleoside Phosphorylase (PNP) System	A. Bzowska; L. Magnowska; B. Wielgus-kutrowska; Z. Kazimierczuk
875-876	Interactions of Calf Spleen Purine Nucleoside Phosphorylase with Antiviral Acyclic Nucleoside Phosphonate Inhibitors: Kinetics and Emission Studies	J. Wierzchowski; E. Kulikowska; A. Bzowska; A. Holy; L. Magnowska; D. Shugar
877-878	Cell Specific Cytotoxicity and Structure-Activity Relationship of Lipophilic 1-B-D-Arabinofuranosylcytosine (Ara-C) Derivatives	G. J. Peters; D. A. Voorn; C. M. Kuiper; C. Van Der Wilt; P. Noordhuis; K. Smid; F. Myhren; M. Sandvold; H. R. Hendriks
879-880	Synthesis and Biological Evaluation of Polyaminated 2′,3′-Dideoxy-3′-thiacytidine Prodrugs	M. Camplo; N. Mourier; J-C Chermann; J-L Kraus
881-882	New Polyazamacrocycle-Nucleoside Conjugates: Synthesis, Anti-HIV Evaluation and Interaction with CXCR-4 Coreceptor	Jean Dessolin; Pascale Galéa; Patrick Vlieghe; Jean-Claude Chermann; Jean-Louis Kraus
883-884	Synthesis of Novel C-5 Substituted d4t Analogues Bearing Linker Arms as Potential Anti-HIV Agents	D. Ladurée; C. Fossey; M. Renoud-grappin; G. Fontaine; F. Camara; D. Gavriliu; A. Ciurea; A. M. Aubertin; A. Kirn
885-889	L-Purine Nucleosides as Selective Antimalarials	Annette M. Gero; Gabriel Perrone; David M. Brown; Simone T. Hall; Chung K. Chu
891-892	Anti-HIV-1 Activities of 1,3-Dioxolane Guanine and 2,6-Diaminopurine Dioxolane	Zhengxian Gu; Mark A. Wainberg; Paul Nguyen-ba; Lucille L'Heureux; Jean-Marc De Muys; Robert F. Rando
893-896	Quantification of Lamivudine (3TC) by Competitive Immunoassay	Fatima Akeb; Christophe Creminon; Marie-Claire Nevers; Jacques Grassi; Danièle Duval; Roger Guedj
897-898	Biological Activity of 1-Deazapurine Nucleosides: Role of Deoxycytidine Kinase?	AM. Bergman; G. Cristalli; S. Vittori; J. Wang; S. Eriksson; Gj Peters
901-906	Antiviral Activity and Resistance Profile of Phosphazid - A Novel Prodrug of AZT	John Machado; Horacio Salomon; Maureen Oliveira; Christos Tsoukas; Alexander A. Krayevsky; Mark A. Wainberg
907-912	CycloSal-2′-ara (ribo)-fluoro-2′,3′-dideoxyadenosine Monophosphates—An Effort to Solve the Structure-Activity Relationship of 2′-Fluoro-dda	C. Meier; T. Knispel; V. E. Marquez; E. De Clercq; J. Balzarini
913-919	Antiviral Nucleoside Drug Delivery via Amino Acid Phosphoramidates	Carston R. Wagner; Shu-Ling Chang; George W. Griesgraber; Heng Song; Edward J. McIntee; Cheryl L. Zimmerman
921-926	DDC- and 3TC-bis(SATE) Monophosphate Prodrugs Overcome Cellular Resistance Mechanisms to HIV-1 Associated with Cytidine Kinase Deficiency	B. Gröschel; N. Himmel; J. Cinatl; C. Périgaud; G. Gosselin; J-L. Imbach; H. W. Doerr; J. Cinatl Jr.
927-932	Novel Mycophenolic Adenine bis(Phosphonate)S as Potent Anticancer Agents and Inducers of Cells Differentiation	Krzysztof W. Pankiewicz; Krystyna Lesiak-watanabe
933-936	Effects of cycloSal-D4TMP Derivatives in H9 Cells with Induced AZT Resistance Phenotype	B. Gröschel; C. Meier; R. Zehner; J. Cinatl; H. W. Doerr; J. Cinatl Jr.

Volume 18, Issue 4-5 (1999)

937-938	Aryl Nucleoside H-Phosphonates—Novel Derivatives of Controlled Reactivity	J. Cieślak; J. Jankowska; M. Szymczak; A. Kers; I. Kers; J. Stawiński; A. Kraszewski
939-940	Synthesis of Analogues of 5′-Mono-,5′-Di-, and 5′-Triphosphate-AZT for the Development of Specific Enzyme Immunoassay for Monitoring of Intracellular Levels of AZT-MP, AZT-DP, and AZT-TP	T. Brossette; M-C. Nevers; C. Creminon; C. Mioskowski; J. Grassi; L. Lebeau
941-942	Phosphoramidite Chemistry for the Synthesis of cycloSal-Pro-Nucleotides	Florence Mugnier; Chris Meier
943-944	Evidence for Cyclophosphate Formation During Hydrolysis of 3-Methyl-cycloSal-PCVMP	Andreas Lomp; Chris Meier; Markus Herderich; Peter Wutzler
945-946	N,O-Selectivity in the Synthesis of 3-Me-CycloSal-ddAMP	Tina Knispel; Chris Meier
947-948	A New Cyclic Phosphoramidate D4T Prodrug Approach cycloAmb-D4T-Phosphoramidates	Martina Lorey; Chris Meier
949-950	Synthesis, In Vitro Anti-HIV and Anti-hepatitis B Activities and Pharmacokinetic Properties of Amphiphilic Heterodinucleoside Phosphates Containing ddC and AZT	R. A. Schwendener; P. A. Peghini; P. S. Ludwig; H. Schott
951-953	Synthesis of Nucleoside 3′-Thiophosphates in One Step Procedure	Maciej B. Szczepanik; Laurent Désaubry; Roger A. Johnson
955-958	Anti-inflammatory Effects of Phosphonomethoxyethyl Analogues of Adenine in a Model of Adjuvant Arthritis	D. Franková; Z. Zidek; E. Buchar; Z. Jiøièka; A. Holý
959-961	Stimulation of Cytokine and Nitric Oxide Production by Acyclic Nucleoside Phosphonates	Z. Zídek; D. Franková; A. Holý
963-964	2′-Deoxynucleoside 5′-Triphosphates with Reporter Groups Modified at α-, β,γ- or γ-Phosphates as Substrates for DNA Polymerases	L. A. Alexandrova; A. Yu. Skoblov; M. V. Jasko; A. A. Murabuldayev; L. S. Victorova; A. A. Krayevsky
965-966	Reinvestigation of 4-Thiothymidine-5′-triphosphate Synthesis	H. Bazin; S. Sauvaigo
967-969	An In Situ Pig Liver Esterase Assay as a Useful Predictive Tool for the Likely In Vitro Anti Viral Activity of Phosphoramidate Pro-Drugs	Carlo Ballatore; Christopher McGuigan; Erik De Clercq; Jan Balzarini
971-972	Prodrugs of Ara-CMP and Ara-AMP with a S-Acyl-2-thioethyl (SATE) Biolabile Phosphate Protecting Group: Synthesis and Biological Evaluation	R. Bazzanini; S. Manfredini; E. Durini; B. Gröschel; J. Cinatl; J. Balzarini; E. De Clercq; J-L. Imbach; C. Périgaud; G. Gosselin
973-975	Anti-HIV Pronucleotides: SATE Versus Phenyl as a Protecting Group of AZT Phosphoramidate Derivatives	T. Beltran; D. Egron; I. Lefebvre; C. Périgaud; A. Pompon; G. Gosselin; A-M. Aubertin; J-L. Imbach
977-978	New Strategies for Chemical Synthesis of Phosphorodithioates Derived from 2′- or 3′- or 5′-Thionucleosides	Izabela Tworowska; Wojciech Dąbkowski
979-980	Synthesis and Biological Evaluation of Nucleoside Triphosphates Incorporating an Oxyamino Function for “Post-amplification Labelling”	E. Trévisiol; E. Defrancq; J. Lhomme; A. Laayoun; A. Hoang; F. Besème; Ph. Cros
981-982	Synthesis and Anti-HIV Activity of Some S-Acyl-2-thioethyl (SATE) Phosphoramidate Derivatives of 3′-Azido-2′,3′-dideoxythymidine	D. Egron; C. Périgaud; G. Gosselin; A-M. Aubertin; J-L. Imbach
983-984	Synthesis, Anti-HIV Activity and Stability Studies of 3′-Azido-2′,3′-dideoxythymidine-5′-fluorophosphate	D. Egron; A. A. Arzumanov; N. B. Dyatkina; A. Krayevsky; J-L. Imbach; A-M. Aubertin; G. Gosselin; C. Périgaud
985-986	Synthesis of New Acyclic Nucleoside Vinyl Phosphonates	Annamaria Esposito; Maurizio Taddei
987-988	Intracellular Metabolism of β-L-ddAMP-bis(tbutylSATE), a Potent Inhibitor of Hepatitis B Virus Replication	A. Faraj; L. Placidi; C. Perigaud; E. Cretton-scott; G. Gosselin; L. T. Martin; C. Pierra; R. F. Schinazi; J. L. Imbach; J. P. Sommadossi
989-990	Synthesis and Biological Application of a New Heterodinucleotide with Both Anti-HSV and Anti-HIV Activity	Palmarisa Franchetti; Ghassan Abu Sheikha; Loredana Cappellacci; Mario Grifantini; Emanuela Balestra; Carlo-Federico Perno; Giorgio Brandi; Luigia Rossi; Mauro Magnani
991-992	³¹P NMR Studies on Oxidative Transformations of Aryl Nucleoside H-Phosphonate Diesters	Annika Kers; Inger Kers; Jacek Cieslak; Adam Kraszewski; Jacek Stawinski
993-994	Synthesis and In Vitro Antiviral Activity of Some Symmetrical Phosphoramidate Dimers of AZT	I. Kers; J-L. Girardet; G. Gosselin; C. Perigaud; J-L. Imbach; J. Stawinski
995-999	Synthesis and Transmembrane Transport Studies of Lipophilic Adenosine 5′-Triphosphate Derivatives	Annett Kreimeyer; François André; Aline Bluzat; Catherine Gouyette; Tam Huynh-dinh
1001-1002	Synthesis of the tBuSATE Pronucleotide of AZT by Two Different Synthetic Approaches	M. Lannuzel; D. Egron; J. -L. Imbach; G. Gosselin; C. Périgaud
1003-1004	Synthesis of New PMEA Diphosphate Mimics	W. H. G. Laux; C. Périgaud; J. -L. Imbach; G. Gosselin
1005-1006	Comparison of Anti-HBV Activity of β-D- and β-L-ddA-5′Monophosphate Prodrugs and Effectiveness in Combination with Lamivudine	A. G. Loi; A. Faraj; C. Pierra; G. Gosselin; J. L. Imbach; S. A. Locarnini; E. V. Groman; R. F. Schinazi; J. P. Sommadossi
1007-1008	Synthesis, Cytostatic Activity and Inhibition of Ribonucleotide Reductase by 5′-Phosphoramidates and 5′-Diphosphates, of 2′-O-Allyl-arabinofuranosyl Nucleosides	S. Manfredini; P. G. Baraldi; E. Durini; J. Balzarini; E. De Clercq; A. Karlsson; V. Buzzoni; L. Thelander
1009-1011	Analysis of DNA Sequencing Reaction Products Made with 7-Halo-7-deaza-2′-deoxyguanosine-5′-triphosphate	Mark G. McDougall; Louis P. Hosta; Shiv Kumar; Carl W. Fuller

Volume 18, Issue 4-5 (1999)

1013-1014	Synthesis and Properties of Novel NTP Derivatives	N. Sh. Padyukova; H. B. F. Dixon; E. V. Efimtseva; B. S. Ermolinsky; S. N. Mikhailov; M. Ya. Karpeisky
1015-1017	Replicative Capability of Anhydrohexitol Analogues of Nucleotides	Sylvie Pochet; Arthur Van Aershot; Piet Herdewijn; Philippe Marlière
1019-1020	Pyridoxal-Catalyzed Release of Nucleotides	Sylvie Pochet; Jean-Jacques Beaussire; Laurence Dugué; Philippe Marlière
1021-1022	Development of a New DNA Sequencing Method: 3′-Ester Cleavage Catalyzed by Taq DNA Polymerase	Isabelle Rasolonjatovo; Simon R. Sarfati
1023-1024	Synthesis of AZT-α-Borano-5′-Diphospho-Hexoses	Simon Sarfati; Catherine Guerreiro; Bruno Canard; Nathalie Dereuddre-bosquet; Pascal Clayette; Dominique Dormont
1025-1026	New Series of Mixed Pronucleotides. Synthesis and Anti-HIV Activities of Mononucleoside Phenyl SATE Phosphotriesters	N. Schlienger; S. Peyrottes; A-M. Aubertin; G. Gosselin; J-L. Imbach; C. Périgaud
1027-1028	Modified Nucleoside 5′-Triphosphonates as a New Type of Antiviral Agents	E. A. Shirokova; A. V. Shipitsin; L. S. Victorova; N. B. Dyatkina; L. E. Goryunova; R. Sh. Beabealashvilli; C. J. Hamilton; S. M. Roberts; A. A. Krayevsky
1029-1030	Novel Series of [ddN]-[TSAO-T] Heterodimers as Potential Bi-Functional Inhibitors of HIV-1 RT. Studies in the Linker and ddN Region	S. Velázquez; V. Tuñón; M. L. Jimeno; M. J. Pérez-Pérez; A. San-Félix; C. Chamorro; E. Lobatón; A. Esteban-gamboa; E. De Clercq; J. Balzarini; M. J. Camarasa
1031-1032	Human DNA Polymerases and Retroviral Reverse Transcriptases: Selectivity in Respect to dNTPs Modified at Triphosphate Residues	L. S. Victorova; D. G. Semizarov; E. A. Shirokova; L. A. Alexandrova; A. A. Arzumanov; M. V. Jasko; A. A. Krayevsky
1035-1053	Determination of the Group Electronegativity of CF₃ Group in 3′-O-CF₃-Thymidine by ¹-NMR	C. Thibaudeau; N. Nishizono; Y. Sumita; A. Matsuda; J. Chattopadhyaya
1055-1056	On the Conformation of UDPG, a Sugar Nucleotide	K. B. Kim; E. C. Behrman; E. J. Behrman
1057-1059	Structure and Properties of 7,9-Diglycosylguanine - an Unstable Intermediate in Transglycosylation of Guanine Nucleosides	Jerzy Boryski; Andrzej Manikowski
1061-1063	Selective Oxidation of 2′-Deoxyguanosine to Imidazolone by the Chemical Nuclease MnTMPyP Associated to KHSO₅ or Sulfite/O_2.	Corine Vialas; Geneviève Pratviel; Jean Bernadou; Bernard Meunier
1065-1066	Radiolabelled Pyrimidine Nucleosides to Monitor the Expression of HSV-1 Thymidine Kinase in Gene Therapy	Leonard I. Wiebe; Edward E. Knaus; Kevin W. Morin
1067-1068	Structural Studies of 5-Ethyl-2′-Deoxyuridine by Selective Pulse ¹H DPFGSE NOE Spectroscopy and PM3 Calculations	L. E. Bailey; M. L. García-Martin; H. Stender; G. Ball
1069-1071	Vibrational Study of a Nucleoside Analogue with Antiviral Activity, 5-Chloro-2′-deoxyuridine, CDU	L. Bailey; R. Navarro; A. Hernanz
1073-1074	Determination Of 2-Chloro-2′-deoxyadenosine (Antileukemic Agent) and Related Compounds by Electrochemical Method	E. Bojarska; Z. Kazimierczuk
1075-1076	Comparative Studies of the Electronic Structure of 2-Chloro-2′-Deoxyadenosine Studied by ³⁵CI-NQR Spectroscopy and Quantum Chemical Calculations	J. N. Latosinska; J. Kasprzak; E. Bojarska; Z. Kazimierczuk
1077-1078	Bicyclonucleosides and Ring-Chain Interconversion	J. M. J. Tronchet; M. Zsély; L. Brenas; O. Lassout; E. Grand; P. Seuret; M. Grigorov; E. Rivara-minten; M. Geoffroy
1079-1082	Unexpected Shift to a 4-Imino Tautomer Upon N⁴-Acylation of 5-Methylcytosin-1-yl Nucleoside Analogues	R. Busson; L. Kerremans; A. Van Aerschot; M. Peeters; N. Blaton; P. Herdewijn
1083-1085	Interaction 3d-and 4d-Group Metal Ions With GMP	V. A. Sorokin; M. V. Degtyar; G. O. Gladchenko; V. A. Valeev; I. V. Sysa; Yu P. Blagoi
1087-1089	Purine Based Combinatorial Chemistry: Solution Phase Simultaneous Addition of Functionalities. Iterative Deconvolution by Orthogonal Protection to a Single Compound with Potent Antibacterial Activity	A. S. Fraser; A. M. Kawasaki; P. D. Cook
1091-1093	NMR Studies of the Tautomerism in Pseudoisocytidine	Lou-Sing Kan; W-C. Lin; R. Dayal Yadav; J. H. Shih; Ito Chao
1095-1096	Reactions of Adenosine with Bromo- and Chloromalonaldehydes in Aqueous Solutions: Kinetics and Mechanism	N. Koissi; K. Ketomäki; K. Neuvonen; S. Kuusela; H. Lönnberg
1097-1098	Trifluoromethyldiazirine-Containing dUTP: Synthesis and Application in DNA/Protein Crosslinking	Galina A. Korshunova; Andrey N. Topin; Natalia V. Sumbatyan; Olga N. Koroleva; Valeriy L. Drutsa
1099-1100	Mechanism of pH-independent Cleavage and Isomerization of 3′-Ribonucleotide Phosphodiesters	Markus Kosonen; Harri Lönnberg
1101-1103	Uniform Band Intensities in Fluorescent Dye Terminator Sequencing	Shiv Kumar; C. W. Fuller; S. Nampalli; M. Khot; I. Livshin; L. Sun; S. Hamilton; S. B. Samols; J. A. Mamone; K. M. Hujer; B. F. McArdle; J. R. Nelson; S. Duthie
1105-1106	Studies on Association of mRNA Cap-analogues with a synthetic Dodecapeptide DGIEPMWEDEKN	A. Niedżwiecka-Kornaś; R. Przedmojski; L. Balaspiri; Z. Wieczorek; J. Stępiński; M. Jankowska; H. Lönnberg; E. Darżynkiewicz; R. Stolarski
1107-1108	Steric and Electronic Properties of the 3′-spiro Moiety of TSAO-T and Analogues	M. J. Pérez-Pérez; R. Alvarez; M. L. Jimeno; A. San-Félix; A. Lozano; M. J. Camarasa
1109-1112	NMR Study on The Tuning of North ⇆ South Equilibrium in Nucleos(t)ides by Metal Ion Interactions	MatjaŽ Polak; Janez Plavec
1113-1117	Synthesis of a New Analog of Thymidine for In Vivo Non-radioactive Labeling of DNA	Ch. Rodríguez-Tanty; R. Pérez; J. Miranda; H. Vélez-Castro; A. Rosado; A. Macias; L. Galán; D. Higginson-clarke; A. M. Riverón
1119-1122	Investigations of Some Nucleic Acid Component Analogs	Yuri Rubin; Jerzy Leszczynski
1123-1124	Manganese Tetraphenylporphyrins Catalyzed Selective Oxidation of Purine Derivatives	Raffaele Saladino; Paola Carlucci; Claudia Crestini; Pietro Tagliatesta; Donato Monti; Tristano Boschi
1125-1126	Hydrolysis of some mRNA 5′-Cap Analogs Catalyzed by the Human Fhit Protein - and Lupin ApppA Hydrolases	E. Bojarska; R. Kraciuk; J. Wierzchowski; Z. Wieczorek; J. Stępiński; M. Jankowska; E. Starzyńska; A. Guranowski; E. Darżynkiewicz
1127-1129	Computer Aided Design of Triplet Forming Artificial Nucleobases	R. Fenyõ; Z. Timár; I. Pálinkó; B. Penke
1131-1133	Synthesis and Preliminary Thermodynamic Investigation of Hypoxanthine-Containing Peptide Nucleic Acids	Zoltán Timár; Sándor Bottka; Lajos Kovács; Botond Penke
1135-1136	Production of Nucleosides by Large-Scale Bioconversion	G. Cotticelli; P. Magrì; M. Grisa; G. Orsini; G. Tonon; G. Zuffi

Volume 18, Issue 3 (1999)

a	Editorial board page for “Nucleosides, Nucleotides & Nucleic Acids”, Volume 18, Number 3
307-310	Preparation of 8-Hydroxy-dGTP and 2-Hydroxy-dATP by a Phosphate Transfer Reaction by Nucleoside-Diphosphate Kinase	Hiroyuki Kamiya; Hiroshi Kasai
311-330	Interaction of the Recombinant Herpes Simplex Virus Type 1 Thymidine Kinase with Thymidine and Aciclovir: A Kinetic Study	Susanna Kussmann-gerber; Christine Wurth; Leonardo Scapozza; Beatrice D. Pilger; Vladimir Pliška; Gerd Folkers
331-335	An Efficient, Short Synthesis, and Potent Anti-Hepatitis B Viral Activity of a Novel Ring-Expanded Purine Nucleoside Analogue Containing a 5:7-Fused, Planar, Aromatic, Imidazo[4,5-E][1,3]diazepine Ring System	Huan-Ming Chen; Ramesh Sood; Ramachandra S. Hosmane
337-351	Synthesis, Lipophilicity, and Anti-HIV Activity of a New Brominated Analog of Zidovudine	Marisa Morura; Horacio Salomón; Guillermo Moroni; Mark Wainberg; Margarita C. Brifiñn
353-361	Synthesis of New Chiral Peptide Nucleic Acid (PNA) Monomers by a Simplified Reductive Animation Method	Bogdan Falkiewicz; Katarzyna Kowalska; Aleksandra S. Kolodziejczyk; Kazimierz Wiśniewski; Leszek łankiewicz
363-376	Synthesis of a Novel C-Nucleoside, 2-Amino-7-(2-deoxy-β- D-erythro-pentofuranosyl)-3H,5H-pyrrolo-[3,2-d]pyrimidin-4-one (2′-Deoxy-9-deazaguanosine)	Eric S. Gibson; Krystyna Lesiak; Kyoichi A. Watanabe; Lorraine J. Gudas; Krzysztof W. Pankiewicz
377-391	Expanding the Catalytic Repertoire of Nucleic Acid Catalysts: Simultaneous Incorporation of Two Modified Deoxyribonucleoside Triphosphates Bearing Ammonium and Imidazolyl Functionalities	David M. Perrin; Thérèse Garestier; Claude Hélène
393-401	Synthesis of a Monocharged Peptide Nucleic Acid (PNA) Analog and Its Recognition as Substrate by DNA Polymerases	M. J. Lutz; D. W. Will; G. Breipohl; S. A. Benner; E. Uhlmann
403-410	Recognition of 2′-Deoxyisoinosine Triphosphate by the Klenow Fragment of DNA Polymerase I	Jean-Jacques Beaussire; Sylvie Pochet
411-423	Molecular Dynamics of Labeled Oligonucleotide Probes Used for the Detection of Point Mutations in DNA	S. Winter; S. Kirschstein; D. P. Millar
425-441	7-Deaza-2′-deoxyinosine: A Stable Nucleoside with the Ambiguous Base Pairing Properties of 2′-Deoxyinosine	Frank Seela; Cathrin Mittelbach
443-456	Chiral Synthons for CARBA-β-D-Ribonucleosides. Synthesis of CARBA-4-Deoxypyrazofurin and Isomeric CARBA-4-Deaza-oxoformycin Analogues	Barbara Mohar; Jože Kobe
457-467	Novel Triazole 2′-Deoxy-4′-thionucleosides: Stereoselective Synthesis and Biological Evaluation	G. Inguaggiato; M. Jasamai; J. E. Smith; M. Slater; C. Simons
469-474	Oligonucleotides Quality Control Analysis in Free Solution by Capillary Electrophoresis at Acidic pH	Maria Flora Mangano; Cristina Battaglia; Giuliana Salani; Luigi Rossi Bernardi; Gianluca De Bellis
475-483	Oligodeoxyribonucleotide Phosphorothioates: Substantial Reduction of (N-1)-mer Content Through the Use of Trimeric Phosphoramidite Synthons	Alessandra Eleuteri; Daniel C. Capaldi; Douglas L. Cole; Vasulinga T. Ravikumar
485-492	Use of Phenylacetyl Disulfide (PADS) in the Synthesis of Oligodeoxyribonucleotide Phosphorothioates	Zacharia S. Cheruvallath; Patrick D. Wheeler; Douglas L. Cole; Vasulinga T. Ravikumar
493-508	Synthesis of DNA-(3′)-PNA Chimeras with Conformationally Restricted Linkers Based on 4-Hydroxyproline	Jeroen C. Verheijen; Anne-Marie van Roon; Alexander van der Laan; Gijsbert van der Marel; Jacques van Boom

Volume 18, Issue 2 (1999)

a	Editorial board page for “Nucleosides, Nucleotides & Nucleic Acids”, Volume 18, Number 2
153-159	Total Synthesis of the Naturally Occurring Antibiotic Toyocamycin Using New and Improved Synthetic Procedures	Anthony R. Porcari; Leroy B. Townsend
161-180	Synthesis and Conformational Analysis of 1,5-Anhydro-2,4-dideoxy-D-mannitol Nucleosides	N. Hossain; I. Luyten; K. Rothenbacher; R. Busson; P. Herdewijn
181-186	Kinetics for the Acid-Catalyzed Hydrolysis of Purine and Cytosine 2′-Deoxy-4′-thionucleosides	Mohamed I. Elzagheid; Mikko Oivanen; Richard T. Walker; John A. Secrist III
187-195	A Practical Synthesis of L-FMAU from L-Arabinose	Jinfa Du; Yongseok Choi; Kyeong Lee; Byoung K. Chun; Joon H. Hong; Chung. K. Chu
197-201	Synthesis of Fluorescent, Photolabile 3′-O-Protected Nucleoside Triphosphates for the Base Addition Sequencing Scheme	Mike B. Welch; Kevin Burgess
203-216	The Synthesis and Antiviral Activity of 4-Fluoro-1-β-D-ribofuranosyl-1H-pyrazole-3-carboxamide	Richard Storer; Claire J. Ashton; Anthony D. Baxter; Michael M. Hann; Clara L. P. Marr; Andrew M. Mason; Chi-Leung Mo; Peter L. Myers; Stewart A. Noble; Charles R. Penn; Niall G. Weir; Jacqueline M. Woods; Paul L. Coe
217-225	Synthesis and Biological Evaluation of a Carbocyclic Azanoraristeromycin Siderophore Conjugate	Arun Ghosh; Marvin J. Miller; Erik De Clercq; Jan Balzarini
227-238	Synthesis and Antiviral Activity of Novel Aza-acyclonucleosides	Stephen C. Bergmeier; Susan L. Fundy; John C. Dracht
239-243	Synthesis of an Enantiomerically Pure Carbocyclic DNA Abasic Site Analogue	Martial Thomas; Bertrand Castaing; Jean-Louis Fourrey; Charles Zelwer
245-262	New N-2-Labelled Fluorescent Derivatives of Guanosine Nucleotides and Their Interaction with GTP-Binding Proteins	Nils Ostermann; Mohammad Reza Ahmadian; Alfred Wittinghofer; Roger S. Goody
263-275	Synthesis of a New Class of HIV-1 Inhibitors	Audrey Farese-Di Giorgio; Sandrine Pairot; Nadia Patino; Roger Condom; Christophe Di Giorgio; André Aumelas; Anne-Marie Aubertin; Roger Guedj
277-289	High Specific Radioactivity Labeling of Oligonucleotides with ³H-Succinimidyl Propionate	Trung Ledoan; Rodolphe Auger; Abdellah Benjahad; Jean-Pierre Tenu
291-305	Synthesis of Achiral Linker Reagents for Direct Labelling of Oligonucleotides On Solid Supports	Carsten Behrens; Otto Dahl

Volume 18, Issue 1 (1999)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 18, Number 1
1-4	Efficient Synthesis of N-4 Alkyl Derivatives of 2′, 3′-Dideoxycytidine (ddC)	E. Dechaux; R. Pontikis; C. Monneret
5-9	6-Thioguanine in Peptide Nucleic Acids. Synthesis and Hybridization Properties	Henrik F. Hansen; Leif Christensen; Otto Dahl; Peter E. Nielsen
11-21	The Cu²-Promoted Cleavage of mRNA 5′-cap Analogs: A Kinetic Study with P¹-(7-Methylguanosin-5′-yl) P³-(Nucleosid-5′-yl) Triphospates and P¹-(7-Methylguanosin-5′-yl) P⁴-(Guanosin-5′-yl) Tetraphosphate	Zbigniew Wieczorek; Edward Darzynkiewicz; Satu Kuusela; Harri Lönnberg
23-37	Synthesis and Utilization of ¹³C(8)-Enriched Purines	Christopher J. Lafrancois; June Fujimoto; Lawrence C. Sowers
39-49	Terminal Diols as Efficient Substrates for Transglycosylational Activity of NAD Glycohydrolase	Shuichi Tono-oka; Ichiro Azuma
51-54	A New Synthesis of Symmetrical P¹,P²-Dinucleoside-5′-pyrophosphates	Kyung Bo Kim; Edward J. Behrman
55-72	Synthesis of 2′-Methylene-Substituted 5-Azapyrimidine, 6-Azapyrimidine, and 3-Deazaguanine Nucleoside Analogues as Potential Antitumor/Antiviral Agents	Mao-Chin Liu; Mei-Zhen Luo; Diane E. Mozdziesz; Tai-Shun Lin; E. Ginger; Dutschman; Yung-Chi Cheng; Alan C. Sartorelli
73-88	8-Amino-2′-deoxyguanosine Incorporation into Oligomeric DNA	Robert A. Rieger; Charles R. Iden; Elena Gonikberg; Francis Johnson
89-93	Stability of Phosphorothioate Oligonucleotides in Aqueous Ammonia in Presence of Stainless Steel	Brett J. Turney; Zacharia S. Cheruvallath; Mark Andrade; Douglas L. Cole; Vasulinga T. Ravikumar
95-111	Synthesis of New Thiolated Acyclonucleosides with Potential Anti-HBV Activity	Ibrahim F. Zeid; A. Adel; H. Abdel-Rahman; Ahmed E. -S. Abdel-Megied; Abd-Allah Sh. Ei-Etrawy
113-123	Synthesis and Anti-HIV Activity of Different Novel Nonclassical Nucleosides	Galal E. H. Elgemeie; Omar A. Mansour; Nadia H. Metwally
125-136	Preparation of N², N²'7-Trimethylguanosine Affinity Columns	Ruth Espuny; Diana Bahia; Regina Maria Barretto Cicarelli; Caries Codony; Amina Khaouja; Anna Maria Aviñó; Ramon Eritja; Montse Bach-Elias
137-151	Synthesis of 2′-Iodo- and 2′-Bromo-ATP and GTP Analogues as Potential Phasing Tools for X-ray Crystallography	Mathias Gruen; Christian Becker; Andrea Beste; Christoph Siethoff; Axel J. Scheidig; Roger S. Goody

Volume 17, Issue 12 (1998)

vii-viii	Contributors to this Issue
2165-2173	Synthesis and Anti-HSV-1 Activity of 6 Substituted Pyrazolo[3,4-d]Pyridazin-7-one Nucleosides	P. G. Baraldi; S. Manfredini; R. Romagnoli; L. Stevanato; A. N. Zaid; R. Manservigi
2175-2187	A Synthetic Approach to Carbocyclic Sinefungin	Adilson D. Da Silva; Edmilson JoseMaria; Pierre Blanchard; Jean-Louis Fourrey; Malka Robert-Gero
2189-2197	A Monoclonal Antibody that Specifically Recognizes m'A Nucleoside	Ruth Espuny; Anna Castro; Carles Codony; Ramon Eritja; Montserrat Bach-Elias
2199-2210	Detailed Studies on Trimethylselyl Triflate Mediated Glycosylation via a 3,5-O-(l,l,3,3-Tetraisopropyl-Disiloxane-l,3-diyl)-2-O-methylribofuranos-l-yl Trichloroacetimidate Intermediate	Koh-ichiroh Shohda; Takeshi Wada; Mitsuo Sekine
2211-2220	Crystal Structure and Molecular Conformation of 4-Thiouracil-2′-Trifluorothioacetamide -3′, 5′-Diacetyl-β-D-Riboside	Thamarapu. Srikrishnan
2221-2239	Synthesis of 4′-Trifluoromethyl Nucleoside Analogs	Janusz Kozak; Carl R. Johnson
2241-2247	Some Aspects on Acyclonucleoside Synthesis	Masaru Ubasawa; Hideaki Takashima; Kouichi Sdciya
2249-2254	The Synthesis of 2′-Deoxy-L-Cytidine-3′-Phosphate	Igor A. Kozlov; Leslie E. Orgel
2255-2266	Quinolone Nucleosides: 6,7-Dihalo-N-β- and α-Glycosyl-l 4-dihydro-4-oxo-quinoline-3-carboxylic Acids and Derivatives. Synthesis, Antimicrobial and Antiviral Activity	Najim A. Al-Masoudi; Yaseen A. Al-Soud; Micheal Ehrmann; Erik de Clercq
2267-2280	3′-Deoxy-3′-C-trifluoromethyl Nucleosides: Synthesis and Antiviral Evaluation	S. Lavaire; R. Plantier-Royon; C. Portella; M. de Monte; A. Kirn; A. -M. Aubertin
2281-2288	The Synthesis of RNA Containing the Modified Nucleotides N²-Methylguanosine and N⁶, N⁶-Dimethyladenosine	Jason P. Rife; Charles S. Cheng; Peter B. Moore; Scott A. Strobel
2289-2310	Synthesis and Antiviral Evaluation of 2′-Deoxy-4′-thio-L-nucleosides and Their Phosphotriester Derivatives Bearing S-Acyl-2-thioethyl Bioreversible Phosphate-Protecting Groups	F. De Valette; J. -L. Barascut; J. -L. Imbach
2311-2322	Extension of the Applicability of δJ-Values for the Configurational Assignment of Diastereomeric Phosphate-Modified Dideoxynucleotides	Daisy Machytka; Eszter Gács-Baitz; Zsuzsa Tegyey
2323-2333	2-Bromoadenosine-Substituted 2′,5′-Oligoadenylates Modulate Binding and Activation Abilities of Human Recombinant RNase L	Yukio Kitade; Masaharu Wakana; Shin-ichi Terai; Takayuki Tsuboi; Masayuki Nakanishi; Chizuko Yatome; Beihua Dong; Robert H. Silverman; Paul F. Torrence
2335-2338	Improved Deproteciton Procedure for DPSE Protected Phosphorothioates	Achim H. Krotz; Zacharia S. Cheruvallath; Douglas L. Cole; Vasulinga T. Ravikumar
2339-2350	Synthesis of Peptidinol Adenylates	Annett Kreimeyer; Philippe Marliere
2351-2365	Improved Targeting of the Flanks of a DNA Stem Using α-Oligodeoxynucleotides.-The Enhanced Effect of an Intercalator	Ahmed F. Khattab; Erik B. Pedersen
2367-2382	Synthesis of 5-Halogeno-6-amino-2′-deoxyurldines and their Analogs as Potential Inhibitors of Thymidine Phosphorylase	Bai-Chuan Pan; Zhi-Hao Chen; Edward Chu; Ming-Yu WangChu; Shih-Hsi Chu

Volume 17, Issue 12 (1998)

2383-2387	Novel Lewis Acid-Catalyzed Rearrangement of a Sugar-Base Hybrid to Afford an Anhydronucleoside	Michael E. Jung; Claire Castro; Saeed I. Khan
2389-2401	Design, Synthesis and Antiviral Activity of α-L-Arabinofuranosyl Derivatives of 2-Substituted-5,6-dichlorobenzimidazoles	Jean-Luc Girardet; John C. Drach; Stanley D. Chamberlain; George W. KosLzalka; Leroy B. Townsend
2403-2416	Chemical Synthesis of 4-Thiouridine-Containing Substrate Analogues of tRNA:Pseudouridine-55 Synthase: Photocross-Linking Studies	Hubert F. Becker; Henri Grosjean; Jean-Louis Fourrey
2417-2427	Catalytically Significant Macrochelate Formation in Zn²Promoted Hydrolysis of Oligoribonucleotides: Model Studies with Chimeric Phosphodiester/Methylphosphonate Oligomers	Satu Kuusela; Harri Lönnberg
2429-2443	Synthesis and Biological Evaluation of Phosphonate Derivatives of Some Acyclic Pyridine-C-Nucleosides	Johan Van hemel; Eddy L. Esmans; Pieter E. Joos; Alex De Groot; Roger A. Dommisse; Jan M. Balzarini; Erik D. De Clercq
2445	Erratum: Synthesis of Novel Bicyclic Nucleosides Related to Natural Griseolic Acids	Lea Pickering; Vasu Nair

Volume 17, Issue 9-11 (1998)

xiii-xvi	Contributors To This Issue
1515-1522	Cloning and Expression of Collagen-Derived Protein in E. Coli And Baculovirus System	S. Schlosser; G. Gröger; O. Holfeld; H. Seliger
1523-1526	1,5-Anhydro-2-Deoxy-D-Altritol Oligonucleotides as Conformationally Restricted Analogues of Rna	Brigitte Allart; Arthur Van Aerschot; Piet Herdewijn
1527-1537	New Building Blocks for the Preparation of Branched Oligonucleotides	Alex Azhayev; Seppo Auriola; Jari Hovinen
1539-1545	Studies on the Interaction of Dna-Ligands with Modified Parallel-Stranded Duplex-Dna Oligomers	I. Förtsch; E. Birch-Hirschfeld; T. M. Jovin; A. Stelzner; C. Zimmer
1547-1556	A Novel Approach to Synthesis of 2′-Deoxy-β-D-Ribonucleosedes Via Transglycosylation of 6-Oxopurine Ribonucleosides	Jerzy Boryski
1557-1566	Penetration and Antiviral Activity of Coxsackievirus B3 (Cvb3)-Specific Phosphorothioate Oligodeoxynucleotides (Ps-Odn)	M. Schmidtke; C. Knorre; L. Blei; A. Stelzner; E. Birch-Hirschfeld
1567-1570	Branched Polyethylene Glycol (Bpeg) Conjugated Antisense Oligonucleotides	B. Burcovich; F. M. Veronese; V. Zarytova; G. M. Bonora
1571-1576	3′-Amidated 3′-Deoxyxylofuranose Analogues of N⁶-^-Cyclopentyladenosines: a New Class of Non-Xanthine Antagonists at the Adenosine A₁ Receptor.	Serge Van Calenbergh; Adriaan P. IJzerman; Piet Herdewijn
1577-1581	Divers Stereoisomers of N-Acetylhydroxyprolinol as Sugar Substitute in Oligonucleotides	G. Ceulemans; A. Van Aerschot; P. Herdewijn
1583-1587	Stability Studies in Biological Media of Dimer Phosphotriesters Bearing Glucuronic Acid Residue	Nathalie Mignet; Carole Chaix; Jean-Louis Imbach
1589-1603	The Information Transmission from the Nucleobase Drives the Sugar-Phosphate Backbone Conformation in the Nucleotide Wire	Christophe Thibaudeau; Jyoti Chattopadhyaya
1605-1611	The Electronic Nature of the Aglycone dictates the Drive of the Pseudorotational Equilibrium of the Pentofuranose Moiety in C-Nucleosides	Ingrid Luyten; Jasenka Matulic-Adamic; Leo Beigelman; Jyoti Chattopadhyaya
1613-1616	The 5′-Purine-Pyrimidine-3′ Stacks are More Stabilizing in a Self-3′-Pyrinudine-Purine-5′ complementary DNA Duplex than the 5′-Purine-Purine-3′ 3′-Pyrimidine-Pyrimidine-5′ Stack	D. Ossipov; E. Zamaratski; J. Chattopadhyaya
1617-1634	Elucidation of the Origin of NOEs And ROEs that Show the Hydration in the Minor and Major Grooves of DNA Duplex with ATTAAT Tract by a Combination of NOESY and ROESY Experiments	T. V. Maltseva; P. Roselt; J. Chattopadhyaya
1635-1637	A simple and efficient synthesis of nucleotides containing 5′-S- or 3′-S-phosphorothioate linkage.	W. Dabkowski; M. Michalska; I. Tworowska
1639-1644	Novel Unique Catalytic Activating Reagents in Synthesis of Biophosphates via the Phosphoramidite Route	Wojciech Dabkowski; Izabela Tworowska; Jan Michaiski; Friedrich Cramer
1645-1649	High Affinity Of Backbone-Modified α-Anomeric Oligodeoxynucleottoes For Dna And Rna Targets	A. Laurent; F. Debart; J. -C. Bologna; J. -J. Vasseur; B. Rayner
1651-1665	Strong, Specific, Reversible Binding Ligands for Transfer Rna: Comparison By Fluorescence and Nmr Spectroscopies with Distamycin Binding for a New Structural Class of Ligand	Elena V. Bichenkova; Seyed E. Sadat-Ebrahimi; Amanda N. Wilton; Niamh O'Toole; Debora S. Marks; Kenneth T. Douglas

Volume 17, Issue 9-11 (1998)

1667-1670	A Novel Concept for the Combinatorial Synthesis of Peptide Nucleic Acids.	Alexander Dömling
1671-1679	Synthesis And Binding Study Of Phosphonate Analogues Of Pnas And Their Hybrids With Pnas	Vladimir A. Efimov; Michael V. Choob; Alla A. Buryakova; Oksana G. Chakhmakhcheva
1681-1684	Disaccharide Nucleosides And Their Enzymatic And Chemical Incorporation Into Oligonucleotides	Ekaterina V. Efimtseva; Lubov S. Victorova; Andrei A. Rodionov; Boris S. Ermolinsky; Marina V. Fomitcheva; Vera L. Tunitskaya; Sergey N. Mikhailov; Mikko Oivanen; Arthur Van Aerschot; Piet Herdewijn
1685-1696	Modified Hammerhead Ribozymes as Potential Therapeutics	Joachim W. Engels; Michaela Scherr; Arnold Ganser; Manuel Grez; Valentin Wittmann
1697-1704	Synthesis of 3′-Azido-3′-Deoxythymidine-Terminated Oligonucleotide	Dmitriy S. Esipov; Olga V. Esipova; Vyacheslav G. Korobko
1705-1708	Quantitative Parametrs of Cooperative Interactions of the Oligodeoxyribonucleotides on the Complementary Template	Abdussalam Adeenah-Zadah; Olga S. Fedorova
1709-1716	Studies on Alternate Strand Triple Helix Formation by Oligodeoxyribonucleotides Containing A 3′-3′ Phosphodiester Bond	L. De Napoli; A. Galeone; L. Mayol; A. Messere; D. Montesarchio; A. Pepe; G. Piccialli
1717-1724	Pna Array Technology in Molecular Diagnostics	Albert Geiger; Ane Lester; Jörg Kleiber; Henrik Ørum
1725-1729	Effect of the Thioalkyl Chain Variation in the Efficiency of Sate Pronucleotides	D. Egron; C. Perigaud; A. -M. Aubertin; J. -L. Imbach; G. Gosselin
1731-1738	Unnatural β-L-Enantiomers of Nucleoside Analogues as Potent Anti-Hepatitis B Virus Agents	G. Gosselin; V. Boudou; J-F Griffon; G. Pavia; C. Pierra; J-L Imbach; A. Faraj; J-P Sommadossi
1739-1745	Asymmetric Synthesis of Optically Active 1,3-Oxathiolane Nucleoside Analogues	Romualdo Caputo; Annalisa Guaragna; Giovanni Palumbo; Silvana Pedatella
1747-1759	Nucleoside 3′-O-(2-Oxo-“Spiro”-4.4-Pentamethylene-1.3.2-Oxathiaphospholane)S: Monomers For Stereocontrolled Synthesis Of Oligo(Nucleoside Phosphorothioate/Phosphate)S	Boleslaw Karwowski; Piotr Guga; Anna Kobylariska; Wojciech J. Stec
1761-1766	Cleavage Of Oligodeoxyribonucleotides From Polymer Supports And Their Rapid Deprotection Under Microwaves	K. C. Gupta; P. Kumar
1767-1773	Oligonucleotide uptake in leukocytes is dependent on extracellular calcium: a hint for the involvement of adhesion molecules?	Gunther Hartmann; Martin Bidlingmaier; Bemd Jahrsdörfer; Anne Krug; Ulrich Hacker; Andreas Eigler; Stefan Endres
1775-1779	Synthesis of 1,5-Anhydro-D-Mannitol Nucleosides with a Purine Base Moeety	Nafizal Hossain; Piet Herdewijn
1781-1786	Facile Synthesis of 3′-C-Branched 1,5-Anhydrohexitol Nucleosides	Nafizal Hossain; Piet Herdewijn
1787-1792	A Versatile Polymer Support Useful for Large-Scale Synthesis of DNA for Biomedical Applications	P. Jaisankar; M. Hinz; E. Happ; H. Seliger
1793-1800	Probability packaging of T4 coliphage DNA driven by oscillatory ATP consumption	Albrecht K. Kleinschmidt; Gerd Baumann; Rainer Martin
1801-1807	DNA Triplex Formation on the Granulocyte-Macrophage Colony-Stimulating Factor Gene Proximal Promoter	Marina Kochetkova; M. Frances Shannon
1809-1812	New Fluorescent Nucleoside Derivatives -5-Alkynylated 2-Deoxyuridines	V. A. Korshun; E. V. Manasova; K. V. Balakin; A. D. Malakhov; A. V. Perepelov; T. A. Sokolova; Yu. A. Berlin

Volume 17, Issue 9-11 (1998)

1813-1821	Chemical Synthesis and Properties of Long-Chain Alkoxymethyl-Nucleobase Derivatives	L. Kovalenko; M. Madre; S. Lindau; C. Bohley; N. Panchenko; W. -V. Meister; R. Zhuk; S. Hoffmann
1823-1834	Influence of P-Chirality of Phosphorothioate Oligonucleotides on the Activity of Amv-Reverse Transcriptase	Agnieszka Krakowiak; Maria Koziolkiewicz
1835-1850	Fluorescence Resonance Energy Transfer (Fret) to Follow Ribozyme Reactions In Real Time	Andreas Hanne; Muktevi V. Ramanujam; Thomas RüUcker; Guido Krupp
1851-1856	Synthesis of Novel Branched Nucleoside Dimers Containing a 1,2,3-Triazolyl Linkage	Hassan. B. Lazrek; Joaachim. W. Engels; Wolfgang Pfleiderer
1857-1860	Synthesis of 2′-Deoxynucleoside 5′-Methylenebis-(phosphonate)s Using 2-(4-Nitrophenyl)ethyl Methylenebis(phosphonate) as the Phosphonylating Agent.	Krystyna Lesiak; Kyoichi A. Watanabe; Krzysztof W. Pankiewicz
1861-1869	Use of Oligonucleotide Conjugates in Creating Self-Assembling Supramolecular Systems	Robert L. Letsinger
1871-1880	Synthesis of A Polyaminooligonucleotide Combinatorial Library	Wojciech. T. Markiewicz; Przemyslaw Godzina; Maria Markiewicz; Anna Astriab
1881-1884	Lessons from the Pseudorotational Cycle: Conformationally Rigid AZT Carbocyclic Nucleosides and Their Interaction with Reverse Transcriptase	Victor E. Marquez; Abdallah Ezzitouni; Pamela Russ; Maqbool A. Siddiqui; Harry Ford Jr; Ron J. Feldman; Hiroaki Mitsuya; Clifford George; Joseph J. Barchi Jr
1885-1894	Properties of Naphtho[2,1-B]pyrans Covalently Linked to Oligonucleotides	M. Mazzei; E. Sottofattori; M. Ibrahim; A. Balbi
1895-1904	Duplex Stabilization by DNA-Hoechst 33258 Conjugates: Effects of Base Pair Mismatches	K. Wiederholt; L. W. McLaughlin
1905-1913	Possibilities of Triplex-Formation by 21-Mer Oligodeoxyribonucleotides as Analogs of Tetrahymena Pre-rRNA Fragments	W-V Meister; S. I. Kargov; E. Birch-Hirschfeld; C. Bohley; G. Burckhardt; G. Bischoff; R. Bischoff; U. Gromann; S. Hoflfmann
1915-1918	Functionally Competent Analogs and Their Use for the Determination of Nucleotide Conformation in the Productive Enzyme-Substrate Complexes	S. N. Mikhailov
1919-1936	Systematic Mutation in the Third Strand of a Purine Motif DNA Triple Helix: a Story of a Molecule Which Hides Its Tail	Martin. Mills; Horst H. Klump
1937-1948	Synthesis and Hybridization Studies of Oligonucleotide Sequences with Modified Fluorescent Nucleoside Analogs	Rajendra KPandey; Snehlata Tripathi; Krishna Misra
1949-1952	Comparative Stability of Triple Helices Containing Modified DNA or RNA Pyrimidine Strands	Francois Morvan; Jean-Louis Imbach; Bernard Rayner
1953-1967	An Improved Synthesis of 1-β-D-Arabinofuranosylcytosine 5′-Phosphate-L-1,2-diacylglycerols	Ágnes Nyilas
1969-1975	Concept of “Binary Oligonucleotide Reagent”	S. I. Oshevski
1977-1982	Application of Oxathiaphospholane Method for the Synthesis of Oligodeoxyribonucleotide 5′-O-Conjugates	Anna Kobyláska; Andrzej Okruszek; Wojciech J. Stec
1983-1986	Synthesis of Derivatives of 3-Methylxantheve and 1-Methyl-3-Isobutylxanthine 7-β-D-Ribofuranosides	Vita Ozola; Yuris Maurinsh; M. Lidaka
1987-1996	New Photolabile Protecting Groups in Nucleoside and Nucleotide Chemistry—Synthesis, Cleavage Mechanisms and Applications	H. Giegrich; S. Eisele-Bühler; Chr Hermann; E. Kvasyuk; R. Charubala; W. Pfleiderer

Volume 17, Issue 9-11 (1998)

1997-2001	DNA-PHONA-PNA Chimeric Molecules: Contributions to Binding Against Complementary DNA	A. Peyman; E. Uhlmann; K. Wagner; S. Augustin; C. Weiser; S. Hein; D. Langner; G. Breipohl; D. W. Will
2003-2009	Imidazole-4-Carboxamide and 1,2,4-Triazole-3-Carboxamide Deoxynucleotides as Simplified DNA Building Blocks with Ambiguous Pairing Capacity	Sylvie Pochet; Laurence Dugué
2011-2020	What Are the Conformational Changes Induced by Hard and Soft Metal Ion Binding to 2′-Deoxyguanosine?	Matjaž Polak; Janez Plavec
2021-2025	6-N-(N-Methylanthranylamido)-4-Oxo-Hexanoic Acid: A New Fluorescent Protecting Group Applicable To A New Dna Sequencing Method	Isabelle Rasolonjatovo; Simon R. Sarfati
2027-2031	A New Approach to Oligonucleotide Synthesis in Solution	Colin B. Reese; Quanlai. Song
2033-2043	New Strategies for the Chemical Synthesis of Biologically Important Nucleic Acid Derivatives	Mitsuo. Sekine; Hiroyuki. Tsuruoka; Koh-ichiro. Shohda; Tomohisa. Moriguchi; Tomohisa. Wada
2045-2052	Parallel-Stranded Duplex DNA and Self-Assembled Quartet Structures Formed by Isoguanine and Related Bases	Frank. Seela; Changfu. Wei; Alexander. Melenewski; Elisabeth. Feiling
2053-2061	Antisense Oligonucleotide Conjugates with Photosensitizers-An Update	H. Seliger; H. Knoller; A. Rück; K. Heckelsmiller; R. Steiner
2063-2072	Activated DNA- And RNA-Duplexes Covalently Cross-Linked to Regulatory Proteins	Zoe A. Shabarova
2073-2080	Nuclear Targeting of Antisense Oligonucleotides: Modification of Pre-mRNA Splicing or Inhibition of Polyadenylation?	Vittorio. Tomasi; Enzo. Spisni; Cristiana. Griffoni; Spartacos. Santi
2081-2084	Synthesis And Anti-HIV Property of Novel Oligo-DNA Phosphorothioate Analogs Bearing an Intercalative Moiety and/Or Polyamine Residues	Kazuo. Shinozuka; Makoto. Matsukura; Tsuyoshi. Okamoto; Hiroaki. Sawai
2085-2086	Synthetic Strategies Towards the Synthesis of 1–(2,4-Dideoxy-4-C-hydroxymethyl-α-L-Lyxopyranosyl)base Nucleosies.	S. J. Turner; P. Herdewijn
2087-2091	Synthesis of Amide Linked Nucleosides at the 6 Position of Deoxy Inosine and Their application to DNA synthesis, Hybridization Studies.	S. Czernecki; G. Viswanadham; J. M. Valery
2093-2102	Crystal Structures of Four A-DNA Decamers that Contain C5-Propyne-Cytosines	Yi-Gui. Gao; Andrew H. J. Wang
2103-2116	The Parallel and Antiparallel Triplex Formation and Stability of Self Complementary Oligonucleotides Containing 2′-Fluoro-arabinosyl Thymine and 5-Methyl-2′-Deoxycytidine	Wu. Yun Ren; Kyoichi A. Watanabe
2117-2125	Enzymatic and Hybridization Properties of Oligonucleotide Analogues Containing Novel Phosphotriester Internucleotide Linkage	D. Wenninger; M. Hinz; S. Hahner; F. Hillenkamp; H. Seliger
2127-2133	Design of the New Molecular Transport Systems for the Nucleosides-Pharmacophores Carrying.	Yu. Berezovskaya; M. Chudinov; Yu. Kirillova; N. Shastina; V. Shvets; A. Yurkevich
2135-2141	New Peptidyl-Anthraquinones: Synthesis and DNA Binding	Giuseppe. Zagotto; Giovanni. Mitaritonna; Claudia. Sissi; Manlio. Palumbo
2143-2147	The Accurate Detection of One Point Mutations by Ligation of Short Oligonucleotides	V. F. Zarytova; D. V. Pyshnyi; A. A. Krivenko; G. M. Dymshitz; E. M. Ivanova
2149-2152	Special Properties of Modification of SsDNA Target by Alkylating Derivatives of Oligonucleotides in Tandem Complexes	D. V. Pyshnyi; S. G. Lokhov; E. M. Ivanova; V. F. Zarytova
2153-2156	Comparative Study of Modification of DNA and RNA by Oligo(2′-O-Methylribonucleotide) Derivatives	Z. A. Sergeeva; A. G. Venyaminova; V. F. Zarytova
2157-2164	Mass Spectrometric DNA Diagnostics	Dirk. vanden Boom; Christian. Jurinke; Scott. Higgins; Thomas. Becker; Hubert. Köster

Volume 17, Issue 8 (1998)

iii-iv	Contributors to this Issue
1299-1308	Activation of c-jun and c-fos Genes in dNTP Imbalance Cell Death Induced With 5-Fluoro-2′-Deoxyuridine in Mouse Mammary Tumor FM3A Cell Line	Toshifumi Kakutani; Yoko Ebara; Kae Kanja; Kazushige Takahashi; Yusuke Wataya
1309-1317	The Characterization of Cell Death Induced by 1-(3-C-Ethynyl-β-D-ribo-Pentofuranosyl)Cytosine (ECyd) in FM3A Cells	Satoshi Takatori; Shinji Tsutsumi; Muneaki Hidaka; Hiroshi Kanda; Akira Matsuda; Masakazu Fukushima; Yusuke Wataya
1319-1324	As-Triazine Derivatives with Potential Therapeutic Action. XXVI.¹ Synthesis of 5-Substituted-6-Azauracil Acyclonucleosides	Carol Cristescu; Francisc Czobor
1325-1331	Effects of 3′-C-Methylation on the Hydrolytic Stability and Hydroxyl pK_a Values of Dinucleoside 2′,5′- and 3′,5′-Monophosphates	Mikko Oivanen; Ekaterina V. Efimtseva; Sergey N. Mikhailov
1333-1345	A Convenient Synthesis of Acyclic Adenosines with an Unsaturated Side Chain by Modification of 9-(2,3-O-Isopropylidene-D-Ribityl)Adenine	Kosaku Hirota; Yasunari Monguchi; Hironao Sajiki; Chizuko Yatome; Akio Hiraoka; Yukio Kitade
1347-1353	New Approach to the Solid Phase Synthesis of N3′→P5′ Phosphoramidate Oligonucleotides	Janina Baraniak; Dariusz Korczyński; Renata Kaczmarek; Ewa Wasilewska
1355-1363	Synthesis of 1-(β-D-Glycopyranosyl)-3-Deazapyrimidines from 2-Hydroxy and 2-Mercaptopyridines	Adel M. Attia; Galal H. Elgemeie; Ibrahim S. Alnaimi
1365-1372	Synthesis and Reactions of Some 3′,4′-Unsaturated 2′,3′-Secouridine Analogues	Shinya KIKUCHI; Tomohiro MAEKAWA; Katsumaro MINAMOTO; Keizo TANIGAWA
1373-1384	Acyclo C-Nucleoside Analogs. Regioselective Annellation of a Triazole Ring to 5-Methyl-1,2,4-Triazino[5,6-b]Indole and Formation of Certain 3-Poly Hydroxyalkyl Derivatives	Nagwa Rashed; Hamida Abdel Hamid; El Sayed Ramadan; El Sayed H. El Ashry
1385-1407	Synthesis of Acyclo C-Nucleosides OF Phenanthro[9,10-e][1,2,4]Triazino[3,4-c]-[1,2,4] Triazoles, and Their Precursors	Atef Hamed; Elham R. Abo-Amaym; El Sayed H. El Ashry
1409-1443	Synthesis and Antiviral Evaluation of Analogs of Adenosine-N¹-Oxide and 1-(Benzyloxy)Adenosine	Cecil D. Kwong; Charles A. Krauth; Anita T. Shortnacy-Fowler; Gussie Arnett; Melinda G. Hollingshead; William M. Shannon; John A. Montgomery; John A. Secrist III
1445-1451	A New Regio-Defined Synthesis of PMEA	Qun Dang; Van Liu; Mark D. Erion
1453-1471	Synthesis of γ-Phosphate-Linked Nucleoside Affinity Chromatography Resins for Protein Purification, Including Ribonucleoside Triphosphate Reductase	Robert K. Suto; Martin A. Whalen; Bruce R. Bender; Richard G. Finke
1473-1487	Synthesis and Antiviral Activity of Apio Dideoxy Nucleosides with Azido or Amino Substituent	Lak Shin Jeong; Young A. Lee; Hyung Ryong Moon; Moon Woo Chun
1489-1504	Potential Antiviral Agents. Part II. Synthesis and Antiviral Evaluation of Pyrazinones Substituted With Acyclic Chains	Jean Davis; Rachida Benhaddou; Olessia Fedoryak; Robert Granet; Pierre Krausz; Christophe Bliard; Michele De Monte; Anne Marie Aubertin
1505-1513	Synthesis and Biochemical Study of N²-(p-n-Butylphenyl)-2′-deoxyguanosine 5′-(α,β-imido)triphosphate (BuPdGMPNHPP): A Non-Substrate Inhibitor of B Family DNA Polymerases	James M. Stattel; Ivan Yanachkov; George E. Wright

Volume 17, Issue 7 (1998)

iii-iv	Contributors to this Issue
1141-1151	Analogues of Azepinomycin as Inhibitors of Guanase	Vasanthakumar P. Rajappan; Ramachandra S. Hosmane
1153-1162	Substrates of DNA polymerases with planar conformation of sugar: model of substrate transition state?	Alexander A. Krayevsky; Kyoichi A. Watanabe
1163-1175	Synthesis of a new Photo-Cross-Linking Nucleoside Analogue Containing an Aryl(Trifluoromethyl)Diazirine Group: Application for Eco RII and Mva I Restriction-Modification Enzymes	Andrey N. Topin; Oxana M. Gritsenko; Maxim G. Brevnov; Elisaveta S. Gromova; Galina A. Korshunova
1177-1182	The Mechanism of Cleavage Under Basic Conditions of Succinyl-Anchored Oligonucleotides	Yolanda Palom; Anna Grandas; Enrique Pedroso
1183-1190	A Simple and Regioselective Synthesis of ¹³C-Methyl-Labeled Thymedine	Mohammad Ahmadian; Donald E. Bergstrom
1191-1207	The Design and Synthesis of N⁴-Anthraniloyl-2′-dC, the Improved Syntheses of N⁴-Carbamoyl-and N⁴- Ureidocarbamoyl-2′-dC, Incorporation into Oligonucleotides and Triplex Formation Testing	Nancy Guzzo-Pernell; Geoff W. Tregear; Jim Haralambidis; John M. Lawlor
1209-1213	A Simple Synthesis of N⁴-(6-Aminohexyl)-2′-Deoxy-5′-O-(4,4′-Dimethoxytrityl)Cytidine	Jari Hovinen
1231-1236	Novel Diastereomeric Thymidine Cyclic 3′,5′-threo- Phosphoramidates	Darinka Katalenić; Mladen Žinić
1237-1253	Novel Carbocyclic Nucleosides Containing A Cyclobutyl Ring. Guanosine and Adenosine Analogues	José E. R. Borges; Franco Fernández; Xerardo García; Antonio R. Hergueta; Carmen López; Graciela Andrei; Robert Snoeck; Myriam Witvrounw; Jan Balzarini; Erik De Clercq
1255-1266	Synthesis, Antiviral and Cytostatic Activities of Carbocyclic Nucleosides Incorporating a Modified Cyclopentane Ring. Part 2:¹ Adenosine and Uridine Analogues	M. I. Nieto; J. M. Blanco; O. CaamañTo; F. Fernández; X. García-Mera; J. Balzarini; E. Padalko; J. Neyts; E. De Clercq
1267-1274	Reverse Action of Ribonuclease T1 Variants In ICE	Marion Haensler; Heike Schuerer; Ulrich Hahn; Hans-Dieter Jakubke
1275-1287	Chirally-Modifiedoligonucleotides and the Control of Gene Expression. The Case of L-DNAS And-RNAS	Anna Garbesi; Massimo L. Capobianco; Francesco P. Colonna; Mauro Maflini; Danieia Niccoiai; Luisa Tondelli
1289-1297	Oligonucleotide Conjugates Designed for Discriminative Hybridization at Physiological Temperature	I. A. Pyshnaya; D. V. Pyshnii; E. M. Ivanova; V. F. Zarytova; G. M. Bonora; C. Scalfi-Happ; H. Seliger

Volume 17, Issue 6 (1998)

iii-iv	Contributors to this Issue
969-985	A Functional Screening of Adenosine Analogues at the Adenosine A_2B Receptor: A Search for Potent Agonists	Maarten de Zwart; Regina Link; Jacobien K. von Frijtag Drabbe Kunzela; Gloria Cristalli; Kenneth A. Jacobson; Andrea Townsend-Nicholson; Ad P. IJzerman
987-1008	Synthesis, In Vitro Anti-HIV Activity, and Biological Stability of 5′-O-Myristoyl Analogue Derivatives of 3′-Fluoro-2′,3′-Dideoxythymidine (FLT) as Potential Bifunctional Prodrugs of FLT	Keykavous Parang; Edward E. Knaus; Leonard I. Wiebe
1009-1018	Quantitation of Cytidine 3′,5′-Cyclic Monophosphate in Aqueous Solution by UV Absorption Spectrophotometry Independent of Direct Determination of Solution pH	Russell P. Newton
1019-1031	Synthesis and Conformational Analysis of A Novel Type of Spin Labelled Bicyclonucleoside Based on A Tetrahydrofurano[2,3-c]Pyrrolidine Sugar Skeleton	Jean M. J. Tronchet; Laetitia Brenas; Françoise Barbalat-Rey; Martina Zsély; Michel Geoffrey
1033-1051	Synthesis of 5′-C-Branched Thymidines and Conversion to Phosphoramidites	Guangyi Wang; Patrick J. Middleton
1053-1075	Heterocyclic Nucleosede Analogues by Cycloaddition Reactions of 1-Vinylthymine with 1,3-Depoles	David R. Adams; Alan S. F. Boyd; R. Ferguson; David S. Grierson; Claude Monneret
1077-1088	Biological Activity and Phosphorylation of 2′-Azido-2′-Deoxyuridine and 2′-Azido-2′-Deoxycytidlne	Shin HongKang; Moo J. Cho
1089-1098	Synthesis and Biological Activity of BIS(Pivaloyloxymethyl) Ester of 2′-Azido-2′-Deoxyuridine 5′-Monophosphate	Shin HongKang; A. K. Sinhababu; Moo J. Cho
1099-1113	Terminal Fluoroolefins. The Synthesis of Novel Carboacyclic Nucleosides	Shawn C. Miller; James R. McCarthy; Jeffrey S. Sabol
1115-1123	Novel Spironucleosides: 1″,3″-Thiazolidine-2″-Spiro-3′-3′-Deoxyuridine Derivatives	Jean M. J. Tronchet; Imre Kovács; Françoise Barbalat-Rey; Margarita VegaHolm
1125-1140	Regio-and Stereoselective Functionalization of Pyrimidinediones by Cohalogenation with Oxygen Nucleophiles	Nathalie Baret; Jean-Pierre Dulcere; Jean Rodriguez

Volume 17, Issue 5 (1998)

iii-iv	Contributors to this Issue
845-853	Analysis of Antiretroviral Nucleosides by Electrospray Ionization Mass Spectrometry and Collision Induced Dissociation	Eva Font; Sonia Lasanta; Osvaldo Rosario; José F. Rodrígúez
855-868	A Synthetic Strategy to a New Class of Cycloalkane Ring-Fused Pyridine Nucleosides as Potential Anti HIV Agents	Galal E. H. EIgemeie; Adel M. E. Attia; Badria A. W. Hussain
869-874	Facile Synthesis of 8, 2′-S-Cyclopurine Nucleoside	Keiko Tekenaka; Tadakazu Tsuji; Masako Muraoka
875-892	Synthesis and Antiviral Evaluation of Pyrazinones Substituted with Acyclic Chains.	Jean Davis; Rachida Benhaddou; Robert Granet; Pierre Krausz; Michele Demonte; Anne Marie Aubertin
895-899	Functionaleation of Nucleoside Analogs: Regiospecific Conversion of 4″-Hydroxyl Groups to Thioesters and Deoxygenation of 3′-Hydroxyl Groups	Zhen Huang; Steven A. Benner
901-910	Synthesis and Anti-HIV Properties of 1,2,4,6-Thiatriazin-3-one 1,1-Dioxtoe Nucleosides	Carmen Ochoa; Rafael Provencio; Maria Luisa Jimeno; Jan Balzarini; Erik De Clercq
911-923	Effect of Acridine with Various Linker Arms Attached to C5 Position of 2′-Deoxyuridine on the Stability of DNA/DNA and DNA/RNA Duplexes	Hiroaki Ozaki; Yoshinori Ogawa; Masayuki Mine; Hiroaki Sawai
925-937	Synthesis and Triplex Forming Properties of an Acyclic N⁷-Glycosylated Guanine Nucleoside	Aimée St. Clair; Guobing Xiang; Larry W. McLaughlin
939-955	Imidazo-oxazaphosphorines as Precursors to Chiral Phosphite Triesters	Eric Marsault; George Just
957-968	Tri-N-Boc-Tetraazamacrocycle-Nucleoside Conjugates: Synthesis and anti-HIV activities	J. Dessolin; P. Vlieghe; M. Bouygues; M. Medou; G. Qúéléver; M. Camplo; J. C. Chermann; J. L. Kraus

Volume 17, Issue 4 (1998)

iii-iv	Contributors To This Issue
697-709	Aldehydo-oligonucleotides for Bioconjugation	M. Dechamps; E. Sonveaux
711-727	Synthesis and Biological Properties of the Four Optical Isomers of 5-o-Carboranyl-2′,3′-didehydro-2′,3′-dideoxyuridine	Jean-Christophe G. Graciet; Junxing Shi; Raymond F. Schinazi
729-744	1-Deaza-3′-O-methyladenosine: A Nucleoside with the Syn-conformation in the Solid State and in Solution	Frank Seela; Harald Debelak; Hans Reuter; Guide Kastner; Igor A. Mikhailopulo
745-758	Stereoselective Synthesis of Some 3-Nitroglucopyranosyladenine Analogues via a Nitroolefin: Intermediate as Potential Therapeutic Agents	Kazunari TSUBOIKE; Katsumaro MINAMOTO; Gen MIZUNO; Kazufumi YANAGIHARA
759-768	Synthesis AND Adenosine Receptor Affinity of 7-β-D-Ribofuranosylxanthine	Peter K. Bridson; Xu Lin; Neli Melman; Xiao-duo Ji; Kenneth A. Jacobson
769-783	Studies ON Epimeric-D-asabino-and-D-ribo-tetritol-1-yl-2-phenyl-2 H-1,2,3-triazoles. Synthesis and Anomeric Configuration of 4-(α-and β-D-Erythrofuranosyl)-2-phenyl-2 H-1,2,3-Triazole C-Nucleoside Analogs	Mohammed A. E. Sallam; Farida F. Louis; John M. Cassady
785-790	What Are THE Practical Limits for Detection of Minor Nucleoside Reaction Products with HPLC (UV Detection), H NMR, and TLC (UV Detection)?	Morris J. Robins; Sanchita Sarker; Stanislaw F. Wnuk
791-814	Conformational Studies on Nucleosides with Furanose Ring Modifications. 1.	Shashidhar N. Rao
815-829	Aminoacyl-tRNA Analogues; Synthesis, Purification and Properties of 3^′-Anthraniloyl Oligoribonucleotides	B. Nawrot; M. Sprinzl
831-841	Structural Characterization of a DNA Duplex Modeled on a DNA:RNA Hybrid of the Polypurine Tract Recognized by a Reverse Transcriptase	Mayumi Kanagawa; Yutaka Okada; Sciichi Uesugi; Hirofumi Doi; Masato Katahira
843	In Memoriam

Volume 17, Issue 1-3 (1998)

xi-xiv	Contributors to this Issue
xv-xxvii	Biography
1-13	Asymmetric Synthesis of Oxazolidine Nucleosides and Related Chemistry	Jinfa Du; Chung K. Chu
15-27	Synthesis of 2-Alkynylcordycepins and Evaluation of Their Vasodilating Activity	Hiroki Kumamoto; Hiroyuki Hayakawa; Hiromichi Tanaka; Satoru Shindoh; Keisuke Kato; Tadashi Miyasaka; Kazuki Endo; Haruhiko Machida; Akira Matsuda
29-38	Efficient Syntheses of (E)-5-(2-Bromovinyl)-2′-deoxy-4-thiouridine; A Nucleoside Analogue with Potent Biological Activity	I. Basnak; G. P. Otter; R. J. Duncombe; N. B. Westwood; M. Pietrarelli; G. W. Hardy; G. Mills; S. G. Rahim; R. T. Walker
39-52	Synthesis of 2′,3′-Didehydro-2′,3′-dideoxyisoinosine and Oxidation of Fluorescent 2-Hydroxypurine Nucleosides by Xanthine Oxidase	Frank Seela; Yaoming Chen; Markus Sauer
53-63	Synthesis of 2′,3′,6′-Trideoxy-β-D-erythro-hexopyranosyl Nucleosides Employing Intramolecular Glycosylation as a Key Step	H. Sugimura; K. Sujino
65-79	Synthesis and Antiviral Activities of 5-Substituted 1-(2-Deoxy-2-C-methylene-4-thio-β-D-erythro-pentofuranosyl)uracilst	Hiroshi Satoh; Yuichi Yoshimura; Mikari Watanabe; Noriyuki Ashida; Katsushi Ijichi; Shinji Sakata; Haruhiko Machida; Akira Matsuda
81-89	Deamination of Cyclaradine by Adenosine Deaminase Under High Pressure	Nobuya Katagiri; Hideaki Kokufuda; Masashi Makino; Robert Vince; Chikara Kaneko
91-97	Facile Method for the Preparation of 7-Methyl-8-oxoguanosines as an Immunomodulator	Yukio Kitade; Naohiro Saito; Atushi Kozaki; Kazumasa Takahashi; Chizuko Yatome; Yoshifumi Takeda; Hironao Sajiki; Kosaku Hirota
99-113	Synthesis of Homologated Halovinyl Derivatives from Aristeromycin and Their Inhibition of Human Placental S-Adenosyl-L-homocysteine Hydrolase	Stanislaw F. Wnuk; Chong- Sheng Yuan; Ronald T. Borchardt; Morris J. Robins
115-122	Synthesis of 8-Substituted Analogs of 3′-Deoxy-3′-fluoroadenosine¹⁾	Tokumi Maruyama; Yoshiko Sato; Takeshi Sakamoto
123-130	Synthesis of Chlorodideoxynucleosides Using Tris(2,4,6-tribromophenoxy)-dichlorophosphorane (BDCP)	R. K. Singh; S. Ohuchi; T. Wada; T. Hata
131-141	Novel Modification of 5-Formyluracil by Cysteine Derivatives in Aqueous Solution	Hiroaki Terato; Hajime Morita; Yoshihiko Ohyama; Hiroshi Ide
143-151	Photosensitized Preparation of Fluorescent Luminarosine and Analogues	A. Burdzy; B. Skalski; S. Paszyc; Z. Gdaniec; R. W. Adamiak
153-159	New Approach to the Synthesis of 2′,3′-dideoxyadenosine and 2′,3′-Dideoxyinosine	K. V. Antonov; I. D. Konstantinova; A. I. Miroshnikov
161-173	Synthesis of 5-Arylthiouridines via Electrophilic Substitution of 5-Bromouridines with Diaryl Disulfides	Kosaku Hirota; Tetsuo Tomishi; Yoshifumi Maki; Hironao Sajiki
175-186	Nucleosides. LXII. Synthesis of 6-Methyl-8-(2-deoxy-β-D-ribofuranosyl)-isoxanthopterin and Derivatives	M. Melguizo; M. Gottlieb; R. Charubala; W. Pfleiderer
187-206	Some 6-Aza-5-substituted-2′-deoxyuridines Show Potent and Selective Inhibition of Herpes Simplex Virus Type 1 Thymidine Kinase	I. Basnak; M. Sun; T. A. Hamor; F. Focher; A. Verri; S. Spadari; B. Wroblowski; P. Herdewijn; R. T. Walker

Volume 17, Issue 1-3 (1998)

207-218	Design and Anti-HIV-1 Activity of Hammerhead and Hairpin Ribozymes Containing a Stable Loop	Makoto Koizumi; Yuji Ozawa; Ryuichi Yagi; Takashi Nishigaki; Masakatsu Kaneko; Shin-ichi Oka; Satoshi Kimura; Aikichi Iwamoto; Yasuo Komatsu; Eiko Ohtsuka
219-231	Synthesis of Chirally Pure Ornithine Based PNA Analogues	Alexander C. van der Laan; Irene van Amsterdam; Godefridus I. Tesser; Jacques H. van Boom; Esther Kuyl- Yeheskiel
233-242	Synthesis and Binding Properties of Oligonucleotides Containing an Azobenzene Linker	Kazushige Yamana; Akira Yoshikawa; Rie Noda; Hidehiko Nakano
243-252	Biologically Active Oligodeoxyribonucleotides. X. Anti-HIV-1 Activity and Stability of Modified Hexanucleotides Containing Glycerol-Skeleton	Hitoshi Hotoda; Makoto Koizumi; Toshinori Ohmine; Hidehiko Furukawa; Takashi Nishigaki; Koji Abe; Toshiyuki Kosaka; Shinya Tsutsumi; Junko Sone; Masakatsu Kaneko; Satoshi Kimura; Kaoru Shimada
253-267	The Reactions of H-Phosphonates with Bifunctional Reagents. V. Functionalization of Support-Bound Oligonucleotides and Synthesis of Nonradioactive Hybridization Probes	Michal Sobkowski; Adam Kraszewski; Jacek Stawiński
269-282	Preparation of Stereoregulated Antisense Oligodeoxyribonucleoside Phoshorothioate and Interaction with its Complementary DNA And RNA	Yutaka Tamura; Hidetaka Miyoshi; Tomoyuki Yokota; Keisuke Makino; Akira Murakami
283-289	Nucleosides and Nucleotides. 165. Chemical Ligation of Oligodeoxynucleotides Having a Mercapto Group at the 5-Position Of 2′-Deoxyuridine via a Disulfide Bond	Yoshihito Ueno; Aiko Nakagawa; Akira Matsuda
291-300	Facile Post-Synthetic Derivatization of Oligodeoxynucleotide Containing 5-Methoxycarbonylmethyl-2′-Deoxyuridine	Kazuo Shinozuka; Akira Umeda; Tsuyoshi Aoki; Hiroaki Sawai
301-308	Two Hydrolase Resistant Analogues of Diadenosine 5′,5″′-P,P-Triphosphate for Studies with FHIT, The Human Fragile Histidine Triad Protein	G. Michael Blackburn; Xiaohai Liu; Angelika Rösler; Charles Brenner
309-316	Synthesis of Novel Oligodeoxynucleotide Conjugates Containing the Anionophoric Moiety of Pamamycin	E. Uhlmann; L. Hornung; D. W. Will; U. Gräfe
317-326	Methylphosphonate Modified DNA Hairpin Loops	Markus Schweitzer; Joachim W. Engels
327-338	The Chemical Synthesis of E. coli tRNA^Lys Anticodon Loop Fragment and Its Analogues	E. Sochacka
339-350	Isopoly-L-ornithine Derivatives of Thymine and Thymidine	Yoshiaki Inaki; Norimitsu Tohnai; Keiko Miyabayashi; Takehiko Wada; Mikiji Miyata
351-364	Stereocontrolled Synthesis of Dithymidine Phosphorothioates by Use of a Functionalized 5′- Protecting Group Bearing an Imidazole Residue	Takeshi Wada; Naotake Kobayashi; Toshiya Mori; Mitsuo Sekine
365-378	A Reinvestigation of Sulfenyl Groups as Amino Protecting Groups for the Synthesis of Oligonucleotides on Solid Support by Phosphoramidite Chemistry	Karine Alvarez; Isabelle Tworkowski; Jean- Jacques Vasseur; Jean- Louis Imbach; Bernard Rayner
379-396	Convenient Approaches to the Synthesis of Oligonucleotide Macrocycles Containing Non-nucleotide Linkers	V. A. Efimov; A. A. Buryakova; A. L. Kalinkina; M. V. Choob; O. G. Chakhmakhcheva; J. O. Ojwang; R. F. Rando
397-410	Intraduplex Photo-cross-linking of p-Azidoaniline Residue and Amino Acid Side Chains Linked to the Complementary Oligonucleotides via a New Phosphorylating Intermediate Formed in the Mukaiyama System	Dmitri G. Knorre; Pave V. Alekseyev; Yulia V. Gerassimova; Vladimir N. Silnikov; Galiya A. Maksakova; Tatyana S. Godovikova
411-424	Studies on Synthesis and Structure of O-β-D-Ribofuranosyl(1″→2′)-ribonucleosides and Oligonucleotides	Wojciech T. Markiewicz; Anna Niewczyk; Zofia Gdaniec; Dorota A. Adamiak; Zbigniew Dauter; Wojciech Rypniewski; Marcin Chmielewski
425-440	Synthesis and Properties of Modified Oligodeoxyribonucleotides Containing 9-(2-Amino-2-deoxy-β-D-arabinofuranosyl)adenine	Eugene M. Zubin; Sergey I. Antsypovich; Tatiana S. Oretskaya; Elena A. Romanova; Eugene M. Volkov; Vadim N. Tashlitsky; Nina G. Dolinnaya; Zoe A. Shabarova
441-449	Electrochemical Removal of Allylic Protecting Groups in Nucleotide Synthesis	Yoshihiro Hayakawa; Rie Kawai; Shigeharu Wakabayashi; Mamoru Uchiyama; Ryoji Noyori

Volume 17, Issue 1-3 (1998)

451-470	Preparation of an Octadeoxyribonucleoside Heptaphosphorothioate by the Phosphotriester Approach in Solution	Colin B. Reese; Quanlai Song; M. Vaman Rao; Ian Beckett
471-478	Inhibition of Influenza Virus Replication by Phosphorothioate and Liposomally Endocapsulated Oligonucleotides	Takayuki Abe; Toshihmi Hatta; Kazuyuki Takai; Hideki Nakashima; Tomoyuki Yokota; Hiroshi Takaku
479-486	Stereospecificity of 6′-C-Neplanocin A Analogues as Inhibitors of S-Adenosylhomocysteine Hydrolase Activity and Human Immunodeficiency Virus Replication	D. Daelemans; Anne- Mieke Vandamme; Satoshi Shuto; Akira Matsuda; Erik De Clercq
487-501	Synthetic Nucleosides and Nucleotides. 40. Selective Inhibition of Eukaryotic DNA Polymerase α by 9-(β-D-Arabinofuranosyl)-2-(p-n-butylanilino)adenine 5′-Triphosphate (BuAaraATP) and Its 2′-Up Azido Analog: Synthesis and Enzymatic Evaluations	Aki Tomikawa; Masaki Seno; Kunie Sato-Kiyotaki; Chizuru Ohtsuki; Toshialu Hirai; Toyofumi Yamaguchi; Takeo Kawaguchi; Shonen Yoshida; Mineo Saneyoshi
503-513	Repair Kinetics of Abasic Sites in Mammalian Cells Selectively Monitored by the Aldehyde Reactive Probe (ARP)	Ayumi Asaeda; Hiroshi Ide; Keizo Tano; Yasuhiko Takamori; Kihei Kubo
515-530	Structurally Altered Substrates for DNA Topoisomerase. I. Effects of Inclusion of a Single 3′-Deoxynucleotide Within the Scissile Strand	Tuncer Arslan; Anil T. Abraham; Sidney M. Hecht
531-539	Ascidian Mitochondrial tRNA^Met Possessing Unique Structural Characteristics	Akiko Kondow; Shin-ichi Yokobori; Takuya Ueda; Kimitsuna Watanabe
541-554	DNA Polymerase Incorporation of Universal Base Triphosphates	C. L. Smith; A. C. Simmonds; I. R. Felix; A. L. Hamilton; S. Kumar; S. Nampalli; D. Loakes; F. Hill; D. M. Brown
555-564	Use of 5-Nitroindole-2′-deoxyribose-5′-triphosphate for Labelling and Detection of Oligonucleotides	C. L. Smith; A. C. Simmonds; A. L. Hamilton; D. L. Martin; A. G. Lashford; D. Loakes; F. Hill; D. M. Brown
565-574	Effect of Cu² on Complex Formation Between a Deoxyribozyme and Its Substrates	Naoki Sugimoto; Noboru Wakizaka
575-584	Characterization of Telomeric Oligonucleotides: Fidelity of Repetitive Nucleotide Sequences	Toshio Shida; Mitsuaki Suda; Junichi Sekiguchi
585-592	Stabilization of Deoxyadenosine/polynucleotide Complexes by 3′,5′-Di-O-Benzoyl Substituents	S. K. Chaturvedi; R. L. Letsinger
593-601	Sequence Selective Interaction Between Nucleotides and Intercalators Bound to Water Soluble Dextran: An Application to the Affinity Chromatography of Dinucleotides	Ryuichi Shirai; Taro Ito; Shigeo Iwasaki; Yuichi Hashimoto
603-611	Interaction of Pyrylium Dye with Self-Complementary DNA Oligomer as Studied by H NMR Spectroscopy	Kenji Kanaori; Kayo Yokoyama; Kunihiko Tajima; Nobuko Yamamoto; Tadashi Okamoto; Keisuke Makino
613-623	Cerium(IV)/Lanthanide(III)/Dextran Ternary Solutions for Efficient and Homogeneous DNA Hydrolysis	Jun Sumaoka; Ayako Kajimura; Takamitsu Imai; Masayuki Ohno; Makoto Komiyama
625-634	Carbocyclic Adenosine Analogues as S-Adenosylhomocysteine Hydrolase Inhibitors and Antiviral Agents: Recent Advances	Erik De Clerq
635-647	Boron Containing Oligonucleotides	Raymond F. Schinazi; Zbigniew J. Lesnikowski
649-662	Design of Functional Diversity in Oligonucleotides via Zwitter-Ionic Derivatives of Deprotected Oligonucleotides	V. Zarytova; E. Ivanova; A. Venyaminova
663-680	Nucleotide Analogues Containing the P-F Bond. An Overview of the Synthetic Methods	Martin Bollmark; Jacek Stawiński
681-693	dNTP Modified at Triphosphate Residues: Substrate Properties Towards DNA Polymerases and Stability in Human Serum	Alexander Krayevsky; Andrey Arzumanov; Elena Shirokova; Natalya Dyatkina; Lyubov Victorova; Maxim Jasko; Ludmila Alexandrova
695	Announcement

Volume 16, Issue 12 (1997)

iii-iv	Contributors to This Issue
2095-2099	A 5′-Noraristeromycin Enantiomer with Activity Towards Hepatitis B Virus	Katherine L. Seley; Stewart W. Schneller; Brent Korba
2101-2110	Solution NMR Conformational Analysis of the Potent Equilibrative Sensitive (ES) Nucleoside Transporter Inhibitor, S⁶-(4-Nitrobenzyl)mercaptopurine Riboside (NBMPR)	John K. Buolamwini; Joseph J. Barchi Jr.
2111-2122	Cytidine Kinase: A Novel Pyrimidine Ribonucleoside Phosphorylating Enzyme in Escherzchza Coli	Tsuguhisa Kaneko; Hiroshi Yamamoto
2123-2131	Trans-Adenosine 3′,5′-Cyclic N,N-Dimethylphosphoramidate Ether Solvate, a Cyclic Nucleotide with an Equatorial Dimethylamino Group on Phosphorus	Sándor Bottka; Jenoö Tomasz; W. B. T. Cruse; Shude Zhang; Olga Kennard
2133-2150	A General Synthetic Method of 5-Carboranyluracil Nucleosides with Potential Antiviral Activity and use in Neutron Capture Therapy	Naganna M. Goudgaon; Yahya A. El-Kattan; Xiaoyang Xia; Jeff McAtee; José Soria; Shiow-Jyi Wey; Dennis C. Liotta; Raymond F. Schinazi
2151-2164	Transprotection of N-Benzoylated Nucleobase Derivatives by Dialkylaminomethylene Group	Magdalena Endová; Milena Masojidková; Ivan Rosenberg
2165-2192	Synthesis of the Optically Active Carbocyclic Analogs of the Four 2′-Deoxyribonucleoside Monophosphates	Laurent Schmitt; Carol A. Caperelli
2193-2218	Study of Creatinine and its 5-Alkoxy Analogs: Structure and Conformational Studies in the Solid and Solution States by X-Ray Crystallography, NMR, UV and Mass Spectrometry	Aruna V. Arakali; J. McCloskeyt; R. Parthasarathy; J. L. Alderfer; G. B. Chheda; T. Srikrishnan
2219-2231	Relationship Between Conformation and Antiviral Activity -IV. 5-Ethyl-2′-Deoxyurldine and 5-Ethyl-2′-Deoxycytidine	Allan L. Stuart; Sashi V. P. Kumar; Sagar V. Gupta; Wajdi M. Zoghaib; Scott Napper; Keith C. Brown; Shajan Mannala; Louis T. J. Delbaere
2233	Announcement

Volume 16, Issue 10-11 (1997)

iii-iv	Contributors to This Issue
1809-1820	The Synthesis of Oligonucleotides Containing Fluoro-2′-Deoxycytidine for Secondary Structure Determination of Tandem Tetraloop DNA Analogs	Caryn Evilia; Xiaolin Zhang; Jean Kanyo; Ponzy Lu
1821-1836	Incorporation of 5′-N-BOC-2′, 5′-Dideoxynucleoside-3′-O-Phosphoramidites Into Oligonucleotides by Automated Synthesis	Kenneth D. James; Guenter von Kiedrowski; Andrew D. Ellington
1837-1846	A New Phosphoramidite Reagent for the Incorporation of Diazaphenoxazinone Nucleoside With Enhanced Base-Pairing Properties into Oligodeoxynucleotides	Nikolay A. Kurchavov; Dmitry A. Stetsenko; Nadezhda V. Skaptsova; Victor K. Potapov; Eugene D. Sverdlov
1847-1854	Calorimetric Evidences for Copper(II)-Regulated Chiral Recognition Between Decanucleotide 5′d(CTGGATCCAG)₂ and ALA-TRP Dipeptides	Vincenzo Cucinotta; Domenico Grasso; Giulia Grasso; Danilo Milardi
1855-1873	A 2′←5′-Adenylate Trimer With a Positively Charged 2′(3′)-Terminal 8-(4-Aminobunl)Aminoadenosine Residue: Synthesis, Conformation and RNase L Binding	Igor A. Mikhailopulo; Elena N. Kalinichenko; Tatjana L. Podkopaeva; Merike Kelve; Mart Saarma; Margeris Y. Lidaks; Helmut Rosemeyer; Frank Seela
1875-1882	Pα-Methyl Deoxynucleoside Triphosphates as Substrates for E. COLI DNA Polymerase I in a Template-Directed Synthesis of DNA	Magda A. Dineval; Ivan G. Ivanov; Dimiter D. Petkov
1883-1891	Polyethylelimine Masks Mitogenic Effect of DNA	Pavel P. Laktionov; Elena Yu. Rykova; Valentin V. Vlassov
1893-1906	Liquid Phase Synthesis of Peptide Nucleic Acid (or Polyamide Nucleic Acid) Dimers	Audrey Farese; Sandrine Pairot; Nadia Patino; Vkronique Ravily; Roger Condom; Andreacute Aumelass; Roger Guedj
1907-1920	Enzymatic Synthesis of 2′,5′-Dideoxv Purine Nucleosides and Related Compounds	Reza Fathi; Kenneth J. Nawoschik; Melissa Zavoda; Alan F. Cook
1921-1932	Synthesis of Unsaturated Analogues of 9-[2(Phosphono- Methoxy)Propyl]Guanine as Antiviral Agents	Palmarisa Franchetti; Ghassan Abu Sheikha; Paolo Perlini; Farhat Farhat; Mario Grifantini; Graziella Perra; Carlo Milia; Monica Putzolu; Paolo La Colla; Maria Elena Marongiu
1933-1950	Synthesis and Incorporation of 5″-Amino- and 5′-Mercapto-5′-Deoxy-2′-O-Methyl Nucleosides Into Hammerhead Ribozymes	Jasenka Matulic-Adamic; Peter Haeberli; Anthony B. DiRenzo; Victor R. Mokler; Lara Maloney; Leonid Beigelman; Nassim Usman; Francine E. Wincott
1951-1959	3′-Terminal Modification of Oligonucleotides Using a Universal Solid Support	Paul S. Nelson; Sylvester Muthini; Mark A. Kent; Thomas H. Smith
1961-1965	Synthesis of a Novel Carbocyclic Nucleoside	George A. Kraus; Todd Begey; Xuemei Wang
1967-1981	Cytldlne Cyclic (3′, 5′) Monophosphate: Cyclic Nucleotide With a Non-Characteristic Ribose Ring Conformation	R. Parthasarathy; T. Srikrishnan
1983-1998	Studies on the Synthesis of S^5′,6-Methano-5′-Thiourldines	Mallela S. P. Sarma; Marianne R. Spada; Sreenivasulu Megati; Robert S. Klein; Brian A. Otter
1999-2012	Novel 2′-Deoxy Pyrazine C-Nucleosides Synthesized VIA Palladium-Catalyzed Cross-Couplings	John A. Walker II; Jiong J. Chen; Jack M. Hinkley; Dean S. Wise; Leroy B. Townsend
2013-2018	Selforganization of Nucleic Acids Visualized by Scanning Force Microscopy	C. Bohley; T. Martini; G. Bischoff; S. Lindau; E. Birch-Hirschfeld; S. Kargov; W. -V. Meister; J. Barthel; S. Hoffmann
2019-2024	Synthesis of 5-Formyluridines	Sidney D. Selvidge III; James Jang; Partha S. Ray

Volume 16, Issue 10-11 (1997)

2025-2033	Ring Opening Reaction of Pyrazolo[3,4-c]Maleimide Nucleosides	Sungjoong Kim; Wooyeon Won; Yonghan Kang
2035-2051	Synthesis of Oligodeoxynucleotides Containing 2-Substituted Guanine Derivatives Using 2-Fluoro-2′-Deoxyinosine as Common Nucleoside Precursor	Antonio R. Diaz; Ramon Eritja; Ramon Guimil Garcia
2053-2068	Synthesis and Stability of Oligonucleotide Duplexes Containing N4 Aralkyl-Substituted Cytosine Bases	Mark P. Wallis; Carl H. Schwalbe; William Fraser
2069-2077	Quantitative One Step Derivatization of Oligonucleotides by a Fluorescent Label Through Abasic Site Formation	Didier Boturyn; Eric Defrancq; Veacute onique Ducros; Catherine Fontaine; Jean Lhomme
2079-2092	Synthesis, Biological Activity and Decomposition Studies of Amino Acid Phosphomonoester Amidates of Acyclovir	Timothy W. Abraham; Edward J. Mclntee; Vidhya V. Iyer; Raymond F. Schinazi; Carston R. Wagne
2093	Announcement

Volume 16, Issue 7-9 (1997)

xxv-xxxv	Contributors to This Issue
xxxvii-xliii	Preface	P. Dan Cook
889-898	Antisense Properties of Morpholino Oligomers	James Summerton; Dwight Weller
899-905	Synthesis and Properties of the Oligonucleotide N3′ →P5′ Phosphoramidates	Sergei M. Gryaznov
907-916	Concept, Discovery and Development of MMI Linkage: Story of a Novel Linkage: for Antisense Constructs	Yogesh S. Sanghvi; Eric E. Swayze; Didier Peoc'h; Balkrishen Bhat; Stuart Dimock
917-926	Second Generation Antisense Oligonucleotides—Inhibition of PKC-α and c-raf Kinase Expression by Chimeric Oligonucleotides Incorporating 6″-Substituted Carbocyclic Nucleosides and 2″-O-Ethylene Glycol Substituted Ribonucleosides	Karl-Heinz Altmann; Pierre Martin; Nicholas M. Dean; Brett P. Mania
927-936	Mixed-Backbone Oligonucleotides Containing Phosphorothioate and Methylphosphonate Linkages as Second Generation Antisense Oligonucleotide	Sudhir Agrawal; Zhiwei Jiang; Qiuyan Zhao; Denise Shaw; Daisy Sun; Carl Saxinger
937-939	A Convenient Synthesis of Deoxynebularine Phosphoramidite	Douglas Picken; Vicki Gault
941-944	Positioning of Functionalities in a Heteroduplex Major Groove: Synthesis of 7-Deaza-2-Amino-2′-deoxyadenosines	Guity Balow; John Brugger; Elena Lesnik; Oscar L. Acevedo
945-949	Oligonucleotide Phosphonates—Solid Phase Synthesis and Biochemical Characterization	D. Bankaitis-Davis; L. Huang; T. Koga; G. Beaton
951-954	Amino-Linked Ribozymes: Post-Synthetic Conjugation of Half-Ribozymes	Laurent Bellon; Christopher Workman; Carolyn Gonzalez; Francine Wincott
955-958	2′-O-Methyl Thiomethyl Modifications in Hammerhead Ribozymes	Alexander Karpeisky; Carolyn Gonzalez; Alex B. Burgin; Nassim Usman; Leonid Beigelman
959-962	Synthesis and Evaluation Of 2″-Modified MMI Linked Dimers in Antisense Constructs	Didier Peoc'h; Eric E. Swayze; Balkrishen Bhat; Stuart Dimock; Richard Griffey; Yogesh S. Sanghvi
963-966	Duplex Stability of Oligonucleotides Containing 7-Substituted 7-Deaza- and 8-Aza-7-Deazapurine Nucleosides	F. Seela; N. Ramzaeva; M. Zulauf
967-970	Synthesis and Properties of Oligoribonucleotide Analogues Having Amide (3″-CH₂-CO-NH-5′) Internucleoside Linkages	Eriks Rozners; Roger Strömberg
971-972	The Synthesis of the Sixteen Possible 2′-O-Methyl MMI Dimer Phosphoramidites: Building Blocks for the Synthesis of Novel Antisense Oligonucleotides	Eric E. Swayze; Balkrishen Bhat; Didier Peoc'h; Yogesh S. Sanghvi
973-976	Hexitol Nucleic Acids (HNA): Synthesis and Properties	B. De Bouvere; L. Kerreinans; C. Hendrix; H. De Winter; G. Schepers; A. Van Aerschot; P. Herdewijn
977-980	Synthesis and Hybridization Properties of Modified Oligonucleotides with PNA-DNA Dimer Blocks	D. Wenninger; H. Seliger
983-992	Therapeutic Potential of HPMPC (Cidofovir), PMEA (Adefovir) and Related Acyclic Nucleoside Phosphonate Analogues as Broad-Spectrum Anttviral Agents	Lieve Naesens; Erik de Clercq
993-1001	Structure-Activity Relationship of Pyrimidine Heterosubstituted Nucleoside Analogues	Tarek S. Mansour; Colleen A. Evans; M. Arshad Siddiqui; Marie Charron; Boulos Zacharie; Nghe Nguyen-Ba; Nola Lee; Brent Korba
1003-1012	Antiviral Nucleoside Analogues with Axial Chirality	Jiri Zemlicka
1013-1021	Design, Synthesis and Anticonvulsant Activity of the Potent Adenosine Kinase Inhibitor GP3269	Mark D. Erion; Bheemarao G. Ugarkar; Jay DaRe; Angelo J. Castellino; James M. Fujitaki; Ross Dixon; James R. Appleman; James B. Wiesner
1023-1032	Synthesis and Properties of Conformationally Rigid Cyclouridylic Acids Having Covalent Bonding Linkers Between the Uracil 5-Position and the 5′-Phosphate Group	Kohji Seio; Osamu Kurasawa; Takeshi Wada; Kensaku Sakamoto; Shigeyuki Yokoyama; M. Sekinea
1033-1036	Novel Analogues of the Anti-HIV-1 Agent TSAO-T Modified at the 3′-Spiro Moiety	Rosa Alvarez; María-Luisa Jimeno; Erik De Clercq; Jan Balzarini; María-José Camarasa
1037-1039	Intracellular Metabolism and Action of an Antitumor Nucleoside, 2′-C-Cyano-2′-Deoxy-1-β-d-arabinofuranosylcytosine (CNDAC)	Atsushi Azuma; Peng Huang; Akira Matsuda; William Plunkett
1041-1044	Vibrational Study of a Nucleoside Analogue with Antitumoral and Antiviral Activity, 5-Fluoro-2′-deoxyuridine, FdU	L. Bailey; A. Hernanz; R. Navarro
1045-1048	Synthesis and Cytotoxic Activity of Selenophenfurin, a New Inhibitor of IMP Dehydrogenase	L. Cappellacci; P. Franchetti; G. Abu Sheikha; H. N. Jayaram; V. V. Gurudutt; T. Sint; B. P. Schneider; B. M. Goldstein; G. Perra; S. Poma; P. La Colla; M. Grifantini
1049-1052	Synthesis of Homo-C-D4T and Homo-C-Thymidine	Bogdan Doboszewski
1053-1057	Irreversible, Tight-Binding Inhibition of Adenosine Deaminase by Coformycins: Inhibitor Structural Features That Contribute to the Mode of Enzyme Inhibition	Mikyung Hong; Ramachandra S. Hosmane

Volume 16, Issue 7-9 (1997)

1059-1062	Synthesis and Anti-HIV Activity of Carbocyclic Ring-Enlarged 4′,1′a-Methano Oxetanocin Analogues	Lak S. Jeong; Min Bae; Moon W. Chun; Victor E. Marquez
1063-1066	Synthesis of Novel 3′-C-Hydroxymethyl Nucleosides by a Convergent Strategy	Pia Nørregaard Jørgensen; Jesper Wengel
1067-1071	Synthesis of the Sulfonylpyrimidine Derivatives as a New Type of Sulfonylcycloureas	Biserka Kašnar; Irena Krizmanić; Mladen Žinić
1073-1077	Synthesis of 3′-Deoxy-3′ and 5′-Deoxy-5′-[4-(Purin-9-yl/Pyrimidin-1-yl) methyl-1,2,3-Triazol-1-yl]thymidine via 1,3-Dipolar Cycloaddition	H. B. Lazrek; M. Taourirte; T. Oulih; Y. Kabbaj; J. L. Barascut; J. L. Imbach; N. A. Almasoudi; W. Pfleiderer
1079-1082	Synthesis of N-Arylinosines	Tokumi Maruyama; Yoshiko Sato; Takeshi Goto; Mitsutoshi Fukuhara
1083-1086	Synthesis and Biological Evaluation of 2′,3′-Dideoxy-3′-Fluororibofuranosyl Purine Nucleosides	Nicolai E. Poopeiko; Natalia B. Khripach; Zygmunt Kazimierczuk; Jan Balzarini; Erik De Clercq; Igor A. Mikhailopulo
1087-1090	Dinucleotides Incorporating Isomeric Nucleosides: Synthesis, Structural and Stereochemical Characterization, and Enzymology	Tamera S. Jahnke; Qi Chao; Vasu Nair
1091-1094	Synthesis of New Dideoxynucleosides Bearing Ring-Extended Nucleobases	Jianzhong Zhang; Vasu Nair
1095-1097	Novel Intramolecular Introduction of Nucleophiles To 2,2′-Anhydrouridine	Danny P. C. McGee; Alecia Vaughn-Settle
1099-1102	4-Substituted Uridine 5′-Triphosphates as Agonists of the P_2Y2 Purinergic Receptor	Sammy R. Shaver; William Pendergast; Suhaib M. Siddiqi; Benjamin R. Yerxa; Dallas K. Croom; Robert W. Dougherty; Michael K. James; A. Neil Jones; Janet L. Rideout
1103-1106	Synthesis and Biological Activities of 2′-Modified 4′-Thionucleosides	Yuichi Yoshimura; Kenji Kitano; Mikari Watanabe; Hiroshi Satoh; Shinji Sakata; Shinji Miura; Noriyuki Ashida; Haruhiko Machida; Akira Matsuda
1107-1110	Addition of 2,3-Dihydrofuran to N₂-Acetyl-8-bromoguanine	M. Madre; R. Zhuk; G. -J. Koomen
1111-1114	Synthesis and Properties of Oligonucleotides Containing 5-Aza-2′-deoxycytidine	Ramon Eritja; Victor E. Marquez; Ramon Güimil García
1115-1118	Synthesis of New 1,2,3-Triazole Acyclonucleoside Analogues of ACV and HBG	H. B. Lazrek; M. Taourirte; T. Oulih; M. Lebtoumi; J. L. Barascut; J. L. Imbach
1121-1127	Delivery of Polynucleotides with Polyamine Lipids and Polymers	B. A. Demeneix; O. Boussif; M. A. Zanta; J. S. Remy; J. P. Behr
1129-1138	Conjugated Antisense Oligonucleotides	Muthiah Manoharan; Kathleen L. Tivel; Thomas P. Condon; Laura K. Andrade; Isabelle Barber-Peoch; Gopal Inamati; Shefali Shah; Venkatraman Mohan; Mark J. Graham; C. Frank Bennett; Stanley T. Crooke; P. Dan Cook
1139-1140	Cholesterol Conjugated Uniform and Gapmer Phosphorothioate Oligonucleotides Targeted Against PKC-α and C-raf Gene Expression	Muthiah Manoharan; Kathleen L. Tivel; Gopal Inamati; Brett P. Monia; Nick Dean; P. Dan Cook
1141-1143	2′- and 3′- Cholesterol-Conjugated Adenosine and Cytosine Nucleoside Building Blocks: Synthesis of Lipidic Nucleic Acids	Muthiah Manoharan; Gopal Inamati; Kathleen L. Tivel; Boyd Conklin; Bruce S. Ross; P. Dan Cook
1145-1153	Preclinical Profiling of Modified Oligonucleotides: Anticoagulation and Pharmacokinetic Properties	Paul L. Nicklin; John Ambler; Andrew Mitchelson; Deborah Bayley; Judy A. Phillips; Sarah J. Craig; Brett P. Mania
1155-1163	Enhanced Antisense Effects Resulting from an Improved Streptolysin-O Protocol for Oligodeoxynucleotide Delivery into Human Leukaemia Cells	R. V. Giles; J. Grzybowski; D. G. Spiller; D. M. Tidd
1165-1168	Modification of a Phosphorothioate Oligonucleotide with Cholesterol Induces Association of the Oligonucleotide to Serum Lipoproteins and Affects Its Biological Fate	Martin K. Bijsterbosch; Muthiah Manoharan; Kathleen L. Tivel; Erik T. Rump; Erik A. L. Biessen; Remco L. A. De Vrueh; P. Dan Cook; Theo J. C. van Berkel
1169-1172	Conjugated Antisense Oligonucleotides for Inhibition of Human Cytomegalovirus In Vitro	Zhaoda Zhang; Jean A. Smith; Adrienne P. Smyth; Warren Eisenberg; Alexandra Nichols; Gregory S. Pari; Jin Yan Tang
1173-1182	Restoration of ß-Globin Gene Expression in Mammalian Cells by Antisense Oligonucleotides That Modify the Aberrant Splicing Patierns of Thalassemic Pre-mRNAs	Halina Sierakowska; Michael Montague; Sudhir Agrawal; Ryszard Kole
1183-1194	Targeted Gene Correction: Synthesis and Characterization of Double-Hairpin 2′-O-Methyl RNA/DNA Chimera Oligonucleotides	Alex Andrus; Ravi Vinayak; Robert G. Kuimelis; Bashar Mullah
1195-1199	Inhibition of 5-α-Reductase (TYPE-II) Expression by Antisense 3′-Deoxy-(2′-5′) Oligonucleotide Chimeras	Purshotam Bhan; Anila Bhan; Mikung Hong; John G. Hartwell; June M. Saunders; Glenn D. Hoke
1201-1204	Synthesis of (2′,5′)-Oligoadenylate Antisense Chimeras Targeting Steroid 5α-Reductase	Hagen Cramer; Paul F. Terrence
1205-1208	Biologically Active Oligodeoxyribonucleotides. VII. Anti-HIV-1 Activity of Hexadeoxyribonucleotides Bearing 3′- and 5′-End-Modifications	Makoto Koizumi; Rika Koga; Hitoshi Hotoda; Kenji Momota; Toshinori Ohmine; Hidehiko Furukawa; Takashi Nishigakit; Koji Abe; Toshiyuki Kosaka; Masakatsu Kaneko; Satoshi Kimura; Kaoru Shimada
1209-1212	Synthesis of 3′,5′-Dithymidylyl-α-hydroxyphosphonate Dimer Building Blocks for Oligonucleotide Synthesis—A New Pro-oliguncleotide	Ralf P. Mauritz; Chris Meier; Eugen Uhlmann
1213-1214	The Pro-Oligonucleotide Approach: Chimeric Dodecamers Bearing Six Bioreversible Protecting Groups	F. Morvan; G. Tosquellas; N. Mignet; I. Barber; B. Rayner; J. -L. Imbach
1215-1219	Enhanced Specificity of Minimally Modified Anti-c-myc Oligonucleotides	A. Peyman; H. Ragg; T. Ulshöfer; D. W. Will; E. Uhlmann

Volume 16, Issue 7-9 (1997)

1221-1222	Targeting HIV mRNA for Degradation: 2,5-A Antisense Chimeras as Potential Chemotherapeutic Agents for AIDS	Mark R. Player; Ratan Maitra; Robert Silverman; Paul F. Torrence
1223-1226	Conjugation of Oligonucleotides with Steroid Structures and Their Interaction with the Low-Density Lipoprotein	Erik T. Rump; Remco L. A. de Vrueh; Erik A. L. Biessen; Theo J. C. van Berkel; Martin K. Bijsterbosch
1229-1233	Beta-L-(-)-dioxolane Cytidine (β-L-(-)-OddC) as a Potent Compound for the Treatment of Cancer	K. L. Grove; X. Guo; S-H. Liu; M. Kukhanova; C-K. Chu; Y-C. Cheng
1235-1240	Resistance Profile of a Novel 2′, 3′ - Dideoxynucleoside Analog with Activity Against HIV-1	Nathalie Richard; Antonietta R. Belmonte; Horacio Salomon; Kazushige Nagai; Tarek Mansour; Mark A. Wainberg
1241-1249	Characterization of GPI2A, a Potent Inhibitor of HIV-1 Gene Expression and Viral Replication	Michael I. Anazodo; Elena Duta; Horacio Salomon; Albert D. Friesen; Mark A. Wainberg; Jim A. Wright
1251-1259	Suicide Gene Therapy for Intrinsically Drug Resistant Solid Tumors	J. Arly Nelson; Bih-Fang Pan; Frank C. Marini III; David Farquhar; Craig A. Mullen
1261-1270	Gemcitabine: Actions and Interactions	William Plunkett; Peng Huang; Varsha Gandhi
1271-1278	Modulation of DNA Triplex Stability Through Nucleobase Modifications	Krishna N. Ganesh; Kallanthottathil G. Rajeev; Pradeep S. Pallan; Vipul S. Rana; Dinesh A. Barawkar; Vaijayanti A. Kumar
1279-1282	Lipophilic Derivatization of the Antiviral Drug 9-(2-Phosphonylmethoxyethyl)adenine and Its Incorporation into a Lactosylated Lipid Carrier to Improve Its Liver Uptake	Remco L. A. de Vrueh; Erik T. Rump; Erik A. L. Biessen; Jan Balzarini; Theo J. C. van Berkel; Martin K. Bijsterbosch
1283-1286	Comparison of the Inhlbitory Effects of 2-Chloro-2′-deoxyadenosine and 9-β-D-Arabinosyl-2-fluoro-adenine on Metabolism of Deoxyadenosine in Human Lymphocytes and Erythrocytes	Krystyna Fabianowska-Majewska; Dorota Wyczechowska
1287-1290	Antiviral Activities of β-Enantiomers of 3′-Substituted-3′-deoxythymidine Analogs	Abdesslem Faraj; M. Abdelaziz El Alaoui; Geraldine Pavia; Gilles Gosselin; Jean-Louis Imbach; Raymond F. Schinazi; Jean Pierre Sommadossi
1291-1294	Anti-Inflammatory Activity of Purine Nucleoside Analogs	Stephanie A. Hartsel; Cecil Chen; John Kennedy; Allison Bendele; Cliff Wright; William S. Marshall
1295-1299	Thiated Pyrimidine Deoxynucleoside Analogues, Potential Chemotherapeutic Agents, and Substrates/Inhibitors in Various Enzyme Systems	M. Bretner; K. Felczak; J. M. Dzik; B. Golos; W. Rode; A. Drabikowska; J. Poznanski; K. Krawiec; A. Piasek; D. Shugar; T. Kulikowski
1301-1302	Derivatives of Imidazole-4-carboxamide as Substrates for Various DNA Polymerases	Christine Le Bec; Pascal Roux; Henri Buc; Sylvie Pochet
1303-1306	Cyclo-saligenyl-2′,3′-dideoxy-2′,3′-didehydroythymidinemonophosphate (cycloSal-d4TMP) — A New Pro-Nucleotide Approach	Chris Meier; Martina Lorey; Eric De Clercq; Jan Balzarini
1307-1310	Cyclo-saligenyl-5-fluoro-2′-deoxyuridinemonophosphate (cycloSal-FdUMP) — A New Prodrug Approach for FdUMP	Martina Lorey; Chris Meier; Eric De Clercq; Jan Balzarini
1311-1314	Di-ddU-α-Hydroxyphosphonate and α-Hydroxy- α- METHYLPHOSPHONATES as Potential Prodrugs of Antiviral Nucleoside Analogues	Lothar W. Habel; Chris Meier
1315-1319	Synergistic Combinations of Nucleoside Analog Drugs with Other Drugs Induce Greater Apoptosis in Human Leukemic T-Cells	Partha Nandy; Antonia P. Periclou; Vassilios I. Avramis
1321-1324	The Pronucleotide Approach. I. Synthesis, Anti-HIV Activity and Preliminary Stability Studies of Mononucleoside S,S′-Bis(O-acyl-2-oxyethyl) Phosphorodithiolates	N. Schlienger; C. Périgaud; G. Gosselin; I. Lefebvre; A. Pompon; A. -M. Aubertin; A. Kirn; J. -L. Imbach
1325-1329	The Pronucleotide Approach. II: Synthesis and Preliminary Stability Studies of Mononucleoside Glycosyl Phosphotriester Derivatives	N. Schlienger; C. Périgaud; G. Gosselin; J. -L. Imbach
1331-1335	The Pronucleotide Approach. III. Synthesis, Anti-HBV Activity and Stability Studies of the Bis(S-pivaloyl-2-thioethyl) Phosphotriester Derivative of Acyclovir	Gilles Valette; Jean-Luc Girardet; Alain Pompon; Christian Périgaud; Gilles Gosselin; Brent Korba; Olivier Hantz; Jean-Louis Imbach
1337-1339	Synthesis and Biological Activity of Some 2-Aminopurine Carbonucleosides	L. Santana; M. Teijeira; E. Uriartea; C. Terán; G. Andrei; R. Snoeck; E. De Clercq
1341-1345	Phosphodiester Amidates of Unsaturated Nucleoside Analogues as Anti-HIV Agents	Holger Winter; Yosuke Maeda; Hiroaki Mitsuya; Jiri Zemlicka
1347-1350	Antileukemic Activities and Mechanism of Action of 2′-Deoxy-4′-methylcytidine and Related Nucleosides	Toyofumi Yamaguchi; Aki Tomikawa; Toshiaki Hirai; Takeo Kawaguchi; Hiroshi Ohrui; Mineo Saneyoshi
1351-1354	Synthesis and Biological Activity of New 2′ 5′-Oligonucleotides	Evgeny I. Kvasyuk; Tamara I. Kulak; Igor A. Mikhailopulo; Robert J. Suhadolnik; Earl E. Henderson; Susan E. Horvath; Ming-Xu Guan; Wolfgang Pfleiderer
1357-1368	Sequence-Specific Cleavage of RNA Using Macrocyclic Lanthanide Complexes Conjugated to Oligonucleotides: A Structure Activity Study	Jonathan Hall; Dieter Hüsken; Robert Häner
1369-1378	Pteridine Nucleosides—New Versatile Building Blocks in Oligonucleotide Synthesis	Ramamurthy Charubala; Juris Maurinsh; Angelika Rösler; Manuel Melguizo; Oliver Jungmann; Margarete Gottlieb; Jörg Lehbauer; Mary Hawkins; Wolfgang Pfleiderer
1379-1388	Potent and Selective Ligands for Adenosine Binding Sites	G. Cristalli; E. Camaioni; E. Di Francesco; A. Eleuteri; S. Vittori; R. Volpini
1389-1398	New Unnatural L-Nucleoside Enantiomers:From Their Stereospecific Synthesis to Their Biological Activities	G. Gosselin; V. Boudou; J. -F. Griffon; G. Pavia; C. Pierra; J. -L. Imbach; A. -M. Aubertin; R. F. Schinazi; A. Faraj; J. -P. Sommadossi
1399-1402	Conformational Studies of 3′-Spironucleosides (TSAO-T and Analogues) by NMR Spectroscopy	Rosa Alvarez; María-Luisa Jimeno; Francisco J. Tomás-Gil; María-Jesús Pérez-Pérez; María-José Camarasa

Volume 16, Issue 7-9 (1997)

1403-1406	A Study Towards Total Synthesis of Antibiotic Agrocin 84	Dmitri Filippov; Cornelis M. Timmers; Gijs A. van der Marel; Jacques H. van Boom
1407-1410	Solid Phase Conjugation Chemistry: Use of Alloc as a Protecting Group for 2′-Aminolinker Containing Oligonucleotides	Isabelle Barber-Peoc'h; Muthiah Manoharan; P. Dan Cook
1411-1413	2′- and 3′- Biotin Conjugated Nucleoside Building Blocks: Synthesis of Biotinylated Oligonucleotides	Muthiah Manoharan; Gopal Inamati; Kathleen L. Tivel; Patrick Wheeler; Kim Stecker; P. Dan Cook
1415-1418	Synthesis and IMP Dehydrogenase (Type I and Type II) Inhibitory Activity of Isosteric NAD Analogs Derived from Thiophenfurin and Furanfurin	P. Franchetti; L. Cappellacci; G. Abu Sheikha; H. N. Jayaram; B. P. Schneider; T. Sint; V. V. Gurudutt; F. R. Collart; E. Hubeman; M. Grifantini
1419-1421	Development of Novel Bridged and Caged Nucleoside Analogs as Biochemical Tools	Michael P. Groziak; Ronghui Lin
1423-1426	1,5-Translocation Strategy for Nucleoside Anomeric Radicals	Atsushi Kittaka; Hiromichi Tanaka; Naoki Yamada; Hajime Kato; Tadashi Miyasaka
1427-1429	The Synthesis of Enantiomerically Pure Pyrazolo[4,3-c]pyridine Carbarzbo C-Nucleoside	Barbara Mohar; Jože Kobe
1431-1434	Conformational Analysis of Nucleosides Constructed on a Bicyclo[3.1.0]hexane Template. Structure-Antiviral Activity Analysis for the Northern and Southern Hemispheres of the Pseudorotational Cycle	Victor E. Marquez; Abdallah Ezzitouni; Maqbool A. Siddiqui; Pamela Russ; Hisafumi Ikeda; Clifford George
1435-1438	Novel Bicyclic Nucleoside Analogues Related to Natural Griseolic Acids	Lea Pickering; Vasu Nair
1439-1442	Synthesis and Evaluation of Novel Oligodeoxynucleotides Containing 3′-C-(3-Benzoyloxypropyl)thymidine and Bicyclo Nucleoside Derivatives	Henrik M. Pfundheller; Poul Nielsen; Jesper Wengel
1443-1446	Properties of Some Diuridine Phosphate Analogues	Bhisma K. Patel; James B. Thomson; Victor Jiménez; Klaus Eckart; Fritz Fxkstein
1447-1451	Steric and Stereoelectronic Effects of 7-Deazapurine Bases on the Sugar Conformation of 2′-Deoxynucleosides	Helmut Rosemeyer; Natalya Ramzaeva; Matthias Zulauf; Horst Thomas; Yaoming Chen; Cathrin Mittelbach; Frank Seela
1453-1456	1,2-Disubstituted Carbocyclic Analogues of Thymine Nucleosides	V. Escuredo; B. Ferro; L. Santana; M. Teijeira; E. Uriarte
1457-1460	2′-C-Alkylribonucleosides: Design, Synthesis, and Conformation	Rogers E. Harry-O'kuru; Emily A. Kryjak; Michael S. Wolfe
1461-1464	New Pyrene Derivatives for Fluorescent Labeling of Oligonucleotides	V. A. Korshun; I. A. Prokhorenko; S. V. Gontarev; M. V. Skorobogatyi; K. V. Balakin; E. V. Manasova; A. D. Malakhov; Yu. A. Berlin
1465-1468	Synthesis of Circular Oligonucleotide Conjugates	O. G. Chakhmakhcheva; A. A. Buryakova; M. V. Choob; A. L. Kalinkina; V. A. Efimov; R. F. Rando
1469-1472	Structural Studies of 2-Thiouridine in RNA	Raju K. Kumar; Darrell R. Davis
1473-1474	Unexpected High Hybridization Properties of α-Anomeric Oligodeoxynucleoside Methylphosphonates	F. Debart-Vasseur; J. -J. Vasseur; J. -L. Imbach; B. Rayner
1475-1480	Synthesis of Novel DNA Analoues Containing Aminomethylphosphonate Internucleoside Linkages	V. A. Efimov; M. V. Choob; A. L. Kalinkina; O. G. Chakhmakkcheva
1481-1485	DNA Duplexes Containing Alpha Anomeric Nucleotides and Polarity Reversals: Coexistence of Parallel and Antiparallel DNA	Markus W. Gerrnann; James M. Aramini; Bernd W. Kalisch; Richard T. Pon; Johan H. van de Sande
1487-1488	Stepwise Solid-Phase Synthesis of Serine-, Tyrosine- and Homoserine-nucleopeptides	Maite Beltrán; Marta Maseda; Yolanda Pérez; Jordi Robles; Enrique Pedroso; Anna Grandas
1489-1490	Novel DNA Damage Mediated by Oxidation of Various Modified Nucleotide Residues	Hideo Inoue; Shiro Koizume; Takahiro Yamauchi; Kouichi Murata; Eiko Ohtsuka
1491-1495	Synthesis, Biophysical Properties, and Stability Studies of Mixed Backbone Oligonucleotides Containing Novel Non-Ionic Linkages	Radhakrishnan P. Iyer; Dong Yu; Theresa Devlin; Nan-Hui Ho; Suzanne Johnson; Sudhir Agrawal
1497-1501	The Synthesis of 2′-C-Functionalised Nucleosides for Incorporation into Catalytic RNA	Anthony J. Lawrence; John B. J. Pavey; Ian A. O'Neil; Richard Cosstick
1503-1505	Comparison of Physicochemical and Biological Properties of (o-Carboran-1-YL)methylphosphonate and Methylphosphonate Oligonucleotides	Zbipniew J. Lesnikowski; Robert M. Lloyd Jr.; Raymond F. Schinazi
1507-1511	Properties of Oligonucleotides Containing the Transition Bases P and K	F. Hill; D. Loakes; D. M. Brown
1513-1514	A Solid-Phase Method for the Synthesis of Small to Medium-Sized Cyclic Oligonucleotides	ElMostafa Alazzouzi; Nuria Escaja; Marcus Straub; Blanca Martí; Anna Grandas; Enrique Pedroso
1515-1518	A Novel Class of 4′-Aza Analogues of 2′,3′-Dideoxynucleosides as Potential Anti-HIV Drugs	Antonella Leggio; Angelo Liguori; Antonio Procopio; Carlo Siciliano; Giovanni Sindona
1519-1522	Amino Acid Nucleic Acids: Synthesis and Hybridization Properties of a Novel Class of Antisense Oligonucleotides	Kanda S. Ramasamy; Wilfried Seifert
1523-1527	Oligonucleotides Containing Consecutive 2′-Deoxy-Isoguanosine Residues: Synthesis, Parallel Duplex Formation and Identification of a d(T₄iG₄T₄) Tetraplex	Frank Seela; Changfu Wei; Alexander Melenewski

Volume 16, Issue 7-9 (1997)

1529-1532	Synthesis and NMR Spectra of Some New Carbohydrate Modified Uridine Phosphoramidites	Pawel J. Serafinowski; Colin L. Barnes
1533-1538	Boranophosphate Oligonucleotides: New Synthetic Approaches	Dmitri Sergueev; Ahmad Hasan; Muthukumar Ramaswamy; Barbara Ramsay Shaw
1539-1542	Oligonucleotides Containing N⁷-Cyanoborane-2′-deoxyguanosine	Ahmad Hasan; Barbara Ramsay Shaw
1543-1545	Synthesis of 3′-Thioribouridine, 3′-Thioribocytidine, and Their Phosphoramidites	Sengen Sun; Joseph A. Piccirilli
1547-1549	Synthesis and Incorporation of 2′-O-Methyl-Pseudouridine into Oligonucleotides	Bruce S. Ross; Guillermo Vasquez; Sheri Manalili; Elena Lesnik; Richard Griffey
1551-1554	Replacement of the Phosphodiester Backbone of Oligodeoxynucleotide Analogues by Non-Ionic Phosphoramidate (P-NH₂)	S. Peyrottes; J. -J. Vasseur; J. -L. Imbach; B. Rayner
1555-1558	Dinucleoside Monophosphate Analogues Containing Disulfide Linkages	Emma M. Witch; Richard Cosstick
1559-1562	Site-Specific Introduction of Functional Groups onto Bases in Synthetic Oligonucleotides for Biological Applications	Yao-Zhong Xu; Qinguo Zheng; Gareth Urwin; Peter F. Swann
1563-1564	The Derivatives of Phosphorothioate Oligonucleotides	N. V. Amirkhanov; V. F. Zarytova
1565-1569	Mini-antisense Oligonucleotides	D. V. Pyshnyi; I. A. Pyshnaya; S. G. Lokhov; E. M. Ivanova; V. F. Zarytova
1571-1574	Oligonucleotide-Peptide Conjjugates for RNA Cleavage	D. Pyshnyi; M. Repkova; S. Lokhov; E. Ivanova; A. Venyaminova; V. Zarytova
1575-1577	Superactive Oligonucleotide Derivatives	D. S. Sergeyev; P. E. Vorobjev; V. F. Zarytova
1579-1582	The Synthesis of 2–5A Antisense Chimeras with Various Non-nucleoside COMPONENTS	Weifeng Zhang; Paul Torrence
1585-1588	Evaluation of Sulfur-Transfer Reagents for Large Scale Synthesis of Oligonucleotide Phosphorothioate Analogues	Zhaoda Zhang; Alexandra Nichols; Jimmy X. Tang; Mazen Alsbeti; Jin Yan Tang
1589-1598	Ultrafast Cleavage and Deprotection of Oligonucleotides Synthesis and Use of C^Ac Derivatives	M. P. Reddy; Naeem B. Hanna; Firdous Farooqui
1599-1608	Structural Correlations of Backbone Modifications in Antisense Oligonucleotide Duplexes	Xiaolian Gao; Jeffrey S. Rice; Collin W. Cross; Xueyong Yang
1609-1615	A Novel Approach for Gene Medicine: Synthetic Poly-L-lysine/serine Copolymer Enhances Bioactivity of Antisense Oligonucleotides	T. Goto; Y. Suzuki; A. Wada; I. Nozawa; S. Sato; S. Kawai; Y. Mizushima
1617-1620	Efforts Toward Synthesis of Oligonucleotides for Commercialization	Mark Andrade; Anthony S. Scozzari; Douglas L. Cole; Vasulinga T. Ravikumar
1621-1624	Phthaloyl Strategy—A New Approach Towards Oligodeoxyribonucleotide Synthesis	Markus Beier; Wolfgang Pfleiderer
1625-1628	Solution Phase Synthesis of an Oligodeoxyribonucleotide Phosphorothioate for Therapeutic Applications	Z. S. Cheruvallath; A. H. Krotz; D. L. Cole; V. T. Ravikumar
1629-1632	An Efficient Multigram Synthesis of Monomers for the Preparation of Novel Oligonucleotides Containing Isosteric Non-Phosphorous Backbones	Stuart Dimock; Balkrishen Bhat; Didier Peoc'h; Yogesh S. Sanghvi; Eric E. Swayze
1633-1636	Synthesis of Oligodeoxynucleoside Phosphoro-Monothioates and Phosphorodithioates by a Phosphotriester Method	Jan Kehler; Ask Püschl; Otto Dahl
1637-1640	Improved Impurity Profile of Phosphorothioate Oligonucleotides Through the Use of Dimeric Phosphoramidite Synthons	Achim H. Krotz; Patrick Klopchin; Douglas L. Cole; Vasulinga T. Ravikumar
1641-1643	A Novel and Economical Synthesis of 2″-O-Alkyl-Uridines	Bruce S. Ross; Robert H. Springer; Zeb Tortorici; Stuart Dimock
1645-1647	An Efficient and Scalable Synthesis of Arabinosylguanine and 2′-Deoxy-2′-Fluoro-guanosine	Bruce S. Ross; Robert H. Springer; Kelly G. Sprankle; Guillermo Vasquez
1649-1652	Protection of 2,6-Diaminopurine 2′-Deoxyriboside	I. Luyten; A. Van Aerschot; J. Rozenski; R. Busson; P. Herdewijn
1653-1656	Automated Chemical Synthesis of PNA and PNA-DNA Chimera on a Nucleic Acid Synthesizer	Ravi Vinayak; Alexander C. van der Laan; Rick Brill; Ken Otteson; Alex Andrus; Esther Kuyl-Yeheskiely; Jacques H. van Boom
1657-1660	An Inverse Approach in Oligodeoxyribonucleotide Synthesis	Thomas Wagner; Wolfgang Pfleiderer
1661-1662	Studies on Nucleoside H-Phosphonothioates as Synthons in the Synthesis of Oligonucleotide Analogues	Rula Zain; Martin Bollmark; Jacek Stawinski
1665-1668	Modulation of Splicing in the DMD Gene by Antisense Oligoribonucleotides	Matthew G. Dunckley; Ian C. Eperon; George Dickson

Volume 16, Issue 7-9 (1997)

1669-1672	Backbone Modified Antisense Oligodeoxynucleotides Directed Against the Hepatitis-C-Virus (HCV)-RNA	S. Eisenhardt; W. Samstag; K. Jahn-Hofman; J. W. Engels; R. Renz; P. H. Hofschneider; W. H. Caselmann; M. Alt
1673-1676	Effects of Intravenous Infusion of Phosphorothioate Oligonucleotides on Coagulation, Complement Activation and Hemodynamics	Scott P. Henry; David Monteith; Doug J. Kornbrust; Arthur A. Levin
1677-1682	Stability of Stereoregular Oligo(Nucleoside Phosphorothioate)s in Human Cells. Diastereoselectivity of Cellular 3′-Exonuclease	Maria Koziokiewicz; Edyta Gendaszewska; Maria Maszewska
1683-1687	Anti-BCL2 Phosphorothioate G3139 Clinical Pharmacology: Plasma Levels During Contwous Subcutaneous Infusion by HPLC Assay	A. V. Lebedev; F. Raynaud; M. Dizik; T. Beck; J. A. Jaeger; B. D. Brown; D. Cunningham; A. Webb; E. McCampbell; T. Riley; I. Judson; M. C. Woodle
1689-1693	Pharmacokinetic Properties of Phosphorothioate Oligonucleotides	Janet M. Leeds; Richard S. Geary; Scott P. Henry; Jo Glover; William Shanahan; Jon Fitchett; Todd Burckin; LoAnne Tmong; Arthur A. Levin
1695-1698	G-Rich Triplex-Forming Oligodeoxynucleotides as Transcription Repressors	Luigi E. Xodo; Marianna Alunni-Fabbroni; Gtorgio Manzini
1699-1702	Pharmacologic Disposition of a Phosphorothioate Oligodeoxynucleotide in Mice	Rosanne M. Orr; Florence I. Raynaud; Phyllis M. Goddard; Ian R. Judson; Terry Beck; Bob Bryant; Finbarr E. Cotter
1703-1707	Inhibition of Tumor Necrosis Factor Alpha (TNFα) Expression and Function In Vitro by Modified Antisense Oligonucleotides	Joshua O. Ojwang; T. Sudhakar Rao; Hélène B. Marshall; Shawn D. Mustain; Nilabh Chaudhary; David A. Walker; Anusch Peyman; Eugen Uhlmann; Ganapathi R. Revankar; Robert F. Rando
1709-1712	4-Cyano-2-butenyl Group: A New Type of Protecting Group in Oligonucleotide Synthesis via Phosphoramidite Approach	Vasulinga T. Ravikumar; Zacharia S. Cheruvallath; Douglas L. Cole
1713-1716	Anti-Influenza Virus Activities of Nicked and Circular Dumbbell RNA/DNA Chimeric Oligonucleotides	Hidefumi Yamakawa; Toshiaki Ishibashi; Takayuki Abe; Toshifumi Hatta; Kazuyuki Takai; Hiroshi Takaku
1717-1720	Enhanced Biological Activity of Antisense Oligonucleotides Containing 5-(1-Hexynyl)-substituted Pyrimidine Nucleotides	E. Uhlmann; L. Homung; S. Hein; S. Augustin; A. Peyman; D. W. Will; M. Helsberg; J. Sági; L. Ötvös; J. O. Ojwang; S. Mustain; R. F. Rando
1721-1725	Cleavage of Leishmania Mini-exon Sequence by Oligonucleotides Conjugated to a Dimidazole Construction	Ludmila Yurchenko; Vladimir Silnikov; Tatyana Godovikova; Gennady Shishlan; Jean-Jacques Toulme; Valentin Vlassov
1727-1730	Immune Cell Involvement in Anti-c-myc DNA Prevention of Tumor Formation in a Mouse Model of Burkitt'S Lymphoma	G. D. Gray; R. Townsend; H. Hayasaka; R. Korngold; E. Wickstrom
1731-1734	Oligonucleotide Pharmacology and Formulation: G3139 Anti-BCL2 Phosphorothioate In Stealth® Liposomes and Gel Implants	M. C. Woodle; F. I. Raynaud; M. Dizik; O. Meyer; S. K. Huang; J. A. Jaeger; B. D. Brown; R. Orr; I. R. Judson; D. Papahadjopoulos
1735-1738	Inhibition of Respiratory Syncytial Virus by Double Termini-Protected 2–5A Antisense Chimeras	Wei Xiao; Guiying Li; Paul F. Torrence; Nick M. Cirino; Robert H. Silverman
1741-1744	Oligonucleotide Conjugates Derived from an Electrophilic Site: Conjugation to Baseless Carbohydrate Residue. Synthesis, Hybridization and Modeling Studies	Muthiah Manoharan; Laura K. Andrade; Venkatraman Mohan; Susan M. Freier; P. Dan Cook
1745-1748	Sequencing Reactions Using 6-Thio-2′-Deoxyguanosine-5′-triphosphate	Mark G. McDougall; Bernie F. McArdle; Shiv Kumar; Carl W. Fuller; Lorraine M. Rellick; Alexei V. Govorine
1749-1752	Ambiguous Base Pairing of 1-(2-Deoxy-β-D-Ribofuranosyl)imidazole-4-carboxamide During PCR	Sylvie Pochet; Laurence Dugué; Monica Sala; Valérie Pézo; Simon Wain-Hobson
1753-1756	Combinatorial Generation of Nucleobase Libraries by MCR	Alexander Dömling; Wolfgang Richter
1757-1760	3′-Modified Nucleotides for DNA Sequencing Without Gel Electrophoresis	Isabelle Rasolonjatovo; Catherine Guerreiro; Robert S. Sarfati
1761-1764	Histological Localization of Phosphorothioate Oligodeoxynucleotides in Normal Rodent Tissue	Madeline Butler; Kim Stecker; C. Frank Bennett
1765-1766	A Convenient Method for Labeling Oligonucleotide Analogs by a Fluorogenic Tag for Direct In Vitro and In Vivo Visualization of Carboxyesterase Activity	A. Laurent; F. Debart-Vasseur; J. -L. Imbach; B. Rayner
1767-1770	Study of the Enantioselectivity of Enzymes Involved in Nucleoside Analogue Metabolism: Deoxycytidine Kinase	M. Shafiee; V. Boudou; J. -F. Griffon; A. Pompon; G. Gosselin; S. Eriksson; J. -L. Imbach; G. Maury
1775-1779	Triplex Formation Between DNA and Mixed Purine-Pyrimidine PNA Analog with Lysines in Backbone	E. Lesnik; F. Hassman; J. Barbeau; K. Teng; K. Weiler; R. Griffey; S. Freier
1781-1784	Synthesis of a 2-Hydroxy-oxolane Derivative as a New Potential Crosslinking Agent of DNA	L. Nzita; S. Ladame; L. Gomez; S. Moreau
1785-1788	Molecular Engine for Transporting Drugs Across Cell Membranes	James Summerton; Dwight Weller
1789-1792	Synthesis of Copper-64 and Technetium-99M Labeled Oligonucleotides with Macrocyclic Ligands	Sven Wagner; Michael Eisenhut; Ramon Eritja; Franz Oberdorfer
1793-1796	Picomole Syntheses of High Quality Oligonucleotide Primers in Combination with the Preparation of Oligonucleotide Arrays	Jan Weiler; Jörg D. Hoheisel
1797-1798	New Photoreactive RNA Analogues	M. N. Repkova; A. G. Venyaminova; V. F. Zarytova
1799-1803	Photochemical Cross-Linking of λ-Cro Repressor to Operator DNA Containing 4-Thiothymine or 6-Thioguanine	Qinguo Zheng; Yao-Zhong Xu; Peter F. Swann
1805-1806	A New Model for the Comparison of the Efficiency and Selectivity of Photoreactive Groups Towards the Nucleic Acid and Protein Functional Groups	Dmitri G. Knorre; Tatyana S. Godovikova; Vera D. Knorre; Vladimir V. Koval
1807-1808	Kinetic Approach for Determination of Affinity Properties of Reactive Oligonucleotide Derivatives to Complementary Regions in Nucleic Acids	Vladimir V. Koval; Dmitri G. Knorre; Olga S. Fedorova

Volume 16, Issue 5-6 (1997)

ix-xii	Contributors to This Issue
517-522	The Application of Uppsala “Nmr-Window” Concept for Conformational Analysis of Biologically Functional Dnas and RNAs by High-Field NMR	A. Földesi; S. I. Yamakage; F. P. R. Nilson; T. V. Maltseva; C. Glemarec; J. Chattopadhyaya
523-529	The Discovery of Intramolecular Stereoelectronic Forces That Drive The Sugar Conformation in Nucleosides and Nucleotides	C. Thibaudeau; J. Chattopadhyaya
531-542	Recognition of Point Mutations in Dna By Means of Time Resolved Fluorescence Methods	S. Winter; S. Kirschstein; G. Löber
543-550	Application of Single Molecule Detection to Dna Sequencing	Peter M. Goodwin; Hong Cai; James H. Jett; Susan L. Ishaug-Riley; Nicholas P. Machara; David J. Semin; Alan Van Orden; Richard A. Keller
551-556	Single-Molecule Detection of Coumarin-120	L. Brand; C. Eggeling; C. A. M. Seidel
557-562	A Fluorescence Detection and Selection Device for Dna-Molecules Bound to Microspheres	Johan Holm; Håkan Elderstig; Ove Kristensen; Rudolf Rigler
563-571	Dna Analysis by Mass Spectrometry: Applications in Dna Sequencing And Dna Diagnostics	H. Köster; D. van den Boom; A. Braun; A. Jacob; C. Jurinke; D. P. Little; K. Tang
573-577	Recent Developments in Mass Spectrometry: Rna Sequencing	K. Wörner; K. Faulstich; J. W. Engels
579-584	Sequence Analysis of Fis Binding Sites Obtained by in Vitro Selection	Karsten Theis; Cornelia Bartsch; Wolfram Saenger
585-589	Enzymatic Fluorescence and Biotin Labelling of Primers for Dna Sequencing and Pcr	Gabor L. Igloi
591-598	Dna Sequencing After the Human Genome Project	Charles R. Cantor; Kai Tang; Joel H. Graber; Maryanne Maloney; Dong Jing Fu; Natalia E. Broude; Fouad Siddiqi; Hubert Koester; Cassandra L. Smith
599-602	Recognition of Double-Stranded Dna by Peptide Nucleic Acid	Pernilla Wittung; Peter Nielsen; Bengt Nordén
603-608	Synthesis of Polyamide Nucleic Acids (Pnas), Pna /Dna-Chimeras and Phosphonic Ester Nucleic Acids (Phonas)	E. Uhlmann; D. W. Will; G. Breipohl; A. Peyman; D. Langner; J. Knolle; G. O'Malley
609-615	Fast Kinetic Studies by Fluorescence Correlation Spectroscopy of Pna-Dna Interactions	Palok Aich; Peter Nielsen; Rudolf Rigler
617-621	Structure of Pna-Nucleic Acid Complexes	Magdalena Eriksson
623-628	Antiviral Activity of Antisense Oligonucleotides Against Various Targets of Herpes Simplex Virus 1 (Hsv1) and Coxsackievirus B3 (Cvb3) Genome	E. Birch-Hirschfeld; C. M. Knorre; A. Stelzner; M. Schmidtke
629-634	Antisense Strategies for Inhibition of Tumor Necrosis Factor-α Synthesis	Gunther Hartmann; Anne Krug; Martin Bidlingmaier; Andreas Eigler; Stefan Endres
635-642	Single Molecule Detection in Microstructures	B. Wagner; H. Mathis; K. Schmidt; G. Kalusche; J. McCaskill

Volume 16, Issue 5-6 (1997)

643-652	Chemical and Photochemical Ligation of Oligonucleotide Blocks	Robert L. Letsinger; Taifeng Wu; Robert Elghanian
653-659	Substrate Specificities, Expression and Primary Sequences of Deoxynucleoside Kinases; Implications for Chemotherapy	Staffan Eriksson; Liya Wang
661-667	Binding of Actinomycin D to Single-Stranded Dna	Elizabeth A. Jares-Erijman; Reinhard Klement; Reinhard Machinek; Randy M. Wadkins; Besik I. Kankia; Luis A. Marky; Thomas M. Jovin
669-674	Oligonucleotides With Purine Nitrogen-7 as Glycosylation Site	Frank Seela; Peter Leonard
675-678	Fpmp-Protected α-Hydroxyphosphonate Diesters for The Synthesis of Pro-Oligonucleotides	Ralf P. Mauritz; Chris Meier
679-684	Studies on Nucleoside Phosphonates and Their Derivatives. a Progress Report	Martin Bollmark; Annika Kers; Inger Kers; Tomas Szabó; Rula Zain; Jacek Stawiński; Jacek Cieślak; Jadwiga Jankowska; Adam Kraszewski
685-696	A New Type of Fluorescence Labeling of Nucleosides, Nucleotides and Oligonucleotides	Harald Sigmund; Thomas Maier; Wolfgang Pfleiderer
697-702	Preparation of Oligonucleotides Containing Non-Natural Base Analogs.	Ramon Eritja; Viviane Adam; Anna AviñTó; Antonio R. Díaz; Carme Fàbrega; Elisenda Ferrer; Morten GrøStli; Ramón Güimil García; Mechtild Hofmann; Víctor E. Márquez; Marten Wiersma
703-710	Synthetic Oligonucleotide Combinatorlal Libraries - Tools For Studying Nucleic Acid Interactions	H. Seliger; R. Bader; M. Hinz; B. Rotte; A. Astriab; M. Markiewicz; W. T. Markiewicz
711-715	Fast Rna-Rna Annealing in Vitro: Single Cycle Selection Versus Multiple Cycle Selection	Volker Patzel; Ralf Kronenwett; Karola Rittner; Georg Sczakiel
717-720	In Vitro Selection, Structural Characteristics, and Photocleavage of an Isoalloxazine Binding Rna Aptamer	C. Huber; P. Burgstaller; M. Famulok
721-725	Role of Metal Ions In The Cleavage Mechanism by The E. Coli Rnase P Holoenzyme	Jens M. Warneckes; Christopher J. Green; Roland K. Hartmann
727-732	Display Of Ribonuclease T1 On The Surface Of Bacteriophage M13	Bernd Hubner; Kerstin Korn; Hans-Heinrich Förster; Ulrich Hahn
733-736	Non-Linear Dynamics in Nucleic Acid Research Using Fractals Ulm Report 1996	Albrecht K. Kleinschmidt
737-742	Multiple Sequence Elements Involved in Polyadenylation at The Murine Igm Secretory Poly(A)Site.	Cathy Phillips; Anders Virtanen
743-750	Determination of The Solution Conformation of A Non-Uniformly Deuterium Labelled (Uppsala ‘Nmr-Window’) 21Mer Rna Hairpin by Nmr Spectroscopy And Computational Methods.	Anders Sandström; Tatiana Maltseva; Jyoti Chattopadhyaya
751-754	Synthesis and Application of 3′-Amino-Dye-Terminators For Dna Sequencing	C. Wojczewski; K. Faulstich; J. W. Engels
755-760	The Chemistry of C-Branched Spermine Tethered Oligo-DNAs and Their Properties in Forming Duplexes and Triplexes	Christian Sund; Nitin Puri; Jyoti Chattopadhyaya
761-768	Synthesis and Enzymatic Studies of Modified Oligonucleotides with Abiological Monomer Units	D. Wenninger; H. Seliger
769-772	5-[2-(2-Methoxy)bornyl]tetrazole as Catalyst for Diastereoselective Synthesis of 2′-Deoxy Dinucleoside (3′, 5′)-Methylphosphonates	Peter Schell; Joachim W. Engels

Volume 16, Issue 5-6 (1997)

773-776	Synthesis and Biological Activity of New Sugar Modified 2′,5′-Oligoadenylate Trimers	Evgeny I. Kvasyuk; Tamara I. Kulak; Olga V. Tkachenko; Svetlana L. Sentyureva; Igor A. Mikhailopulo; Robert J. Suhadolnik; Earl E. Henderson; Susan E. Horvath; Ming Xu Gun; Wolfgang Pfleiderer
777-780	New Developments in Oligomer Array Technologies	Jan Weiler; Nicole Hauser; Jörg D. Hoheisel
781-787	Exonuclease Degradation of DNA Studied by Fluorescence Correlation Spectroscopy	Zeno Földes-Papp; Per Thyberg; Sofie Björling; Arne Holmgen; Rudolf Rigler
789-792	New Synthesis and Antitumor Activity of CycloSal- Derivatives of 5-Fluoro-2′-deoxyuridinemonophosphate	Martina Lorey; Chris Meiera; Eric De Clercq; Jan Balzarini
793-796	Cyclo-Saligenyl-3′-Azido-2′,3′-Dideoxy- Thymidinemonophosphate (cycloSal-AZTMP) - A New Pro-Nucleotide Approach¹ ?-	Chris Meiera; Eric De Clercq; Jan Balzarini
797-800	Incorporation of 2′-Modified Nucleotides into tRNA to Test Importance for Charging	Tina Persson; Claus Stefan Vörtler; Olga Fedorova; Fritz Eckstein
801-808	The (2-Cyano-1-phenyl)ethoxycarbonyl (CPEOC) Group-A New Protecting Group for Oligoribonucleotide Synthesis	Ursula Münch; Wolfgang Pfleiderer
809-814	Synthesis of Novel Fluoro Carbocyclic Purine Nucleoside Analogues	Johanna Wachtmeister; Björn Classon; Ingemar Kvarnströmn; Bertil Samuelsson
815-820	Synthesis and Characterization of Phosphate-modified DNA-Dimers with Fluorine as an uncharged Ligand	Thomas J. Lehmann; Stefan Eisenhardt; Joachim W. Engels
821-828	Stereoelectronic Effects of Modified Purines on the Sugar Conformation of Nucleosides and Fluorescence Properties	Helmut Rosemeyer; Matthias Zulauf; Natalya Ramzaeva; Georg Becher; Elisabeth Feiling; Klaus Mühlegger; Ingo Münster; Anke Lohmann; Frank Seela
829-833	Oligonucleotide Microsynthesis of A 200-mer and of One-Dimensional Arrays on a Surface Hydroxylated Polypropylene Tape	Raoul Bader; Michael Hinz; Bernhard Schu; Hartmut Seliger
835-842	A Rapid Method for the Preparation of a One Dimensional Sequence-Overlapping Oligonucleotide Library	R. Bader; H. Brugger; M. Hinz; C. Rembe; E. P. Hofer; H. Seliger
843-848	MCR III¹. Multicomponent Reactions and Their Libraries, a New Type of Organic Chemistry of the Isocyanides and Phosphorus Derivatives.	Jyoti Chattopadhyaya; Alexander Dömling; Klaus Lorenz; Wolfgang Richter; Ivar Ugi; Birgit Wener
849-854	Specificity of the Receptor-G-Protein Interaction: Assigning Functions TO G-Protein Subunits by the Antisense Technique	Frank Kalkbrenner; Matthias Schroff; Vadim E. Degtiar; Edgar Dippel; Burghardt Wittig; Gunter Schultz
855-861	Acetal Oligonucleotide Conjugates in Antisense Strategy	S. Matysiak; R. Frank; W. Pfleiderer
863-868	Pteridine Nucleosides Analogs of 2′-Deoxyadenosine as Building Blocks for Oligonucleotide Synthesis	Oliver Jungmann; Wolfgang Pfleiderer
869-874	Synthesis of 8-(2-Deoxy-β-D-Ribofuranosyl)-Isoxanthopterins New Fluorescent Analogs of 2′-Deoxyguanosine	Jörg Lehbauer; Wolfgang Pfleidere
875-882	Solid Phase Synthesis, Cloning and Expression of a Synthetic Gene Encoding a Collagen-Like Peptide	A. Seliger; S. Brüninghoff; G. Gröger; J. Ramalho Ortigao; H. Seliger
883-887	Synthesis and Evaluation of Oligonucleotides of High Purity	Emma Jakobsson; Michael Hinz; Hartmut Seliger

Volume 16, Issue 4 (1997)

iii-iv	Contributors to The Issue
347-364	Synthesis of Pyrrolo[2,3-d]pyrimidines that are Structurally Related to Methylated Guanosines from tRNA and the Nucleoside Q Analogs, PreQ₀ and PreQ₁	Chin Shu Cheng; Geoffrey C. Hoops; Robert A. Earl; Leroy B. Townsend
365-377	Synthesis of Duplex DNA Containing a Spin Labeled Analog of 2′ Deoxycytidine	Paula L. Fischhaber; Annabelle W. Reese; Thuc Nguyen; James J. Kirchner; Eric J. Hustedt; Bruce H. Robinson; Paul B. Hopkins
379-401	Synthesis and Biochemical Activity of Hydrophilic Carborane-Containing Pyrimidine Nucleosides as Potential Agents for DNA Incorporation and BNCT	Feng-Guang Rong; Albert H. Soloway; Seiichiro Ikeda; David H. Ives
403-416	Synthesis of Six-Membered Nucleoside Analogs. Part 1: Pyrimidine Nucleosides Based on the 1,3-Dioxane Ring System	Daniel C. Capaldi; Alessandra Eleuteri; Qin Chen; Raymond F. Schinazi
417-432	Diastereoselective Synthesis of 2′-Deoxy and 2′-O-Methyl Dinucleoside (3′ 5′)-Methylphosphonates via Alkoxymagnesium Chloride-Mediated Nucleoside Coupling	William J. Daily; David A. Schwartz; Timothy A. Riley; Lyle J. Arnold Jr.; William B. Marvin; Michael A. Scurria; Stephanie A. Hopkins; Michael B. Atkins; Christine D. Garcia; Michael C. Pirrung
433-444	Glycosylation of 2-Thiouracil Derivatives. A Synthetic Approach to 3-Glycosyl-2, 4-dioxypyrimidines	A. I. Khodair; E. E. Ibrahim; E. El Ashry
445-454	Synthesis and Evaluation of Oligodeoxynucleotides Containing 3′-C-Aminomethyl-and 3′-C-Amethylthymidine	Guangyi Wang; Patrick J. Middleton; Liyan He; Vesna Stoisavljevic; Wiliiied E. Seifert
455-467	Synthesis of 5-Methyl-2′-O-Deoxycytidine Analogs to Determine Monoclonal Antibody Specificity in the Recognition of the 6-(p-Bromobenzoylamino) Caproyl Radical	Chryslaine Rodriguez-Tanty; David Higginson-Clarke; Milenen Hernández; Rafaela Pérez; Hermán Vélez-Castro; Ana Ma. Riverón; Arturo Macías
469-474	A Convenient Synthesis of N⁴,O^3′, O^5′-Triacetyl-2′-Ketocytidine	Douglas P. Kjell; Brian J. Slattery
475-483	Synthesis of a Novel Biotinyl Derivative and its Application to Non-Radioactive Labeling of DNA	Isamu Yamamoto; Yuji Arai; Tsuyoshi Fukuda; Keiko Y-Takihara; Junichi Azuma; Tsunehiro Mukai
485-493	Novel Synthesis of a New Class of Polynuclear Pyridinethione Nucleosides	Galal E. H. Elgemeie; Adel M. E. Attia; Nahed M. Fathy
495-505	Synthesis of Some Pyrrolo[2,3-d]Pyrimidine Isodideoxynucleosides of (S,S)-Stereochemistry	Ratnakar R. Talekar; Richard H. Wightman
507-513	Conformational Analysis of 3′-Deoxy-β-D-Ribonucleosides Using 1D-noe Difference Spectroscopy	Anil Kumar; S. B. Katti; H. Rosemeyer; Frank Seela
515	Erratum

Volume 16, Issue 3 (1997)

iii	Contributors to This Issue
215-225	Synthesis and DNA Duplex Stabilities of Oligonucleotides Containing C-5-(3-Methoxypropynyl)-2′-deoxyuridine Residues	Vladimir V. Tolstikov; Dmitry A. Stetsenko; Victor K. Potapov; Eugene D. Sverdlov
227-237	Carboxyamidation of Purine Nucleosides: New Secondary 8-Carboxamidopurine Nucleosides	Chi Tu; Charlene Keane; Bruce Eaton
239-255	Cis-trans Isomerization of the N-Formyl Amino Group in a Novel Modified Uracil Derivative: 6-Amino-3-methyl-5-(N-Formylamino)uracil	T. Srikrishnan; R. Parthasarathy; W. Pfleiderer; Nimai C. De; Girish B. Chheda
257-263	Selective 5′-O-Acetylation of 2′-Deoxynucleosides and Nucleosides by a Modified Mitsunobu Procedure	Gong-Xin He; Norbert Bischofberger
265-276	Synthesis and Antiviral Activity of Modified 1,2,6-Thiadiazine Dioxide Acyclonucleosides	A. I. Esteban; E. De Clercq; A. Martinez
277-289	Anionic Manganese meso-Tetraphenyl Porphine/Oligonucleotide Conjugates-Synthisis and Utilization in Chemiluminescent DNA-Probe Detection	A. Schubert; T. Klütsch; D. Cech
291-300	Access to a New Type of Homo-C-Nucleosides with a “Split” 8-Deazapurine via a 1,3-Dipolar Cycloaddition Reaction	Serge Van Calenbergh; André De Bruyn; Jan Schraml; Norbert Blaton; Oswald Peeters; Denis De Keukeleire; Roger Busson; Piet Herdewijn
301-303	A Stereoselective Method for the Direct Preparation of 2′-Deoxycytidine	Douglas P. Kjell
305-314	Unexpected Dehalogenation of 3-Bromopyrazolo[3,4-d]pyrimidine Nucleosides During Nucleobase-Anion Glycosylation	Frank Seela; Matthias Zulauf; Georg Becher
315-337	4-Substituted-5(3)-carbamoyl-3(5)-(2-deoxy-β-D-ribofuranosyl)pyrazoles. Application of Palladium Catalyzed Glycal Coupling Methodology to the Synthesis of Pyrazofurin Analogs	Mark D. Erion; Robert M. Rydzewski
339-346	Structural Study of Two 5-Heteroaromatic-2′ deoxyuridines and Their 5-Bromine-heteroaromatic Analogues: Theoretical Conformational Analysis and NMR Experiments	Isabelle Creuven; Florence Lebon; Roger Busson; Piet Herdewijn; François Durant

Volume 16, Issue 1-2 (1997)

iii-iv	Contributors to This Issue
1-10	The Three-Dimensional Structure of 3′-Deoxycytidine	P. Karthe; N. Gautham; Anil Kumar; S. B. Katti
11-22	Synthesis and FAB Mass Spectroscopical Studies on 2′,5′-Dinucleoside-Monophosphates	Anil Kumar; Seturam B. Katti; Kunnath P. Madhusudanan
23-32	Solution Phase Synthesis of Dithymidine Phosphorodithioate Using New S-Protecting Groups in Combination with a Chemoselective Coupling Reagent (PyNOP)	Jan Kehler; Ask Püschl; Otto Dahl
33-40	C1′ Acylated Derivatives of 2′-Deoxyuridine. Photolabile Precursors of 2′-Deoxyuridin-1′-yl	Marc M. Greenberg; Dong Jin Yoo; Brian K. Goodman
41-51	Synthesis of DNA Dumbbells: Chemical vs. Enzymatic Ligation of Self-Complementary Oligonucleotides	Carol S. Lim; C. Anthony Hunt
53-65	Convenient Intermediates for the Preparation of C-4 Modified Derivatives of Pyrimidine Nucleosides	Anwar Miah; Colin B. Reese; Quanlai Song
67-80	Introduction of a Universal Solid Support for Oligonucleotide Synthesis	Claus Schcuer-Larsen; Christoph Rosenbohm; Thomas J. D. Jøgensen; Jesper Wengel
81-85	Conversion of Nucleosides to Cyclic Dinucleoside Dipyrophosphates	Kyung Bo Kim; Edward J. Behrman
87-95	Daunorubicin Derivatives Obtained from Daunorubicin and Nucleoside Dialdehydes	Eugenia N. Olsufyeva; Nikolai A. Brusentsov; Nedyalka Todorova; Jan Balzarini; Erik De Clercq; Maria N. Preobrazhenskaya
97-106	Synthesis and Antiviral Evaluation of N-β-D-Ribosides of Ergot Alkaloids	Vladimír Křen; Alois Pískala; Petr Sedmera; Vladimír Havlíěek; Věra Přikrylová; Myriam Witvrouw; Erik De Clercq
107-114	5-Amido-(carboxyfluorescein)-2′-dU-oligonucloetides: Novel Primers for Fluorescent Detection of PCR Amplified DNA	Vasant R. Jadhav; Dinesh A. Barawkar; Arvind A. Natu; Krishna N. Ganesh
115-128	Synthesis of Some Hydroxamic Acids Related to Uridine: Potential Inhibitors of Ribonucleoside Diphosphate Reductase	Peter Currid; Richard H. Wightman
129-144	6-Methyl-5-Azacytidine-Synthesis, Conformational Properties and Biological Activity. A Comparison of Molecular Conformation with 5-Azacytidine	Naeem B. Hanna; Jaroslav Zajíček; Alois Pískala
145-158	Solution Phase Synthesis of Dithymidine Phosphorothioate by a Phosphotriester Method Using New S-Protecting Groups	Ask Püschl; Jan Kehler; Otto Dahl
159-171	Synthesis and Antiviral and Cytostatic Activities of Carbocyclic Nucleosides Incorporating a Modified Cyclopentane Ring. I: Guanosine Analogues	J. M. Blanco; O. Caamaño; F. Fernández; G. Gómez; M. I. Nieto; J. Balzarini; E. Padalko; E. De Clercq
173-182	The Role of Hydrophobic Versus Hydrophilic Base Character in the Anti-HIV Activity of Purine-Containing Polyribonucleotides	Mayoka G. Tutonda; Heidi D. Fain; Robert W. Buckheit Jr.; Arthur D. Broom
183-191	6-Chloroxanthosine, a Useful Intermediate for the Efficient Syntheses of [6-¹⁵N]-Isoguanosine, Isoinosine and Other Purine Nucleoside Analogues	L. De Napoli; A. Messere; D. Montesarchio; G. Piccialli; M. Varra
193-213	Synthesis of Novel L-Series 2′, 3′-Dideoxy-3′-Hydroxy-Methyl-Nucleosides and a Convenient Method for the Separation of Nucleosede Anomers	Jayne H. M. Gould; John Mann

Volume 15, Issue 11-12 (1996)

iii-iv	Contributors to The Issue
v	Editor's Note
1679-1686	SYNTHESIS OF CYCLIC DINUCLEOTIDES BY AN H-PHOSPHONATE METHOD IN SOLUTION	Fan Zeng; Roger A. Jones
1687-1700	2′-SUBSTITUTED PHOSPHOROTHIOATE CONTAINING OLIGORIBONUCLEOTIDES: AN APPLICATION TO THE SYNTHESIS AND PURIFICATION OF HAMMERHEAD RIBOZYMES	Anthony DiRenzo; Susan Grimm; Kurt Levy; Peter Haeberli; Lara Maloney; Nassim Usman; Francine Wincott
1701-1710	SYNTHESIS AND STRUCTURE DETERMINATION OF A NUCLEOSIDEDERIVED NEW HETEROCYCLIC SYSTEM: 8H,10H,15b(S)-2,3,6,7-TETRAHYDRO-1,5,3-DIOXAZEPINO[3,2-c]INDOLO[3,2-g]PTERIDINE-7-ONE	Ping Ge; Gregory O. Voronin; Thomas I. Kalman
1711-1718	PHOSPHONATE ANALOGS OF CARBOCYCLIC PHOSPHORIBOSYLAMINE AND CARBOCYCLIC GLYCINAMIDE RIBONUCLEOTIDE	Robert Vince; Mei Hua; Carol A. Caperelli
1719-1723	MALDI AND FAB MASS SPECTROMETRY OF NUCLEOSIDE TRIPHOSPHATES: A COMPARATIVE STUDY	Kevin Burgess; David H. Russell; Aroonsiri Shitangkoon; Alex J. Zhang
1725-1739	PHOSPHONOACETATE DERIVATIVES OF OLIGODEOXYRIBONUCLEOTIDES	M Jonathan Rudolph; Michael S. Reitman; Eric W. MacMillan; Alan F. Cook
1741-1749	HYDROLYSIS OF 2′-DEOXY AND 2′-FLUORONUCLEOSIDE-3′-PHOSPHODlESTERS	L. Y. Kuo; K. Travers; J. Chock
1751-1769	SYNTHESIS OF NOVEL BICYCLIC NUCLEOSIDES RELATED TO NATURAL GRISEOLIC ACIDS	Lea Pickering; Vasu Nair
1771-1778	AN IMPROVED SYNTHESIS OF 9-[2-(DIETHOXYPHOSPHONOMETHOXY)ETHYL]ADENINE AND ITS ANALOGUES WITH OTHER PURINE BASES UTILIZING THE MITSUNOBU REACTION	Wei Chen; Michael T. Flavin; Robert Filler; Ze-Qi Xu
1779-1795	SYNTHESIS OF PYRAZOLO[4,3-C]PYRIDINE C-RIBONUCLEOSIDES VIA AN EFFECTIVE TETRAZOLE TO PYRAZOLE TRANSFORMATION	Marija Prhavc; Jože Kobe
1797-1803	REACTION OF ANHYDRONUCLEOSIDES WITH MAGNESIUM ALKOXIDES: REGIOSPECIFIC SYNTHESIS OF 2′-O-ALKYLPYRIMIDINE NUCLEOSIDES.	Danny P. C. McGee; Yansheng Zhai
1805-1819	CRYSTAL STRUCTURE OF 1,3,5-TRIMETHYL-N⁴-HYDROXYCYTOSINE, AND ITS RELEVANCE TO THE MECHANISM OF HYDROXYLAMINE MUTAGENESIS	Karin Bjåmer Birnbaum; Borys Kierdaszuk; David Shugar
1821-1834	SYNTHESES OF 2′,3′-DIDEOXY-D-C-NUCLEOSIDES FROM γ-LACTONE	Yuejun Xiang; Jinfa Du; Chung K. Chu
1835-1847	SYNTHESIS AND BIOLOGICAL ACTIVITY OF 5-SUBSTITUTED ANTI-CONSTRAINED ACYCLIC ANALOGS OF CYTIDINE AND URIDINE	Ling-Yih Hsu; Ya-Mei Chang; Chung-Hsun Lin; John C. Drach
1849-1861	SYNTHESIS OF 3-ALKYL PIPERAZIN-2-ONE NUCLEOSIDES WITH POTENTIAL ANTIRETROVIRAL ACTIVITY	Abdellah Benjahad; Robert Granet; Pierre Krausz; Claudine Bosgiraud; Sylvie Delebassée

Volume 15, Issue 11-12 (1996)

1863-1869	SYNTHESIS OF N⁶-ALKYLATED ADENOSINE DERIVATIVES	E. Lescrinier; C. Pannecouque; J. Rozenski; A. Van Aerschot; L. Kerremans; P. Herdewijn
1871-1889	A COMPARATIVE STUDY OF SUPPORTS FOR THE SYNTHESIS OF OLIGONUCLEOTIDES WITHOUT USING AMMONIA	Anna Aviñó; Ramon Güimil García; Antonio Díaz; Fernando Albericio; Ramon Eritja
1891-1904	Enzymatic Recognition of Acyclic Universal Base Analogues in Oligonucleotides	D. Loakes; A. Van Aerschotl; D. M. Brown; F. Hill
1905-1926	CARBOCYCLIC SUBSTRATES AND INHIBITORS FOR THE BIFUNCTIONAL LYASE OF PURINE NUCLEOTIDE BIOSYNTHESIS	Laurent Schmitt; Carol A. Caperelli
1927-1943	Synthesis of Hydantoin Nucleosides with Naphthylmethylene Substituents in the 5-Position	Ahmed I. Khodair; El-Said E. Ibrahimb
1945-1957	HALOGENATED NUCLEIC ACIDS: STRUCTURE AND CONFORMATIONAL STUDIES OF 5-FLUOROCYTIDINE BY X-RAY CRYSTALLOGRAPHY AND NMR SPECTROSCOPY	Sunil Dutta Soni; T. Srikrishnant; J. L. Alderfer

Volume 15, Issue 10 (1996)

iii-iv	Contributors to This Issue
1561-1566	Substrate Properties of Adenosine- and Uridine- 3′, 5′-bisphenylphosphonates for 3′-Nucleotidase/Nucleases	H. Uchida; T. Oohara; H. Wada; I. Takahashi; A. Nomura
1567-1580	Diazepinone Nucleosides as Inhibitors of Cytidine Deaminase.	G. Cristalli; R. Volpini; S. Vittori; E. Camaioni; G. Rafaiani; S. Potenza; A. Vita
1581-1594	Oligonucleotide Labeling Methods 4. Direct Labeling Reagents with a Novel, Non-Nucleosidic, Chirally Defined 2-Deoxy-β-D-Ribosyl Backbone.	Thomas H. Smith; Mark A. Kent; Sylvester Muthini; Steven J. Boone; Paul S. Nelson
1595-1601	Conformational Analysis of 3′-Deoxyribonucleosides using 1D-Noe Difference Spectroscopy	Anil Kumar; S. B. Katti; H. Rosemeyer; Frank Seela
1603-1610	Fluorescent-Labeled Oligonucleotide Probes with Non-Nucleotide Linker: Detection of Hybrid Formation by Fluorescence Anisotropy	Sucheta V. Patil; Manikrao M. Salunkhe
1611-1617	The RNA World: Functional Diversity in a Nucleoside by Carboxyamidation of Uridine	Torin M. Dewey; Carina M. Zyzniewski; Bruce E. Eaton
1619-1634	Oligodeoxyribonucleosides Containing 1-β-D-Glucopyranosylthymine Synthesis and Substrate Properties	Boris S. Ermolinsky; Marina V. Fomitcheva; Ekaterina V. Efimtseva; Sergey V. Meshkov; Sergey N. Mikhailov; Dmitriy S. Esipov; Elena F. Boldyreva; Vyacheslav G. Korobko
1635-1648	Synthesis of Oligodeoxyribonucleoside Methylphosphonates Containing 2-Aminopurine	Yuanzhong Zhou; Paul O. P. Ts'o
1649-1656	Synthesis of 2,2′-Anhydro Nucleosides with a Modified Sugar Side-Chain	Johann Hiebl; Erich Zbiral
1657-1668	Pyrimidine Deoxyribonucleosides Are Phosphorylated to Triphosphates at Low Temperatures Too, But Are Not Incorporated into DNA or Phospholipids.	Károly Szikla; Mária Sasvári-Székely; Tatjana Spasokukotskaja; Mária Staub
1669-1678	Zn² -Promoted Hydrolysis of 3′,5′-Dinucleoside Monophosphates and Polyribonucleotides. The Effect of Nearest Neighbours on the Cleavage of Phosphodiester Bonds	Satu Kuusela; Harri Lönnberg

Volume 15, Issue 9 (1996)

iii-iv	Contributors to This Issue
1441-1445	Sulfurization Efficiency in the Solution Phase Synthesis of Deoxyribonucleoside Phosphorothioates - Comparison of Sulfur Triethylamine with Various Sulfurizing Agents	Zacharia S. Cheruvallath; Douglas L. Cole; Vasulinga T. Ravikumar
1447-1457	Radical-Mediated Cyclization of A 6-Chloro-9-(2-Deoxy--d erythro-pent-1-enofuranosyl)-8-(2,2-dibromovinyl) purine	Atsushi Kittaka; Naoki Yamada; Hiromichi Tanaka; Kazuo T. Nakamura; Tadashi Miyasaka
1459-1467	Chemoenzymic Synthesis of P^α-Methyl Deoxynucleoside Triphosphates	Magda A. Dineva; Dimiter D. Petkov
1469-1479	Study of Analogues of Thymidine-5′-Monophosphate and Thymidine as Substrates or Inhibitors of Chick Embryo Liver Thymidylate Kinase	Jean-François Navé; Bernhard Neises; Anne Eschbach
1481-1493	Synthesis of 1-Hydroxy-10-methyl-pyrimido [1, 6-C][1, 3]oxazine and the Oxazepine Derivative, Structural Mimicry of Anti-Constrained Acyclic Thymidine	Ling-Yih Hsu; Dean S. Wise; John C. Drach; Leroy B. Townsend
1495-1518	Synthesis of 4-Deoxy-4-C-hydroxymethyl-α-L-Lyxo-Pyranosyl Thymine	Bogdan Doboszewski; Piet A. M. Herdewijn
1519-1529	Synthesis and Analytical Characterization of RNA-Polyethylene Glycol Conjugates	Andres Jäschke; Rolf Bald; Eckhart Nordhoff; Franz Hillenkamp; Dieter Cech; Volker A. Erdmann; Jens P. Fürste
1531-1543	Synthesis of Extended Carbamate and Urea Linked Thymidine Dimers	Shoukath M. Ali; Peter K. Bridson
1545-1558	Interaction of Escherichia Coli Ribonuclease H With Hybrid Duplexes Containing 2′-Deoxyxylotrymidine, 2′-Deoxy-2′ Fluorouridine or Alpha-Thymidine	Y. I. Alekseev; N. F. Krynetskaya; V. N. Tashlytsky; T. S. Oretskaya; N. G. Dolinnaya; F. Morvan; B. Rayner; C. Malvy; Z. A. Shabarova
1559	Erratum

Volume 15, Issue 7-8 (1996)

iii-iv	Contributors to This Issue
1263-1273	Base-Labile Group Protected Biotinphosphoramidite Reagents for Solid Phase Biotinylation of Oligonucleotides	Pradeep Kumar; A. K. Sharma; K. C. Gupta
1275-1285	The Structure of 5-Cyclohexyl-2′-Deoxyuridine as Studied by X-Ray Crystallography and NMR Spectroscopy	I. Basnak; Ming Sun; T. A. Hamor; N. Spencer; R. T. Walke
1287-1305	Synthesis and Mass Spectrometry Analysis of Oligonucleotides Bearing 5-Formyl-2′-Deoxyurldlne in Their Structure	T. Berthod; Y. Pétillot; A. Guy; J. Cadet; E. Forest; D. Molkot
1307-1313	Stereoselective Synthesis of 6-Methyl-9-(2-Deoxy-β-D-Erythro-Pentofuranosyl)purine	Janet E. Anderson-McKay; Gerald W. Both; Gregory W. Simpson
1315-1321	Synthesis of a Fluorinated Ganciclovir Analog	Marcos L. Sznaidman; Lilia M. Beauchamp
1323-1334	Ribosylation of Pyrimidine 2′-Deoxynucleosides	Sergey N. Mikhailov; Erik De Clercq; Piet Herdewijn
1335-1346	Synthesis and Antiviral Activities of Some Novel Carbocyclic Nucleosides	M. Carmen Balo; Franco Fernández; Evangelina Lens; Carmen López; Erik De Clercq; Graciela Andrei; Robert Snoeck; Jan Balzarini
1347-1359	Enzyme-Mediated Protecting Group Chemistry on the Hydroxyl Groups of Nucleosides	Ashok K. Prasad; Jesper Wengel
1361-1368	Convenient Synthesis of 4-C-Branched Lactones and 3′-C-Branched 2′,3′-Dideoxynucleosides	Jesper Wengel; Kirsten Østergaard; Anders Hager
1369-1381	Methodology for the Synthesis of Dinucleoside Monophosphates Containing A 2′-Deoxy-3-Isoadenosine Unit: 3-iso-dApT and Tp(3-iso-dA)	Nelson J. Leonard; Neelima
1383-1395	An Extended Phosphate Linkage: Synthesis, Hybridization and Modeling Studies of Modified Oligonucleotides	Becky Haly; Laurent Bellon; Venkatraman Mohan; Yogesh Sanghvi
1397-1409	Synthesis and Anti-HIV Evaluation of New 5-Substituted-2′,3′-Dideoxy-3′-thiauridine Nucleosides	Nicolas Mourier; Carole Trabaud; Valerie Niddam; Jean-Christophe Graciet; Michel Camplo; Jean-Claude Chermann; Jean-Louis Kraus
1411-1421	Synthesis of 7-(β-D-Glucopyranosyl)-6-Thiotheophylline and 7-(α-D-Arabinopyranosyl)-6-Thiotheopwlline. Conformational Study of the Peracetyl Derivatives.	Rodrigo Rico-Gómez; Ezequiel P. de Inestrosa-Villatoro; Juan Manuel López-Romero; Francisco Nájera; Rafael López-Corpas
1423-1432	Reverse Transcription of 5-Fluorouracil-Substituted RNA	Tim Fisher; L. James Maher III
1433-1437	Thin Layer Chromatography of Radiolabeled Oligonucleotide Analogues: A Rapid and Sensitive Purity Assay	Robert K. DeLong
1439	Erratum

Volume 15, Issue 6 (1996)

iii	Contributors to This Issue
1121-1135	Relationship Between Chemical Structure and Antileishmanial Effect of Sinefungine Analogues	P. Blanchard; M. S. El Kortbi; J. -L. Fourrey; F. Lawrence; M. Robert-Gero
1137-1147	Cyanogen Bromide-Induced Chemical Ligation: Mechanism and Optimization of the Reaction Conditions	O. A. Fedorova; M. B. Gottikh; T. S. Oretskaya; Z. A. Shabarova
1149-1155	Efficiency Of Coupling in the Synthesis of Deoxyribonucleotide Phosphorothioates Via Phosphotriester Approach Utilizing Various Activating Reagents	Vasulinga T. Ravikumar; Zacharia S. Cheruvallath
1157-1167	New Neplanocin Analogues. V. A Potent Adenosylhomocysteine Hydrolase Inhibitor Lacking Antiviral Activity. Synthesis And Antiviral Activity Of 6″-Carboxylic Acid Derivatives Of Neplanocin A	Takumi OBARA; Satoshi SHUUTO; Yasuyoshi SAITO; Minoru TORIYA; Kiyoshi OGAWA; Satoshi YAGINUMA; Shiro SHIGETA; Akira MATSUDA
1169-1178	Influence of a Thiophosphate Linkage on the Duplex Stability - Does Sp Configuration Always Lead to Higher Stability Than Rp?	H. Kanehara; T. Wada; M. Mizuguchi; K. Makino
1179-1187	Synthesis of Cis-1-[(2-Hydroxymethyl) Cyclopentyl]Uridine and Determination of its Conformation by X-Ray Crystallography and Ami Theoretical Calculations	Lourdes Santana; Marta Teijeira; Eugenio Uriarte; Carmen Teran; Umberto Casellato; Rodolfo Graziani
1189-1202	Synthesis of New 5″-Sulfonylamido Derivatives of 3″-Azido-3″-Deoxythymidine (AZT)	Wojciech Urjasz; Lech Celewicz; Krzysztof Golankiewicz
1203-1221	Synthesis and Biological Evaluation of Some Acyclic Pyridine C-Nucleosides. Part Two	Johan Van hemel; Eddy L. Esmans; Alex De Groot; Roger A. Dommisse; Jan M. Balzarini; Erik D. De Clercq
1223-1236	Syntheses of 2″,3″-Dideoxy-L-Glycero-Pentofuranosyl C-Nucleosides	Chang Soo Lee; Jinfa Du; Chung K. Chu
1237-1251	Synthesis and Properties of DNA Dumbbells Containing Chemically Active Substituted Pyrophosphate Internucleotide Groups	Svetlana A. Kuznetsova; Marta Blumenfeld; Marc Vasseur; Zoe A. Shabarova

Volume 15, Issue 5 (1996)

iii-iv	Contributors to This Issue
967-979	Cis (IS,3R)-1-(9-Adenyl)-3-Hydroxycyclopentane Inhibits the Respiratory Burst from Polymorphonuclear Leukocytes and Has In Vivo Efficacy in an Acute and Chronic Model of Inflammation	David R. Borcherding; Brent T. Butler; Matthew D. Linnik; Shujaath Mehdi; Mark W. Dudley; Carl K. Edwards III
981-994	A Direct Approach to the Synthesis of Famciclovir and Penciclovir	Bernadette M. Choudary; Graham R. Geen; Peter M. Kincey; Martin J. Parratt; J. Robert; M. Dales; Graham P. Johnson; Steven O'Donnell; David W. Tudor; Neil Woods
995-1008	New Non-Aromatic Triazinic Nucleosides: Synthesis and Antiretroviral Evaluation of β-Ribosylamine Nucleoside Analogs	Jean Depelley; Robert Granet; Mourad Kaouadji; Pierre Krausz; Salomon Piekarski; Sylvie Delebassée; Claudine Bosgiraud
1009-1028	Structure of the Trinucleotide D-acp³U-A with Coordinated Mg² Demonstrates that Modified Nucleosides Contribute to Regional Conformations of RNA	John W. Stuart; Mufeed M. Basti; Wanda S. Smith; Brian Forrest; Richard Guenther; Hanna Sierzputowska-Gracz; Barbara Nawrot; Andrzej Malkiewicz; Paul F. Agris
1029-1039	A Rapid, High-Yield Method for 5′-Hydroxyl Protection in Very Reactive and Amino Group Modified Nucleosides Using Dimethoxytrityl Tetrafluoroborate	Mahesh K. Lakshman; Barbara Zajc
1041-1057	Definitive Solution Structures for the 6-Formylated Versions of 1-(βD-Ribofuranosyl)-, 1-(2′-Deoxy-β-D-Ribofuranosyl)-, and 1-β-D-Arabinofuranosyluracil, and of Thymidine	Michael P. Groziak; Ronghui Lin; William C. Stevens; Linda L. Wotring; Leroy B. Townsend; J. Balzarini; M. Witvrouw; E. De Clercq
1059-1076	Synthesis of Mimics to Thymidine and 5-(2″-Thienyl)-2′-Deoxyuridine Triphosphates	Ulf Wellmar; Anna-Britta Hörnfeldt; Salo Gronowitz; Nils Gunnar Johansson
1077-1095	Synthesis and ¹H and ¹³C NMR Spectral Characteristics of 8-Bromo-2′,3′-Dideoxyguanosine and 8-Bromo-2′,3′-Dideoxyinosine	Joanna Zeidler; Bożenna Golankiewicz
1097-1111	The Effects of 2-5A on Protein Synthesis in Wheat Germ Extracts and Tobacco Protoplasts	Erkki Truve; Lenne Nigul; Teemu H. Teeri; Merike Kelve
1113-1120	Model Syntheses of Thiazolidine Nucleoside Analogues	Gloria Rassu; Franca Zanardi; Mara Cornia; Giovanni Casiraghi

Volume 15, Issue 4 (1996)

iii-iv	Contributors to This Issue
833-855	Stereoselective Reactions OF 1-(4,6-O-Benzylidene-2,3-Didehydro-2,3-dideoxy-3-nitro-β-D-hexopyranosyl)uracil with some Nucleophiles	N. Ohta; K. Minamoto; Y. Yamamoto; N. Koide; R. Sakoda
857-865	Trifurcated (Four-Center) Hydrogen Bond in Solid State Crystal Structure of 5′-Amino-5′-deoxyadenosine p-Toluenesulfonate	G. S. Padiyar; T. P. Seshadri
867-878	Use of Cyclohexene Epoxides in the Preparation of Carbocyclic Nucleosides	S. N. Mikhailov; N. Blaton; J. Rozenski; J. Balzarini; E. De Clercq; P. Herdewijn
879-888	Express Protocol for Functionalization of Polymer Supports for Oligonucleotide Synthesis	P. Kumar; A. K. Sharma; P. Sharma; B. S. Garg; K. C. Gupta
889-898	Nucleosides Having Quinolone Derivatives as Nitrogenated Base: Regiospecific and Stereospecific Ribosylation of 3-Carbethoxy-1,4-dihydro-4-oxoquinolines	A. D. da Matta; A. M. R. Bernardino; G. A. Romeiro; M. R. P. de Oliveira; M. C. B. V. de Souza; V. F. Ferreira
899-906	An Improved Synthesis of Azidothymidine	M. I. Balagopala; A. P. Ollapally; H. J. Lee
907-921	Preparation of Oligonucleotides Containing 5-Bromouracil and 5-Methylcytidine.	E. Ferrer; C. Fàbrega; R. G. Garcia; F. Azorín; R. Eritja
923-936	Synthesis of Modified Oligonucleotides and Production of Duplexes With Covalently Linked Chains	S. I. Antsypovich; T. S. Oretskaya; E. M. Volkov; E. A. Romanova; V. N. Tashlitsky; M. Blumenfeld; Z. A. Shabarova
937-960	The Novel 6–(N-Pyrrolyl)purine Acyclic Nucleosides: ¹H and ¹³C NMR and X-ray Structural Study	S. Raić; M. Pongraćić; J. Vorkapić-Furać; D. Vikić-Topić; A. Hergold-Brundić; A. Nagl; M. Mintas
961-965	Announcement

Volume 15, Issue 1-3 (1996)

xi-xiv	Contributors to This Issue
xv-xvii	Preface
1-16	Ribosylation of the Base Residue of Inosine Derivatives by Phase-Transfer Catalysis	Keiichi Aritomo; Chihiro Urashima; Takeshi Wada; Mitsuo Sekine
17-30	An Efficient Method for the Synthesis of β-d-Ribonucleosides Catalyzed by Metal Iodides	Teruaki Mukaiyama; Masashi Nagai; Takafumi Matsutani; Naoyuki Shimomura
31-45	Synthesis of 2′,3′-Dideoxypurinenucleosides via the Palladium Catalyzed Reduction of 9-(2,5-Di-O-acetyl-3-bromo-3-deoxy-β-d-xylofuranosyl)purine Derivatives	Hiroshi Shiragami; Yusuke Amino; Yutaka Honda; Masayuki Arai; Yasuhiro Tanaka; Hisao Iwagami; Toshihide Yukawa; Kunisuke Izawa
47-58	Synthesis of 1-(2,3-Dideoxy-β-d-glycero-pent-2-enofuranosyl)thymine (d4T; Stavudine) from 5-Methyluridine	Hiroshi Shiragami; Takashi Ineyama; Yumiko Uchida; Kunisuke Izawa
59-68	Design and Synthesis of Heterocyclic Carboxamides as Natural Nucleic Acid Base Mimics	Donald E. Bergstrom; Peiming Zhang; W. Travis Johnson
69-84	Synthesis and Conformational Studies of New Purine Isodideoxynucleosides	Lawrence B. Zintek; Tamera S. Jahnke; Vasu Nair
85-96	Intramolecular Radical Reactions of 5′-O-Modified 2′,3′-Didehydro-2′,3′-Dideoxyuridine Derivatives	Kaoru Hisa; Atsushi Kittaka; Hiromichi Tanaka; Kentaro Yamaguchi; Tadashi Miyasaka
97-107	Tandem Radical Cyclization-Oxygenation of 6-(2,2-Di-bromovinyl)-1-(2-deoxy-d-erytho-pent-1-enofuranosyl)-uracil: Synthesis of Anomeric Spiro Nucleosides Having Arabino and Ribo Configurations	Atsushi Kittaka; Yasuhiko Tsubaki; Hiromichi Tanaka; Kazuo T. Nakamura; Tadashi Miyasaka
109-119	Synthesis of the Fluoromethyl Derivatives of Carbocyclic Oxetanocin A	Yoshiko Sato; Kenji Ueyama; Tokumi Maruyama; Douglas D. Richman
121-134	The Synthesis of Some 5-Alkyl (Cycloalkyl)-Substituted 2′ -Deoxy-4′-Thiouridines	I. Basnak; M. Sun; P. L. Coe; R. T. Walker
135-148	Some Reactions of 4′-Thionucleosides and Their Sulfones	E. Louise Hancox; Richard T. Walker
149-167	Synthesis of Methylene-Bridged Analogues of Nicotinamide Riboside, Nicotinamide Mononucleotide and Nicotinamide Adenine Dinucleotide	Pawel Lipka; Andrzej Zatorski; Kyoichi A. Watanabe; Krzysztof W. Pankeiwicz
169-181	Nucleosides and Nucleotides. 139. Stereoselective Synthesis of (2′S)-2′-C-Alkyl-2′-deoxyuridines	Tomoharu Iino; Satoshi Shuto; Akira Matsuda
183-204	Synthesis of 2′-C-α-Methyl-2′,3′-dideoxynucleosides	Indrajit Giri; Pascal J. Bolon; Chung K. Chu
205-217	Polydeoxyaminohexopyranosylnucleosides. Synthesis of 1-(2,3,4-Trideoxy-3-nitro-β-D-erythro- and threo-hexopyranosyl)-uracils from Uridine	Akira Matsuda; Kyoichi A. Watanabe
219-233	Electrophilic Amination of Adenines. Formation and Characteristics of N-Aminoadenines	Tetsuya Saga; Toyo Kaiya; Shoji Asano; Kohfuku Kohda
235-250	Synthesis, Conformational Analysis, and Biological Activity of a Rigid Carbocyclic Analogue of 2′-Deoxy Aristeromycin Built on a Bicyclo[3.1.0]hexane Template	Maqbool A. Siddiqui; Harry Ford Jr.; Clifford George; Victor E. Marquez

Volume 15, Issue 1-3 (1996)

251-263	Nucleosides and Nucleotides. 140. Synthesis and Antileukemic Activity of 5-Carbon-Substituted 1-β-d-Ribofuflranosylimidazole-4-Carboxamides	Noriaki Minakawa; Naoshi Kojima; Takuma Sasaki; Akira Matsuda
265-286	Synthesis, In Vitro Biological Stability, and Anti-HIV Activity of 5-Halo (or Methoxy)-6-Alkoxy (Azido or Hydroxy)-5,6-Dihydro-2′,3′-Didehydro-3′-Deoxythymidine Diastereomers as Potential Prodrugs of 2′,3′-Didehydro-3′-deoxythymidine (D4T)	Rakesh Kumar; Lili Wang; Leonard I. Wiebe; Edward E. Knaus
287-304	Synthesis and Biological Evaluation of 4′-C-Methyl Nucleosides	Toshiaki Waga; Hiroshi Ohrui; Hiroshi Meguro
305-324	Synthesis and Biological Evaluation of 1′-C-Cyano-Pyrimidine Nucleosides	Yuichi Yoshimura; Fumitaka Kano; Shuichi Miyazaki; Noriyuki Ashida; Shinji Sakata; Kazuhiro Haraguchi; Yoshiharu Itoh; Hiromichi Tanaka; Tadashi Miyasaka
325-335	Synthesis of 1,5-Anhydrohexitol Nucleosides as Mimics of AZT, D4T and DDC	Ilse Verheggen; Arthur Van Aerschot; Jef Rozenski; Gerard Janssen; Erik De Clercq; Piet Herdewijn
337-347	A Novel Type of Spironucleosides: 2′,5′-O-bis-TBDMS Uridine-3′-spiro-3′-isoxazolidin-5′-one and Its Thymidine Congener	Jean M. J. Tronchet; Imre Kovacs; Françoise Barbalat-Rey; Naz Dolatshahi
349-359	Novel Tsao Derivatives. Synthesis and Anti-HIV-1 Activity of Allofuranosyl-TSAO-T Analogues	Rosa Alvarez; Ana San-Félix; Erik De Clercq; Jan Balzarini; María José Camarasa
361-378	Nucleoside Phosphonates. Development of Synthetic Methods and Reagents	Annika Kers; Inger Kers; Adam Kraszewski; Michal Sobkowski; Tomas Szabó; Mats Thelin; Rula Zain; Jacek Stawinski
379-386	The 1,1-Dianisyl-2,2,2-trichloroethyl Moiety as a New Protective Group for the Synthesis of Dinucleostde Trifluoromethylphosphonates	Rosa Maria Karl; Wolfgang Richter; Roland Klösel; Michael Mayer; Ivar Ugi
387-397	Syntheses of 2′-O-Methylisocytidine Phosphoramidite and Methylphosphonamidite Synthons	Daguang Wang; Paul O. P. Ts'o
399-406	Isolation of Oligodeoxynucleoside Phosphorothioate Diastereomers by the Combination of DEAE Ion-Exchange and Reversed-Phase Chromatography	Hideyuki Kanehara; Masatsugu Mizuguchi; Keisuke Makino
407-417	Stereocontrolled Transesterification for the Synthesis of Chiral Phosphite Triester Backbone	Masatsugu Mizuguchi; Keisuke Makino
419-430	Purification of 5′-O-Trityl-on Oligoribonucleotides. Investigation of Phosphate Migration During Purification and Detritylation.	Bashar Mullah; Alex Andrus
431-443	Nucleosides, LVIII¹ Synthesis of Base - Modified Oligonucleotides Containing 6- and 7-Aryl Lumazines	Yuris Maurinsh; Wolfgang Pfleiderer
445-464	Synthesis of 1-Deazaadenosine Analogues of (2′→5′) ApApA	Igor A. Mikhailopoulo; Elena N. Kalinichenko; Tatjana L. Podkopaeva; Thomas Wenzel; Helmut Rosemeyer; Frank L. Seela
465-475	Synthesis of Oligopeptides as Polynucleotide Analogs	Hiroki Umemiya; Hiroyuki Kagechika; Yuichi Hashimoto; Koichi Shudo
477-488	¹⁹F NMR of RNA. The Structural and Chemical Aspects of 5-Fluoro-cytidine and-uridine Labelling of Oligoribonucleotides	Artur Fischer; Zofia Gdaniec; Ewa Biala; Marek Łożyński; Jan Milecki; Ryszard W. Adamiak
489-503	NMR Studies of a Lead Ribozyme and Its Non-Cleavable Analogue	Masato Katahira; Takashi Sugiyama; Mayumi Kanagawa; Mi Hee Kim; Seiichi Uesugi; Toshiyuki Kohno
505-517	Cleavage of Short RNAs Containing Higher Ordered Structures by Hammerhead Ribozymes	Makoto Koizumi; Tsutomu Ohta; Yasuo Komatsu; Eiko Ohtsuka
519-529	Properties and Anti-HIV Activity of Nicked Dumbbell Oligonucleotides	Hidefumi Yamakawa; Kazumi Hosono; Toshiaki Ishibashi; Hideki Nakashima; Takafumi Inagawa; Naoki Yamamoto; Kazuyuki Takai; Hiroshi Takaku

Volume 15, Issue 1-3 (1996)

539-557	Effects of Psoralen-Derivatized Oligonucleoside Methylphosphonates on Vesicular Stomatitis Virus (VSV) Protein Synthesis In Vitro and in VSV-Infected Cells	Joel T. Levis; Joanne M. Kean; Paul S. Miller
559-567	The Stability of DNA and RNA G-Quartets	Naoki Sugimoto; Tatsuo Ohmichi; Muneo Sasaki
569-584	Polarized Micro Raman Spectroscopic Studies of Nucleic Acid: Local Raman Tensors in Inosine-5′-monophosphoric Acid and the Orientation of Ekypoxanthine Residue in Poly(rI). Poly(rC) Fiber	Koichi Ushizawa; Toyotoshi Ueda; Masamichi Tsuboi
585-598	Comparative Studies of the Thermodynamic Stabilities Between Sheared A:G and Watson-Crick A:U(T) Base Pairs in RNA and DNA	Masato Katahira; Jun-ichi Saeki; Mayumi Kanagawa; Masashi Nagaoka; Seiichi Uesugi
599-605	Drug Binding to Higher Ordered DNA Structures: Ethidium Bromide Complexation with Parallel Quadruple-Stranded DNA	Toshio Shida; Norihito Ikeda; Junichi Sekiguchi
607-618	Synthetic Nucleoside and Nucleotides. XXXIV. Photoaffinity Labeling of HIV Reverse Transcriptase: Synthesis and Utilization of 2′,3′-Dideoxy Uridylate Analogs Bearing Aryl(trifluor0methyl)-Diazirine Moiety	Toyofumi Yamaguchi; Mineo Saneyoshi
619-629	O⁶-(4-Nitrophenyl)inosine and -Guanosine as Chromogenic Substrates for Adenosine Deaminase	Jiri Zemlicka; Takeshi Endo
631-647	Deamination of 9-(Hydroxymethylated cycloalkyl)-9H-adenines (Carbocyclic Adenine Nucleosides) by Adenosine Deaminase: Effect of High-Pressure Upon Deamination Rate and Enantioselectivity	Nobuya Katagiri; Yumiko Ito; Takuya Shiraishi; Tokumi Maruyama; Yoshiko Sato; Chikara Kaneko
649-654	Substrate Properties of Adenosine- and Uridine- 3′- Phenylphosphonates for 3′-Nucleotidase/Nucleases	H. Uchida; Y. -D. Wu; S. Sonoda; S. Fukushima; J. Fukuda; I. Takahashi; S. Maeda; A. Nomura
655-667	Mode of Inhibition of HIV Reverse Transcriptase- Catalyzed DNA Synthesis by 3′-Amino-3′-Deoxythymidine 5′ -Tfiphosphate	Lyubov S. Victorova; Alexander A. Krayevsky
669-682	N²-(p-n-Octylphenyl)dGTP: Synthesis and Inhibitory Activity Against DNA Polymerases	Janis Jansons; James Stattel; Annalisa Verri; Joseph Gambino; Naseema Khan; Federico Focher; Silvio Spadari; George Wright
683-692	Chain Termination With Sugar- Modified Nucleotide Analogs in the DNA Synthesis by DNA Polymerase γ	Shunji Izuta; Shonen Yoshida
693-717	Survey of Nonxanthine Derivatives as Adenosine Receptor Ligands	Suhaib M. Siddiqi; Xiao-duo Ji; Neli Melman; Mark E. Olah; Rahul Jain; Patricia Evans; Marc Glashofer; William L. Padgett; Louis A. Cohen; John W. Daly; Gary L. Stiles; Kenneth A. Jacobson
719-731	A Colorimetric DNA Diagnostic Method for Falciparum Malaria and Vivax Malaria: A Field Trial in the Solomon Islands	Meiji Arai; Kaori Kunisada; Hye-Sook Kim; Hirofumi Miyake; Chiyoko Mizukoshi; Toshifumi Kakutani; Akio Yamane; Satoru Nakagami; Shintaro Kawai; Hiromi Nakano; Fumihiko Kawamoto; Yusuke Wataya
733-738	Efficient Synthesis of 2′-Bromo-2′-Deoxy-3′,5′-O-TPDS-pyrimidine Nucleosides by Boron Trifluoride Catalyzed Reaction of O²,2′-Anhydro-(1-β-D-Arabinofuran0Syl)pyrimidine Nucleosides with Lithium Bromide	Yukio Aoyama; Takeshi Sekine; Yoshiaki Iwamoto; Etsuko Kawashima; Yoshiharu Ishido
739-742	A New Reagent for the Formation of Anhydronucleosides	B. Bennua-Skalmowski; H. Vorbrüggen
743-747	Interactions of 5-(1-Pyrenyl)-10,15,20-tris(4-methylpyridinium)porphine with Double-Helix and Triple-Helix Nucleic Acids	Naoki Sugimoto; Shu-ichi Nakano; Misa Katoh; Muneo Sasaki; Shin-ichi Kugimiya
749-769	An Efficient Method for the Synthesis of [4–¹⁵N]Cytidine, 2′-Deoxy[4–¹⁵N]Cytidine, [6–¹⁵N]adenosine, and 2′-Deoxy [6–¹⁵N]adenosine Derivatives	Kazuo Kamaike; Mihoko Takahashi; Kazuyuki Utsugi; Kazue Tomizuka; Yasunori Okazaki; Yuri Tamada; Kazutomo Kinoshita; Hiroyuki Masuda; Yoshiharu Ishido
771-791	Transglycosylation Reactions of Purine Nucleosides. A Review	Jerzy Boryski
793-807	Conformational Properties of Purine-Like C-Nucleosides	Brian A. Otter; Robert S. Klein
809-820	Configurational Assignment in 2′-Deoxy-4′-Thionucleosides - A Review	David F. Ewing; Grahame Mackenzie
821-831	Herpes Simplex Virus Thymidine Kinase Gene-Transfected Tumor Cells; Sensitivity to Antiherpetic Drugs	J. Balzarini

Volume 14, Issue 9-10 (1995)

1823-1829	Interaction of RKRK Tetrapeptide with Polynucleotides	Ajay Kumar
1831-1852	Synthesis of 5′-Fluoro-5′-deoxy-and 5′-Amino-5′-Deoxytoyocamycin and Sangivamycin and Some Related Derivatives	Moheshwar Sharma; Yi X. Li; Miroslav Ledvina; Miroslav Bobek
1853-1859	Oligonucleotides Containing Acyclic Nucleoside Analogues with Carbamate Internucleoside Linkages	Ivan Habus; Sudhir Agrawal
1861-1871	Kinetic Properties of Adenine Nucleotide Analogues Against Purified 5-Phosphoribosyl-1-pyrophosphate Synthetases from E. coli, Rat Liver and Human Erythrocytes	J. Balzarini; J. F. Navé; M. A. Becker; M. Tatibana; E. De Clercq
1873-1887	Synthesis and Biochemical Activity of 5-Tethered Carborane-Containing Pyrimidine Nucleosides as Potential Agents for DNA Incorporation	Feng-Guang Rong; Albert H. Soloway; Seiichiro Ikeda; David H. Ives
1889-1900	A Simple Method for Synthesis of Spongosine, Azaspongosine, and Their Antiplatelet Effects	Lalit M. Ojha; Deepa Gulati; Neena Seth; Diwan S. Bhakuni; Ram Pratap; Kailash C. Agarwal
1901-1904	Synthesis of 2-Alkyl-3-hydroxy-4-pyridinone-ribonucleosides, Potential Oral Iron Chelators	Gang Liu; Fred W. Bruenger; Amy M. Barrios; Scott C. Miller
1905-1912	Synthesis of a Carboxamide Linked T*T Dimer with an Acyclic Nucleoside Unit and Its Incorporation in Oligodeoxynucleotides	Erik Larsen; Krzysztof Danel; Erik B. Pedersen
1913-1927	Fluorinated Carbaacyclonucleosides: Synthesis and Evaluation of Antiviral Activity	Maureen Lewis; T. Brian; H. McMurry; Erik De Clercq
1929-1945	Enantiospecific Synthesis of Carbocyclic Aminoimidazole Carboxamide Ribonucleotide (C-AICAR), Succinoaminoimidazole Carboxamide Ribonucleotide (C-SAICAR), and a New Intermediate for SAICAR Analogs	Laurent Schmitt; Carol A. Caperelli
1947-1959	Conformational Transitions in Poly d(CGCGCGTTAATT)	Ajay Kumar
1961-1984	Synthesis of 2′-Substituted Sulfide-Linked Dinucleotides	Daguang Wang; Bin; Masad J. Damha; George Just
1985-1996	Synthesis, Conformational and Configurational Studies of Some New Acetylated Glycosides of 2-Thio-3-aryl-4(3H)-quinazolinones, Their Thiono and 3,1-Benzothiazin-2,4-dithione	Mohamed F. Abdel-Megeed; Mohamed A. Saleh; Youssef L. Aly; Ibrahim M. Abdo
1997-2008	Synergistic Effect of 5-Nitro-2′-deoxyuridine with Ganciclovir Against Human Cytomegalovirus In Vitro	T. Sudhakar Rao; Robert F. Rando; John H. Huffman; Ganapathi R. Revankar
2009-2025	Building Blocks for Synthesis of Oligoarabinonucleotides: Preparation of Arabinonucleoside H-Phosphonates from Protected Ribonucleosides	Eriks Rozners; Erika Bizdena
2027-2038	Synthesis of a Carboxamide Linked U^Br*U^Br Dimer–Duplex and Triplex Stabilities of the Corresponding Oligodeoxynucleotides	Abdel Aleem H. Abdel Aleem; Erik Larsen; Erik B. Pedersen
2039-2049	A Short High Yielding Synthesis of the Potent Anti-VZV Carbocyclic Nucleoside Analogue Carba-BVDU	P. G. Wyatt; A. S. Anslow; B. A. Coomber; R. P. C. Cousins; D. N. Evans; V. S. Gilbert; D. C. Humber; I. L. Paternoster; S. L. Sollis; D. J. Tapolczay; G. G. Weingarten
2051-2060	The Synthesis and Biological Evaluation of Sulfamoyl Nucleosides Related to Carbovir and AZT	Robert Vince; Phuong T. Pham
2061-2077	Synthesis and Biological Activity of Cyclohexenyl Nucleosides. cis-5-(9H-Purin-9-yl)-3-cyclohexenyl Carbinols and Their 8-Azapurinyl Analogs	Michael J. Konkel; Robert Vince
2079-2087	Different Mechanisms of Inhibition of DNA Synthesis by (E)-5-(2-Bromovinyl)-2′-deoxyuridine in Cells Transfected with Gene for Thymidine Kinase of Herpes Simplex Virus Type 1 and in Cells Infected with the Virus	Yasuhide Hirota; Yujiro Arao; Akiko Matsumoto; Shiro Nii; Yusuke Wataya
2089-2097	Molecular Mechanism of 5-Fluoro-2′-deoxyuridine-induced dNTP Imbalance Cell Death: Purification of an Endonuclease Involved in DNA Double Strand Breaks During dNTP Imbalance Death	Hwa-shin Hwang; Masashi Ohtani; Tohru Nakazawa; Tatsushi Igaki; Osamu Masui; Shiro Kankawa; Chikao Nakayama; Sei Yoshida; Akiko Yoshioka-Hiramoto; Yusuke Wataya

Volume 14, Issue 8 (1995)

1619-1630	Total Synthesis of the Thymidine Analogue of Sinefungin	Derek H. R. Barton; Stephan D. Gero; Guillerm Negron; Béatrice Quiclet-Sire; Mohammad Samadi; Claire Vincent
1631-1638	Palladium Catalysis in the Synthesis of 8-Position modified Adenosine, 2′-Deoxyadenosine and Guanosine	Chi Tu; Charlene Keane; Bruce E. Eaton
1639-1657	Catalytic Osmylation and Antiviral Activity of Some Garbocyclic 5-Substituted Uridine and Cytidine Analogues	Anne Popescu; Anna-Britta Hörnfeldt; Salo Gronowitz; Nils Gunnar Johansson
1659-1670	Impairment of Streptomyces and Micromonospora Differentiation by Dna-Methylase Inhibitors	Isabel S. Novella; Jesús Sánchez
1671-1674	The ATP ANalogue Containing a Methylene Group in Place of the 5′ Oxygen Serves as a Substrate for Bacteriophage T3 RNA Polymerase	E. J. Higgins; T. J. Miller; P. T. Gilham
1675-1691	Relationship Between Conformation and Antiviral Activity-III. 3′-Azidothymidine (AZT) and 3′-Azido-2′, 3′-dideoxy-5-hydroxymethyluridine	Sagar V. Gupta; Sashi V. P. Kumar; Allan L. Stuart; Ruili Shi; Keith C. Brown; Wajdi M. Zoghaib; Jung Li; Louis T. J. Delbaere
1693-1702	Synthesis and Biological Activity of Some 5-Substituted-6-azauracil-N-1-Nucleosides of 2-Acetamido-2-Deoxy-D-glucose	Najim A. Al-Masoudi; Fadhel B. Issa; Wolgang Pfleiderer; Hassan B. Lazrek
1703-1708	6-Substituted Derivatives of Carbovir: Anti-HIV Activity	Robert Vince; John Kilama; Phuong T. Pham; Scott A. Beers; Bonnie J. Bowdon; Kathy A. Keith; William B. Parker
1709-1724	8-Substituted Adenine β-D-Xylofuranosides and α-L-Arabinofuranosides	Janis Jansons; Yuris Maurinsh; Margeris Lidaks
1725-1735	OLigonucleotide (Cyanomethyl) Phosphonates	Reza Fathi; William Delaney; Qing Huang; Alan F. Cook
1737-1758	4′-Aza-3′,5′-dihomothymidine and Derivatives	Jean M. J. Tronchet; Mohammed Iznaden; Françoise Barbalat-Rey; Istvan Komaromi; Naz Dolatshahi; Gérald Bernardinelli
1759-1783	Synthesis of a Series of Purine 2′,3′-Dideoxy-L-Nucleoside Analogues as Potential Antiviral Agents	Tai-Shun Lin; Mei-Zhen Luo; Ju-Liang Zhu; Mao-Chin Liu; Yong-Lian Zhu; Ginger E. Dutschman; Yung-Chi Cheng
1785-1794	The Preparation of a 3′-(2-Cyanoethyl)phosphoramidite of 5′-O-(3-Thiopropyl)methylphosphorylthymidine	Karen J. Percival; Colin W. G. Fishwick
1795-1801	Nucleopeptidic Bioconjugates Containing a Sulfamide Bridge: Linkage via the Mitsunobu Reaction	Marc Critonl; Georges Dewyntert; Nourreddine Aouf; Jean-Louis Montero; Jean-Louis Imbach
1803-1809	Synthesis of a Difluorophosphonate Analog of the Oxathiolanyl Nucleoside (-)-β-L-(2R,5S)-1,3-Oxathianyl-5-fluorocytosine (FTC)	Richard E. Austin; Darryl G. Cleary
1811-1821	A Novel Approach for Isolation and Mapping of Second-Site Revertants of Intron Mutations in a Ribontjcleotide Reductase Encoding Gene (nrdB) of Bacteriophage T4 Using the White Halo Plaque Phenotype	Heajoon Y. Kwon; Sunil K. Lai; Dwight H. Hall

Volume 14, Issue 7 (1995)

1465-1479	Synthesis of Novel 3′-C-(Hydroxymethyl)thymidines and Oligodeoxynucleotide Analogues Containing Compressed 3′-C-Hydroxymethyl-Linked Phosphodiester Backbones	Jesper Wengel; Margit L. Svendsen; Pia N. Jørgensen; Claus Nielsen
1481-1492	Large Scale Synthesis of Oligoribonucleotides on High-Loaded Polystyrene (HLP) Support	Dean Tsou; Arnold Hampel; Alex Andrus; Ravi Vinayak
1493-1502	Synthesis of 3′,4′-C-Bishydroxymethyl-2′,3′,4′-trideoxy-β-L-threo-pentopyranosyl Nucleosides as Potential Inhibitors of HIV	Åsa Lundquist; Ingemar Kvarnström; Stefan C. T. Svensson; Björn Classon; Bertil Samuelsson
1503-1518	Interaction of (2′ -5′) and (3′ -5′) Linked 2-Aminoadenylyl-3-aminoadenosines with Polyuridylic Acid	Masako Muraoka; Seizo Takahashi; Seiichi Uesugi
1519-1537	Isolation and Characterization of an Unusual Nucleoside, 1-α-D-Ribofuranosyl-4-pyridone-3-carboxamide, from the Urines of Normal Human Individuals and Leukemic Patients	G. B. Chheda; H. B. Patrzyc; H. A. Tworek; S. P. Dutta
1539-1543	A New Synthesis of 2′,3′-Didehydro-3′-deoxy-3-Alkylthymidine	G. Negrón; B. Quiclet-Sire; Y. Diaz; R. Gaviño; R. Cruz
1545-1558	Synthesis, Bioactivation and Anti-HIV Activity of 4-Acyloxybenzyl bis(Nucleosid-5′-yl) Phosphates	Anne Routledge; Ian Walker; Sally Freeman; Alan Hay; Naheed Mahmood
1559-1579	Evaluation of the Kinetics of Hydrolysis of Monoamino Analogues of 2′- or 3′-Deoxyadenosine and of 9-(2-Deoxy-β-D-Threo-pentofuranosyl)Adenine or 9-(3-Deoxy-β-D-threo-pentofuranosyl)Adenine by Liquid Chromatography	Grace Thoithi; Ann Van Schepdael; Roger Busson; Piet Herdewijn; Eugène Roets; Jos Hoogmartens
1581-1590	Synthesis and Antiviral Activity of Some N-Pentopyranosyl-2-Pyridinethiones	Adel M. E. M. Attia; Elsayed I. Ibrahim; Fouad E. A. Hay; Mohammed M. A. Abbasi; Hanaa A. E. Mansour
1591-1600	An Efficient Synthesis of 2-[(4-Amino∼1,2-dihyro-2-oxo-1- pyrimidinyl)methoxyi-l,3-propanediyl-di-L-valinate an Anti-cytomegalovirus Agent	Nabih Ghal; Barbara Johnston; Lilia Beauchamp; Taj Naseree; Tracy Scott; Roy Flanagan; Martha Rodriguez
1601-1612	Synthesis of Certain Acyclic Nucleoside Analogs of 1,2,4-Triazolo[3,4-f][1,2,4]triazine and Pyrimido[5,4-d]pyrimidine	T. Sudhakar Rao; Ganapathi R. Revankar
1613-1617	Note: A Convenient Method for the Preparation of N², N²-Dimethylguanosine	Anna Maria Aviñó; Adrian Mayordomo; Ruth Espuny; Montse Bach; Ramon Eritja

Volume 14, Issue 6 (1995)

1163-1177	Preparation and ¹⁷O NMR Spectra of ¹⁷O-Labeled Thymidine 5′-Phosphate Triesters, Alkylphosphonates, Dialkylphosphinates, and Phosphoramidates	T. Sudhakar Rao; A. E. Sopchik; Wesley G. Bentrude
1179-1193	Conformational Studies on Deoxyribonucleosides of C6-Substituted Pyrimidines	Shashidhar N. Rao
1195-1210	Oligodeoxynucleotides Embodying the Ambiguous Base Z, 5-Amino-imidazole-4-carboxamide	Sylvie Pochet; Laurence Dugué
1211-1218	Nucleic Acid Related Compounds: A Convenient Synthesis of 3-Deazauridine Analogues	Adel M. E. Attia; Galal E. H. Elgemeie
1219-1226	Large-Scale Synthesis of Oligodeoxyribonucleotide Phosphorothioate Using Controlled-Pore Glass as Support	Vasulinga T. Ravikumar; Mark Andrade; Tadeusz K. Wyrzykiewicz; Anthony Scozzari; Douglas L. Cole
1227-1232	Efficient Transformation of Thymidine into 2′,3′-Didehydro-2′,3′-Dideoxy-Thymidine (D4T) Involving Opening of a 2,3′-Anhydro Derivative by Phenylselenol	Stéfan Becouarn; Stanislas Czernecki; Jean-Marc Valéry
1233-1249	Synthesis and Antiviral Activity of Carbocyclic 5-Substituted Uridines and Cytidines	Anne Popescu; Anna-Britta Hörnfeldt; Salo Gronowitz
1251-1258	The X-ray Crystal and Molecular Structure of 5-Amino-1-(2,3:5,6-Di-O-isopropylidene-α-D-mannofuranosyl) Imidazole-4-carboxamide	C. E. Briant; D. W. Jones; G. Shaw
1259-1267	Solid Phase Synthesis of 2′, 5′-Oligoadenylates Containing 3′-Fluorinated Ribose	Teréz Kovács; Arthur Van Aerschot; Piet Herdewijn; Paul F. Torrence
1269-1287	A Practical Synthesis of N1-Methyl-2′-deoxy-ψ-uridine (ψ-Thymidine) and Its Incorporation into G-Rich Triple Helix Forming Oligonucleotides	Birendra K. Bhattacharya; Rodrigo V. Devivar; Ganapathi R. Revankar
1289-1300	Synthesis, Conformation of 3′-(Tetrazole-2″-yl)-3′-deoxythymidine and its 5″-Derivatives. Substrate Properties of 3′-(Tetrazole-2″-yl)-3′-deoxythymidine 5′-Triphosphate	V. A. Ostrovskii; E. P. Studentsov; V. S. Poplavskii; N. V. Ivanova; G. V. Gurskaya; V. E. Zavodnik; M. V. Jasko; D. G. Semizarov; A. A. Krayevsky
1301-1314	Structural Characterization of Cyclic ADP-Ribose by NMR Spectroscopy	Takeshi Wada; Kiyoshi Inageda; Keiichi Aritomo; Ken-ichi Tokita; Hiroshi Nishina; Katsunobu Takahashi; Toshiaki Katada; Mitsuo Sekine
1315-1327	Synthesis and Antiviral (RNA) Evaluation of Nucleoside Analogs of Tiazofurin Modified at the Carboxamide Moiety	Michael J. Phelan; Bjarne Gabrielsen; Jorma J. Kirsi; William M. Shannon; Michael A. Ussery; Louis Barthel-Rosa; Ernst M. Schubert; Ganesh D. Kini; Roland K. Robins
1329-1339	Efficient Synthesis of 2′-Amino-2′-deoxypyrimidine 5′-Triphosphates	Danny P. C. McGee; Chandra Vargeese; Yansheng Zhai; Gary P. Kirschenheuter; Alecia Settle; Colleen R. Siedem; Wolfgang A. Pieken
1341-1348	Synthesis and Reactions of Some Glycosylamine Derivatives of 6-Azauracil Nucleosides	Najim A. Al-Masoudi; Ali A. Al-Atoom
1349-1357	Improved Procedure for the Reduction of N - 1 Content in Synthetic Oligonucleotides	Radhakrishnan P. Iyer; Dong Yu; Zhiwei Jiang; Sudhir Agrawal
1359-1377	Solid State and Solution Structure and Conformation of The Antiviral Acyclonucleoside 9-[4-Hydroxy-2-(hydroxymethyl)-butyl]guanine	Karin Bjåmer Birnbaum; Ryszard Stolarski; David Shugar
1379-1392	Synthesis of New Thiazolidinone Nucleoside Analogues	J. C. Graciet; P. Faury; M. Camplo; A. S. Charvet; N. Mourier; C. Trabaud; V. Niddam; V. Simon; J. L. Kraus
1393-1402	Peptide-Nucleoside Conjugates: Synthesis and Anti-HIV Activities	Nicolas Mourier; Carole Trabaud; Jean Christophe Graciet; Vanessa Simon; Valérie Niddam; Philippe Faury; Anne Sophie Charvet; Michel Camplo; Jean-Claude Chermann; Jean Louis Kraus

Volume 14, Issue 6 (1995)

1403-1414	2-Chloro-2′-deoxyadenosine: Synthesis and Antileukemic Activity of 8-Substituted Derivatives	Zygmunt Kazimierczuk; Juhani A. Vilpo; Frank Seela
1415-1423	Synthesis of N-Glycosylated Pyridines as New Antiviral Agents	E. S. Ibrahim; G. E. H. Elgemeie; M. M. Abbasi; Y. A. Abbas; M. A. Elbadawi; A. M. E. Attia
1425-1435	Synthesis of Racemic 5-Substituted 1-(2,3-Dihydroxypropyl)-6-azauracils and Their Isosteric Isomers	Cherng-Chyi Tzeng; Long-Chih Hwang; Chien-Chi Chen; Dau-Chang Wei
1437-1443	Covalent Attachment of Methylene Blue to Oligonucleotides	F. Schubert; A. Knaf; U. Möller; D. Cech
1445-1452	A New Approach to the Synthesis of 2-Aminopurine-2′-deoxyriboside via Tri-n-butyltin Hydride Reduction	Sabine Schmidt; Dieter Cech
1453-1460	Synthesis of 2′,5′-Dideoxy-adenosine-3′-monophosphate Derivatives as Allosteric Inhibitors of Adenylyl Cyclase	Laurent Désaubry; Ilana Shoshani; Roger A. Johnson

Volume 14, Issue 3-5 (1995)

xxiii-xxiv	Preface	E. De Clercq
279-282	Synthesis of 3′-4′-α-Propylene-2′-3′-dideoxynucleosides	Magnus Björsne; Tomas Szabó; Bertil Samuelsson; Björn Classon
283-286	Synthesis and Anti-viral Properties of 2′,3′-Dideoxy-3′,4′-dihydroxymethyl Substituted Pyrimidine Nucleoside Analogues	Magnus Björsne; Björn Classon; Inger Kers; Bertil Samuelsson; Ingemar Kvarnström
287-290	Tautomerism and Regioselectivity in Ribosylation of Guanine	Jerzy Boryski; Andrzej Manikowski
291-293	The Synthesis of Bicyclic N⁴-Amino-2′-deoxycytidine Derivatives	D. Loakes; D. M. Brown
295-297	Carbocyclic Nucleosides with a Modified Cyclopentane Skeleton	O. Caamaño; F. Fernández; G. Gómez; M. I. Nieto
299-301	Synthesis of [1-[2′,5′-bis-O-(t-Butyldimethylsilyl)-β- L-ribofuranosyl] thymine]-3′-spiro-5″-(4″-amino-1″,2″-oxathiole-2″,2″-dioxide) (L-TSAO-T)	Simon Ingate; Ana San-Félix; Erik De Clercq; Jan Balzarini; Maríia-José Camarasa
303-305	Asymmetric Synthesis of Cyclopropyl Carbocyclic Nucleosides	Y. F. Zhao; M. G. Lee; T. -F. Yang; B. K. Chun; J. F. Du; R. F. Schinazi; C. K. Chu
307-309	Radical Mediated Synthesis of 3′-α-C-Allenyl-2′,3′-dideoxythymidine as a Non-polar Analogue of AZT	S. Becouarn; S. Czernecki; J. M. Valéry
311-312	Simple Synthesis of the 5-O-Benzoylriboside of 1,4-Dihydronicotinic Acid; a Cofactor for DT Diaphorase and Nitroreductase Enzymes	Lawrence C. Davies
313-316	Novel Analogues of Tiazofurin by Lawesson Reagent Effected Cyclization	Bozenna Golankiewicz; Piotr Januszczyk
317-320	Synthesis of the β-2′,3′-Unsaturated Pentopyranosyl Nucleosides and Their 3′-Hydroxymethyl Congeners	Bogdan Doboszewski; Norbert Blaton; Piet Herdewijn
321-324	Synthesis of 1,5-Anhydro-2-(N⁶-Cyclopentyladenin-9-Yl)-2-Deoxy-D-Altrohexitol	I. Verheggen; A. Van Aerschot; N. Pillet; E. M. van der Wenden; A. Ijzerman; P. Herdewijn
325-328	Synthetic Approaches to 5:8-Fused Heterocyclic Systems. A Novel Rearrangement During the Synthesis of Imidazo[4,5-e][1,2,4]triazocine Ring System	Friedrich N. Burnett; Ramachandra S. Hosmane
329-332	Synthesis of Analogues of 3′-Deoxypsicothymidine	Jari Hovinen; Alex Azhayev; Andrei Guzaev; Harri Lönnberg
333-336	Highly Diastereoselective Synthesis of (2′S)-[2′-²H]-2′-Deoxyribonucleosides from the Corresponding Ribonucleosides	Etsuko Kawashima; Yukio Aoyama; Mohamed F. Radwan; Masayoshi Miyahara; Takeshi Sekine; Masatsune Kainosho; Yoshimasa Kyogoku; Yoshiharu Ishido
337-340	Synthesis of 9-(2-Hydroxyethoxymethyl)guanine (Acyclovir) from Guanosine	Hiroshi Shiragami; Yoshihito Koguchi; Yasuhiro Tanaka; Satoshi Takamatsu; Yumiko Uchida; Takashi Ineyama; Kunisuke Izawa
341-344	Synthesis of “Reversed” and “Double Headed” Nucleosides	B. Kašnar
345-347	Synthesis of 3′-C-Phosphono Nucleosides from α,β-Unsaturated Lactone	Thomas Kofoed; Erik B. Pedersen
349-352	Synthesis of Fluorescent Adenosine Analogues¹	R. F. de Boer; D. G. I. Petra; M. J. Wanner; A. Boesaart; G. J. Koomen
353-356	Synthesis of Acycloalkenyl Derivatives of Pyrimidines and Purines	H. B. Lazrek; N. Redwane; A. Rochdi; J. L. Barascut; J. -L. Imbach; E. De Clercq
357-358	Carbocyclic Nucleosides: Synthesis of Analogues of Cyclobut-G	F. Fernández; M. C. López; A. R. Hergueta
359-362	Synthesis of 2-Deoxy-4-thio-D-ribofuranose and Its 3-Azido Analogue from L-Arabinose; Intermediates in the Synthesis of 4′-Thiodeoxynucleosides	H. Ait sir; D. F. Ewing; N. Fahmi; G. Goethals; G. Mackenzie; G. Ronco; B. Tber; P. Villa
363-366	The Synthesis of Novel Transition State Analogues Related to Imidazole and Purine Nucleotides Involved in the De novo Biosynthesis of Purines	A. Scott Frame; Richard H. Wightman; G. Mackenzie
367-368	A Regiospecific and Stereoselective Rearrangement of a 1-β-D-Ribofuranosyl-5-aminoimidazole to a 4-β-D-Ribofuranosylaminoimidazole	David F. Ewing; Graharne Mackenzie; Sean P. N. Rouse; Richard M. Scrowston
369-372	A Novel Synthesis of Mizoribine® and Related Nucleosides from Acyclic Precursors	David F. Ewing; Robert W. Humble; Grahame Mackenzie; Gordon Shaw
373-375	Acyclic Nucleoside and Nucleotide Analogues with Amide Bond	E. V. Efimtseva; S. N. Mikhailov; M. V. Jasko; D. V. Malakhov; D. G. Semizarcv; M. V. Fomicheva; E. R. Kern
377-380	Synthesis of Sugar Modified Nucleosides Containing Nicotinic, Quinaldic, Indol-3-ylpropionic or 1-Nitroanthraquinone-2-carboxylic Acid Residue	S. Ya. Melnik; L. V. Ektova; O. V. Goryunova; E. V. Khorysheva; S. V. Makutova; I. L. Plikhtyak; I. V. Yartseva
381-382	Epimerization at C2 of Methyl 5-O-Benzyl-2-deoxy-2-fluoro-α-D-pentofuranosides upon Oxidation	Igor A. Mikhailopulo; Grigorii G. Sivets; Nicolai E. Poopeiko; Natalia B. Khripach

Volume 14, Issue 3-5 (1995)

383-384	Oxidation-Reduction Sequence for the Synthesis of Peracylated Fluorodeoxy Pentofuranosides	Igor A. Mikhailopulo; Nicolai E. Poopeiko; Grigorii G. Sivets; Natalia B. Khripach
385-388	Base-Transposed Chiral Isomeric Nucleosides	Vasu Nair; Lawrence B. Zintek; Pascal J. Bolon; Todd B. Sells
389-391	Synthesis of Isomeric Dideoxynucleosides with Partial Symmetry	Vasu Nair; Lawrence B. Zintek; Geun S. Jeon
393-396	A Convenient Synthesis of D-Psicofuranosyl Nucleosides¹	Mallela S. P. Sarmastate; Sreenivasulu Megati; Robert S. Klein; Brian A. Otter
397-400	Synthesis of Quinazoline C-Nucleosides: A New Class of 6:6 Bicyclic Purine-Like Analogues.¹	Mallela S. P. Sarma; Phyllis Wilson; Brian A. Otter; Robert S. Klein
401-404	Enzyme Aided Regioselective Acylation of Nucleosides	Shoichiro Ozaki; Kayoko Yamashita; Takako Konishi; Takahiro Maekawa; Mitsuaki Eshima; Atsuliiko Uemura; Lei Ling
405-408	Synthesis of Novel Olefinic Carbocyclic Purine Nucleoside Analogues	Johanna Wachtmeister; Bjorn Classon; Bertil Samuelsson; Ingemar Kvarnström
409-411	Synthesis of 3′-Amino-3′-deoxyadenosine Derivatives as Potential Drugs for the Treatment of Malaria	Johanna Soenens; Guido François; Elfride Van den Eeckhout; Piet Herdewijn
413-416	Stereocontrolled Synthesis of Pyridazine, Pyrazine, and Triazine 2′-DEOXY-β-Nucleosides by Means of Intramolecular Glycosylation	Hideyuki Sugimura; Miho Motegi; Keiko Sujino
417-420	Stereoselective Synthesis of 1′-C-Branched Uracil Nucleosides from Uridine	Kazuhiro Haraguchi; Yoshiharu Itoh; Hiromichi Tanaka; Tadashi Miyasaka
421-425	Alternate Approaches to the Synthesis of 2′-O-Me Nucleosides	Leonid Beigelman; Alexander Karpeisky; Jasenka Matulic-Adamic; Nassim Usman
427-429	Synthesis of (2′S)-1-(2-C-Azidomethyl-2-deoxy and 2-C-Cyanomethyl-2-deoxy-β-D-arabinofuranosyl)cytosines	Yuichi Yoshimura; Hiroshi Satoh; Shinji Sakata; Noriyuki Ashida; Shuichi Miyazaki; Akira Matsud
431-434	Resolution of (±)– Cytallene — A Highly Active Anti-HIV Agent with Axial Dissymmetry	Bryan Colin Nicholas Morgan Jones; Claire Simons; Hisao Nishimura; Jiri Zemlicka
435-437	Synthesis, Solution Conformation and Biological properties of 2′,3′-Dideoxy-3′-fluoro-D-erythro-pentofuranosides of 2-Thiouracil and 2-Thiothymine	N. E. Poopeiko; J. Poznanski; A. Drabikowska; J. Balzarini; E. De Clercq; I. A. Mikhailopulo; D. Shugar; T. Kulikowski
439-447	Rational Approaches to the Design of Mechanism-Based Inhibitors of S-Adenosylhomocysteine Hydrolase	Chong-Sheng Yuan; Siming Liu; Stanislaw F. Wnuk; Moms J. Robins; Ronald T. Borchardt
449-453	Platelet Aggregation Inhibitory Activity of Selective A₂ Adenosine Receptor Agonists	Gloria Cristalli; Emidio Camaioni; Sauro Vittori; Rosaria Volpini
455-458	Analogues of Azepinomycin: Inhibitors of Guanase	Anila Bhan; Ramachandra S. Hosmane
459	From Pro-nucleotides to Pro-oligonucleotides	Jean-Louis Imbach; Gilles Gosselin; Bernard Rayner
461-471	2′-C-Cyano-2′-deoxy-1-β-D-arabinofuranosylcytosine (CNDAC): A Mechanism-Based DNA-Strand-Breaking Antitumor Nucleoside¹	Akira Matsuda; Atsushi Azuma
473-476	Ligand Binding Properties of Bovine Liver Adenosine Kinase	Hélène Pélicano; Gilles Divita; Abdelaziz Elalaoui; Tayeb Daiboun; Manijeh Shafiee; Georges Maury; Roger S. Goody; Jean-Louis Imbach
477-480	Benzimidazoles in the Reaction of Enzymatic Transglycosylation	Igor A. Mikhailopulo; Zygmunt Kazimierczuk; Anatoli I. Zinchenko; Vladimir N. Barai; Valeria V. Romanova; Ludmilla A. Eroshevskaya
481-484	Synthesis and Properties of Some 2′-O-d-Ribofuranosyl-nucleosides	Sergey N. Mikhailov; Andre De Bruyn; Piet Herdewijn
485-493	Ribonucleotide Reductase Targets for Chemotherapy; Mechanistic Aspects and Biologically Active Agents	Morris J. Robins; Mirna C. Samano; Vicente Samano
495-499	5′-Substituted 2′-Deoxycytidines as Non-Substrate Inhibitors of Human Deoxycytidine Kinase	K. Krawiec; B. Kierdaszuk; D. Shugar
501-505	5-Halo-6-alkoxy-5,6-dihydro-pyrimidine Nucleosides: Antiviral Nucleosides or Nucleoside Prodrugs?	Leonard. I. Wiebe; Edward. E. Knaus; A. Majid Cheraghali; Rakesh Kumar; Kevin W. Morin; L. Wang
507-510	Substrate Specificities of Mitochondrial Thymidine Kinase and Cytosolic Deoxycytidine Kinase Against 5-Aryl Substituted Pyrimidine-2′-deoxyribose Analogues	Staffan Eriksson; Jianghai Wang; Salo Gronowitz; Nils Gunnar Johansson
511-515	Yet Another Mechanism of HIV Reverse Transcriptase Inhibition?	Jean M. J. Tronchet; Martina Zséaly; Olivier Lassout; Martin Grigorov; Annie Grouiller
517-520	Substrate/Inhibitor Properties of Tumour Purine Nucleoside Phosphorylase	A. Bzowska; L. Pogosjan; A. V. Ananiev; E. Kulikowska; D. Shugar
521-523	Synthesis and Antiviral Activity of 1,2-Carbonucleosides	L. Santana; M. Teijeira; E. Uriarte; J. Balzarini; E. De Clercq
525-528	Synthesis and Antiviral Activities of Some New 5-Heteroaromatic Substituted Derivatives of 2′-Deoxyuridine	J. Liu; A. Van Aerschot; I. Luyten; P. Wigerinck; C. Pannecouque; J. Balzarini; E. De Clercq; P. Herdewijn

Volume 14, Issue 3-5 (1995)

529-532	Synthesis and Biological Activities of Sugar-Modified 2-(p-n-Butylanilino)-2′-deoxyadenosine Analogues	Toyofumi Yamaguchi; Kunie Sato; Mineo Saneyoshi
533-536	Stereospecific Synthesis and Anti-HIV Activity of (Z)2′- and (E)3′-Deoxy-2′(3′)-C-(chloromethylene) Pyrimidine Nucleosides	Elena N. Kalinichenko; Elena B. Rubinova; Evgueny V. Borisov; Jan Balzarini; Erik De Clercq; Igor A. Mikhailopulo
537-539	Strategically Functionalized Adenosines: Agonists for Adenosine Receptors	Vasu Nair; Steven A. Adah; Seung B. Ha
541-544	Synthesis and Antiviral Evaluation of 3′-Substituted Thymidine Analogues Derived from 3′-Amino-3′-deoxythymidine	C. Pannecouque; K. Van Poppel; J. Balzarini; P. Claes; E. De Clercq; P. Herdewijn
545-547	The Synthesis and Antiviral Activity of Some New S-Adenosyl-L-homocysteine Derivatives and Their Nucleoside Precursors	Pawel Serafinowski; Erwin Dorland; Jan Balzarini; Erik De Clercq
549-550	Synthesis and Antiviral Evaluation of 3′-Deoxy-β-L-erythro-pentofuranosyl Nucleosides of the Five Naturally Occurring Nucleic Acid Bases	C. Mathé; G. Gosselin; M. -C. Bergogne; A. -M. Aubertin; G. Obert; A. Kirn; J. -L. Imbach
551-554	Synthesis and Antiviral Activity of 2 and 3-Substituted Imidazo[1,2-a]pyrimidine	A. Gueiffier; Y. Blache; J. P. Chapat; A. Elhakmaoui; E. M. Essassi; G. Andrei; R. Snoeck; E. De Clercq; O. Chavignon; J. C. Teulade; F. Fauvelle
555-558	Synthesis and Biological Activity of Sugar-Fluorinated 2′,3′-dideoxy-4′-thioribofuranosyl Nucleosides	Victor E. Marquez; Lak S. Jeong; Marc C. Nicklaus; Cliff George
559-562	Combination of Azidothymidine (AZT) and (E)-5-(2-Bromovinyl)-2′-deoxyuridine (BVDU) Inhibits the Replication of Herpes Simplex Virus Type 1 (HSV-1) and Type 2 (HSV-2) and Varicella Zoster Virus (VZV) Strains That Are Deficient in the Expression of the Viral Thymidine Kinase (tk)	G. Andrei; R. Snoeck; J. Balzarini; E. De Clercq
563-565	New Prodrugs of 9-(2-Phosphonomethoxyethyl)adenine [PMEA]: Synthesis and Stability Studies	S. Benzaria; G. Gosselin; H. Pelicano; G. Maury; A. -M. Aubertin; G. Obert; A. Kirn; J. -L. Imbach
567-570	Antiviral Activity of Selected Nucleoside Analogues Against Human Herpes Virus Type 6	D. Reymen; L. Naesens; J. Balzarini; A. Holy; E. De Clercq
571-574	Anti-herpes Activities of Isonucleoside Analogues with Variable Bases at the 2′ Position	T. Kira; A. Kakefuda; S. Shuto; A. Matsuda; M. Baba; S. Shigeta
575-583	Hept Derivatives: 6-Benzyl-1-ethoxymethyl-5-isopropyluracil (MKC-442)	Masanori Baba; Hlromichi Tanaka; Tadashi Miyasaka; Satoshi Yuasa; Masaru Ubasawa; Richard T. Walker; Erik De Clercq
585-594	TSAO Derivatives: Highly Specific Inhibitors of Human Immunodeficiency Virus Type-1 (HIV-1) Replication	Maria J. Camarasa; Maria J. Péarez-Péarez; Sonsoles Velázquez; Ana San-Féalix; Rosa Alvarez; Simon Ingate; Maria Luisa Jimeno; Anna Karlsson; Erik De Clercq; Jan Balzarini
595-598	Synthesis and Anti-HIV-1 Activity of 4- and 5-Substituted 1,2,3-Triazole-TSAO Derivatives	Ana San-Féalix; Rosa Alvarez; Sonsoles Veláazquez; Erik De Clercq; Jan Balzarini; María José Camarasa
599-602	Evidence for the Involvement of the Small Subunit of HIV-1 Reverse Transcriptase (RT) in the TSAO-Resistance	Heidi Jonckheere; Jean-Marc Taymans; Jan Balzarini; Sonsoles Veláazquez; Maria Jose Camarasa; Jan Desmyter; Erik De Clercq; Jozef Annéa
603-606	Inhibitory Effects of 1-Deazaadenosine Analogues on HIV Replication and Adenosine Deaminase	Sauro Vittori; Rosaria Volpini; Emidio Camaioni; Giorgio Palúg; Giorgio Cristalli
607-610	Acyclic Nucleotides Related to Clitocine: Synthesis and Anti-HIV Activity	P. Franchetti; L. Cappellacci; G. Abu Sheikha; M. Grifantini; A. G. Loi; A. De Montis; M. G. Spiga; P. La Colla
611-617	2′-and/or 3Y-Deoxy-β-L-pentofuranosyl Nucleoside Derivatives: Stereospecific Synthesis and Antiviral Activities	Gilles Gosselin; Christophe Mathé; Marie-Christine Bergogne; Anne-Marie Aubertin; Andre Kirn; Jean-Pierre Sommadossi; Raymond Schinazi; Jean-Louis Imbach
619-625	Studies of the Pharmacokinetics and Toxicology of 2′,3′-Dideoxy-β-L-5-fluorocytidine (β-L-FddC) and 2′,3′-Dideoxy-β-L-cytidine (β-L-ddC) In Vivo; and Synthesis and Antiviral Evaluations of 2′,3′-Dideoxy-β-L-5-azacytidine	Tai-Shun Lin; Xin Guo; Mei-Zhen Luo; Mao-Chin Liu; Yong-Lian Zhu; Ginger E. Dutschman; S. Balakrishna Pai; Mao-Mi Li; Yung-Chi Cheng
627-635	Structure-Activity Relationships Among a New Class of Antiviral Heterosubstituted 2′,3′-Dideoxynucleoside Analogues	Tarek S. Mansour; Haolun Jin; Wei Wang; Dilip M. Dixit; Colleen A. Evans; H. L. Allan Tse; Bernard Belleau; John W. Gillard; Elizabeth Hooker; Claire Ashman; Nick Cammack; Horacio Salomon; Antonietta R. Belmonte; Mark A. Wainberg
637-640	Synthesis, Antitumor Activity and Crystallographic Studies of Analogues of Tiazofurin	L. Cappellacci; P. Franchetti; M. Grifantini; L. Messini; G. Abu Sheikha; G. Nocentini; R. Moraca; B. M. Goldstein
641-644	Modulators of Nucleotide Metabolism Inhibit HIV Replication in Lymphoid Cells and Affect Its Inhibition by Dideoxynucleosides	Ranga V. Srinivas; Yi-Fei Gong; Anna Becher; Arnold Fridland
645-647	Synthesis and Antitumor Properties of Some Neutral Triesters of 5-Fluoro-2′-deoxyuridine-5′-monophosphate and 3′,5′-Cyclic Monophosphate	J. -L. Girardet; G. Gosselin; C. Périgaud; J. Balzarini; E. De Clercq; J. -L. Imbach
649-652	Induction of Erythroid Differentiation of Human Leukemia K562 Cells by the Acyclic Nucleoside Phosphonate 9-(2-Phosphonylmethoxyethyl)adenine (PMEA)	S. Hatse; J. Balzarini; E. De Clercq
653-656	Synthesis and Antitumour Properties of 2-Thio-5-chloro-nucleosides	K. Felczak; M. Bretner; M. Balińska; J. M. Dzik; W. Rode; T. Kulikowski
657-660	Synthesis and Biological Activity of 5-Fluoro-2-thiocytosine Nucleosides	M. Bretner; M. Balinska; K. Krawiec; B. Kierdaszuk; D. Shugar; T. Kulikowski
661-664	Three-Dimensional Cell Cultures as a Model System to Evaluate the Biological Activity of Gemcitabine (2′, 2′-Difluoro-2′deoxycytidine)	Godefridus J. Peters; Evelien Smitskamp-Wilms; Gijsbert Veerman; Paulo E. Pizao; Veronique W. T. Ruiz van Haperen; Herbert M. Pinedo
665-669	Studies on 6-Mercaptopurine Cytotoxicity in Molt F4 Human Malignant T-Lymphoblasts	E. H. Stet; R. A. De Abreu; J. P. M. Böukkerink; J. M. F. Trijbels
671-674	Synthesis and Broad-Spectrum Antiviral Activity in Mice of Certain Alkyl, Alkenyl and Ribofuranosyl Derivatives of 7-Deazaguanine	G. R. Revankar; T. S. Rao; K. Ramasamy; D. F. Smee

Volume 14, Issue 3-5 (1995)

675-686	The Synthesis and Biological Activity of Certain 4′-Thionucleosides	John A. Secrist III; William B. Parker; Kamal N. Tiwari; Lea Messini; Sue C. Shaddix; Lucy M. Rose; L. Lee Bennett Jr; John A. Montgomery
689-692	An Improved Synthesis of N⁶-(6-Aminohexyl)FAD	Ashty Saleh; Frans Compernolle; Gerard Janssen
693-694	A Convenient Method for the Synthesis of ATP and Ap₄A	Koichiro Fukuoka; Fuminori Suda; Masahide Ishikawa; Tsujiaki Hata
695-702	Acyclic Nucleotide Analogues and Related Compounds	Antonín Holý; Hana Dvořáková
703-706	Studies on Aryl H-Phosphonates. Synthesis of Nucleoside N-Alkylphosphonamidates	Anna Sobkowska; Michał Sobkowski; Jacek Stawi�ski; Adam Kraszewski
707-710	Phosphonates Derivatives of 2′,3′-Dideoxy-2′,3′-didehydro-pentopyranosyl Nucleosides	María-Jesús Péarez-Péarez; Bogdan Doboszewski; Erik De Clercq; P. Herdewijn
711-714	Conversion of Nucleoside H-Phosphonate Monoesters to the Corresponding H-Phosphonothioates. ³¹P NMR Studies	Jacek Stawiński; Rula Zain
715-716	2-Cyanoethyl H-Phosphonate. A Reagent for the Mild Preparation of Nucleoside H-Phosphonate Monoesters	Tomas Szabóa; Helena Almer; Roger Ströumberg; Jacek Stawinski
717-721	Synthesis and Properties of P¹, P²-, P¹, P³- and P¹, P⁴-Dinucleoside Di-, Tri- and Tetraphosphate mRNA 5′-Cap Analogues	J. Steogon; piński; M. Bretner; M. Jankowska; K. Felczak; R. Stolarski; Z. Wieczorek; A-L. Caipostalcode; R. E. Rhoads; A. Temeriusz; D. Haber; E. Darzynkiewicz
723-726	Synthesis of Four Stereoisomers of Carbocyclic 5′-NOR D4A and Evaluation of Their Triphosphates as Substrates for DNA Polymerases	Natalia Dyatkina; Dniitry Semizarov; Lyubov Victorova; Alexander Krayevsky; Fritz Theil; Martin von Janta-Lipinski
727-729	Synthesis of Dioxolane Analogues of Dideoxynucleotides and Their Substrate Properties in DNA Synthesis Reactions	E. V. Efimtseva; S. N. Mikhailov; L. S. Victorova; T. A. Rosovskaya; R. Sh. Beabealashvilli
731-734	Methylene and Halomethylene Analogues of Diadenosine 5′,5″-P¹, P³-Triphosphate (ApppA) as Substrates or Inhibitors of ApppA-Degrading Enzymes	Andrzej Guranowski; Elżibieta Starzyńska; Lidia Gzik; Steve P. Langston; Paul Brown; G. Michael Blackburn
735-738	Does Interaction of dNTP Glycone with an Active Center of Reverse Transcriptases Takes Place? A Model for a Binding Site	Alexander A. Krayevsky; Natalya B. Dyatkina; Marina K. Kukhanova
739-742	Qualitative and Quantitative Analysis of Cyclic Nucleotides and Related Enzymes by Static and Dynamic Fast Atom Bombardment Mass Spectrometry	James I. Langridge; A. Gareth Brenton; Terry J. Walton; Frank M. Harris; Russell P. Newton
743-747	Cytidine 3′,5′-Cyclic Monophosphate: A Third Cyclic Nucleotide Secondary Messenger?	Russell P. Newton
749-751	Novel Open-Chain Nucleotides Imitating 2′,3′-Dideoxy-2′,3′-Didehydronucleotides: Synthesis and Substrate Properties Toward DNA Polymerases	E. A. Shirokova; N. B. Tarussova; A. V. Shipitsin; D. G. Semizarov; M. Hieber; A. A. Krayevsky
753-757	Investigation of a Proposed Mechanism for Genotoxic Effects Induced by 2-Hydroxyalkylating Agents. Kinetics of Intramolecular Transesterification in Dithymidine 2-Hydroxyethyl-and 2-Hydroxypropyl Phosphate	E. Pettersson; E. Bergmark; U. Rannug; L. Ehrenberg; R. Ströumberg
759-762	Homo Dinucleoside-α-hydroxyphosphonate Diesters as Prodrugs of the Antiviral Nucleoside Analogues 2′,3′-Dideoxythymidine and 3′-Azido-2′,3′-dideoxythymidine	Chris Meier; Lothar Habel; Wolfgang Laux; Erik De Clercq; Jan Balzarini
763-766	Synthesis, Decomposition Pathways and “In Vitro” Evaluation of Bioreversible Phosphotriesters of Azt	Isabelle Lefebvre; Alain Pompon; Christian Périgaud; Jean-Luc Girardet; Gilles Gosselin; Anné-Marie Aubertin; Andre Kirn; Jean-Louis Imbach
767-770	In vivo Antiretroviral Efficacy of Oral bis(POM)-PMEA, the bis(Pivaloyloxymethyl)prodrug of 9-(2-Phosphonylmethoxyethyl) adenine (PMEA)	L. Naesens; J. Neyts; J. Balzarini; N. Bischofberger; E. De Clercq
771-775	Synthesis and Properties of mRNA 5′-Cap Analogues with 7-Methylguanine Replaced by Benzimidazole or 3-Methylbenzimidazole	L. Chlebicka; Z. Wieczorek; R. Stolarski; J. Stepinski; E. Darzynkiewicz; D. Shugar
777-781	Biological Activity of Some Dialkyl α-Anilinobenzylphosphonates and Their Palladium(II) Complexes	Lj. Tušek-Božić; M. Ćurić; J. Balzarini; E. De Clercq
783-787	Synthesis of Nucleotide Lipophilic Prodrugs Containing Two Inhibitors Targeted Against Different Phases of the HIV Replication Cycle	D. Bonnaffé; B. Dupraz; J. Ughetto-Monfrin; A. Namane; T. Huynh Dinh
789-791	bis(S-Acyl-2-thioethyl)esters of 2′,3′-Dideoxyadenosine 5′-Monophosphate Are Potent Anti-HIV Agents in Cell Culture	C. Périgaud; G. Gosselin; S. Benzaria; J. -L. Girardet; G. Maury; H. Pélicano; A. -M. Aubertin; A. Kirn; J. -L. Imbach
795-798	Synthesis of Base-Modified Oligonucleotides Containing 6- and 7-Aryl Lumazines	Yuris Maurinsh; Wolfgang Pfleiderer
799-801	Synthesis of 2′-C-Difluoromethyl Substituted Nucleoside Analogs as Ribonucleoside Replacements in Hammerhead Ribozymes	Martin Dunkel; Vivian Reither; Susanne Ebel-Will; János Ludwig
803-804	Synthesis of Protected 3′,5′-Di-2′-Deoxythymidine-(α-hydroxy-2-nitrobenzyl)-phosphonate Diesters as Dimer Building Blocks for Oligonucleotides	Chris Meier; Ralf Mauritz
805-808	Chemical and Enzymatic Synthesis of 2′-Deoxy-iso-inosine and Its Incorporation into DNA	Jean-Jacques Beaussire; Sylvie Pochet
809-812	The Application of H-Phosphonate Chemistry in the HELP Synthesis of Oligonucleotides	S. Zaramella; G. M. Bonora
813-816	Peptide Analogues of DNA Consisting of l-α-Amino-γ-thymine Butyric Acid and l-Valine Subunits	G. Ceulemans; K. Khan; A. Van Schepdael; P. Herdewijn

Volume 14, Issue 3-5 (1995)

817-820	Phosphoramidites of (Rp) and (Sp)-Configurated Adenosine Methylphosphonate Dimers	Markus Schweitzer; Wendelin Samstag; Joachim W. Engels
821-824	Preparation of Oligonucleotides Containing Non-natural Base Analogues	Ramon Eritja; Montse Acedo; Anna Aviñó; Carme Fà
825-828	Phosphitylation of Primary Carboxamides. Synthesis of Peptide-Oligonucleotide Conjugates with Acylphosphoramidate Linkages	Anna Grandas; Jordi Robles; Enrique Pedroso
829-832	A Rapid Method for the Functionalisation of Polymer Supports for Solid Phase Oligonucleotide Synthesis	K. C. Gupta; Pradeep Kumar; Dimpan Bhatia; A. K. Sharma
833-837	A General Approach for the Hydroxy Group Functionalization of Synthetic Oligonucleotides	Andrei Guzaev; Jan Hovinen; Alex Azhayev; Harri Lönnberg
839-842	Studies on Reactions of Nucleoside H-Phosphonates with Bifunctional Reagents. Part III. Further Studies on Transesterification of Nucleoside H-Phosphonate Diesters with Amino Alcohols	Michal Sobkowski; Jacek Stawińki; Anna Sobkowska; Adam Kraszewski
843-846	How to Synthesize A tRNA?	W. Pfleiderer; K. P. Stengele; F. Bergmann; M. Resmini; C. Henke
847-850	Synthesis of Circular Oligodeoxynucleotide Conjugates VIA Transient Abasic Sites	D. Péoc'h; J. -L. Imbach; B. Rayner
851-853	Synthesis of Oligoarabinonucleotides Using H-Phosphonates	Eriks Rozners; Roger Strömberg; Erika Bizdena
855-857	Synthesis of RNA Fragments Using the H-Phosphonate Method and 2′-(2′-Chlorobenzoyl) Protection	Eriks Rozners; Roger Strömberg; Erika Bizdena
859-862	Synthesis of a New Hydroxyamino Linked Thymidine Dimer via a Radical C-C Bond Formation	Yogesh S. Sanghvi; P. Dan Cook
863-866	2′-Deoxyisoinosine: Synthesis of a Highly Fluorescent Nucleoside and Its Incorporation into Oligonucleotides	Frank Seela; Yaoming Chen
867-870	Aldehyde Functions in Synthetic Oligonucleotides	M. Dechamps; E. Sonveaux
871-874	Solid Phase Synthesis of 5′-Methylenephosphonate DNA	Tomas Szabó; Annika Kers; Jacek Stawinski
875-878	o-Chlorobenzoyl Protected Nucleoside Succinates for Functionalization of the Solid Support Used in Oligoribonucleotide Synthesis	S. Sigurdsson; E. Rozners; E. Westman; E. Bizdena; R. Strömberg
879-881	Chemical Synthesis of RNA-Fragment Analogues That Have Phosphorothioate Linkages of Identical Configuration	Helena Almer; Jacek Stawinski; Roger Strömberg
883-887	RNA-Synthesis Using the H-Phosphonate Approach and an Improved Protecting Group Strategy	Erik Westman; Susannah Sigurdsson; Helena Almer; Mats Thelin; Jacek Stawinski; Eriks Rozners; Roger Strömberg
889-893	Oligodeoxyribonucleotides Covalently Linked via Nucleic Bases with 3′-5′ and 5′-5′ Polarities	Ulysse Asseline; N. T. Thuong
895-899	Synthesis of 6-Aza- & 6-Methyl-pyrimidine Ribonucleoside Phosphoramidites and Their Incorporation in Hammerhead Ribozymes	Leonid Beigelman; Alexander Karpeisky; Nassim Usman
901-905	Synthesis of 5′-C-Methyl-D-allo- & L-Talo-ribonucleoside 3′-O-Phosphoramidites & Their Incorporation into Hammerhead Ribozymes	Leonid Beigelman; Alexander Karpeisky; Nassim Usman
907-910	New Structural Motifs for Hammerhead Ribozymes. Catalytic Activity of Abasic Nucleotide Substituted Ribozymes	Leonid Beigelman; Alexander Karpeisky; Jasenka Matulic-Adamic; Carolyn Gonzalez; Nassim Usman
911-915	Improvements to the Chemical Synthesis of Biologically Active RNA Using 2′-O-Fpmp Chemistry	M. Vaman Rao; K. Macfarlane
917-920	An Improved Method for Large Scale Synthesis of Oligonucleotides Applying the NPE/NPEOC-Strategy	J. Weiler; W. Pfleiderer
921-924	3′-C-Hydroxymethylthymidine: Synthesis and Incorporation into Oligodeoxynucleotide Analogues	Pia Nøncgaard Jørgensen; Margit L. Svendsen; Claus Nielsen; Jesper Wengel
925-928	Synthesis and Characterization of Short Oligonucleotide Segments Containing Nonnatural Internucleoside Amine- and Amide Linkages	Gorm Vang Petersen; Jesper Wengel
929-933	Preparation of Oligodeoxynucleotides Containing 6-Methylthiopurine Residues by Chemical Synthesis or Specific Methylation	Yao-Zhong Xu; Qinguo Zheng; Peter F. Swann
935-937	Synthesis of the 3′-Derivatives of Phosphorothioate Oligonucleotide Analogues	N. V. Amirkhanov; V. F. Zarytova
939-942	An Improved Post-Synthetic Substitution Approach for Synthesis of Oligodeoxynucleotides Containing Labile 4-Substituted Thymines	Qinguo Zheng; Yao-Zhong Xu; Peter F. Swann
943-946	Electrochemically Directed Copolymerization of Pyrrole and Oligonucleotides	A. Roget; T. Livache; J. Marchand; R. Teoule
947-950	Synthesis and Photochemical Conversion of Oligonucleotides Containing 2-Chloro-2′-Deoxyadenosine	Natalya Ramzaeva; Helmut Rosemeyer; Frank Seela

Volume 14, Issue 3-5 (1995)

951-955	Approaches to Enhance the Binding Affinity and Nuclease Stability of Triplex Forming Oligonucleotides	K. Jayaraman; R. H. Durland; T. S. Rao; G. R. Revankar; V. Bodepudi; N. Chaudhary; J. Guy-Caffey
957-960	Hoogsteen-Duplex DNA: Synthesis and Base Pairing of Oligodeoxynucleotides Containing 1-Deaza-2′-deoxyadenosine	Frank Seela; Thomas Wenzel; Harald Debelak
961-965	Synthesis and Properties of New Fluorescein-Labeled Oligonucleotides	Thomas Maier; Wolfgang Pfleiderer
967-968	Diamino-Antraquinone: A New Intercalating Agent. Synthesis and Linking to Oligodeoxynucleotide	Lászió Puskás; József Czombos; Sándor Bottka
969-973	Oligonucleotide Conjugates: Alteration of the Pharmacokinetic Properties of Antisense Agents	Muthiah Manoharan; Kathleen L. Tivel; Laura K. Andrade; V. Mohan; Thomas P. Condon; C. Frank Bennett; P. Dan Cook
975-977	Triple Helix Forming α-Oligonucleotides Containing 5-Methylcytosine and/or 5-Bromouracil	Francęois Morvan; Carole Chaix; Axel Zeissler; Bernard Rayner; Jean-Louis Imbach
979-982	Postsynthetic Transformations of Oligodeoxynucleotides Originated at 6-Methylthio-purine Site	Artur Burdzy; Bohdan Skalski; Ewa Biał; Andrzej Kowalewski; Stefan Paszyc; Rys2ard W. Adamiak
983-984	The Solution NMR Structure of 2′-O-Methyl CGCGCG RNA Duplex	Mariusz Popenda; Jan Milecki; Ewa Biała; Ryszard W. Adamiak
985-990	Enzymatic Synthesis of Stereoregular (All Rp) Oligonucleotide Phosphorothioate and Its Properties	Jinyan Tang; Allysen Roskey; Ying Li; Sudhir Agrawal
991-995	Destabilization of DNA Guanine Quadruplex Structure by Foldback Triplex-Forming Oligodeoxynucleotides	Ekambar R. Kandimalla; Sudhir Agrawal
997-1000	Phosphate-Modified Nucleotides: Conversions in Human Serum	Marina K. Kukhanova; Elena V. Kuznetsova; Andrey A. Arzumanov; Alexander A. Krayevsky
1001-1003	Nitroindoles as Universal Bases	D. Loakes; F. Hill; S. Linde; D. M. Brown
1005-1008	Synthesis and Properties of Oligonucleotide (2-Aminoethyl)Phosphonates	Alan F. Cook; Reza Fathi; Qing Huang; George Coppola; William Delaney; Jia-Lin Syi
1009-1013	Novel Approaches to the Synthesis and Analysis of Branched RNA	K. Ganeshan; T. Tadey; K. Nam; R. Braich; W. C. Purdy; J. D. Boeke; M. J. Damha
1015-1018	Optimization of Antisense Chimeric Oligonucleotides Containing α- and β-Anomeric Deoxynucleotides	F. Debart; G. Tosquellas; B. Rayner; J. -L. Imbach
1019-1022	Autoligation of Oligonucleotides via Nucleophilic Substitution Reaction	Sergei M. Gryaznov
1023-1026	Hybridization Properties of the 5-Methyl-isocytidine/isoguanosine Base Pair in Synthetic Oligodeoxynucleotides	Thomas Horn; Chu-An Chang; Mark L. Collins
1027-1030	4′-Thio-β-D-oligoribonucleotides: Nuclease Resistance and Hydrogen Bonding Properties	C. Leydier; L. Bellon; J. -L. Barascut; J. -L. Imbach
1031-1035	Synthesis and Properties of 2′-O-Methylribonucleotide Methylphosphonate Containing Chimeric Oligonucleotides	Ekambar R. Kandimalla; Jamal Temsamani; Sudhir Agrawal
1037-1040	The N¹-(3′-Deoxythymidin-3′-yl)-N²-cyano-N³-(5′-deoxythymidin-5′-yl) Guanidine Dimeric Building Block in Automated DNA Synthesis and Mass Spectrometric Analysis of Its Integrity	C. Pannecouque; J. Rozenski; B. Devreese; J. Van Beeumen; A. Van Aerschot; P. Herdewijn
1041-1045	Xylose-DNA: Sequence-Dependent Duplex Stability as Function of Backbone Configuration	Helmut Rosemeyer; Frank Seela
1047-1048	Template Activity of Oligoribonucleotides Synthesized by the Phosphoramidite Method Using 2′-O-Tetrahydrofuranyl and 2′-O-Tetrahydropyranyl Protecting Groups	E. Stankevich; V. Kumpins; N. Licis; J. Klovins; V. Berzin
1049-1052	Synthesis and Antibody Mediated Detection of 2,4-Dinitrophenyl (DNP) Labelled Oligonucleotides	A. Davison; G. Duckworth; M. V. Rao; J. McClean; J. Grzybowski; P. Potier; T. Brown; H. Cubie
1053-1056	In Search of Acyclic Analogues as Universal Nucleosides in Degenerate Probes	A. Van Aerschot; C. Hendrix; G. Schepers; N. Pillet; P. Herdewijn
1057-1059	To Wobble or Not to Wobble: Modified Bases Incorporated into DNA	L. Van Meervelt; M. H. Moore; P. K. T. Lin; D. M. Brown
1061-1064	Synthesis and Biophysical Properties of Oligothymidylates Containing Alkoxyphosphoramidate Internucleoside Linkages	Suzanne Peyrottes; Jean-Jacques Vasseur; Jean-Louis Imbach; Bernard Rayner
1065-1068	A New Approach to Potentiate Site-Specific Hybridization: A set of Hydrophobic Heterobifunctional Short Oligodeoxyribonucleotides	D. Pyshnyi; I. Pyshnaya; D. Sergeev; P. Vorobjev; S. Lokhov; E. Ivanova; V. Zarytova
1069-1072	New Photoreactive mRNA Analogues for the Affinity Labeling of Ribosomes	A. G. Venyaminova; M. N. Repkova; T. M. Ivanova; M. I. Dobrikov; K. N. Bulygin; D. M. Graifer; G. G. Karpova; V. F. Zarytova
1073-1076	Targeting RNA for Degradation with a (2′, 5′)-Oligoadenylate Antisense Chimera	Paul F. Torrence; Wei Xiao; Guiying Li; Shahrzad Khamnei; Krystyna Lesiak; Avudaiappan Maran; Ratan Maitra; Aseem Kumar; Beihua Dong; Bryan R. G. Williams; Robert H. Silverman
1077-1081	Enhanced Cellular Uptake of G-Rich Oligonucleotides	A. Peyman; A. Ryte; M. Helsberg; G. Kretzschmar; M. Mag; E. Uhlmann

Volume 14, Issue 3-5 (1995)

1083-1085	Use of Bioreversible Phosphate Protecting Groups for the Intracellular Delivery of Antisense Oligodeoxyribonucleotides	Isabelle Barber; Bernard Rayner; Jean-Louis Imbach
1087-1090	Synthesis, Biophysical and Biological Evaluations of Novel Antisense Oligonucleosides Containing Dephosphono-Internucleosidic Linkages	Yogesh S. Sanghvi; Laurent Bellon; Francęois Morvan; Tomonori Hoshiko; Eric Swayze; Lendell Cummins; Susan Freier; Nicholas Dean; Brett Monia; Richard H. Griffey; P. Dan Cook
1091-1092	5-Methylcytosine and 5-Azacytosine Containing 25Mer Duplexes: Synthesis and Investigation of their Interaction with HeLa Nuclear Protein Extracts	Yacoob Padia; Mario Ariatti; Peter A. Jones
1093-1096	Synthesis and Expression of Some Genes for Human Cytokines	Kiara R. Birikh; Ekaterina N. Lebedenko; Yuri A. Berlin
1097-1100	Evaluation of Oligonucleotides with Novel Modifications	Erik Larsen; Krzysztof Danel; Abdel-Aleem H. Abdel-Aleem; Poul Niclsen; Jesper Wengel; Erik B. Pedersen
1101-1104	Synthesis of Trimeric Cordycepin-Vitamin Conjugates as Improved Antiviral Agents	Marita Wasner; Wolfgang Pfleiderer
1105-1108	Synthesis and Use of (2′,5′)Oligoadenylate Trimers Modified at the 2′-Terminus in Kidney Transplantation in Rabbits and Monkeys	I. A. Mikhailopulo; Z. Yu. Tkachuk; E. A. Baran; L. V. Tkachuk; A. V. Koslov; I. I. Slukvin; E. I. Kvasyuk; T. I. Kulak; G. Kh. Matsuka
1109-1116	Structure-Activity Study of Oligodeoxynucleotides Which Inhibit Thrombin	Steven H. Krawczyk; Norbert Bischofberger; Linda C. Griffin; Veronica S. Law; Regan G. Shea; S. Swaminathan
1117-1127	Novel Guanosine Quartet Structure Binds to the HIV Envelope and Inhibits Envelope Mediated Cell Fusion	David J. Ecker; Jacqueline R. Wyatt; Timothy Vickers
1129-1132	Synthesis and Applications of Oligoribonucleotides Containing N⁴-Methylcytidine	Jane A. Grasby; Mohinder Singh; Jonathan Karn; Michael J. Gait
1133-1144	Synthetic Ribonucleotide Analogues for RNA Structure-Function Studies	Michael J. Gait; Jane A. Grasby; Jonathan Karn; Karin Mersmann; Clare E. Pritchard
1145-1148	Inhibition of Reverse Transcriptase-Mediated cDNA Synthesis by Antisense Oligonucleotides	Toshifumi Hatta; Kazuyuki Takai; Hiroshi Takaku
1149-1152	Properties and Anti-HIV Activity of Circular Sense and Antisense Oligonucleotides	H. Yamakawa; T. Ishibashi; H. Nakashima; N. Yamamoto; K. Takai; H. Takaku
1153-1156	Human Cytomegalovirus Stimulates Thymidylate Synthase in Human Embryonic Lung Cells: A Possible Target for Anti-HCMV Therapy?	J. Neyts; A. Verbiest; A. Meerbach; E. De Clercq

Volume 14, Issue 1-2 (1995)

a	Editorial board page for “Nucleosides, Nucleotides & Nucleic Acids”, Volume 14, Number 1-2
1-12	Incorporation of 2′-Deoxy-9-deazaguanosine and 2′-Deoxy-7-deaza-6-thioguanosine into G-Rich Oligodeoxyribonucleotides	T. Sudhakar Rao; Arthur F. Lewis; Theresa Schmaltz Hill; Ganapathi R. Revankar
13-22	Characterization of Nucleoside Phosphotransferase from Leishmania Tropica	Il-Shik Shin; Yusuke Wataya
23-37	Synthesis, Molecular and Crystal Structure of 3′-N-Alkylamino-3′-deoxythymidines and Some Biochemical Properties of Their Phosphorous Esters	Maxim V. Jasko; lvati I. Fedorov; Alexey M. Atrazhev; Diriiitry Yu. Mozzherin; Nicolay A. Novicov; Alexey V. Bochkarev; Gnliiia V. Gurskaya; Alexander A. Krayevsky
39-44	6-Deoxycarbovir: A Xanthine Oxidase Activated Prodrug of Carbovir	Robert Vince; Jay Brownell; Scott A. Beers
45-63	An Improved Synthesis of 1-(2-Deoxy-β-D-erythro-pentofuranosyl)quinazoline-2,4(3H)-dione and Its Incorporation Into G-Rich Triple Helix Forming Oligonucleotides	Birendra K. Bhattacharya; Mohan V. Chari; Ross H. Durland; Ganapathi R. Revankar
65-76	Synthesis of 2-Azido-1,N⁶-Etheno and 2-Azido Analogs of Deoxyadenosine as Nucleotide Photoaffinity Probes	Diane Flaherty; Preeti Balse; Ke Li; Bob M. Moore; Michael B. Doughty
77-89	Transglycosylation of β-D-RIbofuranosylindazoles	Jerzy Boryski
91-103	Synthesis and Substrate Properties of Thymidine 5′-Triphosphate Analogs with Large Hydrophobic Substituent Groups At α-P Atom	N. Dyatkina; A. Arzumanov; L. Victorova; M. Kukhanova; A. Krayevsky
105-116	Palladium-Mediated Coupling Reactions of an Aminosubstituted Heterocycle. Direct Synthesis of C-Nucleosides Related to Adenosine	Han-Cheng Zhang; Mohamed Brakta; G. Doyle Daves Jr.
117-127	Synthesis of an Uncharged cAMP-Analogue	G. Ceulemans; F. Vandendriessche; J. Rozenski; P. Herdewijn
129-142	Synthesis of 6-Substituted Purine N⁷-(2-Deoxy-β-D-Ribonucleosides) via Anion Glycosylation and Anomerization During the N⁷/N⁹-Glycosyl Transfer	Frank Seela; Holger Winter
143-165	RNA Modified Uridines VII: Chemical Synthesis and Initial Analysis of tRNA D-Loop Oligomers with Tandem Modified Uridines	Barbara Nawrot; Andrzej Malkiewicz; Wanda S. Smith; Hanna Sierzputowska-Gracz; Paul F. Agris
167-173	A Convenient and Efficient Method for the Synthesis of Nucleoside H-Phosphonates Using a Novel Phosphonylating Agent	Zai-Wan Yang; Zu-Sheng Xu; Nan-Zhen Shen; Zhi-Qiang Fang
175-183	The Evaluation OF 2′, 3′-Dideoxy-β-D-Erythro-Hex-2′-Enopyranosyl Nucleosides as Potential Antisense Constructs: Synthesis, Biophysical Properties and Enzymatic Stability of 2′-Deoxyadenosine-(3′–6′)-[1-(2′, 3′-Dideoxy-β-D-Erythro-Hex-2′-Enopyranosyl)thymine] Phosphate	Leslie W. Tari; Krishan L. Sadana; Anthony S. Secco
185-194	3′-C-Trifluoromethyl Ribonucleosides	Carl R. Johnson; Dilip R. Bhumralkar; Erik De Clercq
195-207	Synthesis of (±)-cis-1-[2-(Hydroxymethyl)-1, 3-Oxathiolan-5-yl]cytosine and Its (±)-trans Isomer	Jim J. Huang; Janet L. Rideout; Gary E. Martin
209-218	Synthesis of Pyrimidine 2′,3′-Dideoxy-2-Thionucleosides	Bhalchandra V. Joshi; Colin B. Reese; Chamakura V. N. S. Varaprasad
219-228	Introduction of an Immunochemical Label in a Cytidine Analogue	Chryslaine R. Tanty; Lilia López-Canovas; Adamari López Brauet; Marelys Rivero Paredes; David Higginson Clarke; Herman Vélez Castro; Ana Ma. Riverón Rojas; Arturo Macías Cabrera
229-241	Oligonucleotides and Nucleotide-Peptides. LV. Synthesis and Some Properties of Triesters of Hydroxy Aming Acids and Thymidilyl-(3′ → 5′)-Thymidine¹	B. Juodka; L. Bagdoniene; R. Plaipa
243-253	Preparation of Oligomeric 2′-Deoxy-5-Fluorouridylate of Defined Length and Backbone Composition: A Novel Pro-Drug form of the Potent Anti-Cancer Drug 2′-Deoxy-5-Fluorouridylate	William H. Gmeiner; Parag Sahasrabudhe; Richard T. Pon; Jacque Sonntag; Shashikumar Srinivasan; Patrick L. Iversen
255-273	An Efficient Method for the Isolation and Purification of Oligoribonucleotides	Brian Sproat; Francesco Colonna; Bashar Mullah; Dean Tsou; Alex Andrus; Arnold Hampel; Ravi Vinayak

Volume 13, Issue 10 (1994)

2035-2050	A New Synthesis of Some 4′-Thio-D-ribonucleosides and Preliminary Enzymatic Evaluation	C. Leydier; L. Bellon; J. -L. Barascut; J. Deydier; G. Maury; H. Pelicano; M. A. El Alaoui; J. -L. Imbach
2051-2058	Nucleocyclitols. Synthests of Ethanolamino-Purinyl Inositol Derivatives and Their Reaction With Thionyl Chloride	S. R. Leicach; M. E. Gelpi; R. A. Cadenas
2059-2069	Use of NPE-Protecting Groups for the Preparation of Oligonucleotides Without Using Nucleophiles During the Final Deprotection	A. M. Avino; R. Eritja
2071-2079	Novel Types of Bicyclonucleosides: Isoxazolidinofuranosylthymines	J. M. J. Tronchet; M. Zsely; N. Sultan
2081-2104	Reaction of 2-Deoxy-2-C-(3-bromoacetoxypropyl)-α-D-arabinofuranosides with Oligonucleotide¹	S. Mori; A. Katoh; H. Takenaka; H. Tanaka; H. Kaji; T. Samejima; O. Mitsunobu
2105-2111	Rapid, Stepwise Substitution of Fluorines In 5-Trifluoromethyl-2′-Deoxyuridine by Bisulfite	S. Takatori; A. Matsuda; J. -I. Yamashita; H. Hayatsu; Y. Wataya
2113-2124	Achiral Nucleotide Analogs: 5,5-Disubstituted Pyrimidines Related to Barbituric Acid	M. J. van Vliet; J. Visscher; A. W. Schwartz
2125-2134	Development of Suitable Linkage for Oligonucleotide Synthesis and Preliminary Hybridization Studies on Oligonucleotides Synthesized in Situ	A. Kumar
2135-2149	Synthesis, Base Pairing Properties and Nuclease Resistance of Oligothymidylate Analogs Containing Methoxyphosphoramidate Internucleoside Linkages	S. Peyrottes; J. J. Vasseur; J. L. Imbach; B. Rayner
2151-2168	O^5′,6-Methanocytidine — Synthesis, Conformational Properties and Deamination by Cytidine Deaminase	S. Megati; S. E. Ealick; F. N. M. Naguib; M. H. el Kouni; R. S. Klein; B. A. Otter
2169-2183	Sequence-Dependent Structural Variations of DNA Revealed by Chemical Ligation	N. G. Dolinnaya; I. N. Merenkova; Z. A. Shabarova
2185-2193	Synthesis and Structure Assignment of 1-(2-Acetoxyethoxy)methyl Derivatives of 5-Chloro-6-azauracil and 5-Bromo-6-azaisocytosine	L. -C. Hwang; D. -C. Wei; M. -C. Cheng; Y. Wang; C. -C. Tzeng
2195-2207	Structural Investigation of Model Deadenylated Oligonucleotide Phosphorothioate Analog of Isis 2105	V. T. Ravikumar; T. K. Wyrzykiewicz; V. Mohan; D. L. Cole
2209-2244	Preparation and Utility of 5-β-D-Ribofuranosyl-1H-tetrazole as a Key Synthon for C-Nucleoside Synthesis	J. Kobe; M. Prhavc; M. Hohnjec; L. B. Townsend
2245-2265	New Non Nucleosidic Phosphoramidites for the Solid Phase Multi-Labelling of Oligonucleotides: Comb- and Multifork-Like Structures	M. J. De Vos; A. Van Elsen; A. Bollen
2267-2281	Purine-Substituted Adenosine Derivatives with Small N⁶-Substituents as Adenosine Receptor Agonists	A. P. Ijzerman; J. K. von Frijtag Drabbe Künzel; S. Vittori; G. Cristalli
2283-2305	Novel 4′-Branched Nucleosides	S. A. Surzhykov; A. A. Krayevsky
2307-2320	A Short Synthesis of a Novel Ring-Expanded Purine and Its Nucleoside Analogue Containing the Imidazo[4,5-e][1,3]diazepine Ring Skeleton with Multiple Amino Substituents Attached to the 7-Membered Ring	L. Wang; A. Bhan; R. S. Hosmane; R. D. Guiles
2321-2328	Synthesis and Antiviral Activity of the Cyclopropano Homolog of 2,3-Didehydro-2,3-dideoxythymidine	H. Sard
2329-2344	NMR Studies Show Monomeric 5-Fluorouridine Forms Base Pairs of Increased Stability Compared with Uridine in Non-Aqueous Solvents	W. H. Gmeiner; J. Anderson; P. Sahasrabudhe
2345-2366	Synthesis and Biological Evaluation of Some Acyclic Pyridine C-Nucleosides. Part One	J. Van Hemel; E. L. Esmans; F. C. Alderweireldt; R. A. Dommisse; A. De Groot; J. Balzarini; E. De Clercq

Volume 13, Issue 9 (1994)

1829-1841	Synthesis of Deoxycytidine (dC) Building Blocks for Amide-Linked Dimers or Oligomers: Example of a Deoxycytidine-amide-thymidine Dimer	Evelyne Grunder-Klotz; George Just
1843-1853	Synthesis and Anti-HIV Activity of Alkyl Steroidal 3′-Azido-3′-deoxythymidin-5′-yl Phosphotriesters as Prodrugs of AZT	Meher I. Balagopala; Abraham P. Ollapally; Henry J. Lee
1855-1860	Sequence Specific DNA Purification by Triplex Affinity Capture: Using Solid Support Linked Oligodeoxynucleotide	Ajay Kumar; Suchitra Rustogi
1861-1870	Synthesis of 1-β-L-Arabinofuranosylcytosine (β-L-Ara-C) and 2′-Deoxy-2′-methylene-β-L-cytidine (β-L-DMDC) as Potential Antineoplastic Agents	Tai-Shun Lin; Mei-Zhen Luo; Mao-Chin Liu
1871-1889	Anti-HIV Derivatives of 1-(2,3-Dideoxy-3-N-hydroxyamino-β-D-threo-pentofuranosyl)thymine	Jean M. J. Tronchet; Martina Zsély; Karel Capek; Istvan Komaromi; Michel Geoffroy; Erik De Clercq; Jan Balzarini
1891-1903	A Phosphoramidite-Based Synthesis of Phosphoramidate Amino Acid Diesters of Antiviral Nucleosides	Timothy W. Abraham; Carston R. Wagner
1905-1927	Simplified and Cost Effective Syntheses of Fully Protected Phosphoramidite Monomers Suitable for the Assembly of Oligo(2′-O-allylribonucleotides)	Barbro Beijer; Morten Grøtli; Mark E. Douglas; Brian S. Sproat
1929-1937	Carbocyclic Analogues of 3′,4′-Didehydro-2′-deoxyribofuranosyl-2,4(1H,3H)-pyrimidinediones	C. Allen O'Dell; Y. Fulmer Shealy
1939-1952	Synthesis and Evaluation of Oligodeoxynucleotides Containing 3′-O-Ethyl-4′-C-(hydroxymethyl)thymidine: Introduction of a Novel Class of Phosphodiester Internucleoside Linkages	Lars H. Dreioøe; Jesper Wengel
1953-1976	Adenosine Receptor Classification: Quo Vadimus?	Jill Coates; Mark F. Gurden; Carol Harris; Ian Kennedy; Michael J. Sheehan; Peter Strong
1977-1989	Synthesis of Iodo-aryl-azido Adenosine Analogs as Affinity Ligands for Adenylyl Cyclase	Ilana Shoshani; Howard Qiu; Francis Johnson; Roger A. Johnson
1991-2000	Synthesis of 3′-Fluoro-3′-deoxy-N⁶-cyclopentyladenosine	G. Ceulemans; R. Busson; N. Weyns; F. Vandendriessche; J. Rozenski; A. IJzerman; P. Herdewijn
2001-2011	Synthesis and Biological Activity of 4-Amino-1-(β-D-ribofuranosyl)imidazo[4,5-d]pyridazin-7-one	David A. Berry; Linda L. Wotring; John C. Drach; Leroy B. Townsend
2013-2019	The Synthesis, Fluorescence and Antiviral Studies of 3′-Amino-2′,3′-Dideoxythymidine/substituted 10-Cyano-9-isothiocyanatoanthracene Adducts	Dan Swartling; Mike Fry; Matt Morgan; Ed Biehl; Jan Balzarini; Erik De Clercq
2021-2034	Synthesis of 5-Tethered Carborane-Containing Pyrimidine Nucleosides as Potential Agents for DNA Incorporation	Feng-Guang Rong; Albert H. Soloway

Volume 13, Issue 8 (1994)

1655-1667	Biologic Activity of a Nucleotide Conjugate Between Mitomycin C and Cytarabine Monophosphate	Robert T. Dorr; James D. Liddil; Bhashyam S. lyengar; Alan F. List; William A. Remers
1669-1677	Interaction Between the Guanine Amino Group and the Adenine Six Membered Ring Stabilizes the Unusual Conformation of the CpA Step in B-DNA	J. Šponer; J. Jursa; J. Kypr
1679-1693	Synthesis and Biological Evaluation of Pyrimidine and Purine α-L-2′,3′-Dideoxy Nucleosides	Naina A. Van Draanen; George W. Koszalka
1695-1706	Synthesis of ISIS 2105 Containing the Abasic Site Model Compound 1,4-Anhydro-2-deoxy-D-Ribitol	Vasulinga T. Ravikumar; Tadeusz K. Wyrzykiewicz; Douglas L. Cole
1707-1719	8-Aza-analogues of PMEA and PMEG: Synthesis and In Vitro Anti-HIV Activity	P. Franchetti; G. Abu Sheikha; L. Cappellacci; L. Messini; M. Grifantini; A. G. Loi; A. De Montis; M. G. Spiga; P. La Colla
1721-1738	A Facile Synthesis of the Phosphoramidites of 2-N-Methyl-2′-deoxy (or 2′-O-allyl)-ψ-isocytidine, 1, 3-Dimethyl-2′-deoxy-ψ-uridine and N1-Methyl-2′-O-allyl-ψ-uridine as Synthons Suitable for Oligonucleotide Synthesis	B. K. Bhattacharya; G. R. Revankar
1739-1755	8-Aza-1-deazapurine Nucleosides as Antiviral Agents	P. Franchetti; L. Messini; L. Cappellacci; G. Abu Sheikha; M. Grifantini; P. Guarracino; A. De Montis; A. G. Loi; M. E. Marongiu; P. La Colla
1757-1768	The Stability of Trisubstituted Internucleotide Bond in the Presence of the Vicinal 2′-Hydroxyl. Chemical Synthesis of Uridyl(2′-phosphate)-(3′-5′)-uridine	R. Kierzek
1769-1777	Simplified Analogues of Acyclonucleosides. Synthesis of 6-[N-Alkyl-N-(4-hydroxybutyl)amino]pyrimidine Derivatives	M. Botta; R. Saladino; M. Anzini; F. Corelli
1779-1789	Synthesis and Anti-HIV Activity of 5-Fluorocytallene: N-Dimethylaminomethylene as a Facilitating Group in Acetylene → Allene Isomerization	C. Simons; S. Chokekijchai; H. Mitsuya; J. Zemlicka
1791-1800	2-Hydroxyethoxyethylated Bases as Acyclic Analogues of 1,5-Anhydrohexitol Nucleoside Derivatives	A. Van Aerschot; Z. Ni; J. Rozenski; P. Claes; E. De Clercq; P. Herdewijn
1801-1807	Lipase Catalyzed Diastereoselective Deacetylations of Anomeric Mixtures of Peracetylated 2′-Deoxynucleosides	D. L. Darmkjaer; M. Petersen; J. Wengel
1809-1817	Precursors for the Synthesis of Substituted 1,3,4-Thiadiazolf, C-Nucleosides, Analogues of Tiazofurin and Related Compounds	Hossein S. Khorshidi; Antonio Canas Rodrigez
1819-1828	Synthesis and Biological Activity of 4′-Thionucleosides of 2-Chloroadenine¹	Kamal N. Tiwari; John A. Secrist III; John A. Montgomery

Volume 13, Issue 6-7 (1994)

ix-x	Preface	Eiko Ohtsuka; Seiichi Uesugi; Akira Matsuda
1219-1230	Synthesis and Anti-HIV Activity of 2-Substituted 2′-Deoxy-2′-fluoroadenosines	Tokumi Maruyama; Kunihiko Utsumi; Yoshiko Sato; Douglas D. Richman
1231-1237	Recognition of the Anticodon Loop of tRNA^Ile₁ by Isoleucyl-tRNA Synthetase from Escherichia coli	Tatsuya Niimi; Osamu Nureki; Takashi Yokogawa; Nobuhiro Hayashi; Kazuya Nishikawa; Kimitsuna Watanabe; Shigeyuki Yokoyama
1239-1246	A Newly Devised Method for the Debenzylation of N⁶-Benzyladenosines. A Convenient Synthesis of [6-¹⁵N]-Labeled Adenosines	Magoichi Sako; Hiroaki Ishikura; Kosaku Hirota; Yoshifumi Maki
1247-1258	Synthetic Nucleosides and Nucleotides. XXXI.¹ Inhibitory Effects of 2′-Deoxy-5-styryluridine 5′-Triphosphate Analogues on Retroviral Reverse Transcriptases and Higher Eukaryotic DNA Polymerases	Toyofumi Yamaguchi; Shunji Izuta; Motoshi Suzuki; Shonen Yoshida; Akio Matsukage; Mineo Saneyoshi
1259-1269	Spectroscopic Characterization of the Decadeoxynucleotide Duplex Modified with Dichloroethylenediamineplatinum(II)	Hidehito Urata; Masayuki Urata; Masao Akagi; Hidekazu Hiroaki; Seiich Uesugi
1271-1295	Antiviral Activity Spectrum and Target of Action of Different Classes of Nucleoside Analogues	Erik De Clercq
1297-1309	Rare Earth Metal Ions for DNA Hydrolyses and Their Use to Artificial Nuclease¹	Makoto Komiyama; Naoya Takeda; Tetsuro Shiiba; Yota Takahashi; Yoichi Matsumoto; Morio Yashiro
1311-1317	Application of the Thermodynamic Parameters of DNA Stability Prediction to Double-Helix Formation of Deoxyribooligonucleotides	Naoki Sugimoto; Kei-ichi Honda; Muneo Sasaki
1319-1326	Properties of DNA Duplexes Containing an Abasic Site: Effect of Nucleotide Residue of the Opposite Part of a 2-Deoxyribosylformamide Residue	T. Shida; M. Arakawa; J. Sekiguchi
1327-1335	Conformation of 3-Substituted Purine Nucleoside Studied By X-Ray Crystallography and Theoretical Calculations	Yuriko Yamagata; Masato Kato; Satoshi Fujii; Mitsutoshi Aoyagi; Noriaki Minakawa; Akira Matsuda
1337-1345	Allyl Protection in the Synthesis of Oligodeoxyribonucleotide Phosphorothioates	Yoshihiro Hayakawa; Masaaki Hirose; Ryoji Noyori
1347-1361	Syntheses and Antitumor Activities of D-and L-2′-Deoxy-4′-thio Pyrimidine Nucleosides	Jun'ichi Uenishi; Keiji Takahashi; Mitsuhiro Motoyama; Haruo Akashi; Takuma Sasaki
1363-1374	DNA Diagnosis of Ovale Malaria and Malariae Malaria Using Microtiter Plate-Hybridization	Meiji Arai; Kaori Kunisada; Shintaro Kawai; Mikio Kimura; Yusuke Wataya
1375-1395	Biologically Active Oligodeoxyribonucleotides - II¹: Structure Activity Relationships of Anti-HIV-1 Pentadecadeoxyribonucleotides Bearing 5′-End-Modifications	Hitoshi Hotoda; Kenji Momota; Hidehiko Furukawa; Takemichi Nakamura; Masakatsu Kaneko; Satcshi Kimura; Kawu Shimada
1397-1414	A New Method for Removal of Modified Trityl and Pixyl Groups by Use of an Acid Species Generated by Reaction of Diethyl Oxomalonate with Methanol	Mitsuo Sekine
1415-1423	Change of the Higher Order Structure in a Giant DNA Induced by 4′, 6-Diamidino-2-phenylindole as a Minor Groove Binder and Ethidium Bromide as an Intercalator	Y. Matsuzawa; K. Yoshikawa
1425-1452	Nucleosides. LVI¹ Synthesis and Chemical Modifications of 3′-Deoxy-Pyrimidine Nucleosides	Soo-Young Rhie; Wolfgang Pfleiderer
1453-1465	Reactions of 9-Substituted 1-Aminoadenines with Nucleophiles and Syntheses of 3-Substituted 3H-Imidazo[4, 5-e][1, 2, 4]triazolo[1, 5-c][1, 2, 3]triazines	Shoji Asano; Keiji Itano; Yuriko Yamagata; Kohfuku Kohda

Volume 13, Issue 6-7 (1994)

1467-1481	A Raman Spectroscopic Study on Conformations of DNA Oligomers: A Dominant Effect of an AA:TT Sequence Over Those of AT:AT and TA:TA Sequences on Determining Conformations of DNA Duplexes	Masato Katahira; Yoshifumi Nishimura; Masamichi Tsuboi; Jun-ichi Matsuzaki; Hitoshi Hotoda; Mitsuo Sekine; Tsujiaki Hata
1483-1492	Nucleotide Incorporation Opposite Degenerate Bases by Taq DNA Polymerase	Hiroyuki Kamiya; Naoko Murata-Kamiya; Paul Kong Thoo Lin; Daniel M. Brown; Eiko Ohtsuka
1493-1506	The Synthesis of 4′-t-Butylcarbamyl- and 4′-p-Toluenesulphonamidyl-2′,3′-Dideoxy Pyrimidine Nucleoside Analogues	Lea Pickering; Baljinder S. Malhi; Paul L. Coe; Richard T. Walker
1507-1515	Drastic Difference in G:A Base Pairing Between Two Consecutive G:A Mismatches and a Single G:A Mismatch in DNA	Masato Katahira; Mayumi Kanagawa; Seiichi Uesugi
1517-1534	Synthesis and Thermodynamic Stabilities of Damaged DNA Involving 8-Hydroxyguanine (7,8-Dihydro-8-Oxoguanine) in a ras-Gene Fragments	Shiro Koizume; Hiroyuki Kamiya; Hideo Inoue; Eiko Ohtsuka
1535-1549	Nucleosides and Nucleotides. 130. The Synthesis of Imidazo[4, 5-e][1, 4] Diazepine Nucleosides From N¹-Substituted Inosines	Mitsutoshi Aoyagi; Noriaki Minakawa; Akira Matsuda
1551-1555	The Fluorescence Property of Dinucleoside Monophosphates Containing Ethenoadenosine and 5, 6-Dihydrouridine Derivatives	Kazuo Negishi; Hikoya Hayatsu
1557-1567	Large Scale Synthesis of the Cap Part in Messenger RNA Using a New Type of Bifunctional Phosphorylating Reagent	Koichiro Fukuoka; Fuminori Suda; Ryo Suzuki; Masahide Ishikawa; Hiroshi Takaku; Tsujiaki Hata
1569-1579	Properties of a Hammerhead-Type RNA Enzyme System That Consists of Three RNA Oligomer Strands	Osamu Odai; Hidekazu Hiroaki; Toshiki Tanaka; Seiichi Uesugi
1581-1595	Domains of E. Coli Glutaminyl-tRNA Synthetase Disordered in the Crystal Structure Are Essential for Function or Stability	Jill Conley; Joyce Sherman; Hans-Ulrich Thomann; Dieter Söill
1597-1605	Hybridization of Alternating Cationic/Anionic Oligonucleotides to RNA Segments	Paul M. Jung; Gary Histand; Robert L. Letsinger
1607-1615	Photochemical Cleavage of DNA With Phosphorus(V)porphyrin Derivatives	Takao Saito; Masanori Kitamura; Motomasa Tanaka; Minoru Morimoto; Hiroshi Segawa; Takeo Shimidzu
1617-1626	Inhibition of Restriction Enzyme Ksp 632-I Via Triple Helix Formation by Phosphorothioate Oligonucleotides	Satoru Tsukahara; Hidefumi Yamakawa; Kazuyuki Takai; Hiroshi Takaku
1627-1646	Synthesis of Substituted-Benzyl and Sugar-Modified Analogues of 6-N-(4-Nitrobenzyl)adenosine and Their Interactions with “ES” Nucleoside Transport Systems	Morris J. Robins; Jun-ichi Asakura; Masakatsu Kaneko; Susumu Shibuya; Ewa S. Jakobs; Francisca R. Agbanyo; Carol E. Cass; Alan R. P. Paterson
1647-1654	Facile Synthesis of α-Anomeric Pyrimidine Nucleosides	Hiroaki Sawai; Akiko Nakamura; Hidekazu Hayashi; Kazuo Shinozuka

Volume 13, Issue 5 (1994)

1017-1029	Synthesis and Biologic Evaluation of 8-Substituted Derivatives of Nebularine (9-β-D-Ribofuranosylpurine)	John A. Secrist; Anita Shortnacy-Fowler; L. Lee Bennett Jr.; John A. Montgomery
1031-1037	An Alternative Route for Preparation of α-Methylphosphonyl-β, γ-Diphosphates of Thymidine Derivatives	Aridrey A. Arzumanov; Natalia B. Dyatkina
1039-1047	Synthesis and Separation of Dinucleoside Phenylphosphonate Diastereomers	S. A. Nadeem Hashmi; Anil Kumar; S. B. Kacti
1049-1058	Synthesis and Antifungal Activity of 3′-Deoxyribonucleosides	Anil Kumar; Shoeb I. Khan; Anita Manglani; Z. K. Khan; S. B. Katti
1059-1067	6-N-1 Trobenzotriazol-1-Yloxytris(Dimethylamino)Phosphonium Hexafluorophosphate (NBOP): A New Coupling Reagent in Oligonucleotide Synthesis	S. A. Nadeem Hashmi; M. Adiraj; Anil Kumar; S. B. Katti
1069-1085	The Chemical Synthesis of Biochemically Active Oligoribonucleotides Using Dimethylaminomethylene Protected Purine H-Phosphonates	Gunther Ott; Lubos Arnold; Jiri Smrt; Michal Sobkowski; Stefan Limmer; Hans-Peter Hofmann; Mathias Sprinzl
1087-1111	Rapid and Efficient Syntheses of Phosphorylated Dinucleotides	James P. Ferris; John R. Peyser
1113-1123	Comparative Liquid Chromatographic Stability Study of Thymidine and 1- (2-Deoxy-α-D-Erythro-Pentofuranosyl) Thymine	A. Van Schepdael; F. Heerinckx; A. Van Aerschot; P. Herdewijn; E. Roets; J. Hoogmartens
1125-1133	Synthesis of 4-Amino-8-(2, 2-Difluoro-2-Deoxy-β-D-Ribo Furanosyl Amino)Pyrimido [5, 4-D]Pyrimidine (dFARPP). Stability and Cellular Cytotoxicity	T. E. Mabry; C. D. Jones; T. S. Chou; J. M. Colacino; G. B. Grindey; J. F. Worzalla; H. L. Pearce
1135-1145	Synthesis and Antiviral Study of Dihydrothieno and Thianopyrimidine Diones Acyclic Nucleosides As Potential Anti-HIV Agents	Jacques Renault; Daniel Laduree; Max Robba
1147-1160	Synthesis of Three New Carbocyclic Analogues of 3′-Deoxy Purine Ribonucleosides	Luigi Agrofoglio; Roger Condom; Roger Guedj; S. Richard Challand; John Selway
1161-1168	A Highly Selective and Efficient Access to N-9 Alkylated Purine Derivatives via Radical SRN1 Chemistry	Tawfik Gharbaoui; Rachid Benhida; André Lechevallier; Phillip Maillos; René Beugelmans
1169-1177	Selective N1-Alkylation of Pyrimidine Bases via Radical (SRN1) Mechanism	Rachid Benhida; Tawfik Gharbaoui; Andre Lechevallier; Rene Beugelmans
1179-1188	P-Glycoprotein and the Renal Secretion of Deoxyribonucleosides	Big-Fang Pan; J. Arly Nelson
1189-1199	Conformatzonal Properties of a Novel Modified Nucleoside, 5-Formylcytidine, Found at the First Position of the Anticodon of Bovine Mitochondrial tRNA^Met	Gota Kawai; Takashi Yokogawa; Kazuya Nishikawa; Takuya Ueda; Takeshi Hashizume; James A. McCloskey; Shigeyuki Yokoyama; Kimitsuna Watanabe
1201-1213	Acyclic Nucleosides: Synthesis of 1-[(1-Hydroxy-2-Propoxy) Methyl]Thymine, 6-Azathymine, URACIL, AND 6-Azauracil as Potential Antiviral Agents	Eng-Chi Wang; Hour-Young Chen; Cherng-Chyi Tzeng
1215-1216	A Novel Preparation of Nicotinamide Mononucleotide	Rihe Liu; Johannes Visscher

Volume 13, Issue 4 (1994)

883-889	Synthesis of Acyclic Thieno[3,2-d]Pyrimidine Nucleosides and Azido Derivatives as Potential Anti-HIV Agents	C. Fossey; D. Laduree; M. Robba
891-901	Synthesis and Antiviral Study of Cyclopentano [d] Pyrimidine-2,4-diones and Octahydroquinazoline-2,4-diones Acyclic Nucleosides as Potential Anti-HIV Agents	J. Renault; D. Laduree; M. Robba
903-913	Synthesis and Properties of S-Phosphates of Some Antiviral Acyclonucleosides	Michael R. Harnden; Halina T. Serafinowska
915-923	Synthesis and Anti-HIV Evaluation of 7-Deaza Analogues of Carbovir	Michel Legraverend; Anne-Marie Aubertin; Georges Obert; Christiane Huel; Emile Bisagni
925-937	Synthesis of N-1β-D-Arabinofuranosyl and N-1-2′-Deoxy-β-D-erythro-pentofuranosyl Thieno [3,2-d] Pyrimidine Nucleosides	C. Fossey; H. Landelle; D. Laduree; M. Robba
939-944	Synthesis of 2′-Deoxyuridine Nucleosides with Appended 5-Position Carbonyl Cross-Linking Groups	Gregory J. Crouch; Bruce E. Eaton
945-952	Steric Effect of a Bulky Substituent At 5′-Position on the Regioselectivity of 2′ vs. 3′-O-Methylation of N⁶- Cyclohexyladenosine	Mahavir Prashad; Kapa Prasad; Oijan Repic
953-962	Thermodynamic and NMR Study of Proton Complex Formation of 2′-Deoxyadenylyl-(3′→5′)-2′-Deoxyadenosine in Aqueous Solution	Rosa Chillemi; Annalinda Contino; Vincenzo Cucinotta; Sebastiano Sciuto
963-978	DNA Intercalation and Photoinduced Cleavage by 4-Nitro(N-Hexylamine)1,8-Naphthalimide	Jyoti Mehrotra; Krishna Misra; Rakesh K. Mishra
979-996	Influence of Remote Structure Upon Regioselectivity in the N-Alkylation of 2-Amino-6-Chloropurine: Application to the Synthesis of Penciclovir	Bernadette M. Choudary; Graham R. Geen; Trevor J. Grinter; Fiona S. MacBeath; Martin J. Parratt
997-1005	Interaction of Oligodeoxyribonucleotides Through Formation of Chimeric Duplex/Triplex Complexes	David M. Noll; Jessica L. O'Rear; Cynthia D. Cushman; Paul S. Miller
1007-1010	Synthesis and Antiretroviral Evaluation of Various 5-Alkyl-6-AZA-5,6-Dihydrouridine	Jean Depelley; Robert Granet; Pierre Krausz; Salomon Piekarski; Claudine Bosgiraud; Sylvie Beaussoleil
1011-1013	Straightforward Synthesis of 1-(2,3-Dideoxy-β-D-Glycero-Pent-2-Enofuranosyl)-Thymine	G. Negrón; G. Islas; Y. Díaz; R. Cruz; B. Quiclet-Sire

Volume 13, Issue 1-3 (1994)

1	Memorial Issue Honoring Roland K. Robins
3-16	A Memorial Tribute to Roland Kenith Robins	Leroy B. Townsend
77-94	Derivatives of 1-(2-Deoxy-2-fluoro-β-D-arabinofuranosyl)-5-phenyluracil and 5-Benzyluracil. Synthesis and Biological Properties	Krzysztof Dziewiszek; Raymond F. Schinazi; Ting-Chao Chou; Tsann-Long Su; Jolanta M. Dzik; Wojciech Rode; Kyoichi A. Watanabe
95-107	Synthesis of Triple Helix Forming Oligonucleotides Containing 2′-Deoxyformycin A	T. Sudhakar Rao; Michael E. Hogan; Ganapathi R. Revankar
109-126	Synthesis of Isonucleosides Related to AZT and AZU	David F. Purdy; Lawrence B. Zintek; Vasu Nair
127-153	Photo-Arbuzov Rearrangements of Benzyl Phosphites. Preparation of Acyclic Nucleoside Phosphonates Related to HPMPA	Khairuzzaman B. Mullah; Wesley G. Bentrude
155-162	Design and Synthesis of Regioisomeric Analogues of a Specific Anti-HIV-1 Agent 1-[(2-Hydroxyethoxy)methyl]-6-(phenylthio)thymine (HEPT)	Hiromichi Tanaka; Masanori Baba; Emiko Takahashi; Kouichiro Matsumoto; Atsushi Kittaka; Richard T. Walker; Erik De Clercq; Tadashi Miyasaka
163-175	The Synthesis of Some 5-Substituted-6-aza-2′-deoxyuridines	I. Basnak; P. L. Coe; R. T. Walker
177-196	The Synthesis of Some 5-Substituted and 5,6-Disubstituted 2′-Deoxyuridines	I. Basnak; A. Balkan; P. L. Coe; R. T. Walker
197-211	Nucleosides and Nucleotides. 125. Synthesis and Biological Evaluation of 2′,3′-Dideoxy-3′-fluoro-2′-methylidene Pyrimidine Nucleosides	Abdalla Elsayed A. Hassan; Satoshi Shuto; Akira Matsuda
213-234	Chemistry and Anti-HIV Activity of 2′-β-Fluoro-2′,3′-dideoxyguanosine	Harry Ford Jr.; John S. Driscoll; Maqbool Siddiqui; James A. Kelley; Hioraki Mitsuya; Takuma Shirasaka; David G. Johns; Victor E. Marquez
235-243	Synthesis of 5-Ethyl-2-pyrimidinone-2′-deoxyriboside as a New Potential Antiviral Agent	Smita B. Trehan; Joan E. MacDiarmid; Thomas J. Bardos
245-254	Synthesis of 1-[cis-2-Hydroxy-cis-3-(hydroxymethyl)-cyclobutyl]thymine, a Novel Method for the Synthesis of Cyclobutyl Nucleosides and Related Compounds	Tai-Shun Lin; Mei-Zhen Luo; Mao-Chin Liu
255-273	Synthesis of Triple Helix Forming Oligonucleotides with a Stretched Phosphodiester Backbone	T. Sudhakar Rao; Krishna Jayaraman; Ross H. Durland; Ganapathi R. Revankar
275-292	The Effect of pH on the Covalent Complexes of Thymidylate Synthase	Mary S. Weir; R. Bruce Dunlap
293-295	Structure Determination of 4-Chloro-DRB	R. L. Tolman; G. A. Doss
297-308	A Ribonolactone-Based Approach to the Synthesis of 1′-Carbon-Substituted Thymine Ribonucleosides	Hiroyuki Hayakawa; Michiko Miyazawa; Hiromichi Tanaka; Tadashi Miyasaka
309-323	Synthesis and Biologic Activity of Purine 2′-Deoxy-2′-fluoro-ribonucleosides	H. Jeanette Thomas; Kamal N. Tiwari; Sarah Jo Clayton; John A. Secrist III; John A. Montgomery
325-337	Synthesis and Antiviral Activity of Some Fluorinated Nucleotide Derivatives	Natalia Dyatkina; Andrey Arzumanov; Alexander Krayevsky; Bryan O'Hara; Yacov Gluzman; Penny Baron; Clarinda MacLow; Bruce Polsky

Volume 13, Issue 1-3 (1994)

339-350	Synthesis of the P¹, P²-Methylene Analog of N²- (p-n-Butylphenyl)-2′- deoxyguanosine 5′-Triphosphate: A Non-substrate Inhibitor of DNA Polymerases	Ivan Yanachkov; George E. Wright
351-368	Structure and Stability of an Oligonucleotide Containing 2′-Deoxy-6-thioguanosine	Michael S. Christopherson; Arthur D. Broom
369-378	Nucleophilic Substitution Reactions of 5-Bromo-6-methyluridines	Mallela S. P. Sarma; Robert S. Klein; Brian A. Otter
379-388	Synthesis of a Novel Antiretroviral Thymidine Analog: 1-(2-Deoxy-β-D-ribofuranosyl)-4-acetylimidazolin-2-one (Imidine)	Xiang-Jun Jiang; Thomas I. Kalman
389-403	Nucleic Acid Related Compounds. 82. Conversions of Adenosine to Inosine 5′-Thioether Derivatives with Aspergillus oryzae Adenosine Deaminase or Alkyl Nitrites. Substrate and Inhibitory Activities of Inosine 5′-Thioether Derivatives with Purine Nucleoside Phosphorylase	Stanislaw F. Wnuk; Johanna D. Stoeckler; Morris J. Robins
405-420	Synthesis and Biological Activity of the Novel Adenosine Analogs; 3-Amino-6-(β-D-ribofuranosyl)pyrazolo[3,4-c]pyrazole and 3-Amino-1-methyl-6-(β-D-ribofuranosyl)pyrazolo[3,4-c]pyrazole	David A. Berry; Linda L. Wotring; John C. Drach; Leroy B. Townsend
421-427	Monoclonal Antibodies with Affinity to Self-Complementary Left-Handed DNA Containing Cyclonucleosides with High Anti Conformation	Junji Kawakami; Seiichi Uesugi; Morio Ikehara; Teiji Itoh; Kazunobu Miura; Eiko Ohtsuka
429-435	Relationship Between the Structure of Sangivamycin-Derived Nucleosides and Their Effect on Leukemic Cell Growth and on Protein Kinase A and C Activity	Miroslav Bobek; Alexander Bloch
437-446	Synthesis and Antiviral Evaluation of 2-Mercapto-5,6-dichlorobenzimidazole-β-D-ribofuranonucleoside Derivatives	C. Mathé; C. Périgaud; G. Gosselin; J. -L. Imbach
447-457	Selective Synthesis of 6-Ribo- (and Xylo) Pyrano and Furano Aminopyrimidines¹. Anticancer and Anti-AIDS Activities	M. Nogueras; J. Cobo; M. L. Quijano; M. Melguizo; A. Sánchez; M. Melgarejo
459-479	Synthesis of 2′,3′-Dideoxy- and 3′-Azido-2′,3′-dideoxy-pyridazine Nucleosides as Potential Antiviral Agents	Biserka Kasnar; Dean S. Wise; Louis S. Kucera; John C. Drach; Leroy B. Townsend
481-490	Tautomerism, Protonation, and Ionization of Formycin in Aqueous Solution by the pH Dependence of ¹³C Chemical Shifts and ¹³C-¹H Coupling Constants	Bongsup P. Cho; Michael A. McGregor
491-499	Synthesis of D-Fructofuranosylpurine Nucleosides	Abderrahime Bouali; David F. Ewing; Grahame Mackenzie
501-509	Synthesis of Oligodeoxyribonucleotides Containing 2,6-Diaminopurine	Angeles Canol; Myron F. Goodman; Ramon Eritja
511-525	Synthesis and Biological Evaluation of Some D-Arabino- and D-Lyxofuranosyl-Pyridine C-Nucleosides	F. Verberckmoes; E. L. Esmans; J. Balzarini; E. De Clercq
527-537	Synthesis and Anti-HIV Activity of 6-Substituted Purine 2′-Deoxy-2′-fluororibosides	Tokumi Maruyama; Kunihiko Utzumi; Yoshiko Sato; Douglas D. Richman
539-550	Synthesis of Acyclonucleoside Phosphonates as Antiviral Agents Against Cytomegalovirus	Elmer J. Reist; Wallace W. Bradford III; Beatrice L. Ruhland-Fritsch; Priscilla A. Sturm; Nurulain T. Zaveri; John Huffman; Robert W. Sidwell
551-562	Guanosine Derivatives as Immunostimulants. Discovery of Loxoribine	Robert Chen; Michael G. Goodman; Dennis Argentieri; Stanley C. Bell; Levelle E. Burr; Jon Come; Jacquelyn H. Goodman; Dieter H. Klaubert; Bruce E. Maryanoff; Barbara L. Pope; Marianne S. Rampulla; Mary R. Schott; Allen B. Reitz
563-584	Synthesis of C-6 Pyrimidine Acyclic Nucleoside Analogs as Potential Antiviral Agents	Ling-Yih Hsu; Dean S. Wise; William M. Shannon; John C. Drach; Leroy B. Townsend
585-598	A Convenient Route to 2′-Allenyl Nucleosides	Esa T. Jarvi; James R. McCarthy

Volume 13, Issue 1-3 (1994)

599-605	Construction of a Translation Enhancer-Containing Vector for Gene Expression in a Prokaryotic Two-Cistron System	Klara R. Birikh; Ekaterina N. Lebedenko; Yuri A. Berlin
607-613	Structure-Activity Relationship of Phosphonic Acid Analogs of Acyclovir or Ganciclovir Against Human Cytomegalovirus in MRC-5 Cells	John H. Huffman; Robert W. Sidwell; Ann G. Morrison; Jana Coombs; Elmer J. Reist
615-623	Nucleoside Analogues on the Basis of 4(R),5(R)-Dihydroxymethyl-2-methyl-1,3-dioxolane	Sergey N. Mikhailov; Ekaterina V. Efimtseva; Sergey V. Meshkov; Earl R. Kern
625-636	A Novel Palladium-Catalyzed Deoxygenation of Guanine O⁶-Arenesulfonates. A Practicable Synthesis of 2-Aminopurine Nucleosides and Related Analogs	Anton Štimac; Darja Muhič; Jože Kobe
637-655	¹H NMR Structural Analysis of the Interactions of Proflavine with Self-Complementary Deoxytetranucleosides of Different Base Sequence	D. B. Davies; L. N. Djimant; A. N. Veselkov
657-671	¹H NMR Thermodynamical Analysis of the Interactions of Proflavine with Self-Complementary Deoxytetranucleotides of Different Base Sequence	D. B. Davies; L. N. Djimant; A. N. Veselkov
673-678	The Synthesis of 2-Fluoropurine Nucleosides	K. Krolikiewicz; H. Vorbrüggen
679-688	Synthesis of Bicyclic N⁴-Oxycytidine Derivatives	D. Loakes; D. M. Brown
689-706	X-Ray Crystallographic and Kinetic Analysis of Human Purine Nucleoside Phosphorylase Complexes with 1-β-D-Ribofuranosyl-1,2,4-triazole-3-carobxamide and 1-β-D-Ribofuranosyl-1,2,4-triazole-3-carboxamidine	Richard L. Walter; Jindrich Symersky; Anne F. Poirot; Johanna D. Stoeckler; Mark D. Erionf; Steven E. Ealick
707-717	Synthesis of 3′-Amino and 5′-Amino Hydantoin 2′-Deoxynucleosides	Ahmed A. El-Barbary; Ahmed I. Khodair; Erik B. Pedersen; Claus Nielsen
719-736	Synthesis of Novel Isothiazole and Isothiazolo[4,5-d] Pyrimidine Analogues of the Natural C-Nucleosides Pyrazofurin and the Formycins	Diederik K. Buffel; Lieven Meerpoel; Suzanne M. Toppet; Georges J. Hoornaert
737-751	Conjugates of Fluorescein and Saenta (5′-S-(2-Aminoethyl)-N⁶-(4-nitrobenzyl)-5′-thioadenosine): Flow Cytometry Probes for the ES Nucleoside Transporter Elements of the Plasma Membrane	J. K. Buolamwini; J. D. Craik; J. S. Wiley; M. J. Robins; W. P. Gati; C. E. Cass; A. R. P. Paterson
753-772	Properties of RecA Complexes with Homopolymeric DNA Strands Depend on Sequence Complementarity. Implications for the Mechanism of Strand Exchange	Mikael Kubista; Bengt Nordén; Masayuki Takahashi
773-798	Nucleosides. LIV¹ Synthesis and Properties of 3′-Azido- and 2′,3′-Dideoxy-6,7-diphenyllumazine Nucleosides	Xiaodong Cao; Wolfgang Pfleiderer
799-809	Base Changes and Triple-Helix Hybridization Properties of GT Containing Third Strands: A Systematical Study	Jean-Pierre Clarenc; Bernard Lebleu; Jean-Paul Léonetti
811-817	Synthesis of the Nucleotide Analogue: (R,S)-9-[1-(2-Hydroxyethylthio)-2-phosphonylethyl] Adenine	H. B. Lazrek; H. Khaider; A. Rochdi; J. L. Barascut; J. L. Imbach
819-834	Chemical-Enzymatic Synthesis of 3′-Amino-2′, 3′-dideoxy-β-D-ribofuranosides of Natural Heterocyclic Bases and Their 5′-Monophosphates	Galina V. Zaitseva; Evgenii I. Kvasyuk; Elena V. Vaaks; Vladimir N. Barai; Sergei B. Bokut; Anatolii I. Zinchenko; Igor A. Mikhailopulo
835-848	Synthesis of 2′-Deoxyribonucleoside Derivatives of 1-Deazapurine	G. Cristalli; S. Vittori; A. Eleuteri; R. Volpini; E. Camaioni; G. Lupidi
849-880	Boron Containing Pyrimidines, Nucleosides, and Oligonucleotides for Neutron Capture Therapy	Naganna M. Goudgaon; Geraldine Fulcrand El-Kattan; Raymond F. Schinazi

Volume 12, Issue 10 (1993)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 12, Number 10
1007-1013	A Convenient High Yield Synthesis of N⁴-Isobutyryl-2′-O-Methylcytidine and Its Monomer Units For Incorporation into Oligonucleotides	Morteza M. Vaghefi; Richard I. Hogrefe
1015-1032	Synthesis of an Oligonucleotide Bearing a Phosphate Function at the 5′-Terminus Using a Novel Protecting Group in Terms of a Cellulose Acetate Derivative as a Polymer-Support	Kazuo Kamaike; Tomohiro Ogawa; Yoshiharu Ishido
1033-1046	N-6-Dialkylformamidine-2′-deoxyadenosine Phosphoramidites in Oligodeoxynucleotide Synthesis Raped Deprotection of Oligodeoxynucleotides	Pete Theisen; Christie McCollumy; Alex Andrus
1047-1059	A versatile Solid Phase Method For the Synthesis of Masked 3′-Thiol Group Containing Oligonucleotides	Ajar Kumar
1061-1074	Reactions of Some 2,3-Anhydro Pyrimidine Nucleosides with Dilithium Tetrahalocuprates	Kenji Watanabe; Kazufumi Yanagihara; Katsumaro Minamoto; Hiroshi Iwasaki
1075-1084	The 5′-Hydrogen Phosphonate Analog as a Potential Prodrug of 3′-Azido-2′,3′-dideoxythymidine (AZT)	Jila H. Boal; Radhakrishnan P. Iyer; William Egan
1085-1092	A Simple Multi-Gram Synthesis of 5′-Hydrogenphosphonates and 5′-Phosphorofluoridates of Sugar Modified Nucleosides	J. Matulic-Adamic; I. Rosenberg; A. A. Arzumanov; N. B. Dyatkina; E. A. Shirokova; A. A. Krayevsky; K. A. Watanabe
1093-1109	Synthesis and Some Properties of Modified Oligonucleotides. II. Oligonucleotides Containing 2′-Deoxy-2′-fluoro-β-D-arabinofuranosyl Pyrimidine Nucleosides	Pavol Kois; Zdenek Tocik; Maria Spassova; Wu-Yun Ren; Ivan Rosenberg; Jaume Farras Soler; Kyoichi A. Watanabe

Volume 12, Issue 9 (1993)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 12, Number 9
895-904	Synthesis of (E)-5-(2-cIOdovinyl)-3′-0-(1-Methyl-1,4-Dihydropyridyl-3 -Carbonyl)-2′-Fluoro-2′-Deoxyuridine (Ivfru-Cds) for Brain Targetted Delivery of Ivfru, an Antiviral Nucleoside	Rakesh Kumar; Edward E. Knaus; Leonard I. Wiebe
905-913	Synthesis of 1-(3-Azido-2,3-Dideoxy-Beta-D-Ribo-Hexofuranosyl)Thymine	Merrick R. Almond; Gregory T. Lowen; Gary E. Martin; Janet L. Rideout
915-924	Synthesis of Some New Nucleoside Analogues as Potential Antiviral Agents	M. A. Forestier; A. I. Ayi; R. Condom; B. P. Boyode; J. N. Colin; J. Selway; R. Challand; R. Guedj
925-940	Synthetic and Antiviral Studies on Certain Acyclic Nucleosides of 5-Benzyl-6-Azauracil Derivatives	Yeh-Long Chen; Shwu-Jing Chen; Kuan-Han Lee; Bor-Ruey Huang; Cherng-Chyi Tzeng
941-949	Nucleosides VI: A Novel and Convenient Synthesis of Purine S-Cyclonucleosides Via Mitsunobu Reaction	Ji-Wang Chern; Chia-Chi Kuo; Ming-Jyh Chang; Lee-Tai Liu
951-966	Synthesis of 3′-N-Substituted 3′-Amino-3′-Deoxythymidine Derivatives	Lech Celewicz; Wojciech Urjasz; Krzysztof Golankiewicz
967-971	Predictable and Reproducible Yields in the Anchoring of Dmt-nucleoside-succinates to Highly Loaded Aminoalkyl-Polystyrene Resins	F. Xavier Montserrat; Anna Grandas; Enrique Pedroso
973-980	Synthesis of 1-(β-D-Ribofuranosyl)Thieno[3,2-d] Pyrimidine-2,4-Dione and 4-Substituted Derivatives	C. Fossey; H. Landelle; D. Ladureey; M. Robba
981-992	Improved Synthesis of 2′,3′-Dideoxycytidine (d2C) and Its Correlated Nucleoside Analogues	L. De Napoli; A. Messere; D. Montesarchio; G. Piccialli; C. Santacroce
993-1005	Use of a Base-Labile Protected Derivative of 6-Mercaptohexanol for the Preparation of Oligonucleotides Containing a Thiol Group at the 5′-End	Beatriz G. de la Torre; Anna Maria Aviñó; Mónica Escarceller; Miriam Royo; Fernando Albericio; Ramon Eritja

Volume 12, Issue 8 (1993)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 12, Number 8
785-792	Syntheses and Interactions of Oligodeoxyribonucleotides Containing 2′-Amino-2′-Deoxyuridine	Paul S. Miller; Purshotam Bhan; Lou-Sing Kan
793-802	Enantioselective Synthesis of the Carbocyclic Tetrazole C-Ribonucleosides	Barbara Mohar; Anton Štimac; Jože Kobe
803-814	α-Trifluoromethyl-β-Ureido-Propionic Acid (F₃MUPA): A New Metabolite of Trifluridine (F₃TdR)	Manju Tandon; Piyush Kumar; Leonard I. Wiebe
815-826	Analysis of Modified Deoxynucleosides by Electrospray Ionization Mass SPECTROMETRY	Dasari M. Reddy; Charles R. Iden
827-839	Synthesis of 8-Substituted Theophyllineβ-D-Ribofuranosides	Vita Ozola; Natalya Ramzaeva; Yuris Maurinsh; Margeris Lidaks
841-846	The Synthesis and Biological Activity of 1-(2-Deoxy-4-Thio-α;-L-Threo-Pentofuranosyl)Thymine	Kamal N. Tiwari; John A. Montgomery; John A. Secrist III
847-852	A Reinvestigation of the Synthesis of 4-Thio-Pentofuranosides for Further Nucleosidic Synthesis	L. Bellon; C. Leydier; J. L. Barascut; J. L. Imbach
853-864	Synthesis of Cholesteryl Supports and Phosphoramidite for Automated DNA Synthesis of Triple-Helix Forming Oligonucleotides (Tfos)	Huynh Vu; Pradeep Singh; Laurie Lewis; Joseph G. Zendegui; Krishna Jayaraman
865-877	Synthesis of 2′,3′-Didehydro-2′,3′-Dideoxy-3′-C-Methyl Substituted Nucleosides	Panagiotis Ioannidis; Björn Classon; Bertil Samuelssony; Ingemar Kvarnström
879-893	5′-Phosphonates of Ribonucleosides and 2′-Deoxyribonucleosides: Synthesis and Antiviral Activity	Maxim Jasko; Alexander Shipitsin; Elena Shirokova; Alexander Krayevsky; Bruce Polsky; Penny Baron; Clarinda MacLow; Michael Ostrander; Brian O'Hara

Volume 12, Issue 7 (1993)

a-b	Editorial board page for “Nucleosides & Nucleotides”, Volume 12, Number 7
675-685	Synthesis of Some Novel Acyclolumazine N-1 Nucleosides	Najim A. Al-Masoudi; Wolfgang Pfleiderer; Wasfi A. Al-Masoudi
687-699	Synthesis of Some Novel 1-(5-Thio-ß-D-glucopyranosyl)-6-azauracil Derivatives - Thiosugar Nucleosides	Najim A. Al-Masoudi; Wolfgang Pfleiderer; Hassan B. Lazrek
701-711	Metal Carbonate-Mediated Complete Deacylation of Polyacyl Protected Nucleosides	Jun-ichi Asakura
713-728	Approaches to Nuclease Models: Synthesis and Conformational Studies of dT_prA Conjugated with Histamine AT C8(A) and Ethylenediamine at C5′(T)	T. P. Prakash; R. Krishnakumar; K. N. Ganesh
729-736	A Rapid Solid Phase Method for the Synthesis of 3′-Thiol Group Containing Oligonucleotides	Ajay Kumar
737-755	A Stereoselective Synthesis of α - and β-2′-Deoxy-2-thiouridine	Robert G. Kuimelis; Håkon Hope; Krishnan P. Nambiar
757-771	Synthesis of 8-Bromo- and 8-Azido-2′-deoxyadenosine-5′-O-(1-thiotriphosphate)	Norbert Ettner; Ute Haak; Michael Niederweis; Wolfgang Hillen
773-784	Cyclohexenyl Nucleosides and Related Compounds	J. H. Arango; A. Geer; J. Rodriguez; P. E. Young; P. Scheiner

Volume 12, Issue 6 (1993)

a	Editorial board page for “Nucleosides & Nucleotides” Volume 12, Number 6
565-584	Improved Methods for 3′-O-Succinylation of 2′-Deoxyribo- and Ribonucleosides and Their Covalent Anchoring on Polymer Supports for Oligonucleotide Synthesis	P. Kumar; N. N. Ghosh; K. L. Sadana; B. S. Garg; K. C. Gupta
585-596	Determination of N⁶-Threoninocarbonyladenosine, N², N²-Dimethylguanosine, Pseudouridine and Other Ribonucleosides in Human Breast Milk	H. Topp; H. Groß; G. Heller-Schöch; G. Schöch
597-604	N, N-Diisopropyl-O-Methyl-O-4-Nitrophenyl Phosphoramidite. New Flexible Phosphitylating Reagent in the Synthesis of Thio- and Seleno- Oligonucleotides	Jan Heliński; Wojciech Dabkowski; Jan Michalski
605-614	Solution and Solid State Structure of 2′,5′-BIS-(O-Trityl)-3′-Oximinouridine	Peter Agback; A. Papchikhin; S. Neidle; Jyoti Chattopadhyaya
615-629	Spin Labeled Nucleoside Analogues: 4′-Hydroxymorpholin-2′-Ylpurines and Pyrimidines	Jean M. J. Tronchet; Martina Zsély; Daniel Cabrini; Chantal Jorand; Françoise Barbalat-Rey; Istvan Komaromi; Alessandra Ricca; Michel Geoffroy
631-641	Synthesis and Biological Evaluation of a New N⁴-(N-Formyl Peptide)- 2′,3′-Dideoxy-3′-Thiacytidine as Anti-Hiv Prodrug	Michel Camplo; Philippe Faury; Anne-Sophie Charvet; Florence Lederer; Jean-Claude Chermann; Jean-Louis Kraus
643-648	A Practical Synthesis of The Antibiotic Toyocamycin	Moheshwar Sharma; Alexander Bloch; Miroslav Bobek
649-670	Possibility for the Existence of a General Conformational Motif in the Active Sites of Enzymes Which are Involved in Nucleic Acids Metabolism	Alexander A. Krayevsky; Kyoichi A. Watanabe

Volume 12, Issue 5 (1993)

a-b	Editorial board page for “Nucleosides & Nucleotides”, Volume 12, Number 5
431-439	Nucleosides, I Ribosylation of 8-Substituted Theophylline Derivatives	Mosselhi A. N. Mosselhi
441-447	A New Solid Phase Method for the Synthesis of Oligonucleotides with Terminal -3′-Phosphate	Ajay Kumar
449-462	Synthesis of 2′,3′-Didehydro-2′,3′-dideoxy-2′-C-methylsubstituted Nucleosides Using a Novel S_N2′ Type Reaction	Panagiotis Ioannidis; Björn Classon; Bertil Samuelsson; Ingemar Kvarnström
463-477	A New Approach for the Efficient Synthesis of Oligodeoxyribonucleotides Containing the Mutagenic DNA Modification 7,8-Dihydro-8-oxo-2′-deoxyguanosine at Predefined Positions
479-486	Synthesis of 8-Substituted 7-(α-L-Arabinofuranosyl)theophyllines	Vita Ozola; Natalya Ramzaeva; Yuris Maurinsh; Margeris Lidaks
487-498	An Improved Synthesis of 2′-Deoxy-9-deazaadenosine and an N-7 Blocked Derivative Useful for the Synthesis of Modified Oligonucleotides Containing 2′-Deoxy-9-deazaadenosine	Lech A. Ciszewski; Pawel Lipka; Wu-Yon Ren; Kyoichi A. Watanabe
499-528	Synthesis of 2′,3′-Dideoxy-3′-nitro-2′,3′-didehydrothymidine. Its Use as a General Intermediate for the Preparation of Various 2′,3′-Substituted Nucleosides	N. Hossain; A. Papchikhin; N. Garg; I. Fedorov; J. Chattopadhyaya
529-536	Synthesis of Mimics to Thymidine Triphosphate and 3′-Deoxy-3′-fluorothymidine Triphosphate	Magnus Björsne; Björn Classon; Ingemar Kvarnström; Bertil Samuelsson
537-545	Synthesis and Antiviral Activity of 1-β-D-Arabinofuranosyluracils and Uridines Containing 5-[2-Bromo-2-chloro (or Bromo)-1-Hydroxy (or Methoxy) Ethyl] Substituents	Rakesh Kumar; Leonard I. Wiebe; Edward E. Knaus
547-558	Synthetic and Antiviral Studies of Carboacyclic 6- and 2,6-Substituted Purine Nucleosides	Renée Pontikis; Claude Monneret

Volume 12, Issue 3-4 (1993)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 12, Number 3-4
267-278	Enantiospecific Synthesis of 5′-Noraristeromycin and its 7-Deaza Derivative and A Formal Synthesis of (-)-5′-Homoaristeromycin	Suhaib M. Siddiqi; Xing Chen; Stewart W. Schneller
279-294	Studies Towards the Synthesis of the Saturated and Unsaturated Carbocyclic Methylene Phosphonate Analogs of Dideoxyadenosine	D. Wolff-Kugel; S. Halazy
295-304	Synthesis of 5′-Substituted Derivatives of the Pyrrolo[2,3-d]-Pyrimidine Nucleoside Sangivamycin and Their Effect on Protein Kinase A and C Activity	Moheshwar Sharma; Hanna Wikiel; Rosemary Hromchak; Alexander Bloch; Miroslav Bobek
305-321	Synthesis of Uridylyl (3′-5′) Uridine Derivatives Containing 5-(Methylamino-Methyl) Uridine as A Modified Nucleoside Found from E. COLI Minor tRNA^Arg	Mitsuo Sekine; Kouji Seio; Takahiko Satoh; Kensaku Sakamoto; Shigeyuki Yokoyama
323-329	Photo-Induced P-Methylbenzylation of 1,3-Dimethylthymine and 1, 3-Dimethyluracil in the Presence of Trifluoroacetic Acid	Koh-ichi Seki; Kazue Ohkura
331-350	Synthesis of Glucuronides of Fluoropyrimidine Drugs: N- and O-Glucuronides of 5-Fluorocytosine and 5-Fluorouracil	N. Chouini-Lalanne; J. P. Vialaneix; S. Mansouri; M. C. Malet-Martino; R. Martino
351-358	Automated Synthesis of Cyclic Oligodeoxyribonucleotides via Phosphoramidite Method	M. R. Conte; L. Mayol; D. Montesarchio; G. Piccialli; C. Santacroce
359-368	A New Facile Synthesis and Antiviral Activity of Oxazofurin	P. Franchetti; L. Messini; L. Cappellacci; M. Grifantini; P. Guarracino; M. E. Marongiu; G. Piras; P. La Colla
369-380	Synthesis and Anti-HIV-1 Activity of Base Modified Analogues of 3′-Azido-2′,3′-Dideoxythymidine (AZT)	S. Czernecki; T. Le Diguarher; J. M. Valéry
381-401	Synthesis of Oligodeoxynucleotides Containing the C-Nucleoside and 2′- Deoxy-2′-Fluoro-ara-Nucleoside Moieties by the H-Phosphonate Method.^1,2	Ivan Rosenberg; Jaume Farras Soler; Zdenek Tocik; Wu-Yon Ren; Lech A. Ciszewski; Pavol Kois; Krzysztof W. Pankiewicz; Maria Spassova; Kyoichi A. Watanabe
403-416	Synthesis of Several 2′-Deoxy-3-Alkyl(ARYL)-3-Deazaguanosines: Mild Alkylation of a Cyanomethyl Imidazole with Electrophiles	Oscar L. Acevedo; Robert S. Andrews; P. Dan Cook
417-422	Synthesis of 2-Chloro-2′-Deoxyadenosine by Microbiological Transglycosylation	I. A. Mikhailopulo; A. I. Zinchenko; Z. Kazimierczuk; V. N. Barai; S. B. Bokut; E. N. Kalinichenko
423	Erratum

Volume 12, Issue 2 (1993)

a-b	Editorial board page for “Nucleosides & Nucleotides”, Volume 12, Number 2
115-123	Improved Synthesis of (E)-2′-Deoxy-2′-(fluoromethylene)cytidine - A Potent Inhibitor Of Ribonucleotide Diphosphate Reductase	Donald P. Matthews; Rose A. Persichetti; Jeffrey S. Sabol; Kenneth T. Stewart; James R. McCarthy
125-137	Nucleosides LII¹, Synthesis and Properties of Quinazoline-3′-azidonucleosides	Martin Dunkel; Wolfgang Pfleiderer
139-147	A Facile Synthesis of 4′-Thio-2′-deoxypyrimidine Nucleosides and Preliminary Studies on Their Properties	Baoguo Huang; Yongzheng Hui
149-155	A Short Synthesis of 2′,3′-Didehydro-3′-deoxythymidine	Nicholas D. P. Cosford; Raymond F. Schinazi
157-162	New Phosphonate Analogues of 3′-Thia-2′,3′-dideoxycytidine(BCH-189) Synthesis and Anti-HIV Evaluation	Jean-Louis Kraus
163-173	Studies with 2-(Butyldiphenylsiloxymethyl)-benzoyl Protected Oligodeoxyribonucleotides	M. Jonathan Rudolph; Ching-Hsuan Tung; Yon Ebright; Ziping Wei; Stanley Stein
175-183	Reaction of Epichlorohydrin with Adenosine and Uridine- 5′-monophosphates	Khurshid Alam Khan; Kaniz Fizza
185-198	S-Adenosyl-L-homocysteine Hydrolase Inhibitors as Anti-Viral Agents: 5′-Deoxyaristeromycin	Suhaib M. Siddiqi; Stewart W. Schneller; Satoru Ikeda; Robert Snoeck; Graciela Andrei; Jan Balzarini; Erik De Clercq
199-213	Synthesis of C-1′-Branched Acyclic Nucleosides	James A. Linn; James L. Kelley
215-224	Imidazole Nucleosides IV Nucleosides of 5 (4)-Formamido-imidazole-4 (5)carboxamide	Hans Guglielmi; Klaus Albert
225-236	The Resolution and Absolute Stereochemistry of the Enantiomers of cis-1-[2-(Hydroxymethyl)-1,3-oxathiolan-5-yl)cytosine (BCH189): Equipotent Anti-HIV Agents	Richard Storer; Ian R. Clemens; Brian Lamont; Stewart A. Noble; Christopher Williamson; Bernard Belleau
237-243	Triple Helix Binding of Oligodeoxyribonucleotides Containing 8-Oxo-2′-deoxyadenosine	Edwin C. Davison; Kai Johnsson
245-261	High-Yield Regioselective Thiation of Biologically Important Pyrimidinones, Dihydropyrimidinones and Their Ribo, 2′-Deoxyribo and 2′, 3′-Dideoxyribo Nucleosides	Krzysztof Felczak; Maria Bretner; Tadeusz Kulikowski; David Shugar
263	Erratum

Volume 12, Issue 1 (1993)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 12, Number 1
1-20	Synthesis and Biological Activity of Novel 2-Thio Derivatives of ATP	J. Zimmet; L. Järlebark; T. Hammarberg; P. J. M. Van Galen; K. A. Jacobson; E. Heilbronn
21-30	PEG-Supported Synthesis of Cyclic Oligodeoxyribonucleotides	L. De Napoli; A. Messere; D. Montesarchio; G. Piccialli; C. Santacroce; G. M. Bonora
31-37	Effects of Polyamines on the Binding of Hoechst 33258 to Calf Thymus DNA	Ronald D. Snyder
39-53	Synthesis of 1, 7-Dideazapurine Ribonucleosides and Deoxyribonucleosides	G. Cristalli; S. Vittori; A. Eleuteri; R. Volpini; D. Cola; E. Camaioni; P. V. Gariboldi; G. Lupidi
55-71	Novel Types of N⁶,2′-Cyclonucleosides	Jean M. J. Tronchet; Rachid Benhamza; Gérald Bernardinelli
73-82	Synthesis of 2′-Deuterio Tubercidin and Adenosine and the Corresponding Arabino Analogs	Michael E. Perlman
83-93	Acyclic 2′, 3′-Dideoxy-2′,3′-didehydronucleoside 5′-Triphosphates as Termination Substrates of Broad Set of DNA Polymerases	Alexander A. Krayevsky; Ljubov S. Victorova; Dmitrii Ju. Mozzherin; Marina K. Kukhanova
95-106	Chain Cleavage During Deprotection of RNA Synthesized by the 2′-O-Trialkylsilyl Protection Strategy	Matthew H. Lyttle
107-114	Synthesis of Acyclic Nucleoside Analogs Related to Barbituric Acid	J. Visscher; Alan W. Schwartz

Volume 11, Issue 10 (1992)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 11, Number 10
1683-1694	RNA Modified Uridines VI: Conformations of 3-[3-(S)-Amino-3-Carboxypropyl]Uridine (acp³U) from tRNA and 1-Methyl-3-[3-(S)-Amino-3-Carboxypropyl]Pseudouridine (m¹acp³Ψ) from rRNA	Wanda S. Smith; Barbara Nawrot; Andrzej Malkiewicz; Paul F. Agris
1695-1701	Modified Nucleosides. II.¹ Economical Synthesis of 2′,3′-Dideoxycytidine	Sebastian M. Marcuccio; Bryan C. Elmes; George Holan; E. John Middleton
1703-1711	A New Method of Synthesis of Fluorescently Labelled Oligonucleotides and Their Application in DNA Sequencing	Wojciech T. Markiewicz; Gabriele Gröger; Rudi Rösch; Anna Zebrowska; Hartmut Seliger
1713-1730	Syntheses and Properties of Dansylated Deoxycytidine 3′,5′-Bisphosphate Derivatives Useful for 3′-Labeling of Oligoribonucleotides	Mitsuo Sekine; Hiroshi Kusuoku
1731-1738	Synthesis of Thymidine Derivatives 3′-Modified with a Polar Three-Atom Group as Potential Anti-HIV-1 Agents	Kosaku Hirota; Hiroshi Hosono; Yukio Kitade; Yoshifumi Maki; Chung K. Chu; Raymond F. Schinazi; Osamu Muraoka
1739-1747	Synthesis of Some Purine Carbocyclic Isosteres of 2′,3′-Dideoxy-3′-C-Hydroxymethyl Nucleosides as Potential Inhibitors of HIV	Marianne Janson; Lars Svansson; Stefan C. T. Svensson; Ingemar Kvarnström; Björn Classon; Bertil Samuelsson
1749-1763	Aminolysis of 2′-Deoxyinosine Aryl Ethers: Nucleoside Model Studies for the Synthesis of Functionally Tethered Oligonucleotides	Ann E. Ferentz; Gregory L. Verdine
1765-1779	Synthesis of 1,3-Dl-O-Acetyl-5-O-Benzoyl-2-O -(O-Carboran-1-Ylmethyl)- D-Ribofuranose. A General Precursor for the Preparation of Carborane-Containing Nucleosides for Boron Neutron Capture Therapy	Werner Tjarks; Abul K. M. Anisuzzaman; Albert H. Soloway
1781-1793	Inhibition of Cytidine Deaminase by Derivatives of 1-(β-D-Ribofuranosyl)-Dihydropyrimidin-2-One (Zebularine)	Joseph J. Barchi Jr; Alberto Haces; Victor E. Marquez; John J. McCormack

Volume 11, Issue 9 (1992)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 11, Number 9
1575-1578	A Rapid Method for Purification of Oligonucleotides	Ajay Kumar; Hema Dawar; Sudhakar Mathur
1579-1593	Synthesis of Oligoribonucleotides by the H-Phosphonate Approach Using Base Labile 2′-O-Protecting Groups. V. Recent Progress in Development of the Method	Eriks Rozners; Regina Renhofa; Marina Petrova; Juris Popelis; Viktors Kumpins; Erika Bizdena
1595-1606	Synthesis and Antiviral Properties of New Cycloalkanol Derivatives of Guanine	S. Halazy; M. Kenny; J. Dulworth; A. Eggenspiller
1607-1620	1′, 2′-Seco-2′,3′-Dideoxynucleoside Analogues: Synthesis and Antiviral Evaluation of Racemic Trans-[1′, 5′-Dihydroxy 3′, 4′-methylenylpent-2′-oxy)methyl] Nucleosides	Muhammad Azymah; Claude Chavis; Alain Fruchier; Marc Lucas; Jean-Louis Imbach
1621-1638	The First Stereocontrolled Synthesis of Thiooligoribonucleotide: (RpRp)- and (SpSp)-U_psU_psU	Zbigniew J. Lesnikowski
1639-1649	A Dihydropyridine Carrier System for Delivery of 2′,3′-Dideoxycytidine (DDC) to the Brain	Eduardo Palomino; David Kessel; Jerome P. Horwitz
1651-1660	Synthesis of Thymine Nucleosides Derived from 1-Deoxy-D-psicofuranose	Véronique Faivre-Buet; Annie Grouiller; Gérard Descotes
1661-1666	Structural Determination of Silicon-Containing Oligonucleotides by ¹H^-29Si Long-Range Heteronuclear Multiple Quantum Correlation NMR Spectroscopy	James M. Hewitt; William C. Lenhart; Richard N. Moore; Ashis K. Saha; Alexander L. Weis
1667-1671	Synthesis of an Octameric Phosphodiester of 2, 3-dideoxy-ß-D-erythro-hex-2-eno-pyranosyl-thymine and Its Interactions with Poly-rA and Poly-dA	Eduard Felder; Raphael Gattlen; Flavio Ossola; Gerhard Baschang
1673-1682	Condensation Reaction Between 2,2-Diphenylthio-2,3-Dideoxyribose and Silylated Pyrimidine Bases	Hiroshi Kawakami; Takashi Ebata; Koshi Koseki; Katsuya Matsumoto; Koji Okano; Hajime Matsushita

Volume 11, Issue 8 (1992)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 11, Number 8
1445-1453	Oligonucleotides and Nucleotide-Peptides. LIV. The Synthesis and Hydrolytic Properties of Adenylyl-(5′→N_ε)-lysylpeptides — Model Compounds of the AMP-RNA Ligase Covalent Complex	Benediktas Juodka; Sofija Sasnauskiene; Ruta Petniunaite
1455-1461	RNA Modified Uridines. V. An Improved Synthesis of 3-[3-(S)-Amino-3-carboxypropyl]uridine (acp³U) and Its 5′-Phosphate	Barbara Nawrot; Andrzej Malkiewicz
1463-1466	An Efficient Synthesis of N²-Isobutyryl-O⁶-[2-(4-nitrophenyl)ethyl]-5′-O-Dimethoxytrityl-2′-deoxyguanosine	Andrey P. Guzaev
1467-1479	Efficient Synthesis of 4-Thio-D-ribofuranose and Some 4′-Thioribonucleosides	L. Bellon; J. -L. Barascut; J. -L. Imbach
1481-1488	Synthesis of Tetrazole Oxathiolane Nucleoside Analogues and Their Evaluation as HIV-1 Antiviral Agents	Philippe Faury; Michel Camplo; Anne-Sophie Charvet; Jean-Claude Chermann; Jean-Louis Kraus
1489-1505	Synthesis of Racemic Carboacyclonucleosides Derived from Butane-1, 4-Diol and Hexane-1, 6-Diol	Michel Perbost; Marc Lucas; Claude Chavis; Jean-Louis Imbach
1507-1527	Synthesis, Antiproliferative, and Antiviral Evaluation of Certain Acyclic 6-Substituted Pyrrolo[2,3-D]-pyrimidine Nucleoside Analogs Related to Sangivamycin and Toyocamycin	Eric E. Swayze; William M. Shannon; Robert W. Buckheit; Linda L. Wotring; John C. Drach; Leroy B. Townsend
1529-1537	An Expeditious Synthesis of Homochiral (R) 2-(9-Purinyl)butane-1, 4-Diols from (S) Butane-1, 2, 4-Triol	Michel Perbost; Marc Lucas; Claude Chavis; Jean-Louis Imbach
1539-1547	Synthesis of Nucleoside Analogues Containing an Oxetane Ring Fused to the Furan Ring	Robert J. Hambalek; George Just
1549-1559	A Practical and Stereospecific Approach to the Synthesis of 3′-Deoxy-2′,3′-didehydrothymidine (D₄T)	Chandra Vargeese; Elie Abushanab
1561-1574	Straightforward Synthesis of 6-Thiodeoxyguanosine and Its Incorporation into Oligodeoxynucleotides	Timothy R. Waters; Bernard A. Connolly

Volume 11, Issue 7 (1992)

a-b	Editorial board page for “Nucleosides & Nucleotides”, Volume 11, Number 7
1297-1303	Synthesis of an Acyclic Analogue of Azidothymidine	G. J. Koomen; L. M. Provoost; D. A. H. van Maarschalkerwaart; N. P. Willard
1305-1324	Time-of-Flight Secondary Ion Mass Spectrometry of Isomeric O-Alkylthymidines	Francois Lafortune; Garry W. Buchko; Frank E. Hruska; Krishan L. Sadana; Kenneth G. Standing; John B. Westmore
1325-1332	A Potential Suicide Inhibitor of Adenylosuccinate Lyase	W. A. Hartgers; R. F. de Boer; M. J. Wanner; G. J. Koomen
1333-1351	Synthesis of Suitably-Protected Phosphoramidites of 2′-Fluoro-2′-Deoxyguanosine and 2′-Amino-2′-Deoxyguanosine for Incorporation Into Oligoribonucleotides	Fritz Benseler; David M. Williams; Fritz Eckstein
1353-1366	Synthesis of Some 2′,3′-Dideoxy-3′-C-Fluoromethyl and 3′-C-Azidomethyl Nucleosides	Lars Svansson; Ingemar Kvarnström; Björn Classon; Bertil Samuelsson
1367-1370	Synthesis of 2′,3′-Dideoxy-3′-C-Hydroxymethyl Nucleosides Having the L-Configuration as Potential Inhibitors of HIV	Ingemar Kvarnström; Lars Svansson; Carina Svensson; Stefan; C. T. Svensson; Björn Classon; Bertil Samuelsson
1371-1381	Chiral 1′, 2′-Seco-Nucleosides: Synthesis of D and L-Threitol-2′-O-Methylenyl Nucleosides	Muhammad Azymah; Claude Chavis; Marc Lucas; Jean-Louis Imbach
1383-1391	Synthesis and Activities of the Phosphonate Isostere of the Monophosphate of (±)Cyclobut-G	Daniel W. Norbeck; Hing L. Sham; William Rosenbrook; Thomas Herrin; Jacob J. Plattner
1393-1409	9-(2-Deoxy-ß-D-xylofuranosyl)adenine and 1-(2-Deoxy-ß-D-xylofuranosyl)thymine: Phosphorylation and Stability	Marcela Krecmerova; Frank Seela
1411-1424	Synthesis of 1′-Deoxypsicofuranosyl-deoxynucleosides as Potential Anti-HIV Agents	Véronique Faivre-Buet; Annie Grouiller; Gérard Descotes
1425-1442	The Synthesis of 5-Substituted-2, 4-dimethoxypyrimidines and Some Related Nucleoside Analogues	R. F. Whale; P. L. Coe; R. T. Walker

Volume 11, Issue 6 (1992)

a-b	Editorial board page for “Nucleosides & Nucleotides”, Volume 11, Number 6
1123-1135	Synthesis and Biological Study of the Cyclopentenyl Carbocyclic Nucleoside Analogue of 5-Azacytidine	Benjamin B. Lim; Victor E. Marquez; Kathryn A. Dobyns; David A. Cooney; Erik De Clercq
1137-1149	The Synthesis of Novel Regioisomeric Ring-Expanded Xanthine Nucleosides Containing The 5:7-Fused Imidazo[4,5-e][1,2,4]Triazepine Ring System	Vishweshwar S. Bhadti; Anila Bhan; Ramachandra S. Hosmane; Martin Hulce
1151-1173	Synthesis and Antiviral Activity of Various 5-Substituted 2′-Deoxyuridines and -Cytidines	Dan Peters; Anna-Britta Hörnfeldt; Salo Gronowitz; Nils Gunnar Johansson
1175-1200	The Synthesis, Structure, and Conformation of 2′-Deoxy Analogues of „Fat“ Xanthine Nucleosides, Containing the Imidazo[4,5-e][1,4]Diazepine Ring System	Anila Bhan; Ramachandra S. Hosmane
1201-1204	A Convenient Preparation of Protected 2′-0-Methylguanosine	Thomas E. Leonard; Purshotam Bhan; Paul S. Miller
1205-1218	Synthesis of Some 2′,3′-Dideoxy-2′-C-Methyl-Substituted Nucleosides	Panagiotis Ioannidis; Björn Classon; Bertil Samuelsson; Ingemar Kvarnström
1219-1228	Synthesis and Anti-Hiv Activity of 3′-0-Formyl Derivatives of Thymidine and 2′-Deoxyuridine	Rakesh Kumar; Edward E. Knaus; Leonard I. Wiebe
1229-1239	The Crystal and Molecular Structure of the Complex of 2′3′-Didehydro-2′3′-Dideoxyguanosine with Pyridine	Patrick Van Roey; C. K. Chu
1241-1255	Isotactic Glycero Oligothymidylate. a Convenient Preparation of (R) and (S) 1′, 2′-Seco 2′-Nor Thymidine	Muhammad Azymah; Claude Chavis; Marc Lucas; François Morvan; Jean-Louis Imbach
1257-1261	N²-Isobutyryl-O⁶-[2-(p-Nitrophenyl)Ethyl]Guanine: A New Building Block for the Efficient Synthesis of Carbocyclic Guanosine Analogs	Thomas F. Jenny; K. Christian Schneider; Steven A. Benner
1263-1273	Regioselective 2′/3′-O-Allylation of Pyrimidine Ribonucleosides Using Phase Transfer Catalysis	Vidhya Gopalakrishnan; Vaijayanti Kumar; K. N. Ganesh
1275-1292	The Identification of 5′-Deoxy-5′-Methylthioguanosine in Human Urine by Gas Chromatography/Mass Spectrometry	William M. Hammargren; Debra R. Luffer; Karl H. Schram; Mark L. J. Reimer; Katsuyuki Nakano; Toshio Yasaka; Allan R. Moorman

Volume 11, Issue 5 (1992)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 11, Number 5
961-983	The Chemistry of 2′-Deoxyribo-C-Nucleosides	Lars J. S. Knutsen
985-998	Straightforward Synthesis of 6-Thiodeoxyguanosine and Its Incorporation into Oligodeoxynucleotides	Timothy R. Waters; Bernard A. Connolly
999-1002	A Simple Method for Introducing -SH/COOH Group at 5′-OH end of Oligonucleotide	Ajay Kumar; Sonia Advani
1003-1007	A Simple Method for Introducing -SH Group at 5′OH Terminus of Oligonucleotide	Ajay Kumar; Sonal Malhotra
1009-1038	Synthesis and Biological Activities of Unsaturated Ketohexopyranosyl Nucleosides of Pyrimidines	Arun P. Sharma; Abraham P. Ollapally; Willishea Jones; Tracey Lemon
1039-1046	Solvent Dependent Changes in the Proton NMR Spectra of 2′-Deoxyadenosine and Its Derivatives	Mahesh K. Lakshman; Roland E. Lehr
1047-1057	Crystal Structure of Sodium Deoxyinosine Monophosphate	R. Krishnan; T. P. Seshadri
1059-1076	8-Aza Analogues of Deaza Purine Nucleosides. Synthesis and Biological Evaluation of 8-Aza-1-deazaadenosine and 2′-Deoxy-8-aza-1-deazaadenosine	Palmarisa Franchetti; Loredana Cappellacci; Mario Grifantini; Giulio Lupidi; Giuseppe Nocentini; Anna Barzi
1077-1088	Synthesis of a Potent A₁ Selective Adenosine Agonist: N⁶-[1-R-[(3-Chloro-2-thienyl)methyl]propyl]adenosine, RG 14718(-)	Cynthia A. Fink; Alfred P. Spada; Dennis Colussi; Luz Rivera; Linda Merkel
1089-1101	Influence of Acetyl and Bromine Substitutions on Stacking. Crystal and Molecular Structures of 8-Bromo 2′,3′,5′-Triacetyl Adenosine and 8-Bromo 2′,3′,5′-Triacetyl Guanosine	Sharmila S. Mande; H. N. Lalitha; S. Ramakumar; M. A. Viswamitra
1103-1114	Conformational Variability in Modified Nucleosides. Crystal and Molecular Structure of 2′,3′-O-Isopropylidene Inosine	Sharmila S. Mande; N. Shamala; T. P. Seshadri; M. A. Viswamitra
1115-1121	Expeditious and Stereoselective Synthesis of α-Guanosine	Allen B. Reitz; Mary C. Rebarchak

Volume 11, Issue 2-4 (1992)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 11, Number 2-4
xiii	Memorial Issue Honoring Prof. Tohru Ueda
xv-xxvii	Biography
177-196	5′-Hydrogenphosphonates and 5′-Methylphosphonates of Sugar Modified Pyrimidine Nucleosides as Potential Anti-HIV-1 Agents.¹	Alexander A. Krayevsky; Natalie B. Tarussova; Qing-Yu Zhu; Pedro Vidal; Ting-Chao Chou; Penny Baron; Bruce Polsky; Xiang-Jun Jiang; Jasenka Matulič-Adamič; Ivan Rosenberg; Kyoichi A. Watanabe
197-226	Nucleosides and Nucleotides. 104. Radical and Palladium-Catalyzed Deoxygenation of the Allylic Alcohol Systems in the Sugar Moiety of Pyrimidine Nucleosides^§,1
227-235	Nucleosides and Nucleotides. 105. DNA Bending in d(A)₄ - d(T)₄ TRACTS Containing 3-Deazaadenine or 7-Deazaadenine Substituted for Adenine^§,1	Akira Ono; Chie Ohdoi; Akira Matsuda; Tohru Ueda
237-246	Nucleosides and Nucleotides. 106. Synthesis and Biological Activity of 1-(2-Deoxy-2-hydroxyimino- or Methoxyimino-β-D-erythro-pentofuranosyl)-thymine and -Cytosine^§,1
247-260	Mutation Induced by Deoxyxanthosine in Codon 12 of A Synthetic c-Ha-ras Gene	Hiroyuki Kamiya; Miho Shimizu; Masayuki Suzuki; Hideo Inoue; Eiko Ohtsuka
261-272	NMR Studies of a DNA Containing 8-Methoxydeoxyguanosine	Yasushi Oda; Seiichi Uesugi; Masaya Orita; Hideo Inoue; Yasutoshi Kawase; Eiko Ohtsuka; Morio Ikeharay
273-278	Formation of an Unexpected 2-Deoxy-α-D-Threo-Pentofuranosyl Azide by Reaction of O²,3′-Anhydro-5′-O-trityl-2′-deoxycytidine with Lithium Azide	I. A. Mikhailopulo; G. V. Zaitseva; E. V. Vaaks; H. Rosemeyer; F. Seela
279-293	The Synthesis of Novel Carbohydrates Amenable to the Synthesis of 2′,3′-Dideoxy-3′-Branched Nucleosides	Jeffrey S. Pudlo; Leroy B. Townsend
295-310	Synthesis and Biological Action of a New Cyclic AMP Analogue	Toshiaki Fujihashi; Takahiro Ogata; Tetsuo Ohkuma; Tohru Endo; Akira Kaji
311-317	Quantification Analysis of Human α- and δ-Globin Genes. Mutations in 5′-Splice Junction Sequence and α- and δ- Thalassemias	Yôichi Iida
319-328	Synthesis of 6-Methyluridine via Palladium-Catalyzed Cross-Coupling Between A 6-Iodouridine Derivative and Tetramethylstannane	Hiromichi Tanaka; Hiroyuki Hayakawa; Sachiko Shibata; Kazuhiro Haraguchi; Tadashi Miyasaka; Kosaku Hirota
329-340	Synthesis of 2′,3′-Dideoxy-2′-methylene Pyrimidine Nucleosides as Potential Anti-Human Immunodeficiency Virus (HIV) Agents	Tai-Shun Lin; Mei-Zhen Luo; Mao-Chin Liu
341-349	A Convenient and Stereoselective Synthesis of 2′-Deoxy-β-L-Ribonucleosides	Shizuyoshi Fujimori; Naoko Iwanami; Yuichi Hashimoto; Koichi Shudo
351-363	The Controlled Stereospecific Reduction of Cyclopentenyl Cytosine (CPE-C) to Carbodine and Isocarbodine	Pamela L. Russ; Lajos Hegedus; James A. Kelley; Joseph J. Barchi Jr.; Victor E. Marquez
365-372	Oxidative Cyclization of 2′,3′-O-Isopropylidene-Adenosines into 5′-O,8-Cycloadenosines with Lead Tetraacetate: Remarkable Effect of N⁶-Substituents on the Oxidation	Yukio Kitade; Tohru Makino; Kosaku Hirota; Yoshifumi Maki
373-382	Synthetic Nucleosides and Nucleotides. XXX.¹ Synthesis and Antiviral Activity of 3′-Azido, 2′,3′-Unsaturated and 2′,3′-Dideoxy Derivatives of E-5-Styryl-2′-Deoxyuridine on Human Immunodeficiency Virus	Toyofumi Yamaguchi; Mineo Saneyoshi

Volume 11, Issue 2-4 (1992)

383-390	Enhanced Fluorescence in the Binding of Oligonucleotides With a Pyrene Group in the Sugar Fragment to Complementary Polynucleotides	Kazushige Yamana; Tadao Gokota; Hiroaki Ozaki; Hidehiko Nakano; Osamu Sangen; Takeo Shimidzu
391-400	A Novel Method for the Synthesis of ddA and F-ddA Via Regioselective 2′-O-Deacetylation of 9-(2,5-DI-O-Acetyl-3-bromo-3-deoxy-β-D-xylofuranosyl)adenine	Hiroshi Shiragami; Yasuhiro Tanaka; Yumiko Uchida; Hisao Iwagami; Kunisuke Izawa; Toshihide Yukawa
401-416	Synthesis of Novel Fluorinated 2′,3′-Dideoxynucleosides	P. Kumar; L. I. Wiebe
417-436	Oxetanocin—Oxetanose Chemistry: Lewis Acid Promoted Glycosidations of the D-Erythrooxetanose Derivatives	Shigeru Nishiyama; Tadaaki Ohgiya; Shosuke Yamamura; Kuniki Kato; Tomohisa Takita
437-446	New Neplanocin Analogues II. Enzymatic One-Step Synthesis and Antitumor Activity of 6′-(3-sn-Phosphatidyl)Neplanocin a Derivatives	Satoshi Shuto; Hiromichi Ito; Takumi Obara; Keiji Nakagami; Masao Yaso; Satoshi Yaginuma; Masatoshi Tsujino; Tetsu Saito; Akira Matsuda; Tohru Ueda
447-456	Synthesis of Some Analogues Of 1-[(2-Hydroxyethoxy)-methyl]-6-(phenylthio) Thymine (HEPT) which have Different types of Acyclic Structures	Hiromichi Tanaka; Tadashi Miyasaka; Kouichi Sekiya; Hideaki Takashima; Masaru Ubasawa; Issei Nitta; Masanori Baba; R. T. Walker; E. De Clercq
457-471	Synthesis of 2,2′-Anhydro-1 - (3′ -deoxy -3′ -iodo-β-D-arabino-furanosyl) thymine and Its Derivatives as Versatile Synthetic Intermediates	Katsumaro Minamoto; Yuji Hamano; Yoji Matsuoka; Kenji Watanabe; Toyohiko Hirota; Shoji Eguchi
473-482	Chiral Phosphoromorpholidate Derivatives of Oligothymidylate and Their Hybridization Abilities	Masanori Kitamura; Hiroaki Ozaki; Kazushige Yamana; Takeo Shimidzu
483-493	Pummerer Rearrangement of Selenium-Containing Uracil Nucleosides	Kazuhiro Haraguchi; Shigeru Saito; Hiromichi Tanaka; Tadashi Miyasaka
495-513	Synthesis and Antitumor Activity of Acyl and Benzyl Types of Prodrugs of 2′-Deoxy-2′-methylidenecytidine	Takanori Miyashita; Noriyuki Ashida; Kazuhiko Kondoh; Shinji Sakata; Haruhiko Machida; Akihiro Fujii; Tohru Ueda; Akira Matsuda
515-520	Melting Behavior and Stability of (dA)₈·(dT)₈ Double Helix	Naoki Sugimoto; Muneo Sasaki
521-527	Acid-Catalyzed Photosubstitution of 5-Fluoro-1,3-Dimethyluracil with Substituted Benzenes	Koh-ichi Seki; Kazue Ohkura
529-549	Carbocyclic Purine Nucleosides Derived from Aristeromycin Through Two Key Intermediates, Carbocyclic 5-Amino-4-Imidazolecarboxamide Riboside and 2′-Deoxyriboside	Yoshio Taniyama; Tsunehiko Fukuda; Ryuji Marumoto
551-569	Synthesis of Fused Cyclopropane-Containing Nucleosides by [1,2]-Hydride Shift Rearrangements and B-Elimination Reactions of Sulfonylated Ribonucleosides	Masajiro Kawana; Hiroyoshi Kuzuhara
571-582	Synthesis of 6-Sulfur Analogues of Oxanosine and Closely Related Derivatives Thereof	Sumiko Hara; Chisato Kaneko; Hiroatsu Matsumoto; Takeshi Nishino; Tadao Takeuchi; Takeo Mori; Yoshihisa Mizuno; Kazuyoshi Ikeda
583-594	The Synthesis and Biological Properties of some Aryl bis(Nucleosid-5′-yl) Phosphates Using Nucleosides with Proven Anti-HIV Activity	S. I. Shimizu; J. Balzarini; E. De Clercq; R. T. Walker
595-602	The Synthesis and Antiviral Activity of (E)-5-(2-Nitrovinyl)uridine and (E)-5-(2-Nitrovinyl)-2′-deoxyuridine	R. F. Whale; V. Bou; P. L. Coe; R. T. Walker
603-613	A Stereospecific Synthesis of Pyrimidine β-D-2′-Deoxyribonucleosides	Hussein I. El Subbagh; Li-Jen Ping; Elie Abushanab
615-635	Synthesis and Conformational Studies of O^5′, 6-Methanouridine—A New Type of Pyrimidine Cyclonucleoside	Brian A. Otter; Shirish A. Patil; Marianne R. Spada; Linda A. Jelicks; Yuichi Yoshimura; Akira Matsuda; Robert S. Klein
637-668	Partial Protection of Carbohydrate Derivatives. Part 27.¹ Further Improvement in the Protecting Procedure for Oligonucleotide Synthesis in Terms of a Cellulose Acetate Derivative as a Polymer-Support	Kazuo Kamaike; Tomohiro Ogawa; Yasushi Inoue; Yoshiharu Ishido

Volume 11, Issue 2-4 (1992)

669-678	Synthesis of Oligodeoxyribonucleotide Analogues by Use of Deoxyribonucleoside-3′-yl O-bis(1,1,1,3,3,3-Hexafluoro-2-Propyl) Phosphites as New Key Intermediates	Hideo Hosaka; Yoshikazu Suzuki; Hiroyuki Nakamura; Hidenori Funakoshi; Hideki Nakashima; Naoki Yamamoto; Hiroshi Takaku
679-691	Synthesis of Adenosine, Guanosine and Cytidine Monomer Building Units Bearing the [[2-(Methylthio)-phenyl]thio]methyl (MPTM) Group as The 2′-Hydroxyl Protecting Group	Mitsuo Sekine; Takashi Nakanishi
693-705	Practical Synthesis of AZT and AZDU from Xylose: Efficient Deoxygenation via Nucleoside 2′-Xanthates	Yaoquan Chen; John G. Bauman; Chung K. Chu
707-718	Synthesis and Biological Evaluation of 9-(f-2, c-3-Bishydroxymethyl-r-cyclopropylmethyl)-9H-adenine (A Lower Methylene Homolog of Carbocyclic Oxetanocin) and Related Compounds	Nobuya Katagiri; Hiroshi Sato; Chikara Kaneko
719-730	Recognition of the Nucleoside in the First Position of the Anticodon of Isoleucine tRNA by Isoleucyl-tRNA Synthetase from Escherichia Coli	Tomonari Muramatsu; Tatsuo Miyazawa; Shigeyuki Yokoyama
731-738	Conformation Analysis of Two Anti-HIV Nucleoside Analogues 2′,3′-Dideoxy-3′-fluorocytidine and Its N⁴-Dimethylaminomethylene Prodrug Derivative	Vivian Cody; Thomas I. Kalman
739-748	Synthesis of 1′,2′-Seco-nucleoside Analogues of AZT	Purushotham Vemishetti; Hussein I. El Subbagh; Elie Abushanab; Raymond P. Panzica
749-757	O-Alkylation of Dialkyl Phosphates and O-Alkyl Phosphonates via the Stannyl Intermediates	Shokichi Ohuchi; Takashi Imada; Tsujiaki Hata
759-771	Conformational Rigidity of N⁴-Acetyl-2′-O-methylcytidine Found in tRNA of Extremely Thermophilic Archaebacteria (Archaea)	Gota Kawai; Takeshi Hashizume; Masayuki Yasuda; Tatsuo Miyazawa; James A. McCloskey; Shigeyuki Yokoyama
773-785	Divalent Metal Ion-Catalyzed Pyrophosphate Bond Formation in Aqueous Solution. Synthesis of Nucleotides Containing Polyphosphate	H. Sawai; M. Shimazu; H. Wakai; H. Wakabayashi; K. Shinozuka
787-819	Nucleosides. IL. Synthesis and Properties of 2,4-Quinazolinedione N-1-2′ Deoxy-, 3′-Deoxy- and 2′,3′-Dideoxynucleosides	Martin Dunkel; Wolfgang Pfleiderer
821-834	Nucleic Acid Related Compounds. LXXXI. Efficient General Synthesis of Purine (Amino, Azido, and Triflate)-Sugar Nucleosides	Morris J. Robins; S. D. Hawrelak; Amelia E. Hernández; Stanislaw F. Wnuk
835-853	Molecular Conformation of 2′-Deoxy-2′-methylidene-cytidine: A Potent Antineoplastic Nucleoside	Yuriko Yamagat; Ken-ichi Tomita; Nobuhiro Marubayashi; Ikuhiko Ueda; Shinji Sakata; Akira Matsuda; Kenji Takenuki; Tohru Ueda
855-864	Synthesis of Methylenecyclobutyl- and Cyclobutenyl Adenine, Potent Antiviral Carbocyclic Analogues of Oxetanocin A	Tokumi Maruyama; Yasuaki Hanai; Yoshiko Sato
865-887	Studies on Griseolic Acid Derivatives X. Synthesis and Phosphodiesterase Inhibitory Activity of 2-Substituted Derivatives of Griseolic Acid	Masakatsu Kaneko; Misako Kimura; Yoshinobu Murofushi; Takashi Yasumoto; Yasuteru Iijima; Mitsuo Yamazaki
889-901	Spin-Labeled Oligonucleotides Site Specifically Labeled at the Internucleotide Linkage. Separation of Stereoisomeric Probes and EPR Spectroscopical Detection of Hybrid Formation in Solution	Shunji Nagahara; Akira Murakami; Keisuke Makino
903-945	Nucleoside Analogues as Chemotherapeutic Agents: A Review	C. Périgaud; G. Gosselin; J. L. Imbach
947-956	Syntheses of Phosphonate Analogues of Dideoxyadenosine (DDA)-, Dideoxycytidine (DDC)-, Dideoxyinosine (DDI)-, and Deoxythymidine (DDT)-5′-Monophosphates	John A. Secrist III; Robert M. Riggs; Robert N. Comber; John A. Montgomery

Volume 11, Issue 1 (1992)

a-b	Editorial board page for “Nucleosides & Nucleotides”, Volume 11, Number 1
1-9	Structural Features Of 2′,3′-Riboanhydroadenosine, A Conformationally Restricted Termination Substrate Of DNA Polymerases	Galina Gurskaya; Alexey Bochkarev; Alexander Zdanov; Alexander Papchikhin; Alexander Krayevsky
11-21	Synthesis and Anti-HIV Activity of a New Hexopyranoside Analogue of AZT	Ferenc Sztaricskai; Zoltán Dinya; Gyula Batta; Lajos Gergely; Béla Szabó
23-35	Utilization of 2′-Deoxy-6-thioguanosine 5′-Triphosphate In DNA Synthesis Catalyzed by DNA Polymerase I Klenow Fragment of Escherichia Coli	Yi-He Ling; J. Arly Nelson; David Farquhar; Kenneth L. Beattie
37-47	Reactions Of 2′-Deoxy-2′-halouridines and O²,2′-Cyclouridine with Lithium Dialkylamides: Formation of 1′,2′-Unsaturated Derivatives	Atsushi Kittaka; Hiromichi Tanaka; Tadashi Miyasaka; Kentaro Yamaguchi
49-60	Synthesis Of 6-Alkoxy-5-bromo-5,6-dihydropyrimidine Nucleosides Using Dibutyltin Alkoxide-Bromine	A. George Samuel; Hari Babu Mereyala; K. N. Ganesh
61-83	Synthesis of the Pyrido[4,3-D]pyrimidine Congeners of Inosine and of Adenosine - A New Class of 6:6 Bicyclic C-Ribofuranosides	Kambhampati V. B. Rao; Robert S. Klein; Mallela S. P. Sarma; Brian A. Otter
85-95	Synthesis of Protected 8-Substituted Deoxyribonucleosides and Its Helix Stability in Oligodeoxyribonucleotides Containing the Eco RI Recognition Site	Hiroshi Komatsu; Takashi Ichikawa; Michiaki Nakai; Hiroshi Takaku
97-119	Synthesis Of 9-(1-Deoxy-1-phosphono-β-D-psicofuranosyl)-1,9-dihydro-6H-purin-6-one as a Potential Transition State Analog Inhibitor of Purine Nucleoside Phosphorylase	Robert D. Elliott; Shri Niwas; James M. Riordan; John A. Montgomery; John A. Secrist III
121-139	Reaction of 5-αChloroacetyl-4-glycosylaminopyrimidines with Thiourea. Synthesis of 4-Glycosylaminofuro[2,3-d]pyrimidines and 4-Glycosylamino-5-(2-amino-4-thiazolyl)pyrimidines	M. L. Quijano; M. Nogueras; A. Sánchez
141-156	Stereoselective Synthesis of Ribonucleoside 3′,5′-Cyclic Methyl(phenyl)phosphonates and Phosphonothioates	H. C. P. F. Roelen; E. de Vroom; A. H. J. Wang; G. A. van der Marel; J. H. van Boom
159-166	Computer Graphics Modelling and Molecular Dynamics Simulation of the Core of the Self Splicing Intervening Sequence of the T4 NrdB mRNA in the Presence of the Guanosine Cofactor	Lenoart Nilsson; Agneta Ahgren-Stålhandske; Ann-Sofie Sjögren; Solveig Hahne; Britt-Marie Sjöberg
167-173	Free Energy Calculations Predict Sequence Specificity in DNA-Drug Complexes	T. Härd; L. Nilsson

Volume 10, Issue 8 (1991)

a	Editorial board page for “Nucleosides, Nucleotides & Nucleic Acids”, Volume 10, Number 8
1625-1640	Structure and Conformation of 5′-Chlorocyclocytidine, a Potent Inhibitor of Nucleic Acid Synthesis: X-Ray, ¹H and ¹³C NMR Analyses	George I. Birnbaum; Miloś Budéšínsk; Ladislav Novotn
1641-1655	Thiopurine Nucleosides: Variations in Hydrophobicity Among N^l Suhstituents	Peter C. Ratsep; Nrusingha C. Mishra; Arthur D. Broom
1657-1665	Synthesis of N-Aminopyrazinium Analogs of Cytidine and 2′-Deoxycytidine	Miroslav Bobek; Pittaya Tuntiwachwuttikul; M. Mohsen Ismail; Thomas J. Bardos
1667-1675	Covalent Nucleoside Adducts of Aspidosperma Alkaloids	B. Danieli; G. Lesma; G. Palmisano; D. Passarella; B. Pyuskyulev
1677-1692	Inhibition and Substrate Specificity of Adenosine Deaminase. Interaction with 2′-, 3′- and/or 5′-Substituted Adenine Nucleoside Derivatives	G. Maury; T. Daiboun; A. Elalaoui; C. Génu-Dellac; C. Périgaud; C. Bergogne; G. Gosselin; J. -L. Imbach
1693-1706	Synthesis of Ring-Expanded Xanthines and Xanthosines Containing the Imidazo[4,5-d][1,3]diazepine Ring System	Ramachandra S. Hosmane; Vijayvithal P. Vaidya; Mi Kyung Chung; Upali Siriwardane; Hongming Zhang; Narayan S. Hosmane
1707-1717	Synthetic Studies on the Isomeric N -Methyl Derivatives of C-Ribavirin	Giin-Yuan Shen; Roland K. Robins; Ganapathi R. Revankar
1719-1728	Synthesis of 4-Substituted Pyrimidine 2′,3′-Dideoxynucleosides	L. De Napoli; A. Messere; D. Montesarchio; G. Piccialli; C. Santacroce
1729-1742	Effect of 2-Amino Substitution on the Antiviral Effects of 5-Ethyl-2′-Deoxyuridine and (E)-5-(2-bromovinyl)-2′-Deoxyuridine and Their Incorporation into DNA	J. Sági; A. Szabolcs; K. Ebinger; L. Ötvös; J. Balzarini; E. De Clercq
1743-1757	Synthesis and Biological Properties of 2-Amino-3-fluoro-2,3-Dideoxy-D-Pentofuranosides of Natural Heterocyclic Bases	Igor A. Mikhailopulo; Grigorii G. Sivets; Tamara I. Pricota; Nicolai E. Poopeiko; Jan Balzarini; Erik De Clercq
1759-1769	Imidazole Ring Opening of 7-Methylguanosine at Physiological pH	G. Barbarella; V. Tugnoli; M. Zambianchi
1771-1787	Synthesis and Biological Evaluation of Some D-Xylofuranosyl-Pyridine C-Nudeosides	F. Verberckmoes; E. L. Esmans; R. A. Dommisse; J. A. Lepoivre; F. C. Alderweireldt; J. Balzarini; E. De Clercq

Volume 10, Issue 7 (1991)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 10, Number 7
1431-1449	Synthesis And Antiviral Evaluation Of 2′,3′-Secothymidine Analogs of ddT and AZT	Annie-Fransoise Maggio; Valerie Boyer; Anne-Marie Aubertin; Georges Obert; André Kirn; Jean-Louis Imbach
1451-1463	Synthesis and Biological Activity of 5-halo-2-Pyrimidinone 3′-Azido-2′,3′-Dideoxyribosides	S. M. N. Efange; A. K. Dutta
1465-1475	Phosphonoformate Esters of Anti-HIV Nucleosides: 3′-Azido-3′-deoxythymidine and 2′,3′-Dideoxycytidine Derivatives Containing a Small 5′-(0-Alkoxycarbon-ylphosphinyl) or 5′-(O-Cholesterylcarbonylphosphinyl) Substituent	Jayanta Saha; Ruth M. Ruprecht; Andre Rosowsky
1477-1483	A Direct and Efficient Synthesis of 5′-Deoxy-2′, 3′-	James G. Davidson; Phillip J. Fiore
1485-1498	Synthesis of a Non-Hydrolyzable Dinucleoside Analogue	Stephen H. Kawai; George Just
1499-1505	Strategy for Industrial Scale Production of Dideoxyinosine: Enzymatic Deamination of Dideoxyadenosine by Adenosine Deaminase	Carol M. Beach; Robert K. Evans; Mary Sue Coleman
1507-1524	N²-Substituted-2′-deoxyguanosine 5′-Triphosphates as Substrates for E. coli DNA Polymerase I	Stephen Freese; Jörg Hoheisel; Hans Lehrach; George Wright
1525-1549	Synthesis of 2′-Deoxy-2′ -Fluoro-D-Arabinopyranopyranosyl Nucleosides and Their 3′,4′-Seco analogues	P. Herdewijn; A. Van Aerschot; R. Busson; P. Claes; E. De Clercq
1551-1562	Synthesis and Evaluation of Anti-HIV-1 and Antitumor Activity of 2′,3′-didehydro-2′,3′-dideoxy-3-deazaadenosine, 2′,3′-dideoxy-3-Deazaadenosine and Some 2′,3′-dideoxy-3-deaza-adenosine 5′-dialkyl Phosphates¹	P. Franchetti; L. Cappellacci; G. Cristalli; M. Grifantini; A. Pani; P. La Colla; G. Nocentini
1563-1572	Coronary Vasoactivity of Novel N⁶-Substituted Adenosines	Shozo Kusachi; Robert D. Thompson; William J. Bugni; Nobuyuki Yamada; Ray A. Olsson
1573-1598	Synthesis and Biological Evaluation of 2-(2-Deoxy-D-erythro-pent-1-enofuranosyl)pyridine C-Nucleosides	E. De Vos; E. L. Esmans; J. A. Lepoivre; F. C. Alderweireldt; R. A. Dommisse; P. François; R. Touillaux; J. Balzarini; E. De Clercq
1599-1614	3′/5′-Regioselectivity of Introduction of the 9-Fluorenyl-Methoxycarbonyl Group to 2′-o-Tetrahydropyran-2-YL-and 2′-O-(4-Methoxytetrahydropyran-4-YL-)-Nucleosides: Useful Intermediates for Solid-Phase-Rna-Synthesis	Christian Lehmann; Yao-Zhong Xu; Chris Christodoulou; Michael J. Gait; Luc Van Meervelt; Madeleine Moore; Olga Kennard
1615-1624	The Synthesis of Some 5-Vinyluracil-Nucleoside Analogues	R. F. Whale; P. L. Coe; R. T. Walker

Volume 10, Issue 6 (1991)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 10, Number 6
1257-1275	The Synthesis of 5′-O-Triphosphate-4N-(ω-aminoalkyl)deoxycytidine A Useful Precursor to the Generation of Differently Labeled Triphosphates	Ryszard Kierzek; Wojciech T. Markiewicz
1277-1283	Cytidlne Nucleosides I: Photochemical Approach for the Synthesis of C-5 Aryl and Heteroaryl Substituted 2′-Deoxycytidine	Mohamed E. Hassan
1285-1293	Solid-Liquid Phase-Transfer Catalysis I: Studies of the N-Alkylation of Purines and Pyrimidines	H. B. Lazrek; M. Taourirte; J. -L. Barascut; J. -L. Imbach
1295-1303	Studies on Glycosides of 3, 4, 6-Trisubstituted Pyrazolo-[3, 4-D]Pyrimidines. Synthesis of 2′-Deoxyribonucleosides	Lydmila D. Garaeva; Irina V. Yartseva; Stalina Ya. Melnik
1305-1316	NMR Studies of N¹- and N³-(D-2′-Deoxyribofuranosyl) Nucleosides from Ethyl 5-Aminoimidazole-4-Carboxylate	David F. Ewing; Robert W. Humblet; Graham Mackenzie
1317-1332	Synthesis and Properties of 2′4′- and 3′-5′-Linked Ribodinucleoside Monophosphates Containing 2-Aminoadenosine and Uridine	Masako Muraoka; Akiko Iida; Seizo Takahashi; Tomohiko Ebata; Seiichi Uesugi
1333-1344	Synthesis of 2,2′-Anhydro-2-Hydroxy- and 6,2′-Anhydro-6-Hydroxy-1-β-D-Arabindfuranosylnicotinamide as Conformationally Restricted Nicotinamide Nucleoside Analogs¹	Krzysztof W. Pankiewicz; Lech A. Ciszewski; Anna T. Ptak
1345-1376	Systematic Synthesis and Antiviral Evaluation of α-L-Arabinofuranosyl and 2′-Deoxy-α-L-Erythro-Pento-Furanosyl Nucleosides of the Five Naturally Occurring Nucleic Acid Bases	Corinne Génu-Dellac; Gilles Gosselin; Frédéric Puech; Jean-Claude Henry; Anne-Marie Aubertin; Georges Obert; André Kirn; Jean-Louis Imbach
1377-1390	Synthesis of Fused Oligoribonucleotides with Trideoxyribonucleotide Containing Phosphorothioate to Stabilize Against Nuclease Activity	Masahide Ishikawa; Kazunori Ikebukuro; Ichiro Hirao; Kin-Ichiro Miura
1391-1406	Synthetic Studies on the Acyclic Nucleosides of 5-Substituted-6-Azauracils	Chein H. Han; Yeh L. Chen; Cherng C. Tzeng
1407-1416	Synthetic and Antiviral Studies of Certain Acyclic 3′-Azido-3′-Deoxythymidine (AZT) Analogues	Kuan-Han Lee; Yeh-Long Chen; Bor-Ruey Huang; Qing-Yu Zhu; Ting-Chao Chou; Cherng-Chyi Tzeng
1417-1427	In Vivo Antiviral Activity of 5-Amino-1-Methyl-3-β-D-Ribofuranosyl-Pyrazolo[4,3-d]Pyrimidin-7(6H)-One and Related Guanosine Analogues Prepared from Formycin	Yogesh S. Sanghvi; Steven B. Larson; Donald F. Smee; Ganapathi R. Revankar; Roland K. Robins

Volume 10, Issue 5 (1991)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 10, Number 5
xi-xii	Preface	A. P. Ijzerman; P. J. M. van Galen
917-930	Distribution and Roles of Purinoceptor Subtypes	G. Burnstock
931-943	Role of Adenosine in Energy Supply/Demand Balance	Robert F. Bruns
945-953	On the Adenosine Receptor Involved in the Excitatory Action of Adenosine on Respiration: Antagonist Profile	J. A. Ribeiro; E. C. Monteiro
955-964	Pharmacological Implications of A Multiplicity of Adenosine Actions in the CNS	Bertil B. Fredholm; Montse Ballarin; Pär Genvins; Ping-Sheng Hu; Ingeborg van der Ploeg; Fiona Parkinson
965-973	Nucleoside Transport in Neurons. Regulation by Secretagogues and Effectors of Protein Kinases A and C	M. T. Miras-portugal; R. P. Sen; E. G. Delicado
975-982	Comparative Pharmacology of Nucleoside Transport Inhibitors	H. Van Belle; P. A. J. Janssen
983-991	Recent Progress in the Purification of Adenosine Receptors	Hiroyasu Nakata
993-1001	Autoradiographic Localization and Characterization of Adenosine Receptor Subtypes in Mammalian Brain	Michael F. Jarvis
1003-1017	Transduction Mechanisms of P₂ Purinergic Receptors Role of Phospholipase C and Calcium	S. Pirotton; J. M. Boeynaems
1019-1028	Design, Syntheses and Pharmacology of ATP Analogues Selective for Subtypes of P₂-Purinoceptors	Noel J. Cusack; Susanna M. O. Hourani
1029-1038	Purine Functionalized Congeners as Molecular Probes for Adenosine Receptors	Kenneth A. Jacobson; John W. Daly
1039-1047	Molecular Modelling of the Antagonist Binding Site on the Adenosine A, Receptor	A. P. Ljzerman; P. J. M. Van Galen; H. W. Van Vlijmen; W. Soudijn; P. Nissen; I. Van Wijngaarden
1049-1055	Synthesis and Cardiac Pharmacology of 2-(AR)Alkoxyadenosines	Ray A. Olsson; Robert D. Thompson; Masayuki Ueeda; Luis H. Arroyo
1057-1066	Adenosine Receptors in Isolated Tissue Preparations	Michael G. Collis
1067-1076	Selective A₁-Antagonists for Treatment of Cognitive Deficits	G. Schingnitz; U. Küfner-Mühl; H. Ensinger; E. Lehr; F. J. Kuhn
1077-1086	Adenosine and Neuropsychiatric Disease	Jürgen Deckert; Paul J. Marangos
1087-1099	Purinergic Pharmaceuticals for the 1990s	Michael Williams

Volume 10, Issue 5 (1991)

1103-1106	Modulation of [³H]Nitrobenzylthioinosine Binding Kinetics	James R. Hammond
1107-1111	Recognition of Adenosine Receptors by Amiloride and Its Analogues	A. Garritsen; M. W. Beukers; A. P. Ijzerman; W. Soudijn
1113-1116	Adenosine Receptor Modulation of Inositol Phospholipid Turnover in the Central Nervous System	Stephen Ph Alexander; Stephen J. Hill; David A. Kendall
1117-1120	Suramin is a Competitive But Slowly-Equilibrating Antagonist at P_2x-Receptors in the Rabbit Ear Artery	P. Leff; B. E. Wood; S. E. O'connor; N. T. Fear
1121-1124	A Computer Generated Model of Adenosine Receptors Rationalising Binding and Selectivity of Receptor Ligands	Ronald J. Quinn; Michael J. Dooley; Andre Escher; Fiona A. Harden; Hiranthi Jayasuriya
1127-1129	Cardiovascular Effects of Adenosine Derivatives in Conscious Normotensive Rats	M. Milavec-krizman; H. Wagner; A. Kralj; J. P. Evenou; F. Gadient
1131-1133	Antinociceptive Effect Following Peripheral Administration of Adenosine Analogs in the Formalin Test in Mice	R. Karlsten; C. Post
1135-1137	Solubilized Rat Brain Adenosine Receptors Have Two Binding Sites For 1,3-Dipropyl-8-Cyclopentylxanthine	J. C. Oliveira; A. M. Sebastião; J. A. Ribeiro
1139-1140	Ligand Binding to A₁ Adenosine Receptors is Influenced by Protonation	Edmund Hoppe; Martin Reddington
1141-1143	Effect of Endogenous Phospholipids on the [³H]R-Pia Binding to A₁ Adenosine Receptors from PIG Cerebral Cortex	V. Casadó; J. Mallol; C. Lluis; E. I. Canela; R. Franco
1145-1147	Autoradiographical Studies of in Vitro and Chronic in Vivo Effects of Propentofylline on Adenosine A₁ and A₂ Receptors and NBMPR-Sensitive Nucleoside Transporters	F. E. Parkinson; B. Johansson; K. Rudolphi; B. B. Fredholm
1149-1150	Possible Agonistic Interaction of Defibrotide, A DNA Derivative, with Adenosine Receptors “In Vitro”	G. Bianchi; M. Mantovani; G. Prino; L. Salvetti; D. Barone
1151-1153	R-N⁶-Phenylisopropyladenosine Produces Tracheal Contraction Through A₁ Adenosine Receptor and Challenges Prostanoid Mechanisms	G. Froldi; M. De Biasi; G. Fassina; L. Puglisi
1155-1159	Effects of Adenosine Agonists on Camp Accumulation in Adult and Newborn Rat Aortic Smooth Muscle Cell Cultures	Valerie Querol-ferrer; Bror Jonzon; Anna Hultgårdh-Nilsson
1161-1163	Adenosine Inhibition of ⁴⁵Ca Uptake by Synaptosomes as Function of Time of Electrical Stimulation	M. L. Gonçalves; F. Pinto; J. A. Ribeiro
1165-1167	Regional Difference of Purinergic Modulation on Adrenergic Neurotransmission in Isolated Rabbit Pulmonary Artery	Kazumasa Shinozuka; Yuta Kobayashi; Keiko Shimoura; Keisuke Hattori
1169-1171	Effects of Adenosine (ADO) and A₁ and A₂ Ado Agonists on Calcium Uptake and cAMP Levels in Cultured Rat Mesangial Cells (MC)	A. Olivera; M. Tomás; J. M. López-Novoa
1173-1174	GTP and IAP Shifts Adenosine A₁-Agonist Binding in Smooth Muscle Membranes to the Low Affinity State, Similar to the one Found in Intact Cells	Pär Gerwins; Christer Nordstedt; Bertil B. Fredholm
1175-1176	Unilateral Entorhinal Cortex Lesion - An Animal Model For Cognitive Impairment in Human Disease: Effects on Adenosine Receptors and Second Messengers	J. Deckert; M. B. Jorgensen
1177-1179	The Inhibition of Nucleoside Transport in Human Erythrocytes by Mioflazine Analogues	Irene M. Pirovano; Adriaan P. Ijzerman

Volume 10, Issue 5 (1991)

1181-1182	Effects of Suramin on the ATP- and α,β-Methylene-ATP-induced Constriction of the Rabbit Ear Artery	Ivar von Kügelgen; Klaus Starke
1183-1184	Characteristics of Adenosine-Mediated Inhibition of Tachykinin Release from Perifused Myenteric Plexus Synaptosomes	M. A. Cook; R. M. Broad
1185-1186	Calcium Antagonists Modulate ³H-Purine Release from Rat Striatum Glial Cultures Via Vscc-Dependent and Independent Mechanisms	P. Ballerini; R. Cccarelli; P. Di Iorio; H. Di Huzio; S. Ferrari; F. Caciagli
1187-1188	Regional Changes in Rat Brain Adenosine A1 Receptors Following Seizures	J. L. Daval; M. C. Werck
1189-1190	Relative Contribution of Nerve Endings to the Release of Adenine Nucleotides in the Innervated from Sartorius Muscle	R. A. Cunha; A. M. Sebastião; J. A. Ribeiro
1191-1193	Xanthine-7-Ribosides as Adenosine Receptor Antagonists: Further Evidence for Adenosine'S Anti Mode Of Binding	P. J. M. van Galen; A. P. Ijzerman; W. Soudijn
1195-1197	Effect of ATP and ADP on U-937 Promonocyte Cell Adhesiveness and Intracellular Ca Levels	M. A. Ventura; P. Thomopoulos
1199-1200	Mapping the Xanthine CS-Region of the Adenosine A, Receptor with Computer Graphics	E. M. van der Wenden; P. J. M. van Galen; A. P. Ijzerman; W. Soudijn
1201-1202	Characterization of the Binding of a Novel Non-Xanthine Adenosine Antagonist Radioligand, [³H]CGS 15943, to Multiple Affinity States of the Adenosine A₁ Receptor in the Rat Cortex	Michael F. Jarvis; Michael Williams; Un Hoi Do; Matthew A. Sills
1203-1205	Amppcp Acts Via P₁ and Not P₂ Receptors in Some Isolated Smooth Muscle Preparations	S. M. O. Hourani; S. J. Bailey; J. Nicholls; I. Kitchen
1207-1208	P_2x-Receptor Characterisation in Rabbit Isolated Ear Artery	S. E. O'connor; B. E. Wood; P. Leff
1209-1210	Age-Elated Impairment of Relaxation To ATP in Rabbit Aortas	A. Chinellato; L. Pandolfo; E. Ragazzi; L. Caparrotta; G. Fassina
1211-1212	APEC, An A₂-Selective Adenosine Agonist, is a More Potent Locomotor Depressant Than N⁶-Cyclohexyladenosine	Kenneth A. Jacobson; Olga Nikodijevic; David de la Cruz; John W. Daly
1213-1214	Ascorbate-Induced Lipid Peroxidation and Inhibition of [³H] Adenosine Binding to Rat Brain Synaptosomes	E. Fonseca; J. A. Ribeiro
1215-1216	Potentiation of ATP Responses by α,β-Methyleneadp in the Rabbit Ear Artery	B. E. Wood; J. E. Steptoe; S. E. O'connor; P. Leff
1217-1218	P₁-Purinergic Receptor-Mediated Modulation of TSH Actions on FRTL-5 Thyroid Cells: Possible Switching From cAMP Pathway to Inositol Phosphate-Ca System	Y. Kondo; K. Sho; M. A. Majid; F. Okajima
1219-1220	The Influence of Adenosine Receptor Antagonists Ahinophylline (AMP) and Caffeine (CAF) on Seizure Protective Ability of Antiepileptic Drugs (AEDs) in Rats	Chanda Kulkarni; Thangam Joseph; Joy David
1221-1222	Circadian Fluctuation in 3H-CHA Binding to Mouse Cerebral Cortex Membranes	C. Florio; A. M. Rosati; U. Traversa; R. Vertua
1223-1224	[³H]R75231; A New Radiolabelled Nucleoside Transporter Probe Related to Mioflazine and Lidoflazine	M. Kruidering; A. P. Ijzerman; H. Van Belle
1225-1226	Effects of Caffeine and/OR L-Phenylisopropyladenosine (LPIA) on Local Cerebral Blood Flow and Glucose Utilization in the Rat	A. Nehlig; A. Pereira de Vasconcelos; S. Boyet

Volume 10, Issue 5 (1991)

1227-1229	Involvement of Adenosine in the Acute Action of Progesterone on Glucose Metabolism In Rat Adipocytes	P. Cordoba; J. Sutter; M.-Th. Sutter-Dub
1231-1233	Adenosine-induced dilation of rat thoracic aorta is mediated by cyclic GMP and is age-dependent	Hideki Moritoki; Tetsuhiro Hisayama; Haruyasu Ueda
1235-1236	Influence of Phospholipase A₂-Prostaglawdin System Linked to A1 Adexosine Becepmb on Protein Kinase C Activity of Cultubed Glial Cells	R. Ciccarelli; M. Di Muzio; P. Di Iorio; P. Ballerini; F. Caciagli
1237-1238	A₁ and A₂ Adenosine Receptors Involvement in Controlling Purine and Acetylcholine Release From Rat Hippocampal Slices	P. Di Iorio; P. Ballerini; R. Ciccarelli; M. Di Muzio; U. Traversa; F. Caciagli
1239-1240	P₂-Purinoceptor Mediated Inhibition of Adenylate Cyclase Activity	A. M. Van Rhee; A. P. Ijzerman; W. Soudijn
1241-1243	Characterization and Photoaffinity Labeling of A₁ - Adenosine Receptors in Coated Vesicles from Bovine Brain	G. Gonzalez-calero; A. Cubero; K. N. Klotz
1245-1246	Affinity of Ionic Species of Nucleoside Transport Protein Inhibitors	AH Voorschuur; Ap Ijzerman
1247-1251	Purinergic Receptors, Past and Future (Closing Remarks)	Robert F. Bruns

Volume 10, Issue 4 (1991)

a	Editorial Board Page for “Nucleosides & Nucleotides”, Volume 10, Number 4
739-753	Synthesis and Antiherpetic Activities of Several Acyclic Analogues Of Guanosine	Hirofumi Furusho; Takahiro Ogata; Akihisa Kato; Yoshie Sato; Tohru Endo; Akira Kaji
755-761	An Improved Method for The Preparation Of The Phosphoramidites Of Modified 2′-Deoxynucleotides: Incorporation Of 8-Oxo-2′-Deoxy-7H-Guanosine Into Synthetic Oligomers	Veeraiah Bodepudi; Charles R. Iden; Francis Johnson
763-779	Synthesis of Modified Nucleosides. Palladium-Catalysed Couplings of Organostannanes or Organoboranes with Pyrimidine Nucleosides	Bernard L. Flynn; Vilma Macolino; Geoffrey T. Crisp
781-798	Synthesis of 9-(2-Deoxy-2-Fukuoro-β-D- Abinoruranosyl)Hypoxhine. The First Direct Introduction of A 2′-β-Fldoro Substituent in Ppepormed Purine Nucleosides. Studies Directed Toward the Synthesis of 2′-DEOXY-2′-Substituted Arabppmocebosides. 8.¹	Jacek Krzeminski; Barbara Nawrot; Krzysztof W. Pankiewicz; Kyoichi A. Watanabe
799-817	Nucleosides, XLVIII. Syntheses and Properties of Quinazoline N-1-Ribofuranosides	Martin Dunkel; Wolfgang Pfleiderer
819-836	Synthetic, Structural, and Conformational Studies of Methylated Ring-Expanded Nucleosides Containing the Ihidazo[4, 5-e][1, 4]Diazepine Ring System	Ramachandra S. Hosmane; Anila Bhan; Martin Hulce; Hongming Zhang; Narayan S. Hosmane
837-851	Synthesis of the 2′-,3′-Didehydro-2′-,3′-dideoxy and 2′-,3′-Dideoxy Derivatives of 6-Azauridine and a New Route to 2′-,3′-Didehydro-2′-,3′-dideoxy-5-chlorouridine	Andre Rosowsky; Niranjan N. Pai
853-866	Synthesis of Bridged Pyrimidine Nucleosides and Triazo [4, 3-c] Pyrimidine Nucleoside Analogues	Stefania Barbato; Gennaro Piccialli; Ciro Santacroce; Lorenzo De Napoli; Luciano Mayol
867-882	Solid-Phase Synthesis of Oligodeoxyribonucleotide Analogues Containing 5, 6-Dihydroimidazo [1, 2-c] Pyrimidin-5-One as a Base Moiety	Stefania Barbato; Gennaro Piccialli; Ciro Santacroce; Lorenzo De Napoli; Luciano Mayol
883-894	Synthesis and Biological Evaluation of 4-Carbamoyl-2-β-D-Ribofuranosyl-Pyridine	Pieter E. Joos; Eddy L. Esmans; Roger A. Dommisse; Walter Van Dongen; Jozef A. Lepoivre; Frank C. Alderweireldt; Jan Balzarini; Erik De Clercq
895-909	Introduction of 5′-Terminal Amino and Thiol Groups into Synthetic Oligonucleotides	R. K. Gaur
911-912	Erratum
913	Erratum

Volume 10, Issue 1-3 (1991)

Proceedings of the 9th International Round Table

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 10, Number 1-3
3-24	Polymorphism, Packing, Resolution, and Reliability in Single-Crystal DNA Oligomer Analyses	Richard E. Dickerson; Kazimierz Grzeskowiak; Maria Grzeskowiak; Mary L. Kopka; Teresa Larsen; Andrei Lipanov; Gilbert G. Privé; Jordi Quintana; Peter Schultze; Kazunori Yanagi; Hanna Yuan; Hyo-Chun Yoon
25-36	2′-O-alkyloligoribonucleotides Synthesis and Applications in Studying RNA Splicing	Brian S. Sproat; Adolfo Iribarren; Barbro Beijer; Uwe Pieles; Angus I. Lamond
37-46	Antisense Oligonucleoside Methylphosphonates and Their Derivatives	Paul S. Miller; Purshotam Bhan; Cynthia D. Cushman; Joanne M. Kean; Joel T. Levis
47-59	Chemical and Biochemical Studies with Dithioate DNA	Marvin H. Caruthers; Graham Beaton; Lendell Cummins; Douglas Dellinger; Darla Graff; Yun-Xi Ma; William S. Marshall; Henri Sasmor; Paula Shankland; John Van Wu; Eric K. Yau
61-80	High Resolution NMR Studies of DNA Hairpins with Four Nucleotides in the Loop Region	C. W. Hilbers; M. J.J. Blommers; F. J.M. Van de Van; J. H. Van Boom; G. A. Van Der Marel
81-97	Studies in the Solid Phase Synthesis of Oligo- and Poly-Ribonucleotides	Colin B. Reese; M. Vaman Rao; Halina T. Serafinowska; Elizabeth A. Thompson; Pak Sang Yu
99-105	An Attempt to Design and Chemical Synthesis of a Eukaryotic Messenger RNA	Reiko Iwase; Tsujiaki Hata
107-117	Derivatization of Oligonucleotides Through Abasic Site Formation	J.-J. Vasseur; D. Peoc'h; B. Rayner; J.-L. Imbach
119-127	Synthesis of Pyranose Nucleosides	P. Herdewijn; A. Van Aerschot; J. Balzarini; E. De Clercq
129-139	Nucleic Acids Probes in Diagnostic	Robert Teoule; Hervé Bazins; Brigitte Fouqué; André Roget; Sylvie Sauvaigo
141-153	Synthesis and Properties of Non-Hammerhead RNA Using 1-(2-Chloroethoxy)-ethyl Group for the Protection of 2′-Hydroxyl Function	Osamu Sakatsume; Takashi Ogawa; Hideo Hosaka; Masahiko Kawashima; Makoto Takaki; Hiroshi Takaku
155-166	Phosphorothioate Oligonucleotides as Potential Antiviral Compounds Against Human Immunodeficiency Virus and Herpes Viruses	Yung-chi Cheng; Wen-yi Gao; Fu-sheng Han
167-180	Antiviral Activity Spectrum of Nucleoside and Nucleotide Analogues	Erik De Clercq
181-193	Stereochemical Analysis of the Enzymic Synthesis and Hydrolysis of Ap₄A	Gordon Lowe
195-205	DNA Interaction with Chiral Metal Complexes	Bengt Nordén; Naina Patel; Catharina Hiort; Astrid Gräslund; Seog Kyu Kim
215-227	Metal-Catalyzed RNA Strand Scission	Barbara J. Carter; Chris E. Holmes; Reuel B. Van Atta; V. Dange; Sidney M. Hecht
231-234	Hybridization Properties of a DeoxyoIigonucleotide Containing Four Formacetal Linkages	Mark Matteucci
235-238	Design, Synthesis and Tumor Specificity of Azomycin Ribo- and Acyclonucleosides	Prem C. Srivastava; Donald J. Buchsbaum; Ahmad Hasad
239-244	Effect of Antisense Oligonucleotides Linked to Alkylating Agents on In Vitro Translation of Rabbit β-Globin and Typuaosomu brucei mRNAs	C. Boiziau; A. S. Boutorine; N. Loreau; P. Verspieren; N. T. Thuong; J. J. Toulmé
245-248	Synthesis of the 6′-Fluoro Derivatives of Carbocyclic 2′,3′-Dideoxy-3′-oxa-adenosine	Steve Tam; Michael Holman; Donna Huryn; Andrew Cislo
249-252	Synthesis and ¹⁵N NMR Study of N-7/N-9 Substituted Glyoxal-Guanine Adducts	J. Plavec; J. Kobe
253-257	Synthesis and Antitumor Activity of 6–Substituted Purine and Deazapurine Nucleosides	Gloria Cristalli; Sauro Vittori; Alessandra Eleuteri; Palmarisa Franchetti; Mario Grifantini; Giulio Lupidi; Laura Capolongo; Enrico Pesenti
259-262	Synthesis and Biophysical and Biological Evaluation of 2′-Modified Antisense Oligonucleotides	C. J. Guinosso; G. D. Hoke; S. Frier; J. F. Martin; D. J. Ecker; C. K. Mirabelli; S. T. Crooke; P. D. Cook
263-267	Deoxyluminarosine: New, Photochemically Prepared Fluorophore for the Sequence-Specific Oligonucleotide Labelling	Sllawornir Mielewczyk; Graźyna Dominiak; Zofia Gdaniec; Edyta Krzymańska-Olejnik; Ryszard W. Adamiak; Bohdan Skalskiy
269-273	Large-Scale, PEG-Supported DNA Synthesis	G. M. Bonora; C. L. Screminl; F. P. Colonna; A. Garbesi
275-278	Unsaturated Analogues of Acyclic Nucleoside Phosphonates an Unusual Arbuzov Reaction with Unactivated Triple Bond	Shashikant Phadtare; Jiri Zemlicka
279-282	New Prodrugs of Aciclovir with Antiviral Activity	M. Madre; R. Zhuk; M. Lidaks

Volume 10, Issue 1-3 (1991)

Proceedings of the 9th International Round Table

283-286	Stereoselective Synthesis of Nucleoside Phosphorofluoridates	J. Michalski; W. Dabkowski; A. Topusi�ski; F. Cramer
287-290	Deoxyoligonucleotides with Inverted Polarity Synthesis and Use in Triple-Helix Formation	S. McCurdy; C. Moulds; B. Froehler
291-294	Synthesis and Antiviral Evaluation of 3′-Branched Nucixoside Analogues	Roman Z. Sterzycki; J. C. Martin; M. Wittman; V. Rrankovan; H. Yang; M. J. Hitchcock; M. M. Mansuri
295-298	Steroid and N-(2-Hydroxyethyl)phenazinium Oligodeoxynucleotides	V. F. Zarytova; E. M. Ivanova; A. S. Levina
299-302	Controlled Chemical Cleavage of Synthetic DNA at Specific Sites	Thomas Horn; Kristina Downing; Yougen Gee; Mickey S. Urdea
303-306	Specific Intrachain Introduction of Reporter Groups into Oligonucleotides as Substituents at Internucleotidic Linkages	H. Seliger; B. Krist; S. Berner
307-310	Approaches to New Dideoxynucleosides	Vasu Nair; Greg S. Buenger
311-314	Psicoplanocin A. A Synthetic Carbocyclic Nucleoside with the Combined Structural Features of Neplanocin A and Psicofuranine	Victor E. Marquez; Michael Bodenteich
315-318	Solid Phase Synthesis of Oligodeoxynucleotides Containing O⁶-Alkylguanine and O⁴-Alkylthymine	Yao-Zhong Xu; Peter F. Swann
319-322	Assignment of Absolute Configuration at Phosphorus in Dithymidylyl(3′,5′)phosphormorpholidates and -Phosphormorpholidothioates	A. Wilk; B. Uzanski; W. J. Stec
323-324	Synthesis of Some Pyridine-C-Nucleosides	P. E. Joos; E. L. Esmans; R. A. Dommisse; J. A. Lepoivre; F. C. Aldenveireldt
325-327	Studies on the Interaction between HIV-1 Reverse Transcriptase and Templateoligo α-Thymidylate Duplexes	Georges Maury; Bernard Rayner; Jean-Louis Imbach; Barbara Müller; Tobias Restle; Roger S. Goody
329-332	Stereoselective Synthesis of 6-Amln0-5,6dideoxy-D-ribo-heptafuranouronates with the Aid of Glycine. Chiral Templates	L. W. Dudycz
333-337	Oligonucleotide-Polyamide Conjugate Probes with Multiple Non-Radioactive Labels: Applications and Comparison to Radiolabelled Probes	J. Haralambidis; L. Violaris; G. W. Tregear
339-343	Substrate Properties of C′-Methylnucleoside and C′-Methyl-2′-deoxynucleoside 5′-Triphosphates in RNA and DNA Synthesis Reactions Catalysed by RNA and DNA Polymerases	S. N. Mikhailov; N. Sh. Padyukova; Yu P. Lysov; L. P. Savochkina; Z. G. Chidgeavadze; R. Sh. Beabealashvilli
345-346	Synthesis and Biological Evaluation of Antisense Oligonucleotides Containing Modified Pyrimidines	Y. S. Sanghvi; G. D. Hoke; M. C. Zounes; S. M. Freier; J. F. Martin; H. Chan; O. L. Acevedo; D. J. Ecker; C. K. Mirabelli; S. T. Crooke; P. D. Cook
347-350	Diastereoselective Synthesis of Thymidine-Methylphosphonate Dimers	Joachim W. Engels; Thomas Löschner; Albrecht Frauendorf
351-354	Inhibition of Human Immunodeficiency Virus (HIV) Production by 5′-Hydrogenphosphonates of 3′-Azido-2′,3′- dideoxynucleosides	Natalya B. Tarussqva; Marina K. Kukhanova; Alexander A. Krayevsky; Edward K. Karamov; Vladimir V. Lukashov; Galina B. Kornilayeva; Mariana A. Rodina; Georgii A. Galecov
355-358	1-(5-Amino-1-β-D-Ribofuranosylimidazol-4-carbonyl)-3,5-dimethylpyrazole, a new Intermediate for the Preparation of Aicar Analogs	Peter K. Bridson; Rogers E. Harry O'Kuru
359-362	Synthesis of Oligonucleotides Covalently Linked to Intercalating Agents and to Reactive Groups	Ulysse Asseline; Nguyen T. Thuong
363-366	Phosphoramidite Reagents for the Easy Preparation of Polylabelled Oligonucleotide Probes	Bazin Hervé; Roget André; Téoule Robert
367-370	Inhibition of the First Stage of RNA Ligase Reaction by ATP Analogues	B. Juodka; D. Labeiltyte
371-375	Phosphonate Isosteres of 2′,3′-Didehydro-2,3-dideoxynucleoside Monophosphates: Synthesis and Anti-HIV Activity	Choung Un Kim; Bing Y. Luh; Peter F. Misco; John C. Martin
377-382	Model Studies Towards the Automated Synthesis of tRNAs	W. Pfleiderer; M. Pfister; S. Farkas; H. Schirmeister; R. Charubala; K. P. Stengele; M. Mohr; F. Bergmann; S. Gokhale
383-388	Chemical Synthesis and Biological Activity of 2′-5′-Phosphorothioate Tetramer Cores	R. Charubala; W. Pfleiderer; R. J. Suhadolnik; R. W. Sobol
389-392	Improved Methods for the Synthesis of Branched DNA (bDNA) for use as Amplification Multimers in Bioassays	Chu-an Chanz; Thomas Horn; David Ahle; Mickey S. Urdea
393-396	Synthesis and Biological Activity of Carbocyclic Clitocine	Anthony D. Baxter; Charles R. Penn; Richard Storer; Niall G. Weir; Jacqueline M. Woods
397-400	Lithiation of Uracilnucleosides and its Application to the Synthesis of a New Class of Anti-HIV-1 Acyclonucleosides	Hiromichi Tanaka; Masanori Baba; Hiroyuki Hayakawa; Kazuhiro Haraguchi; Tadashi Miyasaka; Masaru Ubasawa; Hideaki Takashima; Kouichi Sekiya; Issei Nitta; Richard T. Walker; Erik De Clercq
401-404	Biological and Biochemical Studies on Ro31-6840 (2′βFddC), a Dideoxynucleoside Analogue Active Against Human Imhunodeficiency Virus Type 1 (HIV-1)	P. Wong-Kai-In; K. E. B. Parkes; D. Kinchington; S. A. L. Hope; N. A. Roberts; J. A. Martin; J. H. Herrett; P. Machin; G. Thomas
405-408	New Strategies in the Synthesis of 3′-Azido-2′,3′-dideoxy-nucleosides with Furanose Configuration	Jesper Wengel; Jesper Lau; Krzysztof Walczak; Erik B. Pedersen

Volume 10, Issue 1-3 (1991)

Proceedings of the 9th International Round Table

409-412	Base-Modifled Purine 2′,3′-Dideoxyribonucleosjdes: Synthesis via Deoxygenation or Direct Nucleobase Anion Glycosylation	F. Seela; H. Rosemeyer; R. Gumbiowski; K. Mersmann; H.-P. Muth; A. Röling
413-414	A Simple Preparation of 5′-Biotinylated Oligonucleotides and Their use as Primers in Dideoxy-Sequencing of DNA	Anthony J. Cocuzza; Robert J. Zagursky
415-418	Properties of Trialkoxysilyl Grows	Wojciech T. Markiewicz; Katarzyna Adrych-Rozek
419-422	Anti-HIV Activity of the Antisense Oligonucleotides Bearing Lipophilic and Alkylating Groups at the 5′-Terminus	T. V. Abramova; V. M. Blinov; V. V. Vlassov; V. V. Gorn; V. F. Zarytova; E. M. Ivanova; D. A. Konevets; O. A. Plyasunova; A. G. Pokrovsky; L. S. Sandahchiev; F. P. Svinarchuk; V. P. Starostin; S. R. Chapligina
423-426	Stereoselective Synthesis of 2′,3′-Dideoxy-and 2,3′-Didehydro-2′,3′-dideoxy-nucleosides	Chung K. Chu; J. Warren Beach; J. Ramesh Babu; Lak Shin Jeong; Heaok Kim; Jeong; Soon Kil Ahn; Qamrul Islam; Sang Joa; Yaoquan Chen
427-430	9-[2-(Phosphonomethoxy)alkoxy]purines, A New Series of Antiviral Acyclonucleotides	D. M. Duckworth; M. R. Harnden; R. M. Perkins; D. N. Planterose
431-455	Biologically Important Nucleosides: A General Method for the Synthesis of Unsaturated Ketonucleosides of Uracil and its Analogs	Dimitri Komiotis; Sylvie Delatre; Leonard Holt; Abraham P. Ollapally; Jan Balzariei; Erik De Clercq; Masaaki Iigo
457-460	Abasic Oligodeoxyribonucleoside Phosphorothioates as Inhibitors of the Human Immunodeficiency Virus-1 (HIV-1) Phosphorothioate Inhibition of HIV-1 Reverse Transcriptase and Interactions with Syrian Hampster Fibroblast (V79) Cells	William Egan; Jila Boal; Radhakrishnan P. Iyer; Christy Storm; Samuel H. Wilsont; Anita Meyer; Patrick Iversenq
461-464	Preparation and Properties of Oligodeoxynucleoside Phosphorodithioates	Kirsten Bjergarde; Bjarne H. Dahl; Otto Dahl
465-468	Enzymatic Sywmesis of Dideoxyribonucleosides	D. Betbeder; C. M. Heath; D. U. Hutchinson
469-475	Oligonucleotide Analogues with Terminal 3′-3′- and 5′-5′-Internucleotidic Linkages as Antisense Inhibitors of Viral Gene Expression	H. Seliger; A. Fröhlich; M. Montenarh; J. F. Ramalho Ortigao; H. Rösch
479-481	3′/5′-Regioselectivity of Introduction of the 9-Fluorenyl-Methoxycarbonyl Group to 2′-O- Tetrahydropyran-2-Yl- and 2′-O-(4- methoxytetrahydropyran-4-Yl-)-nucleosides Useful Intermediates for Solid-Phase-RNA-Synthesis	Christian Lehmann; Yao-Zhong Xu; Chris Christodoulou; Michael J. Gait; Luc Van Meervelt; Madeleine Moore; Olga Kennard
483-485	Phosphonate Isosteres of Acyclovir and Ganciclovir Honophosphates Synthesis and Anti-Herpesvirus Activity	Choung Un Kim; Bing Y. Luh; Peter F. Misco; John C. Martin
487-490	Synthesis and Biological Evaluation of Carbocyclic Analogues of Ribavirin	Stewart A. Noble; Nicola E. Beddall; Alison J. Beveridge; Clara L.P. Marr; Chi L. Mo; Peter L. Myers; Charles R. Penn; Richard Storer; Jacqueline M. Woods
491-493	Synthesis of Some 2′,3′-Didehydro-2′,3′-dideoxynucleosides and 2′,3′- dideoxynucleosides	Pawel Serafinowski
495-496	Solid Phase -Nucleotide Links Cleavable by Mild Acid Treatments: Phosphoramidates, Phosphoesters and Ethers	Eduard R. Felder
497-498	Novel Analogues of the Nucleoside Antibiotics Coroyepin	Vasu Nalr; David F. Purdy; Arthur G. Lyons
499-500	Metal Mediated Reactions in Nucleside Synthesis	Vasu Nalr; Todd B. Sells
501-502	Novel Inhibitor-Probes of DNA Polymerase III Based on DGTP Analogues of the H₂·HPURA Type: Redesign of the Inhibitor Structure Using an N²-Benzylguanine Format	M. Butler; L. W. Dudycz; N. N. Khan; G. E. Wright; N. C. Brown
503-505	The Synthesis and Interaction of Novel GTP Derivatives with Ras Oncogene Proteins	Timothy P. Noonan; Lech W. Dudycz; George E. Wright
507-509	Biotinylation of Oligonucleotides and Their Use as Polymerase Chain Reaction Primers	M. Bengtström; L. Harju; A-C. Syvhen
511-514	Some Chemical and Stereochemical Aspects of Ribonucleoside H-Phosphonate and H-Phosphonothioate Diester Synthesis	Jacek Stawinski; Roger Stromberg; Mats Thelin
515-516	Studies on the Conversion of Nucleoside H-Phosphonate Monoesters into the Corresponding H-Phosphonothioates	Jacek Stawinski; Roger Stromberg; Rula Zain
517-518	Studies on Sulfurization of Nucleoside H-Phosphonate and H-Phosphonothioate Esters Using 3H-1,2-Benzodithiol.3-one 1,1-dioxide	Jacek Stawinski; Mats Thelin; Erik Von Stedingk
519-520	Ribonucleoside H-Phosphonates. Pyridine vs Quinoline - Influence on Condensation Rate	J. Stawinski; R. Strömberg; E. Westman
521-522	2,3′-Anhydro-[l- (6′- O-benzoyl-2′,5′- dideoxy-β-D-glucofuranosyl)thymine], a Versatile Starting Material for Homo - Nucleosides	Johann Hiebl; Erich Zbiral; Jan Balzarinib; Eric De Clercq
523-525	Oligonucleotide Derivatives in Organism: Distribution Among Organs, Rates of Release and Degradation	O. M. Bazanova; V. V. Vlassov; V. F. Zarytova; E. M. Ivanov; E. A. Kuligina; L. A. Yakubov; M. N. Abdukayumov; V. N. Karamyshev; G. Zon
527-529	More Efficient Alkylating Oligonucleotide Derivatives for the Sequence Specific Chemical Modification of dsDNA	V. V. Vlassov; A. A. Godovikov; A. A. Gall; E. M. Ivanova; A. U. Semeryanova
531-533	The Chemical Synthesis of ATP-Derivative of Phosphoglyceric Acid	Lucyna A. Wozniak; Halina Serafinowska; Colin B. Reese
535-536	Inhibition of the Reverse Transcriptase of HIV-1 by 3′-Azidothymidine Triphosphate and 3′-Azido-oligothymidylate	Olaf Heidenreich; Fritz Eckstein

Volume 10, Issue 1-3 (1991)

Proceedings of the 9th International Round Table

537-539	Nuclear Accumulation of Microinjected Antisense Oligonucleotides	Jean Paul Leonetti; Nadir Mechti; Geneviève Degols; Bernard Lebleu
541-542	Ethidium Oligodeoxynucleotide Derivatives. Stability Against Cellular Nuclease Hydrolysis and Photochemical Modification of Cellular Proteins in the Living Cells	A. A. Koshkin; A. V. Lebedev; A. S. Ryte; V. V. Vlassov
543-545	Synthesis of 3-Deazaclitocwe [2-Amino-3-nitro-4-(β-D-ribofuranosylamino)pyridine] as Cytotoxic Agent	Palmarisa Franchetti; Loredana Cappellacci; Gloria Cristalli; Mario Grifantini; Sauro Vittori
547-548	Interaction of a Minor Groove Binder with a Fluorescent DNA Oligomer Containing the Eco RI Recognition Sequence	N. Patel; A. Grälund; H. Berglund; L. Nilsson; R. Rigler; L. W. McLaughlin
549-551	Synthesis, Physical, Chemical, and Enzyme Studies on bis-2,β-Diaminopurine β-D-Ribofuranoside p1, p4-Tetraphosphate	G. Michael Blackburn; Mao-Jun Guo
553-554	Synthesis of Oligodeoxynucleoside Phosphorodithioates by a Phosphortriester Method	Bjame H. Dahl; Kirsten Bjerghde; John Nielsen; Otto Dahl
555-561	Synthesis of Base Modified Phosphorothioate Oligodeoxynucleotides as Inhibitors of HIV-1	O. Kemal; T. Brown; S. Burgess; J. D. Bishop; A. J. Leigh-Brown
563-564	Hydrogen Fluoride Mediated Alkylation and Dimerization of the Base Moiety of the cis Diastereoisomers of 5,6-Dihydroxy-5,6-dihydrothymidine	Michel Polverelli; Maurice Berger; Jean Cadet
565-566	Synthesis of Oligodeoxynucleotides Bearing a Radiation Induced DNA Damage: Deoxyribosylurea and Deoxyribosylformamide	André Guy; Hervé Bazin; Robert Teoule
567-568	Conformation of 3′-Substituted 2′,3′-Dideoxyribonucleosides in Aqueous Solution; Nucleoside Analogues with Potential Antiviral Activity	Pentti Oksman; Ryszard Stolarski; Alex Azhayev; Harri Lönnberg
569-570	Interconversion and Hydrolysis of Monoalkyl Esters of Adenosine 2′- and 3′-Monophosphates: Kinetics and Mechanisms	Mikko Oivanen; Ralf Schnell; Wolfang Pfleiderer; Harri Lönnberg
571-572	Kinetics and Mechanism for Acid-Catalyzed Hydrolysis of Regioisomeric 2′-Deoxyribonucleosides of 8-Azaadenine and Substituted Benzotriazoles	Rainer Käppi; Zygmunt Kazimierczuk; Frank Seela; Harri Lönnberg
573-574	A New Support For Automated Oligonucleotide Synthesis	Christie McCollum; Alex Andrus
575-577	Synthesis and Properties of Daunomycin Mono- and Oligonucleotide Derivatives	V. F. Zarytova; T. S. Godovikova; T. V. Maltseva; D. S. Sergeyev
579-580	Investigation of the C-Myc and C-Fos Genes Functions with Retroviral Vectors Producing Antisense RNA	V. V. Vlassov; F. P. Svinarohuk; D. A. Konevets; E. J. Frolova; M. Markelov; V. A. Lavrovsky; A. Ustinov
581-582	Interaction of Oligonucleotide Derivativts with Animal Cells	V. V. Vlassov; E. A. Deeva; M. N. Nechaeva; E. N. Rykova; L. A. Yakubov
583-584	Synthesis of Thymidine Analogues with a Cyanoimido Substituent	P. Wigerinck; A. Van Aerschot; L. Kerremans; J. Balzarini; E. De Clercq; P. Claes; P. Herdewijn
585-586	5-(Thien-2-yl)-2′-deoxyuridine: A New and Potent Inhibitor of Herpes Simplex Virus Type 1 Replication	P. Wigerinck; A. Van Aerschot; E. De Clercq; P. Herdewijn
587-588	Sugar Modified Oligonucleotides	K. Augustyns; A. Van Aerschot; P. Herdewijn
589-590	Synthesis and Anti-HIV Activity of Dideoxycytidine Analogues Containing a Pyranose Carbohydrate Moiety	A. Van Aerschot; L. Kerremans; J. Balzarini; E. De Clercq; P. Herdewijn
591-592	Synthesis and Antiviral Activity of 1.4-Dioxane, 1.4-Oxathiane and 1,4-Morpholine Nucleoside Analogues	A. Van Aerschot; J. Balzarini; E. De Clercq; P. Herdewijn
593-594	Intermolecular Association of Deoxycytidylyl-(3′,5′)deoxy-guanosine and Thymidylyl-(3′,5′)-deoxyadenosine in Dimethylsulfoxide	Giovanna Barbarella; Luisa Tondelli; Vitaliano Tugnoli
595-597	Synthesis and Application of N(6)-Phenoxycarbonyl-deoxy-adenosine Derivatives in Oligonucleotide Probes Chemistry	Edyta Krzymańska-Olejnik; Ryszard W. Adamiak
599-600	First, Solid Support-Aided Introduction of Isopentyladenosine, Hypermodified Nucleose of TRNA, into Oligoribonucleotide Chain	Piotr Sacute; widerski; Wieslaw Z. Antkowiak; Ryszard W. Adamiak
601-602	Silyloxyphosphanes. New Phosphitylating Reagents in Nucleotide Chemistry	W. Dabkowski; J. Michalski; Q. Wang
603-605	X-Ray Crystal Structure of Luminarine - Aglycone of Highly Fluorescent Luminarosine	Dorota A. Adamiak; K. Surma; Marian Gawron; Bohdan Skalski
607-608	Mechanism of Initiation of Transcription in Escherichia Coli	Rakesh K. Mishra; Dipankar Chatteji
609-613	Sequence Specific Chemical Recognition Of DNA	Jyoti Mehrotra; Krishna Misra; Rakesh K. Mishra
615-617	Synthesis of Aryl Phosphorodichloridothioates from ARYL Phosphorodichloridites via Arbuzov-Type Rearrangement	Antonio Procopio; Giovanni Sindona; Nicola Uccella
619-620	Synthesis of Nucleosides Using Trimethylsilyl Perfluoroethoxyethanesulphonate as Catalyst	J. A. Maurinsš; J. J. Jansons; M. J. Lidaks

Volume 10, Issue 1-3 (1991)

Proceedings of the 9th International Round Table

621-622	Synthesis of L-Threo- and D-Erythro-apiofuranosylcytidines	Johann-Peter Polsterer; Erich Zbiral; Jan Balzarini; Erik De Clerq
623-624	Syhthesis of Oligonucleotides Containing 4-0-Ethylthymidine	E. Pedroso; D. Fernández; Y. Palom; R. Eritja
625-626	Pyrazolo[3, 4-b]pyridine Nucleosides: Total Synthesis of the Guanosine, Isoguanosine and Xanthosine Analogues	Yogesh S. Sanghvi; Roland K. Robins; Ganapathi R. Revankar
627-629	HIV Inhibition by Antisense Oligodeoxynucleotides	M. Mag; J. Muth; S. Lücking; L. Biesert; J. Engels
631-632	Approach to the Synthesis of Functionally Active Polydeoxynucleotides Using DNA Amplification In Vitro	E. N. Lebedenko; O. V. Plutalov; Yu. A. Berlin
633-634	A Novel Approach to Sequence Specific Cross-Linking in Oligonucleotides	R. Cosstick; M. E. Douglas
635-638	Studies on the Synthesis of O-Ribosyl-Adenosine – a new Minor Nucleoside Of tRNA	Anna Niewczyk; Andrzej Krzyzaniak; Jan Barciszewski; Wojciech T. Markiewicz
639-640	The Effect of Oligodeoxyribonucleotide Terminal Phosphate and Ribose Modification on the Interactions of Oligonucleotides with Cells and Intracellular Stability	T. V. Abramova; V. V. Vlassov; V. F. Zarytova; E. M. Ivanova; E. A. Kuligina; A. S. Ryte
641-643	Photoactivatable Porphyrin Oligonucleotide Derivatives for Sequence Specific Chemical Modification and Cleavage of DNA	V. V. Vlassov; E. A. Deeva; E. M. Ivanova; D. G. Knorre; T. V. Maltseva; E. I. Frolova; G. V. Ponomariov; G. V. Kirillova
645-647	Suppression of Transcription and Translation of the Influenza Virus RNAs by Oligonucleotide Derivatives	V. V. Vlassov; E. I. Frolova; T. S. Godovikova; E. M. Ivanova; A. A. Koshkin; N. B. Ledovskikh; G. A. Nevinsky; L. V. Yurchenko; V. F. Zarytova
649-650	Inhibition of the Influenza Virus M Protein MRNA Translation in vitro with Complementary Oligonucleotides	V. V. Vlassov; V. V. Gorn; N. Yu. Nomokonova; T. N. Fokina; L. v. Yurchenko
651-652	Synthesis and Anti-HIV Activity of Modified 2′,3′-Dideoxy-3′-Fluoro Pyrimidine Nucleosides	M. Von Janta-Lipinski; K. Gaertner; J. Schildt; E. Matther; D. Scholz; P. Langon
653-655	Nonenzymatic Hydrolysis of an RNA-DIMER Containing a Thiophosphate Linkage	Helena Almer; Roger Strömberg
657-658	Differentiation of Anomeric & Positional Isomers of Acyclic & Cyclic Nucleosides by FAB Tandem Mass Spectrometry & NMR	J. H. Banoub; D. F. Ewing; R. W. Humble; G. Mackenzie; M. Becchi; D. Fraisse; G. Descotes; G. Shaw
659-661	Analysis of Urinary Nucleosides from AIDS Patients Using GC/MS	William M. Hammargren; Karl H. Schram; Katsuyuki Nakano; Toshio Yasaka; Michael Katz; Esklid Petersen
663-664	Synthesis of 5′-Dithiotriphosphate Derivatives of 3′-Deoxy 3′-Azidothymidine	János Ludwig; Fritz Eckstein
665-667	Interaction of Restriction Endonucleases with Phosphorothioate-Containing DNA	D. B. Olsen; J. R. Sayers; G. Kotzorek; F. Eckstein
669-670	Effect of length and netropsin binding on base-pair lifetimes of oligonucleotides with the center core GCGAATTCGC	M. Leijon; A. Gräslund
671-672	A New Multiple Labelling Method for Synthetic Oligonucleotides and Increased Sensitivity in DNA Detection	Konrad Misiura; Ian Durrant; Michael R. Evans; Michael J. Gait
673-674	Acetaldehyde Adducts of DNA	Pekka Sillanaukee; Leena M. Vilpo; Juhani A. Vilpo
675-677	Synthesis and Stability of Oligonucleotides Containing Purine Base Analogues	Paul Kong Thoo Lin; Daniel M. Brown
679-680	Oligoribonucleotides and Their 2′-O-Me-Analogs Carrying Alkylating and Intercalating Groups	V. F. Zarytova; A. G. Venjaminova; Z. A. Sergeyeva; M. N. Repkova; L. Arnold; J. Smrt
681-683	Synthesis of [5′-Phosphoryl-N(α)]-oligonucleotidyl-peptides	V. F. Zarytova; E. M. Ivanova; S. I. Yarmolyuk
685-688	Periodic-Catastrophic Transport of an Adenosine 5′-Monophosphate Amantadine Conjugate Through a Model Liquid Membrane	Donald E. Bergstrom; Julie K. Abrahamson; Michael Y.-M. Chan
689-691	Recent Advances in Palladium-Mediated Reactions of Nucleosides	Donald E. Bergstrom; Xiaoping Lin
693-697	Evaluation of Thymidine, Dideoxythymidine and Fluorine Substituted Deoxyribonucleoside Geometry by the MIND0/3 Technique The Effect of Fluorine Substitution on Nucleoside Geometry and Biological Activity	D. E. Bergstrom; D. J. Swartling; A. Wisar; M. R. Hoffmann
699-700	Interaction of the Deoxy-Oligonucleotide Duplex d(CGCGATCGCG)₂ and Anti-Herpes Virus Active Indolo [2,3-b]-quinoxaline Derivatives	N. Patel; J. Bergman; A. Gräslund
701-709	Free Energy Calculations Predict Sequence Specificity In DNA-drug Complexes	T. Härd; L. Nilsson
711-712	Stereospecific Oxidation of R_p- and S_p-Dinucleoside H-Phosphonates to Phoephorothioates	F. Seela; U. Kretschmer
713-714	Synthesis of Pyrrolo[3,2-c]pyridine and Pyrazolo[3,4-d]pyrimidine β-D-Arabinonucleosides via Nucleobase Anion Glycosylation	F. Seela; W. Bourgeois; H. Winter

Volume 10, Issue 1-3 (1991)

Proceedings of the 9th International Round Table

715-717	DNA-Fragments Resistant to Endodeoxyribonuclease Hydrolysis PCR-Amplification using 7-Deaza-2′-deoxyguanosine Triphosphate in Place of dGTP	F. Seela; A. Röling
719-721	A New Synthesis of 3′-Fluoro-3′-deoxyadenosine	A. Giordani; A. Ermoli; C. Battisthi
723-725	High Stereoselectivity in the Formation of the Inter-Ribonucleotidic Phosphorothioate Bond	C. Battisthi; M. G. Brasca; S. Fustinoni
727-728	The Synthesis of v-Triazolo[4,5-c]pyridine Nucleosides	A. Sscaron; timac; L. B. Townsend; J. Kobe
729-730	Reactions of 5-β-D-Ribofuranosyl Tetrazoles with Dipolarophiles	M. Prhavc; L. B. Townsend; J. Kobe
731-732	Synthesis of 5′-H-Phosphonates of 3′-Substituted Purine Deoxynucleosides	Natalia B. Dyatkina; Andrey A. Arzumanov; Natalia B. Tarussova
733-736	Stereospecific Synthesis of P-Chiral Di(2′-O-Deoxyribonucleoside)methanephosphonates	Zbigniew J. Lesnikowski; Maria M. Jaworska-Maslanka; Wojciech J. Stec

Volume 9, Issue 8 (1990)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 9, Number 8
1001-1013	8-Diazoguanosine, 2,8-Diaminoadenosine and Other Purine Nucleosides Derived from Guanosine	Peter C. Ratsep; Roland K. Robins; Morteza M. Vaghefi
1015-1019	Synthesis of Two 2′-Deoxyuridine Analogs Substituted in Position 5 with 2-Atom Tethered Nitroxide Radicals	David D. Kryak; Albert M. Bobst
1021-1043	Studies on the Synthesis of Furo[3,2-d]pyrimidine C-Nucleosides: New Inosine Analogues with Antiprotozoan Activity	Birendra K. Bhattacharya; Brian A. Otter; Randolph L. Berens; Robert S. Klein
1045-1060	Synthesis of Branched-Chain and Bicyclic Thiosugar Nucleosides	Stephen H. Kawai; Jik Chin; George Just
1061-1065	An Improved Synthesis of 2′,3′-Dideoxycytidine	V. Bhat; B. C. Ugarkar; K. Grirara; E. Stocker; P. A. Domenico; V. A. Sayeed; N. Kosora
1067-1078	Nucleosides and Nucleotides. 98. Synthesis and Antitumor Activities of 5-Ethynylimidazole-4-carboxamide and -carbonitrile Derivatives	Noriaki Minakawa; Akira Matsuda; Tohru Ueda; Takuma Sasaki
1079-1086	5′-Phosphorylation of Oligonucleotides with Phosphorous Acid in Automated DNA Synthesis	James C. Marsters; Peter Ng; Parkash Jhurani; Mark Yasser; Norbert Bischofberger
1087-1098	Studies on the Formation of the Internucleotidic Bond in RNA Synthesis Using Dialkylamino Phosphoroamidites	D. Gasparutto; D. Molko; R. Teoule
1099-1112	Novel 2.6-Disubstituted Adenosine Analogues: Potential Agonists for Adenosine Receptors	Vasu Nair; Allen J. Fasbender
1113-1122	Synthesis and Properties of an Initiation Codon Analog Consisting of 2′-O-Methyl Nucleotides	Ichiro Hirao; Mitsuharu Okubo; Masahide Ishikawa; Kin-Ichiro Miura

Volume 9, Issue 7 (1990)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 9, Number 7
875-884	The Synthesis of Aminopyri Dine-Based Phosphonoacetates as ADP Analogs	Michael D. Ennis; Mark E. Baze
885-897	The Use of Acetyl Bromide for the Multigram Synthesis of the Anti-HIV Agent 2′,3′-Didehydro-2′,3′-Dideoxycytidine (d4C)	John E. Starrett Jr; David R. Tortolani; David C. Baker; Mahrooud T. Omar; Anna K. Hebbler; John A. Wos; John C. Martin; Muzammil M. Mansurl
899-905	The Synthesis of 2-Nitro-1-[(2-Hydroxyethoxy)Methyl]Imidazole (Azomycin Acyclonucleoside)	Prem C. Srivastava; Ahmad Hasan
907-912	1,3,5-Tri-O-acetyl-2-deoxy- α, β-D-ERYTHRO-Pentofuranose from 2-Deoxy-D-ERYTHRO-Pentose	Avram Gold; R. Sangaiah
913-922	The Synthesis of Two Novel Ring-Expanded Xanthine Nucleosides Containing the Imidazo[4,5-e][1,4]Diazepine Ring System	Ramachandra S. Hosmane; Anila Bhan
923-935	Synthesis and Anticancer Activity of 3-(3-Oxoprop-1-enyl)-Substituted Analogues of Carbocyclic Pyrimidine Nucleosides and 2′,3′-Dideoxy Pyrimidine Nucleosides	Tai-Shun Lin; Ji-Yu Guo; Xiao-Hui Zhang
937-956	C-Glycosylation of Substituted Heterocycles Under Friedel-Crafts Conditions (II): Ribosylation of Multi-Functionalized Thiophenes and Furans for the Synthesis of Purine-Like C-Nucleosides	Shirish A. Patil; Brian A. Otter; Robert S. Klein
957-966	Selective Attachment of Oligonucleotides to Interleukin-1β and Targeted Delivery to Cells	André Chollet
967-983	Differentiation of Isomeric Purine and Pyrimidine Mononucleotides by Fast Atom Bombardment Tandem Mass Spectrometry	Terence J. Walton; Dipankar Ghosh; Russell P. Newton; A. Gareth Brenton; Frank M. Harris
985-1000	5′-O-[N-(Amnoacyl)Sulfamoyl]Nucleosides. Synthesis and Antiviral and Cytostatic Activities	Julia Castro-pichel; Ma. Teresa García-López; Rosario Herranz; Concepción Pérez

Volume 9, Issue 6 (1990)

a	Editorial board page for “Nucleosides, Nucleotides & Nucleic Acids”, Volume 9, Number 6
745-769	A New Synthesis of the Potent and Selective Anti-Herpesvirus Agent (S)-1-[3-Hydroxy-2-(Phosphonylmethoxy)Propyl]Cytosine	Joanne J. Bronson; Louis M. Ferrara; Henry G. Howell; Paul R. Brodfuehrer; John C. Martin
771-785	Synthesis of 5′-Deoxy-5′-nucleosideacetic Acid Derivatives	Kazuo Harada; Leslie E. Orgel
787-791	Carbocyclic Nucleoside Analogues. Synthesis and Properties of 1-(4-Hydroxymethyl-2-cyclopenten-1-YL)-Thymine	D. van Maarschalkerwaart; N. P. Willard; G. J. Koomen
793-802	The tRNA “Wobble Position” Uridines. IV. The Synthesis of 2′-O-Methyl-5-methoxycarbonylmethyluridine and its Derivatives	Elżbieta Sochacka; Andrzej Małkiewicz
803-813	1, N²-Ethenoguanosine: Three Methods of Synthesis	Jerzy Boryski
815-826	Synthesis and Antiviral Activity of the 3-Deaza Analogue of 9-((1, 3-Dihydroxy-2-propoxy)Methyl)Guanine	Danny P. C. McGee; John C. Martin; Donald F. Smee; Julien P. H. Verheyden
827-836	Conformation of Diastereomers of Adenosine Cyclic 3′, 5′-Phosphorothioate	K. S. Bruzik; A. Grajkowski; Z. J. Lesnikowski; G. M. Salamonczyk; W. J. Stec
837-846	Studies on Nucleosides: Part XXVIII¹. Synthesis of 4-Amino (or Hydroxy)-6-Methylthio-1-(3′-Deoxy-β- D-ribofuranosyl)-1-H-pyrazolo[3, 4-d]Pyrimidines	Shalini Misra; Sudha Jain; K. Avasthi; D. S. Bhakuni
847-859	The Synthesis of Novel 5-Trifluoroethyl Ethers of Thymidine	P. Kumar; L. I. Wiebe
861-873	The Synthesis of Novel 5-Trifluoroethoxy Pyrimidine Nucleosides	P. Kumar; L. I. Wiebe

Volume 9, Issue 5 (1990)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 9, Number 5
629-637	3-(3-Azido-2,3-Dideoxy-β-D-erythro pentofuranosyl)-thymine from 3′-Azido-3′-deoxythymidine (AZT). An Intriguing Rearrangement	Joanna M. Zeidler; Moon Hwan Kim; Kyoichi A. Watanabe
639-647	Synthesis and Antiviral Evaluation of Two New Carbocyclic Pyrrolo [2,3-d] Pyrimidine Nucleosides	Michel Legraverend; Christiane Huel; Aurelio Zerial; Marc Lemaitre; Emile Bisagni
649-662	Preparation and Antiviral Activity of Several Deoxygenated Ribavirin and Tiazofurin Derivatives	Krishna Upadhya; Jay Dare; Ernst M. Schubert; Gwendolyn N. Chmurny; Bjarne Gabrielsen
663-677	Synthesis and Biological Activity of Ara and 2′-Deoxycyclopentenyl Cytosine Nucleoside Analogues	Sung K. Kim; Richard W. Fuller; Victor E. Marquez
679-695	Natural and Phosphorothioate-Modified Oligodeoxyribonucleotides Exhibit a Non-Random Cellular Distribution	Marion Ceruzzi; Kenneth Draper; Jerome Schwartz
697-712	Acid-Catalyzed Hydrolysis of 2-Amino-9-(α-D-Ribofuranosyl)-purine and its Acyclo and 2-Methyl Analogues: Competition Between Depurination and Opening of the Imidazole Ring	Jari Hovinen; David Shugar; Harri Lönnberg
713-720	Synthesis of 5-Fluoro-1-(3-O-benzoyl-4, 6-dideoxy- β-L-GLYCERO-hex-3-enopyranos-2-ulosyl)uracil	Arun P. Sharma; Merilyn Blair; Abraham P. Ollapally
721-730	Synthesis and Murzne P388 Antitumor Activity of Uridine Mustard: A Preliminary Report	Abdol H. Talebian; Philip S. Schein; Dianna C. Green
731-744	Crystal Structure of 1-(2′,3′,5′-Tri -O-Acetyl-β-D-ribofuranosyl)-3-acetoxy-2-pyridone: An Antitumour Agent	A. K. Das; M. Ghosh; A. K. Basak; S. K. Mazumdar; R. A. Palmer

Volume 9, Issue 4 (1990)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 9, Number 4
479-488	The Effect of Exocyclic Substituents on Base-Pair Propeller Twist	C. C. Wilson
489-497	Pseudo-ADP: Darstellung und Biomimetische Eigenschaften	Martina Kinzig; Karl-Siegfried Boos
499-513	Crystal and Molecular Structures of the Antiviral Acyclonucleoside 9-[4-Hydroxy-3-(hydroxymethyl)butyl]guanine (BRL 39123, Penciclovir) and its Prodrug 9-[4-Acetoxy-3-(acetoxymethyl)butyl]-2-aminopurine (BRL 42810, Famciclovir)	Michael R. Harnden; Richard L. Jarvest; Alexandra M. Z. Slawin; David J. Williams
515-531	Dinucleoside Phosphates Containing Arabinose or Deoxyxylose. Hydrolysis by Exonucleases and Stacking Properties	N. I. Sokolova; N. G. Dolinnaya; N. F. Krynetskaya; Z. A. Shabarova
533-546	Aldol Reaction of Nucleoside 5′-Carboxaldehydes with Acetone. Synthesis of 5′-C-Chain Extended Thymidine Derivatives	María-José Camarasa; Federico G. De las Heras; María Jesús Pérez-Pérez
547-557	Synthesis and Structure of 2′,3′-Dideoxy-3′-fluoro-5-cyanouridine	A. A. Van Aerschot; D. H. Everaert; O. M. Peeters; N. M. Blaton; C. J. De Ranter; P. A. Herdewijn
559-568	Synthesis of (R - and (S)-1-[[2-Hydroxy-1-(aminomethyl)ethoxy]methyl]-5- benzyluracil, Potent Inhibitors of Uridine Phosphorylase	Tai-Shun Lin; Shi-Ping Xu; Mao-Chin Liu; William R. Mancini
569-577	The Enzymatic Synthesis of Imidazole Deoxynucleosides: 1-β-D-2′-Deoxyribofuranosyl-5-aminoiinidazole-4-carboxamide and 1-β-D-2′-Deoxyribofuranosylbenzimidazole	Didier Betbeder; David W. Hutchinson
579-585	Synthesis of 9-[(Phosphonomethoxy)methyl]guanine and 9-[2-Hydroxy-1-(phosphonomethoxy)ethyl]guanine	Choung Un Kim; Peter F. Misco; John C. Martin
587-597	Synthesis and Biological Activities of 3′-Deoxy-3′-Isocyano, -Isothiocyano, and -Isoselenocyano-thymidines	Akira Matsuda; Mutsumi Satoh; Tohru Ueda; Haruhiko Machida; Takuma Sasaki
599-618	Synthesis, Conformation and Hydrolytic Stability of p¹,p³-Dinucleoside Triphosphates Related to mRNA 5′-cap, and Comparative Kinetic Studies on their Nucleoside and Nucleoside Monophosphate Analogs	Edward Darzynkiewicz; Janusz Stepinski; Stanley M. Tahara; Ryszard Stolarski; Irena Ekiel; Dorota Haber; Kari Neuvonen; Pertti Lehikoinen; Imre Labadi; Harri Lönnberg
619-627	5′-C-Chain-Extended Adenosine Derivatives Related to Sinefungin. Synthesis and Biological Activity	John A. Secrist III; Ratnakar R. Talekar

Volume 9, Issue 3 (1990)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 9, Number 3
297-301	Structural Studies on Nucleic Acids: From Nucleotides to the Double Helix	Wolfram Saenger
303-310	NMR Analyses of Structures and Functions of Modified Nucleosides in Transfer Ribonucleic Acids	Shigeyuki Yokoyama; Tomonari Muramatsu; Gota Kawai; Tatsuo Miyazawa
311-317	Mass Spectrometry: Applications in the Analysis of Nucleosides, Nucleotides and Oligonucleotides	Karl H. Schram
319-330	High-Performance Electrophoresis Including Separation of Nucleic Acids and their Degradation Products. Interplay Between Theory and Practical Experiments	Stellan Hjertén
333-344	Fast Atom Bombardment and Tandem Mass Spectrometry for the Identification of Nucleoside Adducts with Phenyl Glycidyl Ether	J. Claereboudt; E. L. Esmans; E. G. Van den Eeckhout; M. Claeys
345-348	Comparison of the Molecular Structural Parameters in the Spermine-Bound and Spermine-Free DNA Octamer d(GTGTACAC). The Conformational Plasticity of DNA	M. Sundaralingam; S. Jain; G. Zon
349-354	X-Ray Studies of DNA Aiming at Elucidating the Sequence-Structure Code	Udo Heinemann
355-359	Applications of LC/MS and Tandem Mass Spectrometry to the Characterization of Nucleosides in Mixtures	Takeshi Hashizume; Chad C. Nelson; Steven C. Pomerantz; James A. McCloskey
361-364	Low Level, Detection of Modified DNA Bases and Nucleosides by FAB MS/MS	E. De Pauw; E. Marafante; J. Riego; C. Leuratti
365-368	Application of Fast Atom Bombardment Mass Spectrometry and Mass-Analysed Ion Kinetic Energy Spectrum Scanning to Studies of Cyclic Nucleotide Biochemistry	Russell P. Newton; A. Gareth Brenton; Terence J. Walton; Frank M. Harris; Dipankar Ghosh; Andrea M. Jenkins; Eric E. Kingston
369-372	N-Dimethylaminomethylene-O-trialkylsilyl Derivatives of Nucleosides for Chromatography and Mass Spectrometry	E. Y. Osei-twum; O. A. Mamer; M. A. Quilliam; R. Gergely
373-377	Unimlecular Depurination of Substituted Deoxyadenosines by Fast Atom Bombardment Mass Spectrometry/Mass Spectrometry	Angelo Liguori; Giovanni Sindona; Nicola Uccella
379-382	A High Field NMR Study of 2′-Deoxyribo-C-Nucleosides	P. Francois; E. Sonveaur; R. Touillaux
383-388	New Methods for the Solid-Phase Sequence Analysis of Nucleic Acid Fragments Using the Sanger Dideoxy Procedure	H. Seliger; G. Groger; G. Jirikowksi; F. Ramalho Ortigao
389-393	An Automated Coupled-Column HPLC-System for the Direct Analysis of Ribonucleosides and Ribonucleotides in Biological Fluids	K. -S. Boos; B. Wilmers; E. Schlimme; R. Sauerbrey
395-405	Determination of Nucleosides and their Adducts with RP-HPLC and (Laser-)Fluorescence Detection	D. Alders; R. M. Hoefnagel; M. M. Rhernrev-boom
407-410	Dual Column HPLC Analysis of Modified Ribonucleosides as Urinary Pathobiochemical Markers in Clinical Research	E. Schlimme; K. -S. Boos; E. Schwarzenau; H. Frister; F. -G. Ott; K. -P. Raezke; B. Wilmers
411-415	Base-Modified 2′-Deoxyribonucleosides in Bended DNA Fragments: Differential Bending at 3′- and 5′- Junctions of H- and B-DNA	F. Seela; H. Rosemeyer; T. Grein

Volume 9, Issue 3 (1990)

417-418	Configurational and Conformational Analysis of Regular and Modified Nucleosides by 1D-NOE Difference Spectroscopy	Helmut Rosemeyer; Frank Seela
419-422	Biodistribution of [⁷⁷Br]-5-Bromo-2-Deoxyuridine in Rats	E. Poupeye; P. Goethals; M. Coene; M. Van Eykeren; A. De Leenheer
423-427	Isolation and Characterization of Diastereomeric 2′-Oeoxy-ribonucleoside-3′-phosphoramidites	Klaus-Peter Stengele; Wolfgang Pfleiderer
431-434	Comparison of FAB and FD Mass Spectrometry in the Analysis of Unusually Linked Nucleotides	E. Arlandini; B. Gioia; M. G. Brasca; S. Fustinoni
435-436	Determination of 5-Fluorouracil and its Main Metabolites by Ion-Pair Liquid Chromatography on a Microbore Column	M. Barberi; J. L. Merlin; B. Weber
437-438	Electroanalytical Study on Nicotinamide 7-Methylguanine Dinucleotide (Nm⁷GD), Analog of Coenzyme NAD and Related Compounds	Elzbieta Bojarsk; Edward Darzynkiewicz; Piotr Ostapczuk; Jean-Marie Sequaris; Barbara Czochralsk
439-440	Comparison of Acid- and Enzyme-Catalyzed Cleavage of the Glycosidic Bond of N(7)-Substituted Guanosines	Agnieszka Bzowska; Ewa Kulikowska; David Shugar
441-442	Evaluation of 5-Carbamoylmethyluridine as an Indicator of Tumor Burden in Lung Cancer Patients	G. B. Chheda; J. G. Antkowiakt; H. Takitat; A. K. Bhargava; H. A. Tworek
443-444	Electrochemical Analysis of 3′-Azidothymidine (AZT)	Barbara Czochralska; Bozena Sapok; David Shugar
445-446	Time-of-flight Secondary Ion Mass Spectrometry of Branched RNA Fragrants: Messenger RNA Splicing Intermedistes	Francois Lafortune; Masad J. Damha; Xuejun Tang; Kenneth G. Standing; John B. Westmore; Kelvin K. Ogilvie
447-448	Combined UV and Liquid Scintillation Detection in HPLC. Formation and Depurination of Substitution Inert Pt(II) Complexes of Purine Nucleosides	Jorma Arpalahti; Rainer Käppi; Pejtti Lehikoinen; Harri Lönnberg
449-450	HPLC as a Tool to Study the Kinetics of Parallel and Consecutive Reactions: Competitive Interconversion, Dephosphorylation, Deamination and Depyrimidination of Cytidine 2′- and 3′-Monophosphates in Aqueous Acid	Mikko Oivanen; Harri Lönnberg
451-452	Acidic Hydrolysis of the N-Glycosidic Bonds of Deoxyribo-nucleic Acid by Hydrogen Fluoride Stabilized in Pyridine	M. Polverelli; M. Berger; J. -F. Mouret; F. Odin; J. Cadet
453-454	HPLC and Synthesis Strategy in Nucleoside and (Oligo)Nucleotide Chemistry	A. Pompon; F. Puech; G. Gosselin; J. L. Imbach
455-456	Chlorotetrolic Acid Ester as a Structural Probe of RNA	P. Roques; M. Olomucki
457-458	Rapid Ahalysis of Pseudouridine in Serum of Patients with Chronic Renal Failure, Using Phenylboronic Acid (PBA) Solid-Phase Extraction and HPLC	A. C. Schoots; J. H. M. Peeters
459-460	Computerized Interpretation of the Electron Ionization Mass Spectra of Nucleoside TMS Derivatives	Thomas D. McClure; Karl H. Schram
461-462	Mass Spectrometric Study of Modified Uridines and Their N³—Isomers	Marek Sochacki
463-465	Chromatography and Characterization of Phenylglycidyl Ether Nucleoside Adducts	E. G. Van den Eeckhout; E. L. Esmans; J. Claereboudt; J. Coene; M. Claeys
467-469	Molecular and Crystal Structure of d(CGCGmo⁴CG): N⁴-Methoxy-cytosineguanine Base Pairs in Z-DNA	L. Van Meervelt; M. H. Moore; P. Kong Thoo Lin; D. M. Brown; O. Kennard
471-472	Quantitative Analysis of Orotic Acid in Urine by RP-HPLC	B. Giordano; A. T. Cracco; V. Ferrari; N. Dussini; L. Chiandetti; F. Zacchello
473-477	NMR Study and Improvement of H-Phosphonate Oligonucleotide Synthesis	V. A. Efimov; I. Y. Dubey; O. G. Chakhmakhcheva

Volume 9, Issue 2 (1990)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 9, Number 2
151-162	Synthesis and Biological Activity of 6-Hydroxyguanidino-and 6-Hydroxyureidopurine And Their Ribonucleosides	Shib P. Dutta; Ralph J. Bernacki; Alexander Bloch; Girish B. Chheda
163-171	A Procedure for Analysing Nucleic Acid Fragment Geometry and Stacking Interactions	C. C. Wilson
173-177	A Possible Mechanism for the Base-Catalyzed Hydrolysis of Nucleoside Cyclic 3′,5′-Monophosphates	J. Tomasz
179-187	Detection of 5-Hydroxymethyl-2′-Deoxyuridine in Dna from Calf Thymus, Hela Cells, and Rat Liver Nuclei	Russell C. Cattley; Susan R. Dietze; Frank C. Richardson; James A. Popp
189-195	Convenient Regioselective Formation of 2′-O-Tosyladenosine	B. M. Ratnayake Bandara; Carl Bernofsky
197-204	Introduction of Fluorine Into the C8 Position of Purine Nucleosides	Peter C. Ratsep; Roland K. Robins; Morteza M. Vaghefi
205-221	Synthesis and Properties of Dinucleoside Monophosphates Containing 2-Aminoadenine 8,2′-S- and Uracil 6,2′-O-Cyclonucleosides	Masako Muraoka; Seizo Takahashi; Naoko Yamaguchi; Yasushi Oda; Seiichi Uesugi
223-233	8-Hydroxydeoxyguanosine in dna Inhibits Restriction Endonuclease Digestion	David S. Jones; Fumiko Nemoto; Yoshiyuki Kuchino; Eiko Ohtsuka; Susumu Nishimura
235-243	Crystal and Molecular Structure of ( )-Carba-Thymidine, C₁₁ H₁₀ N₂ O₆	Alajos Kálmán; Tibor Yoritsánszky; József Béres; Gyula Sági
245-258	A new Synthesis of 1-(2,3-Dideoxy-β-D-Glycero-Pent-2-Enofuranosyl)- Thymine. A Highly Potent and Selective Anti-Hiv Agent	J. -M. Vial; P. Agback; J. Chattopadhyaya
259-273	Solid Phase Non Isotopic Labelling of Oligodeoxynucleotides Using 5′- Protected Aminoalkyl Phosphoramidites: Application to the Specific Detection of Human Papilloma Virus Dna	Marie-Joelle De Vos; Alfredo Cravador; Jean-Pierre Lenders; Sophie Houard; Alex Bollen
275-291	Xanthine-7-Ribosides as Adenosine A_l Receptor Antagonists: Further Evidence for Adenosine's Anti Mode of Binding	Philip J. M. van Galen; Adriaan P. Ijzerman; Willem Soudijn

Volume 9, Issue 1 (1990)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 9, Number 1
1-19	Synthese de Tetrathymidylates Lies de Facon Covalente a des Derives de L'ellipticine	Claudie Gautier; Philippe Sizun; Tam Huynh-dinh; Abdelkader Namane; Claude Paoletti; Jean Igolen
21-34	Nucleocyclitols. Coupling of Heterocyclic Bases to Cyclitol Oxiranes	Raúl A. Cadenas; Margarita Yaber Grass; Jorge Mosettig; Maria E. Gelpi
35-41	An Unexpected Nucleophilic Displacement Involving 6-Bromo-4- chloro-5-cyanopyrrolo[2,3-d]pyrimidine with Methanolic Ammonia	Pranab K. Gupta; Sauro Vittori; Leroy B. Townsend
43-49	¹³C NMR Spectra of Some Ribose Alkylated Adenosine-5′-monophosphate Derivatives	Khurshid Alam Khan; Kaniz Fizza; Viqar-Uddin Ahmed
51-67	Syntheses of Triazole and Pyrimidine Homo-C-nucleosides	M. S. Pino González; F. J. López Herrera; R. Pabón Aguas; C. Uraga Baelo
69-79	Glycosides of Pyrido [2,3-c]-1,2,6-thiadiazine 2,2-Dioxides	A. de la Cruz; P. Goya; A. Martínez; J. A. Páez
81-87	Stereospecific Synthesis and Biological Evaluation of 9-α-D-Ribofuranosylguanine (α-Guanosine)	Gilles Gosselin; Marie-Christine Bergogne; Jean-Louis Imbach
89-96	The Synthesis of 5′-Homo-2′-deoxycytidine	Thomas E. Rawson; Thomas R. Webb
97-108	Synthesis of 2′,3′-Unsaturated and 2′, 3′-Dideoxy Analogs of 6-Azapyrimidine Nucleosides as Potential Anti-Hiv Agents	Tai-Shun Lin; Jing-Hua Yang; You-Song Gao
109-121	Synthesis of an Epoxide Derivative of Thymidine as a Potential Enzyme Inhibitor	H. Jeanette Thomas; Robert D. Elliott; James M. Riordan; John A. Montgomery
123-127	Biotinylation of Oligonucleotides Using a Water Soluble Biotin Ester	M. Bengtström; A. Jungell-nortamo; A-C. Syvänen
129-135	Nucleoside H-Phosphonates. XI. A Convenient Method for the Preparation of Nucleoside H-Phosphonates	Jacek Stawinski; Mats Thelin
137-149	Reaction of Glycosylisothiocyanates with 2-Chloroethylamine. Synthesis and Structure of N-Nucleoside Analogues	M. Avalos; R. Babiano; P. Cintas; J. Fuentes; J. L. Jimenez; J. C. Palacios

Volume 8, Issue 8 (1989)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 8, Number 8
iii-x	In Memory	Gary L. Grunewald; Robert P. Hanzlik
1379-1385	Preparation and Properties of the 5,6- and 4,6(5,7)-Dinitro Derivatives of Benzimidazole and their 1-β-D-Ribofuranosides	Zygmunt Kazimierczuk; David Shugar
1387-1398	Adducts of Mannose 6-Phosphate with 5-Iodo-2′-Deoxyuridine and 2-5A as Potential Antiviral Agents	Krystyna Lesiak; Erik De Clercq; Paul F. Torrence
1399-1415	Identification and Synthesis Of 5′-Deoxyxanthosine, a Novel Nucleoside in Normal Human Urine1	Thomas D. McClure; Karl H. Schram; Katsuyuki Nakano; Toshio Yasaka
1417-1426	3-Methyluridine in Normal Human Urine	Thomas D. McClure; Karl H. Schram
1427-1440	Novel Approach to the Ligation of Single-Stranded DNA Fragments by T₄ DNA Ligase—DNA Mobile Multiple-Restriction Fragments: “UNI-LINKERS” for Cloning of Genes	Fawzy Georges; Ravindra N. Chibbar; W. Jay Newsted; Friedrich Constabel
1441-1451	C-1′-Branched Acyclovir Derivatives. Synthesis and Antiviral Evaluation	Peter Scheiner; Aloma Geer; Ann Marie Bucknor; Hakan Gadler; R. W. Price
1453-1462	Labelling of DNA with a Non-Radioactive Analogue of dGTP	I. C. Gillam; G. M. Tener
1463-1471	A Short Syhthesis of 3′-(Methylsulfinyl)-3′-Deoxythymidine and Related Analogues	Muzammil M. Mansuri; John A. Wos; John C. Martin
1473-1483	The Behaviour of 2′-Deoxy-2′-Fluorouridine Incorporated into Oligonucleotides by the Phosphoramidite Approach	A. Krug; T. S. Oretskaya; E. M. Volkov; D. Cech; Z. A. Shabarova; A. Rosenthal
1485-1498	Nucleosides, XLVI¹ Syntheses and Reactions of 6- and 7-p-Chlorophenyllumazine Nucleosides	Najim A. Al-masoudi; Wolfgang Pfleiderer
1499-1512	The tRNA “WOBBLE POSITION” Uridines. III.¹ the Synthesis of 5-[S-Methoxycarbonyl (Hydroxy)Methyl] Uridine and its 2-Thio Analogue	Barbara Nawrot; Andrzej Malkiewicz
1513-1517	Determination of the Tautomeric Populations of the Y-Base	C. Glemarec; G. Remaud; J. Chattopadhyaya
1519-1528	Aminopyrimidines and Derivatives. 27¹.-Synthesis, Anticancer and Antimicrobiological Activities of 7-Glycopyranosyl-Pyrrolo[2,3-D]Pyrimidines²	M. L. Quijano; M. Nogueras; M. Melguizo; G. Alvarez de Cienfuegos; M. Melgarejo; A. Sánchez
1529-1535	An Improved Synthesis of 3′-Keto-5′-Tritylthymidine	M. L. Froehlich; D. J. Swartling; R. E. Lind; A. W. Mott; D. E. Bergstrom

Volume 8, Issue 7 (1989)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 8, Number 7
1179-1188	Nucleosides. 145. Synthesis of 2,5′-Anhydro-2-Thiouridine and its Conversion to 3′-O-Acetyl-2,2′-Anhydro-5′-Chloro-5′-Deoxy-2-Thiouridine. Studies Directed Toward the Synthesis of 2′-Deoxy-2′-Substituted arabino Nucleosides (7)	Ling-Ching Chen; Tsann-Long Su; Krzysztof W. Pankiewicz; Kyoichi A. Watanabe
1189-1200	Conformation and Antiherpes Activity of 3′- and 5′-Azido and Amino Analogs of 5-Methoxymethyl-2′-Deoxyuridine	Guy Tourigny; Allan L. Stuart; Irena Ekiel; Philip J. Aduma; Sagar V. Gupta
1201-1216	Synthesis of Tubercidin, 6-Chlorotubercidin and Related Nucleosides	Jack D. Anderson; Roger J. Bontems; Stewart Geary; Howard B. Cottam; Steven B. Larson; Steven S. Matsumoto; Donald F. Smee; Roland K. Robins
1217-1229	Evidence for the Stereoelectronic Control of the Acid Hydrolysis of Adenosine Cyclic 3′,5′-Phosphoramidate Diastereoisomers	S. Bottka; L. Radics; J. Tomasz
1231-1257	Synthesis and Biological Activity of the Mono- and Diamino Analogues of 2′-Deoxyadenosine, Cordycepin, 9-(3-Deoxy-α-D-Threo-Pentofuranosyl)-Adenine (A Structural Component of Agrocin 84) and 9-(2-Deoxy-α-D-Threo-Pentofuranosyl)Adenine	Piet Herdewijn; Jan Balzarini; Rudi Pauwels; Gerard Janssen; Arthur Van Aerschot; Erik De Clercq
1259-1269	Structural Features of 2′,3′-Dideoxy-2′,3′-Didehydrocytidine, A Potent Inhibitor of the HIV (AIDS) Virus	George I. Birnbaum; Jerzy Giziewicz; Tai-Shun Lin; William H. Prusoff
1271-1280	Ribosylation of 3-Methylguanine and the Relative Stability of its 7- and 9-α-D-Ribofuranosides	Jerzy Boryski; Tomasz Ostrowski; Bożenna Golankiewicz
1281-1285	An Unusual Iodine Monochloride Chlorination of an Imidazole Nucleoside	P. C. Srivastava; A. Hasan; R. Pratap; D. S. Bhakuni
1287-1296	An Unusual Reaction Observed in Sulfonylation and Acylation of 2′,3′-O-Isopropylidenenebularine	Hiroyuki Hayakawa; Hiroshi Ashizawa; Hiromichi Tanaka; Tadashi Miyasaka; Kentaro Yamaguchi
1297-1303	³¹P-¹⁵N One-Bond Couplings of Diastereoisomeric Adenosine Cyclic 3′,5′-Phosphoramidates	J. Tomasz; S. Bottka; L. Radics
1305-1317	9-(6-Deoxy- β -D-Allofuranosyl)Adenine Cyclic 3′,5′ -Phosphor-Amidate: A New Cyclic AMP Amide Derivative Containing an Equatorial Methyl Group at the 5′-Position	L. Radics; S. Bottka; J. Tomasz
1319-1324	Conversion of Methylthioadenosine Into its Naturally Occurring 3′-Isomer	Margherita Gavagnin; Guido Sodano
1325-1334	Synthesis of 5′-C-Chain-Extended Uridines by Reaction of 5′-Halonucleosides with Malonic Acid Type Derivatives	José Fiandor; María Teresa García-López; Federico G. De las Heras
1335-1343	Crystal and Molecular Structure of a Cytosine Analog; 5-Bromo-6-Benzylamino Isocytosine	Biswas Goutam; I. Iitaka; D. Shugar; Banerjee Asok
1345-1358	Nucleoside, XLV¹) Synthese von 8-β-D-Ribofuranosyl-Leukopterin	Leonidas Kiriasis; Wolfgang Pfleiderer
1359-1367	Efficient Preparation of Cyclic 3′,5′-Phosphoramidites and -Amidates of Antiviral and Antitumor 5-X-2′-Deoxyuridines (X = H, CH₃, I, F, CF₃, trans-CH=CHBr)	Wesley G. Bentrude; Mamunur R. Khan; M. R. Saadein; Alan E. Sopchik
1369-1377	Synthesis of 2′-Deoxyformycin B and 2′-Deoxyoxoformycin B	Vishnu C. Solan; Andre Rosowsky

Volume 8, Issue 5-6 (1989)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 8, Number 5-6
627-648	Sugar-Modified Oligonucleotides: Synthesis, Physicochemical and Biological Properties	Jean-Louis Imbach; Bernard Rayner; François Morvan
649-657	Synthesis and Properties of Novel 5′-Linked Oligos	Kenya Mori; Chris Subasinghe; C. A. Stein; Jack S. Cohen
659-671	Anti-Hiv-1 Activity of 2′,3′-Dideoxinucleoside Analogues : Structure-Activity Relationship	Erik De Clercq; Arthur Van Aerschot; Piet Herdewijn; Masanori Baba; Rudi Pauwels; Jan Balzarini
673-688	Phosphonylalkoxyalkyl and Phosphonylalkyl Derivatives of Heterocyclic Bases	Antonln Holý; Ivan Rosenberg
689-698	Elucidation of the Mechanism by Which 9-(Trans-2′, Trans-3′-Dihydroxycyclopent-4′-enyl)-Adenine Lnactivates S-Adenosylhomocysteine Hydrolase and Elevates Cellular Levels of Sadenosylhomocysteinew	Steven D. Paisley; Masahide Hasobe; Ronald T. Borchardt
699-708	Development of Methodologies for the Strategic Modification of Purim Ribonwxeoside System	Vasu Nair
709-724	USE OF THE SODIUM SALT GLYCOSYLATION HETBOD IN NUCLEOSIDE SYNTHESIS	Ganapathi R. Revankar; Roland K. Robins
725-741	Synthesis, Transformation Chemistry, and Biological Activity of Guanine Nucleosides and Analoges	Moms J. Robins; Ruiming Zou; Fritz Hansske; Danuta Madej; David L. J. Tyrrell
743-752	SYNTHESIS AND BIOLOGICAL ACTIVITY OF BRANCHED CHAIN-SUGAR NUCLEOSIDES¹	Tohru Ueda; Akira Matsuda; Yuichi Yoshimura; Kenji Takenuki
753-764	New Potent and Selective Inhibitors of Herpes Simplex Virus Tbyhidine Kinase	J. A. Martin; I. B. Duncan; M. J. Hall; P. Wong-Kai-In; R. W. Lambert; G. J. Thomas
765-774	Membrane Transport of Nucleoside Analogues in Mammalian Cells	Thomas P. Zimmerman; Barbara A. Domin; William B. Mahony; Karen L. Prus
775-785	2′,2′-Difluorodeoxycytidine Metabolism and Mechanism of Action In Human Leukemia Cells	William Plunkett; Varsha Gandi; Sherri Chubb; Billie Nowak; Volker Heinemann; Shin Mineishi; Alina Sen; Larry W. Herte; Gerald B. Grindey
789-792	Pyrazolo[3,4-d)Pyrimidine 2′-Deoxyribo and 2′,3′-Dideoxyribo-Furanosides: Synthesis and Application to Oligonucleotide Chemistry	F. Seela; H. Driller; K. Kaiser; H. Rosemeyer; H. Steker
793-797	Synthesis of Branched Oligoribonucleotides (“Lariat”)	N. Balgobin; X-X. Zhou; J-M. Vial; A. Nyilas; A. Földesi; J. Chattopadhyaya
799-803	The H-Phosphonate Method for Constructing Phosphodiester Linkages. A Progress Report	Jacek Stawiński; Roger Strömberg; Ingvar Lindh; Tor Regberg; Thomas Szabó; Mats Thelin; Erik Westman; Per J. Garegg
805-813	5-Bromouridinylated Oligonucleotide for Hybridization Analysis of DNA and RNA on Membranes and in Situ	J. F. Ramalho Ortlgao; G. F. Jirikowski; H. Seliger
815-818	The Intracellular and Extracellular Fate of Oligodeoxyribonucleotides in Tissle Culture Systems	Marion Ceruzzi; Kenneth Draper
819-823	Phosphoramidate, Phosphorothioate, and Methylphosphonate Analogs of Oligodeoxynucleotide : Inhibitors of Replication of Human Immunodeficiency Virus	Sudhir Agrawal; John Goodchild; Maria Civeira; Prem S. Sarin; Paul C. Zamecnik
825-828	Antiviral activity of antisense oligonucleotides linked to poly(L-lysine):targets on genomic RNA and/or mRNA of Vesicular Stomatitis Virus	Jean-Paul Leonetti; Genevieve Degols; Pierre Milhaud; Corinne Gagnor; Marc Lemaitre; Bernard Lebleu
829-832	Acycloadenosine Derivatives as Inhibitors of 5′-Deoxy-5′-Methylthioadenosine Phosphorylase (MesADo PASE)	Shih-Hsi Chu; Zhi-Hao Chen; Todd M. Savarese; Charles E. Nakamura; Robert E. Parks Jr.; Elie Abushamb
833-836	EFFECT OF PHOSPHONIC ACID ANALOGS OF ACYCLOVIR AND GANCICLOVIR ON IN VITRO CYTOMEGALOVIRUS INFECTIONS	Robert W. Sidwell; John H. Huffman; Dale L. Barnard; Elmer J. Reist
837-840	Synthesis and Evaluation of Antiviral Activity of 3′-C-Cyano-3′-Deoxynucleosides	María-José Camarasa; Angel Díaz-Ortíz; Ana Calvo-hateo; Pederico G. De las Heras; Jan Balzarini; Erik de Clercq
841-844	Synthesis, Anti-Hiv Activity, and Biological Properties of 2′,3′-Didehydro-2′,3′-Dideoxythwidine (d4T)	John C. Martin; Muzammia M. Mansuri; John E. Starrett Jr.; Jean-Pierre Sommadossi; Vera Brankovan; Ismail Ghazzouli; H-T. Ho; Michael J. M. Hitchcock
845-848	Pharmacokinetics of A New Anti-HIV Ageht: 2′,3′-Dideoxy-2′,3′-Didehydrothymidine (d4T)	J. W. Russell; V. J. Whiterock; D. Marrero; L. J. Klunk
849-853	Synthesis and Biological Applications of 2′,3′-Dideoxynucleoside-5′-O-(α-thio)Triphosphates	M. Auer; C. Kriege; M. Gautel; S. Labeit; G. Sczakie; S. Weisz; R. S. Goody
855-858	Synthesis and Biological Properties of ( ) and (-)-(E)-5-(2-bronovinyl)-2¹ -deoxy-1¹ a-Carbauridine	Jan Balzarini; Harald Baumgartner; Michael Bodenteich; Erik De Clercq; Herfried Griengl
859-862	Synthesis of Novel Polycyclic Nucleoside Analogs	Norbert Bischofberger; Mark D. Matteucci
863-866	Apurinic DNA: Modelisation and Reactivity Towards 9-Aminoellipticine and Related Amines	Jean-Jacques Vasseur; Bernard Rayner; Jean-Louis Imbach; Jean-Remi Bertrand; Claude Malvy; Claude Paoletti

Volume 8, Issue 5-6 (1989)

867-870	Regiocontrolled General Synthesis of Branch-Type 2′-5′-Linked Oligoadenylates	Y. Hayakawa; M. Hirose; R. Noyori
871-874	Base Analogues Related to N⁴-Hydroxicytosine	Paul V. S. Kong; Thoo Lin; D. M. Rrown
875-877	The Synthesis of Branched Oligonucleotides as Signal Amplification Multimers for Use in Nucleic Acid Assays	Thomas Horn; Brian D. Warner; Joyce A. Running; Kristi Downing; Jennifer Clyne; Mickey S. Urdea
879-883	Site-Specific ¹³C Labeling of DNA to Deduce DNA Repair Mechanisms of Uracil-DNA Glycosyiase and UV Endonuclease V	M. Manoharan; S. C. Ransom; A. Mazumder; J. A. Gerlt
885-886	Synthesis of Glycofuranosyl - formamides, -isocyanides and - isocyanates - Useful synthons for new approaches to nucleosid analogues	Johann Hebl; Johann Polsterer; Erich Zbiral
887-890	Synteesis of Certain C-4 Substituted Pyrazolo[3,4-b]-Pyridine Nucleosides Structurally Related to Adenosine and Inosine by Tee Sodiw Salt Glycosylation Procedure	Yogesh S. Sanghvi; Steven B. Larson; Roland K. Robins; Ganapathi R. Revankar
891-894	Synthesis and Biological Evaluation of 2-Carbamoyl-5-D-Ribofuranosylpyridine	F. C. Alderweireldt; I. Vrijens; E. L. Esmans; L. L. Wotring; L. B. Townsend; J. Balzarini; E. De Clercq
895-898	Sulfur Isosteres of Orotidine	Subhasish Purkayastha; Gabriel Menichi; Raymond P. Panzica
899-902	Novel Acyclic Derivatives of Aica-Riboside (1-(β-D-Ribopuranosyl)5-Amino-4-Imidazolecarboxamide), Potential Antiviral Agents	Thomas I. Kalman; D. Michael Houston
903-906	A General Synthetic Method for 2′,3′-Dideoxynucleosldes: Total Synthetic Approach	Chung K. Chu; Ramesh Raghavachari; J. Warren Beach; Yoshiyuki Kosugi; Giliyar V. Ullas
907-910	Unsaturated Nucleoside Analogues: Synthesis and Antitumor Activity	Shashikant Phadtare; David Kessel; Jiri Zemlicka
911-913	8-Substituted Purine Ribosides: Synthesis and Biological Activity	Anita T. Shortnacy; John A. Montgomery; John A. Secriist III
915-917	Synthesis and Antiviral Evaluation of Adenosine-N¹-Oxide and 1-(Benzyloxy) Adenosines	Charles A. Krauth; Anita T. Shortnacy; John K. Montgomery; John A. Secrist III
919-922	Synthesis of Phosphonic Acid Analogs of Acyclovir (ACV) and Canciclovir (DHPG)	Elmer J. Reist; Priscilla A. Sturm; Ronald Y. Pong; Robert W. Sidwell
923-926	Synthesis and Antiherpesvirus Activity of (S)-1-((3-Hydroxy-2-Phosphon-Ylmethoxy)Propyi.)Cytosine (HPMPC) and Related Nucleotide Analogues	John C. Martin; Joanne J. Bronson; Robert R. Webb II; Michael M. J. Hitchcock; Ismail Ghazzouli
927-931	Synthesis and Biological Activities of Phosphonylalkylpurine Derivatives	Choung Un Kim; Bing Yu Luh; Peter F. Misco; Joanne J. Bronson; Michael J. M. Hitchcock; Ismail Ghazzouli; John C. Martin
933-937	Some Examples of the Use of Trifluoromethane Sulfonic Anhydride in Nucleic Acid Chemistry	P. Herdewijn; A. Van Aerschot
939-941	Isomerization of Cytidine 2′,3′-Thionocarbonates	L. W. Dudycz
943-946	Synthesis of Some 2-Alkylated-5-Aminoimidazoles Related to Intermediates in Purine Nucleotide de novo and Thiamine Biosynthesis	Grahame Mackenzie; Hilary A. Wilson; Robert W. Humble; Fawzy Hewedi; Gordon Shaw; David Ewing
947-950	The Synthesis of 1-[7,8-Anhydr0-2,5,6-trideoxy-β-D-allo (and α-L-Talo)-Octofuranosyl]-Thymine as a Potential Enzyme Inhibitor	H. Jeanette Thomas; James M. Riordan; Robert D. Elliott; John A. Montgomery
951-955	Synthesis, Cytotoxicity and Metabolism of the 2′,2′-Difluoro-Analogs of Deoxyadenosine (dFdA)and Deoxyguanosine (dFdG)	L. W. Hertel; C. S. Grossmana; J. S. Kroina; S. Mineishi; S. Chubb; B. Nowak; W. Plunkett
957-960	An Unusual Dephosphorylation Reaction	Anne F. Cichy; Purushotham Vemishetti; Elie Abushanab
961-965	Syntiiesis of New 3′-Amino-2′,3′-Dideoxynucleosides in Five Steps Starting from Peracetylated Clycals	Jesper Lau; Erik B. Pedersen; Jesper Wengel
967-968	Synthesis of Anti-Sense Phosphorothioate Analogues for Pharmacokinetic and Pre-Clinical Studies	Alex Andrus; Timothy Geiser; Gerald Zon
969-973	Renal Deoxyadenosine Transport and Immunodeficiency Associated with Adenosine Deaminase Deficiency	J. Arly Nelson
975-978	Control of Differentiation by GTP	Ernst Freese
979-982	Enzymatic Synthesis of Radioactive 5-Methyl-2′-Deoxycytidine 5′-Monophosphate by Using ³²P-Postlabeling	Juhani A. Vilpo; Leena M. Vilpo
983-986	Biosynthesis of the Naturally Occurring Nucleoside Antibiotics from Adenosine	Robert J. Suhadolnik; Jeffery C. Hanvey; Somchai Pornbanlualap; Joseph M. Wu; Kamal N. Tiwari; Anna K. Hebbler; David C. Baker
987-990	Phosphorothioate Analogs OF 2-5A: Activation / Inhibition of Rnase L and Inhibition of HIV-1 Reverse Transcriftase	Robert J. Suhadolnik; Bernard Lebleu; Wolfgang Pfleiderer; Ramamurthy Charubala; David C. Montefiori; William M. Mitchell; Robert W. Sobol Jr.; Shi Wu Li; Katalin Kariko; Nancy L. Reichenbach
991-994	Design and Chemoenzymatic Synthesis of A Tissue Plasminogen Activator Gene with Unique Restriction Sites: A Model for Studying Protein Domain Function	N. Theriault Hatzenbuhler; E. F. Rehberg; J. B. Carter; D. P. Palermo; E. V. Hubert; P. W. Bergum; L. A. Erickson; K. R. Marotti

Volume 8, Issue 5-6 (1989)

995-1000	Alpba-Oligodeoxynucleotides as Inhibitors of HIV Reverse Transcriptase	R. Pauwels; Z. Debyser; J. Balzarini; M. Baba; J. Desmyter; B. Rayner; F. Morvan; J. L. Imbach; E. De Clercq
1001-1006	New Results in Oligoribonucleotide Synthesis	Magdalena Pfister; Wolfgang Pfleiderer
1007-1010	Stereochemical Problems in Oligonucleotide Synthesis	R. Charubala; K. P. Stengele; W. Pfleiderer
1011-1014	Synthesis of Oligodeoxynlicleotides Containing Specific Methylphosphonothioate and Dithioate Moieties	W. K. -D. Brill; M. H. Caruthers
1015-1018	Synthesis of Oligonucleotides Containing 5,6-Dihydro-5-Azacytosine and 5-Azacytosine at Specific CpG Sites	Amanda J. Goddard; Victor E. Marquez
1019-1022	General Synthesis of 2′(3′)-O-Aminoacyl Oligoribonucleotides Related to the 3′-Terminus of aa-tRNA	Michael D. Hagen; Stanislav Chlàdek
1023-1027	Synthetic Approaches to Oligodeoxyribonucleoside Phosphorodithioates Using Tervalent Phosphorus Monomers	Bjarne H. Dahl; Kirsten Bjergårde; Vibeke B. Sommer; Otto Dahl
1029-1032	Recent Studies in Nucleoside Phosphonate Chemistry	Jacek Stawinski; Roger Strömberg; Tomas Szabó; Erik Westman
1033-1036	Use of New Phosphonylating and Condensing Agents in The Synthesis of Oligonucleotides Via The H-Phosphonate Approach	Osamu Sakatsume; Hiroshi Yamane; Hiroshi Takaku
1039-1040	Inhibition of Purine Nucleoside Phosphorylase by Phosphonoalkylpurines ¹	Charles E. Nakamura; Shih-Hsi Chu; Johanna D. Stoeckler; Robert E. Parks Jr.
1041-1042	Rapid Synthesis of 2′ and 3′ Fluorinated Nucleotides and Their Use in ¹⁹F-NMR-Spectroscopy of Nucleotide-Binding Enzymes	M. Auer; P. Röisch; G. Sczakiel; R. S. Goody
1043-1044	2 and 8-Azido ATP: Photoaffinity Labeling of 2-5A Synthetase, Enzymatic Synthesis of 2 and 8-Azido Anamgs of 2-5A for Use as Photoaffinity Probes of Rnase L	Shi Wu Li; Robert W. Sobol Jr.; Nancy L. Reichenbach; Katalin Kariko; Boyd E. Haley; Robert J. Suhadolnik
1045-1046	Use of A Uridine Nucleotide as an Affinity Handle and 5′ Phosphorylating Agent for Synthetic DNA	E. Higgins; J. S. Debear; P. C. Andrews; G. R. Gough
1047-1048	Large Scale HPLC Purification of Oligodeoxyribonucleotides for Studies of the Binding of CC-1065 to DNA by NMR Spectroscopy	S. P. Pulaski; N. Theriault Hatzenbuhler; T. A. Scahill; N. Richter
1049-1050	Sequence Preference of Acridine Interaction with Single and Double Stranded Octadeoxyribonucleotides	I. Lassalle; P. A. Hoyos; S. R. Byrn; H. L. Weith
1051	The Incorporation of 2,6-Diaminopurine Into Oligodeoxyribonucleotides by the Phosphoramidite Method	Tom Brown; Alister G. Craig
1053-1054	The Synthesis of αβ Imidothymidine Diphospate	Lawrence C. Davies
1055-1056	A Solid-Phase Synthesis of 2′,5′-Linked Oligoadenylates (2-5A)	Krystyna Lesiak; Bogdan Uznanski; Paul F. Terrence
1057-1059	Synthesis of (Dicarbonyl)(η⁵-cyclopentadieny1)iron -Derived Nucleoside Phosphonate Esters	Don Bergstrom; Theresa Schmaltz
1061-1063	Synthesis of (Dicarbonyl)(η⁵-cyclopentadienyl)Manganese Complex Stabilized Nucleoside Phosphite Esters	Don Bergstrom; Peter; Robert Lind
1065-1068	Deprotecton Studies of Ethanoic Acid 5,6,7,9-Tetrahydro-3-/2-(Acetoxyemxy Iethyl-5-0-Acetyl-9-OXO-3H-IMIDAZO/1,2a/ Purine-6,7-Dioyol Ester (1) and Related Glyoxal-Guaniee Adduts	J. Plavec; A. Štimac; A. Šmidovnik; J. Kobe
1069-1070	2,3-Dideoxy-3-Phthalimidopentoses in the Synthesis of 3′-Amino-2′,3′-Dideoxynucleosides	Erik B. Pedersen; Mohammed S. Motawia; Erik S. Andreassen; Jesper Wengel; Jesper Lau
1071-1072	Photochemistry of the O-Nitrobenzyl Protecting Group in RNA Synthesis	J. A. Hayes; G. R. Gough; P. T. Gilham
1073-1074	C-5 Substituted Pyrimidine Nucleosides, Synthesis of 5-Alkylglycoside Deoxyuridine and Uridine Analogs VIA Organopalladium Intermediates	Sylvie Pochet; Simon R. Satfati; Jean Igolen
1075-1076	Synthesis of 2′ -Deoxypyrihidine Nucleosides Via Copper (I) Iodide Catalysis	John N. Freskos
1077-1078	The Role of Molecular Oxygen in the Catalytic Hydrogenation of Hydrazinonucleosides to the Corresponding Aminonucleosides	Vaidyanathan K. Iyer
1079-1080	The Synthesis of Pyrazol0[3,4-c]Pyridine C-Nucleosides	Daryl R. Sauer; Stewart W. Schneller
1081-1082	The Synthesis of the Carbocyclic Derivative of lin-Benzo-Separated 2′,3′-Dideoxyinosine	James W. Leahy; Stewart W. Schneller
1083-1084	A Convenient Synthesis of 9-(5′-DEOXY-β-D-Allofuranosyl)-Adenine (5′-Homoadenosine)	Ellen M. Salcines; Stewart W. Schneller
1085-1086	The Synthesis of Derivatives of 2-Arylamino ara-Carbocyclic Purine Nucleosides as Potential Anti-Viral Agents	Masakazu Koga; Stewart W. Schneller

Volume 8, Issue 5-6 (1989)

1087-1088	Synthesis Of Pyrrolo[2,3-b]Pyridine Nucleosides by Solid-Liquid Phase-Transfer Clycosylation and Deoxycenation of 4-Chloropyrrolo[2,3-d]Pyrimidine 2′-Deoxyribofuranosides	F. Seela; R. Cumbiowski; H. -P. Muth; W. Bourgeois
1089-1090	Synthesis of Pyrrolo[3,2-C]Pyridine 2′-Deoxy-D-Ribo-, 2′,3′-Dideoxy-D-Ribo-, and D-Arabinofuranosyl Nucleosides	F. Seela; W. Bourgeois; T. Jürgens
1091-1092	Unambiguous Assignment of Anomeric Configuration of Nucleosides by Noe-Difference Spectroscopy	Cábor Tóth; Helmut Rosemeyer; Frank Seela
1093-1095	Novel Acyclic Analogues of 3′-Azido-3′ Deoxythymidine 1-Hydroxy-3-Azido-2-Propoxymethyl Derivatives	H. B. Lazrek; M. Taourirte; J. -L. Barascut; J. -L. Imbach
1097-1100	Synthesis of Acyclic Nucleoside Using Potassium Iodide as Catalyst	H. B. Lazrek; N. Redwane; J. -L. Barascut; J. -L. Imbach
1101-1102	Investigation of the Synthesis of 2-Carbamoylmethyl-6-D-Ribofuranosylpyridine	E. De Vos; E. L. Esmans; F. C. Alderweireldt; J. A. Lepoivre
1103-1105	Progress in the Synthesis of A Potential PNP Transition State Inhibitor	Robert D. Elliott; Shri Niwas; John A. Montgomery; John A. Secrist III
1107-1108	Synthesis of 3′-C-Substituted-2′,3′-Dideoxynucleosldes as Potential Antcaids Agents	J. Fiandor; D. M. Huryn; B. Sluboski; L. J. Todaro; S. Tam
1109-1110	Synthesis and Evaluation of 2′,3′-Dideoxy-9-Deazaadenoslne and Some Related Derivatives	S. Tam; M. Holman; R. S. Klein; M. Mitsuya; S. Broder
1111-1114	Synthesis and Biological Evaluation of Dideoxunucleosides Containing A Difluoromethylene Unit	Esa T. Jarvi; Prasad S. Sunkara; Terry L. Bowlin
1115-1117	1-(2,3-Dideoxy-3-Fluoro-β-D-Ribofuranosyl)Tine (FDDT). Improved Preparation and Evaluation as a Potential Anti-Aids Agent	R. Sterzycki; M. Mansuri; V. Brankovan; R. Buroker; I. Ghazzouli; M. Hitchcock; J-P. Somrnadossi; J. C. Martin
1119-1120	Phosphate Modified Analogues of 5′-O-Phosphorylated 2′,3′-Dideoxynucleosides: Synthesis and Anti-HIV Activity	Robert M. Rigs; Robert N. Comber; John A. Montgomery; John A. Secrist III; Janet M. Leeds; Sara Chaffee; Michael S. Hershfield
1121-1122	Influence of Fluorination of the Sugar Moiety on the Anti-HIV-1 Activity of 2′,3′-Dideoxynucleosides	Arthur Van Aerschot; Jan Balzarini; Rudi Pauwels; Luk Kerremans; Erik De Clercq; Piet Herdewijn
1123-1124	Synthesis of 3′-Fluoro-3′-Deoxyribonucleosides; Anti-HIV-1 and Cytostatic Properties	Arthur Van Aerschot; Jan Balzarini; Erik De Clercq; Piet Herdewijn
1125-1126	Sugar and Base-Modified 2′,3′-Dideoxynucleosides as Potential Anti-Aids Drugs	Arthur Van Aerschot; Jan Balzarini; Rudi Pauwels; Piet Wigerinck; Erik De Clercq; Piet Herdewijn
1127-1128	Carbovir: A Carbocyclic Nucleoside with Potent and Selective Activity Against Human Immunodeficiency Virus (HIV) in Vitro	Robert Vince; Mel Hua; Jay Brownell; George C. Lavelle; Jeanine Qualls; William M. Shannon
1129-1130	6,6′-Bis-[1-(6-Deoxy-β-D-Galacopyranosyl) Uracil] - A Tunicaminyl Uracil Analogue : Synthesis and Preliminary Biological Evaluation	M. Ariatti
1131-1133	Cyclopentenyl Cytosine (CPE-C). A Carbocyclic Nucleoside with Antitumor and Antiviral Properties	John S. Driscoll; Victor E. Marquez; Jacqueline Plowman
1135-1140	Synthesis and Biological Activity of Various Selenenyl and Tellurenyl-Substituted Deoxyuridines and Deoxyuridylates	Ralph J. Cisneros; Louis A. Silks III; Jerome D. Odom; R. Bruce Dunlap
1141-1142	Synthesis and Biological Activity of Certain 4-Substituted Imidazo[4,5-d]Pyridazine Nucleosides	Kakarla Ramesh; Raymond P. Panzica
1143-1144	Synthesis and Biological Evaluation of 4-Amino-1-β-D-Ribofuranosylpyrrolo[3,2-c]Pyriding (3-Deazatubercidin)	P. Franchetti; G. Cristalli; M. Grifantini; E. Nasini; S. Vittori
1145-1146	Synthesis of O-Benzyl Derivatives of 2′-Deoxy-5-Trifluoromethyluridine for Antitumor Agents	Jun-Ichi Yamashita; Hiroshi Matsumoto; Kazuhiro Kobayashi; Kazuharu Noguchi; Mitsugi Yasumoto; Tohru Ueda
1147-1151	Comparative Efficacy of Nucleoside Analogues Against African Swine Fever Virus “in Vitro”	Alessandra Pani; M. Elena Marongiu; Paolo La Colla
1153-1154	Synthesis of 5′-Substituted Analogues of Carbocyclic 3-Deazaadenosine as Potential Antivirals	J. A. Secrist; R. M. Brash; R. J. Gray; R. N. Comber; J. A. Montgomery
1155-1156	The Synthesis and Preliminary Biological Evaluations of Selected Analogues of the Potent Broad-Spectrum Antiviral Agent Ganciclovir 1′,3′-Cyclic Monophosphate¹ (2′-Nor-cGMP)	M. Maccoss; A. F. Wagner; C. L. Cantone; R. A. Strelitz; A. Chen; W. T. Ashton; J. Hannah; R. L. Tolman; R. Bostedor; J. Germershausen; J. D. Karkas; H. C. Perry; A. K. Field
1157-1158	A Potent, Selective, Non-Substrate Inhibitor of HSV-I Thymidine Kinase: (±)-9-[[(Z)-2-(Hydroxymethyl)Cyclohexyl]Methyl]Guanine and Related Compounds	W. T. Ashton; L. C. Meurer; R. L. Tolman; J. D. Karkas; R. Liou; H. C. Perryt; S. M. Czelusniak; R. J. Klein
1159-1160	In Vitro and in Vivo Phlebovirus Inhibition by Nucleosides Related to Ribavirin	John H. Huffman; Robert W. Sidwell; Roland K. Robins; Ganapathi R. Revankar; Dominique Y. Pifat
1161-1163	Synthesis and Use of New Digoxicenin- Meled Hucleotides in Non-Radioactive Labeling and Detection of Nucleic Acids	K. Mühlegger; H. -G. Batz; S. Böhm; H. V. D. Eltz; H. -J. Höltke; Ch. Kessler
1165-1167	A New Option in Solid Phase Synthesis of DNA-Fragments	S. Berner; G. Gröger; K. Mühlegger; H. Seliger
1169-1173	Queuine Content of Hematopoietic and Neuronal Tissues	W. R. Farkas; B. J. Lifsey; T. J. Siard
1175-1176	Synthesis of Reagents for Fluorescence-Tagging of DNA	George L. Trainor; Frank W. Hobbs; Anthony J. Cocuzza; Pat N. Confalone
1177-1178	2-Deoxy-D-Ribofuranosylation of Ethyl 5-Aminoimidazole-4-Carboxylate by Biotransformation and Chemical Methods	David Ewing; Robert W. Humble; Antonin Holy; Grahame Mackenzie; Gordon Shaw; Ivan Votruba

Volume 8, Issue 4 (1989)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 8, Number 4
449-461	Adenosine Receptor Agonists. X-Ray Crystal Structure of Neca 1-(6-Amino-9H-Purin-9-Yl)-1-Deoxy-N-Ethyl-β-D-Ribofuranuronamide	Walter H. Moos; Harriet W. Hamilton; Daniel F. Ortwine; Michael D. Taylor; Andrew T. McPhail
463-474	On the Application of t-Butyldimethylsilyl Group in Chemical RNA Synthesis. Part I. ³¹P NMR Study of 2′-O-t-BDMSi Group Migration During Nucleoside 3′-OH Phosphorylation and Phosphitylation Reactions	Jan Milecki; Piotr Dembek; Wieslaw Z. Antkowiak; Zofia Gdaniec; Slawomir Mielewczyk; Ryszard W. Adamiak
475-489	Acyclic Nucleosides. Synthesis and Antiherpetic Activity of 9-[[[2-Hydroxy-1-(Hydroxymethyl)Ethyl]Thio]Methyl]Guanine and 1-[[[2-Hydroxy-1-(Hydroxymethyl)Ethyl]Thio]Methyl]Cytosine	James L. Kelley; James A. Linn; Lilia Beauchamp; Peter Collins; J. W. T. Selway; Karen K. Biron; Howard J. Schaeffer
491-497	Synthesis of 3′-O-Propargylthymidine as a Candidate Antiretroviral Agent	Andre Rosowsky; Ruth M. Ruprecht; Vishnu C. Solan
499-504	A Convenient Approach to the Synthesis of Azido-Acyclic Nucleosides	Takashi Ogawa; Hiroshi Takaku; Naoki Yamamoto
505-514	Synthesis and Biological Effects of 5′-Deoxy-5′-(Cyclo-Propylmethylthio)Adenosine	Janice R. Sufrin; Arthur J. Spiess; John F. Karny; Debora L. Kramer; Robert G. Hughes Jr; Ralph J. Bernacki; Carl W. Porter
515-528	Synthesis of Bridged Pyrimidine Nucleosides and Triazo [4, 3-c] Pyrimidine Nucleoside Analogues	Stefania Barbato; Gennaro Piccialli; Ciro Santacroce; Lorenzo De Napoli; Luciano Mayol
529-536	Application of the Transpuriation Reaction to Synthesis of Acyclic Guanosine Analogues	Jerzy Boryski; Bożenna Golankiewicz
537-547	Hydrogen Atom Location in the Modified Nucleic Acid Base 3-Deazauracil by Neutron Powder Diffraction	J. W. Wadsworth; C. C. Wilson; W. I. F. David
549-555	Synthesis of 2′-Deoxypyrimidine Nucleosides via Copper (I) Iodide Catalysis	John N. Freskos
557-567	Synthesis of Cytidylyl(3′→5′)cytidylyl(3′→5′)-(2′)3′-O-[Lα-alanyl]adenosine	A. Nyilas; A. Földesi; J. Chattopadhyaya
569-586	Differential Sensitivities of Normal and Malignant Murine Lymphocytes to Purine Nucleosides	J. Arly Nelson; Ellen R. Richie; Osama Kandil; Elena Vidale; Bih Fang Pan
587-597	Assignment of Anomeric Configuration of D-Ribo-, Arabino-, 2′-Deoxyribo-, and 2′,3′-Dideoxyribonucleosides by Noe Difference Spectroscopy	H. Rosemeyer; G. Tóth; F. Seela
599-617	Nucleosides, XLIV¹ Synthesis, Properties and Biological Activity of Indazole Nucleosides	Zygmunt Kazimierczuk; Harri Lönnberg; Juhani Vilpo; Wolfgang Pfleiderer
619-624	The Bis-Trityl Route to (S)-HPMPA	Robert R. Webb II

Volume 8, Issue 3 (1989)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 8, Number 3
307-315	Synthesis and Biological Evaluation of a Series of Substituted Pyridine-C-Nucleosides. Part V: 3-Chloro-4-(D-Ribofuranosyl)Pyridine and 3-(D-Ribofuranosyl)-2-Pyridone	M. Belmans; I. Vrijens; E. L. Esmans; R. A. Dommisse; J. A. Lepoivre; F. C. Alderweireldt; L. B. Townsend; L. L. Wotring; J. Balzarini; E. De Clercq
317-326	Use of the 2-(4-Pyridyl)Ethyl Protecting Group in the Synthesis of DNA Fragments Via Phosphoramidite Intermediates	Shoji Hamamoto; Yoshiharu Shishido; Mitunori Furuta; Hiroshi Takaku; Masahiko Kawashima; Makoto Takaki
327-337	Preparation of 2,3′-Anhydropyrimidine Nucleosides using N,N-Diethylaminosulfur Trifluoride (DAST)	Kwasi Agyei-aye; Shijia Yan; Anna K. Hebbler; David C. Baker
339-348	Sodium Thiosulfate and Potassium Selenosulfate as Reagents to Prepare Thio-and Selenopurine Nucleosides	Aleksander J. Jankowski; Dean S. Wise Jr.; Leroy B. Townsend
349-356	AS Triazine Acyclonucleosides: Potential Inhibitors of Pyrimidine Enzymes¹	Subhasish Purkayastha; Bihi H. Lazrek; Raymond P. Panzica; Fardos N. M. Naguib; Mahmoud H. el Kouni
357-366	A Synthesis of the Potent A₂ Selective Adenosine Agonist N⁶-[2-(3,5-Dimethoxyphenyl)-2-(2-Methylphenyl)Ethyl]Adenosine, and Its 5′-N-Ethyl Ribofuranuronamide Derivative	Alexander J. Bridges
367-382	Bis (2,4,6-Tribromophenyl) Phosphorochloridate: A New Type of Condensing Reagent in Oligonucleotide Synthesis	Jun-Ichi Matsuzaki; Hitoshi Hotoda; Mitsuo Sekine; Tsujiaki Hata
383-405	The Acidic Hydrolysis of Nucleosides and Nucleotides	Ewa Zielonacka-lis
407-414	N-Cyanoimidazole and Diimidazole Imine: Water-Soluble Condensing Agents for the Formation of the Phosphodiester Bond	James P. Ferris; Chun-Hsien Huang; William J. Hagan Jr.
415-430	Isolation and Identification of 1-Ribosyl Pyridone Nucleosides from Human Urine	Gordon C. Mills; Nora J. Davis; Khingkan Lertratanangkoon
431-448	The Synthesis of 2-Amino 7-Substituted Purines	Jonathan L. Sessler; Darren J. Magda; Vincent Lynch; Gilbert M. Schiff; David I. Bernstein

Volume 8, Issue 2 (1989)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 8, Number 2
159-178	Double Protection of the Heterocyclic Base of Xanthosine and 2′-Deoxyxanthosine	A. Van Aerschot; M. Mag; P. Herdewijn; H. Vanderhaeghe
179-183	A Simple and Convenient Method for the Selective N-Acylations of Cytosine Nucleosides	V. Bhat; B. G. Ugarkar; V. A. Sayeed; K. Grimm; N. Kosora; P. A. Domenico; E. Stocker
185-200	Phosphate-Modified Oligonucleotides. The Synthesis, Stereochemistry and ECO Ri Endonuclease Substrate Ability of Decanucleotides d[GGGAATTCCC] Bearing Altered Internucleotide Phosphate Function Between A and A¹	Maria Koziolkiewicz; Bogdan Uznanski; Wojciech J. Stec
201-211	Synthesis of Chiral 1′,2′-SECO-Nucleosides OF Guanine AND Uracil	Purushotham Vemishetti; Elie Abushanab; Robert W. Leiby; Raymond P. Panzica
213-223	Structure of Ethyl Hydrogen P(R), 5′-Anhydro-2′,3′-O-Isopropylidene-Adenosine-8-Phosphonate Hemiethylacetate Solvate	Yuriko Yamagata; Ken-Ich Tomita; Tokumi Maruyama; Mikio Honjo
225-256	Studies on the Alkylation of Derivatives of Guanines	Jonas Kjellberg; Nils Gunnar Johansson
257-271	Synthesis and Antiviral Activity of 5′-O-Sulfamoyluridine Derivatives	José Fiandor; María Teresa García-López; Federico G. De las Heras; Paloma P. Méndez-Castrillón; Carmen Gil-Fernández; Sara Pérez; Pilar Vilas; Concepción Pérez; Angel García Gancedo
273-284	Synthesis and Biological Activity of a Bis-Substituted 3′-Deoxyadenosine Analog of 2–5A	Ramamurthy Charubala; Wolfgang Pfleiderer; David Alster; Danuta Brozda; Paul F. Torrence
285-295	The Cyclic Dimer of 5-Fluoro-2′-Deoxyuridylic Acid: A Potent Anticancer Agent	G. Hamoir; E. Sonveaux; M. Iigo; E. De Clercq
297-303	The Inhibition of Adenosine Kinase by α,ω-Di (Adenosin - N⁶- YL) Alkanes¹

Volume 8, Issue 1 (1989)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 8, Number 1
1-21	7-Deaza-2′-Deoxy-O⁶-Methylguanosine: Selective N²-Formylation Via a Formamidine, Phosphoramidite Synthesis and Properties of Oligonucleotides	F. Seela; H. Driller
23-34	Preparation of Imino and Amino N-15 Enriched 2-Aminopurine Deoxynucleoside	Lawrence C. Sowers; Dhananjaya N. Mhaskar; Tasneem A. Khwaja; Myron F. Goodman
35-41	Synthesis of 2′,3′-Dideoxyuridine Via the Corey-Winter Reaction	L. W. Dudycz
43-48	The Oxidative Chlorination of Pyrimidine and Purine Bases, and Nucleosides Using Acyl Chloride-Dimethyl-Formamide-m-Chloroperbenzoic Acid System¹	E. K. Ryu; J. N. Kim
49-64	Synthesis of Novel Isocytosine Pseudonucleotide Analogues	Sharon M. Bennett; Kelvin K. Ogilvie; Jean Paul Roduit
65-96	Synthesis of Nucleosides Fluorinated in the Sugar Moiety. The Application of Diethylaminosulfur Trifluoride to the Synthesis of Fluorinated Nucleosides	P. Herdewijn; A. Van Aerschot; L. Kerremans
97-115	2′,3′-Dideoxyadenosine Analogs of the Nucleoside Antibiotics Tubercidin, Toyocamycin and Sangivamycin	Steven H. Krawczyk; Leroy B. Townsend
117-132	Aminopyrimidines and Derivatives. 22¹. Synthesis of 3-Glycopyrano-Syl-vic-Triazolo [4,5-d]Pyrimidines, 7-Glycopyranosyl-Pyrrolo [2,3-d]PY-Rimidines and 4-Glycopyranosylamino-Furo [2,3-d]Pyrimidines²	Manuel Nogueras; M Luisa Quijano; Adolfo Sanchez; Miguel Melgarejo
133-144	Mechanism for Acid-Catalyzed Hydrolysis of Nucleoside and Acyclonucleoside Analogues of Benzimidazole	Mikko Oivanen; Harri Lönnberg; Zygmunt Kazimierczuk; David Shugar
145-156	Nucleosides. 140. Stereoselectivity of the Reaction of 1-(2,3-Anhydro-5-O-Benzoyl-β-D-Lyxofuranosyl)Uracil with Ammonium Azide. Isolation and Characterization of 2-Azido-XYLO-Nucleoside Derivatives.¹	Michael E. Perlman; Kyoichi A. Watanabe

Volume 7, Issue 5-6 (1988)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 7, Number 5-6
551-554	Synthesis and Transport of a Specific Premessenger RNP Particle	U. Skoglund Mehlin; A. Lönnroth; B. Daneholt
555-558	On the Self-Splicing Complex of Tetrahymena Pre-rRna	Siegfried Hoffmann
559-564	Antisense RNA in Replication Control of the INC FII Plasmid R1	E. G. H. Wagner; C. Persson; M. Öhman; K. Nordstrom
565-569	Test System for Measurement of Translational Activity in Vivo	Asgeir Björnsson; Leif A. Isaksson
571-576	Effects on the Activity of the Enzyme Phosphoribosyl-Aminoimidazole Carboxylase, Involved in the Biosynthesis of Purine Nucleotides De Novo by Bi-Valent Metal Complexes of the Natural Substrate 5-Amino-1-β-D-Ribofuranosylimidazole-4-Carboxylic Acid 5′-Phosphate	J. R. Chipperfiel; R. W. Humble; G. Iveson; K. Kadir; G. Mackenzie; G. Shaw
577-580	Glycosylation of Mono- and Bicyclic Dicarbonic Acid Imides	E. Schlimme; H. Frister; K. -P. Raezke
581-584	7-Carbapurine Ribofuranosides: Synthesis by Solid-Liquid Phase-Transfer Glycosylation and ¹⁵N-NMR Spectra	F. Seela; H. Rosemeyer; A. Biesewig; T. Jorgens
585-588	the Influence of Modifications on the Cleavage of Oligonucleotide Duplexes by Eco R II and Mva I Endonucleases	D. Cech; C. -D. Pein; E. A. Kubareva; E. S. Gromova; T. S. Oretskaya; Z. A. Shabarova
589-593	C-Nucleoside Analogues of Nicotinamide Mononucleotide (NMN)	Krzysztof W. Pankiewicz; Marek M. Kabat; Elzbieta Sochacka; Lech Ciszewski; Joanna Zeidler; Kyoichi A. Watanabe
595-600	Recent Progress in Oligoribonucleotide Synthesis	Magdalena Pfister; Silke Farkas; Ramamurthy Charubala; Wolfgang Pfleiderer
601-604	Reactions of Nucleoside Hydrogenphosphonates with Diphenyl Chlorophosphate and Sterically Hindered Aromatic Acyl Chlorides	J. Stawinski; R. Stromberg; M. Thelin; E. Westman
605-608	Phosphite Oxidation and the Preparation of Five-Membered Cyclic Phosphorylating Reagents Via the Phosphites	I. Ugi; P. Jacob; B. Landgraf; C. Ruppf; P. Lemmen; U. Verfürth
609-612	Glycal Ethers as Starting Materials in C-Nucleoside Synthesis	Andrew Kaye; Colin B. Reese; Stephen Neidle
613-617	Selective Inhibition of DNA Chain Elongation Catalyzed by DNA Polymerases	A. A. Krayevsky; M. K. Kukhanova; A. M. Atrazhev; N. B. Dyatkina; A. V. Papchikhin; Z. G. Chidgeavadze; R. Sh. Beabealashvilli
619-623	Expression of Ribonuclease T1 in Escherichia Coli and Rapid Purification of the Enzyme	Rainer Quaas; Hans-Peter Grunert; Makoto Kimura; Ulrich Hahn
625-628	Phosphorothioate-Based Site-Directed Mutagenesis: Extending the Basic Methodology	Jon R. Sayers; Walter Schmidt; Fritz Eckstein
629-638	Approaches to Solid Phase DNA Sequencing	Thomas Hultman; Stefan Ståhl; Tomas Moks; Mathias Uhlen
639-643	Affinty Electrophoresis for the Separation of Oligo- and Polynucleotides	Gabor L. Igloi; Hans Kössel

Volume 7, Issue 5-6 (1988)

645-650	Rational Methods of DNA Synthesis, Exemplified for the Preparation of Parts of the Human Proopiomelanocortin Gene	H. Seliger; H. Fancelli; G. Gröger; S. Klein; U. Kotschi; R. Schlenk; G. Schmidt; E. Schwichtenberg
651-653	Synthesis of Modified Building Blocks Containing Amino or Thiol Moieties: Application of Modified Oligodeoxyribonucleotides	Brian S. Sproat; Barbro Beijer; Peter Rider; Philippe Neuner
655-659	Construction of Europium (Eu³)-Labelled Oligo DNA Hybridization Probes	C. Sund; J. Ylikoski; P. Hurskainen; M. Kwiatkowski
661-665	Enantioselective DNA Binding Geometries of Δ and Λ Ru(phenanthroline)₃² Studied with Linear Dichroism	Catharina Hiort; Bengt Nordén
667-670	Synthesis and Evaluation of Acyclic Nucleotide Analogs	Antonin Holy; Ivan Rosenberg; Hana Dvofakova; Erik Declercq
671-674	Simultaneous Protection of 3′- and 5′-Hydroxyls of Ribonucleosides with Di-t-Butoxydichlorosilane	Wojciech T. Markiewicz; Katarzyna Adrych
675-678	Synthetic Approach to D-Psicofuranosyl Nucleosides and Their 1-Deoxy Analogues	Annie Brouiller; Anne-Dominique Lespinasse; Jean-Marc Ricca
679-682	Synthesis Aitd Properties of C'-Methylhuclsosides and Their Phosphoric Esters	Sergey H. Mikhailov
683-686	The Construction, Cloning, and Expression of Synthetic Genes Coding for Totally Artificial Proteins	H. Itoster; J. Biernat; H. Hasselmanr; B. Hofer; N. Kennedy
687-691	Chemical Synthesis of Proteinase Inhibitor Genes	Michael Strauß; Jürgen Stollwerk; Klaus-Dieter Jany; Hans Günter Gassen
693-697	Cloning and Sequence Analysis of a cDNA from Seminal Vesicle Tissue Encoding the Precursor of the Major Protein of Bull Semen	Michael Kemme; Karl Heinz Soheit
699-702	X-Ray Crystallographic Studies of the A-Form of DNA	U. Heinemann; H. Lauble; R. Frank; H. Blöcker
703-706	The Chemical Syntheses of (2′-5′)-P-Thioadenylate Dimers, Trimers and Tetramers	R. Charubala; W. Pfleiderer
707-711	On the Influence of the Nature of 2-N-Protecting Acyl Groups on the Stability of Deoxyguanosine Derivatives	Peter Lemmen; Mirjana Baumgartner-rupnik
713-716	The Use of Synthetic Oligo-RNA and -DNA as Defined Templates for the Determination Of Catalytic Properties of RNA-Directed RNA Polymerase from Tomato Leaf Tissue	Bernd Haas; Winfried Schiebel; Snezan Marinkovic; Andrea Klanner; Heinz L. Sanger
717-720	Structure of a Covalent Complex Between Benzo(_a)Pyrene Diol Epoxide and DNA	Magdalena Eriksson; Bengt Nordeh; Bengt Jernström
721-723	Antibody Cell-Targeting of Liposomes Carrying Ara C Derivatives	H. Schott; W. Heβ; B. Leitner; R. A. Schwendener
725-728	Phosphoramidate Analogs of Dinucleotides: Synthesis and ¹H Assignment by Two Dimensional NMR Spectroscopy (¹H,¹H-COSY)	Matthias Mag; Joachim W. Engels
729-732	Methylphosphonamidites: Preparation and Application in Oligodeoxynucleoside Methyl-Phosphonate Synthesis	Thomas Löschner; Joachim W. Engels
733-736	Synthesis and ¹-NMR Studies of DNA-RNA Hybrids for Structural Analysis	C. Scalfi Happ; E. Happ; A. M. Gronenborn; G. M. Clore

Volume 7, Issue 5-6 (1988)

737-740	Site Directed Mutagenesis on the Restriction Endonuclease Eco RI Using Mixed Oligonucleotides	Andreas Dusterhöft; Manfred Kroger
741-744	Oligonucleotide Directed Mutagenesis of the E. coli hisS Gene: Introduction of an Ncoi Restriction Site at the Initiating GTG and Cloning of the Mutated Gene to the Expression Vector pKK 233–2	Thomas Glade; Uwe Englisch
745-749	NMR Investigation of Palindromic LAC Operator DNA Sequences of Varying Size: Influences of Complex Formation with the LAC Repressor Headpiece on the DNA ¹H Resonances	Brian Fera; Friedrich Buck; Heinz Rüterjans
751-755	Synthesis of Dumbbell-Shaped Circular DMA-Molecules	H. Schieferdecker; G. L. Igloi; H. Kossel
757-761	Solution Structure of Rnase T₁ and Its Complexes with Nucleotides	E. Hoffmann; J. Schmidt; J. Simon; H. Ruterjans
763-767	The reaction of Tetrazole with Phosphoramidites as a Model for the Nucleotide Coupling Step	S. Berner; K. Mtihlegger; H. Seliger
769-771	In Situ Hybridization with Antisense Oligonucleotide: Estradiol Stimulates Transcription and Translation in Oxytocin Producing Hypothalamic Neurons	F. Ramalho-ortigao; G. F. Jirikowski; H. Seliger
773-778	A Polymeric Support for Chemical and Enzymatic Nucleic Acid Synthesis (1)	G. Groger; H. Seliger
779-782	Evaluation of the Use of the t-Butyldimethylsilyl Group for 2′-Protection in RNA-Synthesis Via the H-Phosphonate Approach	Jacek Stawinski; Roger Sternberg; Mats Thelin; Erik Westman
783-786	Competitive Binding Between Unmodified and Etheno DNA Provides Information About Structure and Stoichiometry of RECA-DNA Complexes	Mikael Kubista; Masayuki Takahashi; Bengt Nordén
787-793	Arenesulfonylethoxycarbonyl- a Set of Amino Protecting Groups for DNA and RNA Synthesis	A. Nyilas; A. Földesi; J. Chattopadhyaya
795-799	The 4-Decyloxytrityl Group as an AID in the Affinity Chromatography of Synthetic Oligonucleotides	G. Schmidt; R. Schlenk; H. Seliger
801-804	On the Structure and Reactivity of Y-Nucleoside [Wyosine]	C. Glemarec; J-C. Wu; H. Bazin; G. Remaud; M. Oivanen; H. Lönnberg; J. Chattopadhyaya
805-811	Fluorescence Properties of Y-Nucleoside Derivatives	T. M. Nordlund; R. Rigler; C. Glemarec; J. -C. Wu; H. Bazin; G. Remaud; J. Chattopadhyaya
813-816	New Trityl-Based Protecting Groups with a Mild Two-Step Removal	Erwin Happ; Claudia Scalfi Happ
817-820	Chemical Synthesis and Cloning of a Gene Coding for Bacillus Subjilis Hbsu Protein	N. Groch; R. Quaas; U. Hahn; U. Heinemann
821-825	¹⁵N-Labeled Oligodeoxynucleotides -Useful Probes for ¹H-NMR Investigations	Ingo Kieper; Thomas Schmidt; Brian Fera; Heinz Rüterjans
827-830	Conformation of Lariat Structures Formed in the Splicing of Pre-mRNA by NMR Spectroscopy	A. Sandström; N. Balgobin; A. Nyilas; G. Remaud; J. -M. Vial; X. -X. Zhou; J. Chattopadhyaya

Volume 7, Issue 4 (1988)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 7, Number 4
409-416	Synthesis of 6,3′-Methanothymidine from a Ribofuranos-3-Ulose and 2,4-Dimethoxy-5,6-Dimethylpyrimidine	Yuichi Yoshimura; Akira Matsuda; Tohru Ueda
417-429	Isolation and Characterization of 3-(3-Amino-3-Carboxypropyl)Uridine from Human Urine	Girish B. Chheda; Henry A. Tworek; Arvind K. Bhargava; Elliot Rachlin; Shib P. Dutta; Helen B. Patrzyc
431-455	Oligothymidylates Substitues Par Un Derive De L'Acridine en Position 5′, A La Fois En Position 5′ et 3′ Ou Sur Un Phosphate Internucleotidique	U. Asseline; N. T. Thuong
457-477	Preparation of New Glycoheptofurano[2,1-d]Imidazolidine-2-Thiones., Isomerizations to Acyclic-Sugar C-Nucleoside Analogues of Imidazole	J. Fuentes Mota; J. I. Fernández García-Hierro; P. Areces Bravo; F. Rebolledo Vicente; J. A. Galbis Pérez
479-495	Characterization of a Novel 2′-5′ Oligoadenylate in Stimulated Lymphocytes	J. Marti; D. Roux; J. Favero; J. Dornand; H. Cailla
497-510	Construction of Genes or Gene Fragments by Use of Two Long Synthetic Oligonucleotides Representing the Coding and Noncoding Strands	Friedrich Hein; Hans W. Jansen; Eugen Uhlmann
511-517	Potential Antiviral Agents. Synthesis and Properties of Glutarimide-Nucleosides	M. J. Wanner; G. J. Koomen
519-536	Protection of the Lactam Function of 2′-Deoxyinosine with A 2-(4-Nitrophenyl)-Ethyl Moiety	A. Van Aerschot; P. Herdewijn; G. Janssen; H. Vanderhaeghe
537-547	Nucleosides, IV¹ Synthesis and Properties of 2-Metylthio-Naphthimidazole-Ribonucleoside	Abdullah Hijazi

Volume 7, Issue 3 (1988)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 7, Number 3
271-294	¹⁸O-Labeled Adenosine and 9-(β-D-Arabinofuranosyl)Adenine (ARA-A): Synthesis, Mass Spectrometry, and Studies of ¹⁸O-Induced ¹³C NMR Chemical Shifts	Cong Jiang; Robert J. Suhadolnik; David C. Baker
295-306	Hydrolysis of Adenosine Cyclic 3′,5′-(R_p)- and (S_p)-Phosphoramidates. Stereoelectronic Effects in the Acid Hydrolysis	J. Tomasz; S. Bottka
307-319	Improved Synthesis of Adenosine Cyclic 3′, 5′-Phosphoramidates via Anhydrides. Preparation of Adenosine Cylic 3′, 5′-(R_p) - and (_p)-N-Methylphosphoramidate	S. Bottka; J. Tomasz
321-337	Studies on Ribonucleoside Hydrogenphosphonates. Effect of a Vicinal Hydroxyl Function on the Stability of H-Phosphonate Diester Bond	Sophie Huss; Gilles Gosselin; Jacek Stawinski; Roger Stromberg; Jean-Louis Imbach
339-346	Studies in the Protection and Selective Deprotection of 5-Amino-1-β-D-Ribofuranosylimidazole-4-Carboxamide (Aica-Riboside)	R. D. Chambers; M. R. Bryce; S. T. Mullins; A. Parkin
347-363	Dodecanucleotides Containing (E)-5-(2-Bromovinyl)-2′-Deoxyuridine: Influence of a Bulky Major Groove Substituent on Duplex Stability and Endodeoxyribonuclease Eco Ri Recognition	Frank Seela; Hansjürgen Driller; Wilhelm Herdering; Erik De Clercq
365-374	Synthesis of 4′-(Hydroxymethyl)Guanosine and a Phosphonate Analogue of Guanylic Acid	John C. Martin; Julien P. H. Verheyden
375-383	Triaryl(Oxy)Phosphine Dibromide- A Convenient Reagent for the Preparation of S-Arylthioinosines and N⁶, 5′-Disubstituted Adenosine Derivatives from Inosine	Alexander J. Bridges
385-392	Synthesis of Brunfelsamidine Ribonucleoside and Certain Related Compounds by the Stereospecific Sodium Salt Glycosylation Procedure	Kandasamy Ramasamy; Roland K. Robins; Ganapathi R. Revankar
393-402	Studies Toward Synthesis of C2-Substituted Adenosines: An Efficient Synthesis of 2-(Phenylamino)Adenosine [CV-1808]	Bharat K. Trivedi
403-408	Synthesis of Bis(Aziridinyl) Phosphinic Amide Derivatives of Thymidine as Potential Anticancer Agents	Tai-Shun Lin; Guo-Lin Cai; Alan C. Sartorelli

Volume 7, Issue 2 (1988)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 7, Number 2
129-135	Inhibition of the Herpes Simplex Virus Thymidine Kinase by 5 Substituted Thymidine Analogues. Comparison of the Types 1 and 2 Enzymes	Iain S. Sim; Colin Picton; Richard Cosstick; A. Stanley Jones; Richard T. Walker; Albert Jaxa Chamiec
137-145	Cyclic AMP Diphenyl Phosphoric Mixed Anhydride: Synthesis, P NMR Characterization and Reaction with Dimethylamine	S. Bottka; I. Pelczer; J. Tomasz
147-153	Synthesis of 2′,3′-Dideoxyinosine	Robert R. Webb II; John A. Wos; John C. Martin; Paul R. Brodfuehrer
155-165	Synthesis and Anti-Herpetic Activity of A 2′-Fluoroarabinosyl Analog of Trifluridine	Donald F. Smee; Marlene Chernow; Monica Kraft; Patricia M. Okamoto; Ernest J. Prisbe
167-179	An Assessment of Electronic Properties of Pyrimidine and Purine Nucleosides by ¹⁵N-NMR Spectroscopy	G. Remaud; C. J. Welch; X. X. Zhou; J. Chattopadhyaya
181-193	The Synthesis of Ribosides of Asymmetrically-Substituted Aminohalogenobenzimidazoles	Maria José Camarasa; Richard T. Walker; A. Stanley Jones
195-202	Synthesis of 5′ -0-Succinyl-2′, 3′-Cyclic Adenosine Monophosphate	Charles E. Dreiling; Joanne B. Pachuta; John P. Hamlin
203-211	Photochemical Synthesis of Phosphonopyrimidine and Phosphonopurine Ribonucleosides	Tokumi Maruyama; Mikio Honjo
213-225	1,4:3,6-Dianhydrohexitol Nucleosides	Peter Stoss; Elmar Kaes
227-244	Studies on the Dehydration of New 2- (Pentitol-1-YL) Pyridines Having D-Gulo, D-IDO, and L-Manno Configurations	M. Bueno Martínez; E. Román Galán; J. A. Galbis Pérez
245-248	A Mild Procedure for O-Deacylation of the Fully Acylated Sugar Moiety of Nucleosides in the Presence of Cyanide	Jun-Ichi Asakura; Takanori Tomura
249-269	3′-Deoxy-3′-Hydroxyamino-β-D-Xylofuranosyluracil and Derivatives Thereof	Jean M. J. Tronchet; Rachid Benhamza; Naz Dolatshahi; Michel Geoffroy; Hans Türler

Volume 7, Issue 1 (1988)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 7, Number 1
1-21	Reaction of 5-Halocytosine Derivatives with Cysteine	Bimal C. Pal; Chandrakanta Ghosh; Satinder K. Sethi; Bruce E. Suttle; James A. McCloskey
23-35	Nucleoside H-Phosphonates. IX. Possible Side-Reactions During Hydrogen Phosphonate Diester Formation	Tor Regberg; Jacek Stawinski; Roger Ströberg
37-43	A Simple, Preparative Procedure for N³-Anisoyluridine and O⁶-Diphenylcarbamoylguanosine 2′-O-(Tetrahydropyran-2-YL) Derivatives via The Corresponding 3′,5′-Dibenzoates	Kazuo Kamaike; Yoshihiro Hasegawa; Yoshiharu Ishido
45-60	Structure and Conformation of 1-β-D-Ribofuranosylpyridin-4-One-3- Carboxamide, A Novel Nucleoside from Human Urine with a Rare Ribose Pucker	T. Srikrishnan; R. Parthasarathy; J. L. Alderfer; S. P. Dutta; G. B. Chheda
61-73	Synthesis, Molecular Cloning and Expression of Genes Coding for Atrial Natriuretic Factors from Rat and Human	Hans Sachse; Gerd Hagendorff; Klaus Dieter Preuβ; Hari S. Sharma; Karl Heinz Scheit
75-90	Silica Gel Functionalised with Different Spacers as Solid Support for Oligonucleotide Synthesis	Arthur Van Aerschot; Piet Herdewijn; Hubert Vanderhaeghe
91-102	Synthesis of 5-Benzyl and 5-Benzyloxybenzyl 2,2′-Anhydrouridines and Related Nucleoside Analogs as Inhibitors of Uridine Phosphorylase	Shih Hsi Chu; Zum Yao Weng; Zhi Hao Chen; Elizabeth C. Rowe; Edward Chu; Fardos N. M. Naguib; Mahmoud H. el Kouni; Sungman Cha; Ming Y. Chu
103-115	Probing the Thymidylate Synthase Active site with Bisubstrate Analog Inhibitors	Said M. M. Bayomi; Diana I. Brixner; Hassan Eisa; Arthur D. Broom; Takamori Ueda; Yung-Chi Cheng
117-120	An Improved Preparation of Rp and Sp N⁶, N⁶, O²′ - Tri-Benzoyl-Adenosine-3′, 5′-Cyclic Phosphoranilidates	Marcel K. Eberle; Leszek Brzechffa
121-128	Preparation of 8-Chloropurine Nucleosides Through the Reaction Between their C-8 Lithiated Species and p-Toluenesulfonyl Chloride	Hiroyuki Hayakawa; Hiromichi Tanaka; Kazuhiro Haraguchi; Masami Mayumi; Masako Nakajima; Takashi Sakamaki; Tadashi Miyasaka

Volume 6, Issue 5 (1987)

a	Editorial board page for “Nucleosides, Nucleotides & Nucleic Acids”, Volume 6, Number 5
815-820	Iodine and Iodine Catalysed Phosphorylation of Nucleosides by Phosphorodiester Derivatives	Roger Strömberg; Jacek Stawinski
821-830	A Universal Glass Support for Oligonucleotide Synthesis	J. S. Debear; J. A. Hayes; M. P. Koleck; G. R. Gough
831-840	Synthesis of 2-S-Dioxo Isosteres of Purine and Pyrimidine Nucleosides. V. ¹³ CDNMR Study of SYN-ANTI Equilibrium in a Glucoside of a N-Substituted Barbituric Acid Isostere	A. Cuberta; M. L. Jimeno; C. Ochoa
841-852	Partial Protection of Carbohydrate Derivatives. Part 24.¹ Synthesis of Adenylyl-(2′–5′)-Adenylyl-(2′–5′)-Adenosine Using a 3′-O-(Tetrahydropyran-2-YL) Adenosine Derivative	Kazuo Kamaike; Shun-Ichi Yamakage; Yoshiharu Ishido
853-863	Synthesis of Pyrazolo[3, 4-d]Pyrimidine Ribonucleoside 3′, 5′-Cyclic Phosphates Related to cAMP, cIMP and cGMP¹	Jack D. Anderson; Roland K. Robins; Ganapathi R. Revankar
865-876	Analysis of Substituted Pyridine-C-Nucleosides by Direct Liquid Introduction Liquid Chromatography/Mass Spectrometry	E. L. Esmans; M. Belmans; I. Vrijens; Y. Luyten; F. C. Alderweireldt; L. L. Wotring; L. B. Townsend
877-885	Crystal Structure of a Tightly Bound Inhibitor of Adenosine Transport N⁶-(4-Nitrobenzyl)-β-D-2′-Deoxyadenosine Methanol Solvate, C₁₇H₁₈N₆O₅.1/2 CH₃OH	J. Wilson Quail; Louis T. J. Delbaere; Alan R. P. Paterson
887-899	Aminopyrimidines and Derivatives. 20. On the Acetylations of 5-Amino-4-Glycosylmino Pyrimidines	M. Rodríuez; C. Rodríguez; M. Melgarejo; R. Asenjo; M. Nogueras; A. Sánchez
901-911	Nucleoside Peptides. 8. Synthesis of Certain Peptide Derivatives of Ribavirin and Tiazofurin	Kandasamy Ramasamy; Ganesh D. Kini; Roland K. Robins; Ganapathi R. Revankar
913-934	Modification of Oligo (Poly) Nucleotide Phosphomonoester Groups in Aqueous Solutions	M. G. Ivanovskaya; M. B. Gottikh; Z. A. Shabarova

Volume 6, Issue 4 (1987)

a	Editorial board page for “Nucleosides, Nucleotides & Nucleic Acids”, Volume 6, Number 4
663-678	Synthesis and Biological Activity of C-Acyclic Nucleosides of Imidazo [1,5-a]-1,3,5-Triazines	Bozenna Golankiewicz; Joanna Zeidler; Erik De Clercq
679-689	The Large Scale Synthesis and Chromatographic and Spectral Properties of a Series of Alkylated Thymine and Uracil-Containing Nucleosides. O²-, 3- and O⁴-Alkylpyrimidine Derivatives	Roy Saffhill
691-698	Ribonucleoside Diphosphate Adducts with Elliptinium Acetate, an Antitumor Agent	T. B. Tam Ha; Jean Bernadou; Bernard Meunier
699-736	Partial Protection of Carbohydrate Derivatives. Part 23.¹ Simple, Efficient Procedure for the Preparation of 3′- and 2′-0-(Tetrahydropyran-2-YL)Ribonucleoside Derivatives Involving Highly Regioselective 2′,5′-DI-O-Acylation or that Followed by Acyl Migration on Silica Gel and Subsequent O-(Tetrahydropyran-2-YL)Ation	Kazuo Kamaike; Fumihiko Uemura; Shun-Ichi Yamakage; Shigeyoshi Nishino; Yoshiharu Ishido
737-759	Synthesis of Certain 4-Substituted-1-β-D-Ribofuranosyl-3-Hydroxypyrazoles Structurally Related to the Antibiotic Pyrazofurin	Yogesh S. Sanghvi; Krishna G. Upadhya; N. Kent Dalley; Roland K. Robins; Ganapathi R. Revankar
761-774	Synthesis of 2′,3′-Dideoxyribavirin	Yogesh S. Sanghvi; Naeem B. Hanna; Steven B. Larson; Roland K. Robins; Ganapathi R. Revankar
775-783	Conformations of Acyclonucleosides: Crystal Structure of 9-(4-Hydroxybutyl)Guanine, an Analogue of Acyclovir	George I. Birnbaum; Nils Gunnar Johansson; David Shugar
785-792	A ³¹P NMR Study of the Reaction of Adenosine 3′ 5′-Cyclic Monophosphate with 2, 4, 6-Triisopropylbenzenesulfonyl Chloride	J. Tomasz; S. Bottka; I. Pelozer
793-802	Synthesis and Biological Evaluation of some Acyclic Nucleoside Cyclic Phosphoramidate Derivatives	Hiroshi Takaku; Tsunehiko Ito; Shiro Yoshida; Tomoni Aoki; Erik De Clercq
803-814	Synthesis of Oligonucleotides Containing the Abasic Site Model Compound 1,4-Anhydro-2-Deoxy-D-Ribitol	Ramon Eritja; Peter A. Walker; Sandra K. Randall; Myron F. Goodman; Bruce E. Kaplan

Volume 6, Issue 3 (1987)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 6, Number 3
543-554	Synthetic Templates and the RNA Polymerase of Influenza a Virus	Zainub Khan; Mario Ariatti; Arthur Hawtrey
555-574	Novel Acyclonucleosides. Part 2. 2, 3-Dihydroxy-1-Methoxypropyl-and 3-Hydroxy-1-Methoxypropyl-Substituted Purines	Stuart Bailey; Michael R. Harnden
575-580	Facile 5′-Halogenation of Unprotected Nucleosides	Tadakazu Tsuji; Keiko Takenaka
581-587	A New Synthesis of 7-Methyl-8-Oxoguanosine	Ganesh D. Kini; William J. Hennen; Roland K. Robins
589-595	An Improved Method for the Preparation of Methyl dichlorophosphite. A Key Reagent In the Phosphite Method of Oligonucleotide Synthesis	Z. Tashma; I. Ringel; J. Deutsch; S. Cohen; M. Weisz; J. Katzhendler
597-611	Isolation and Characterization of a Novel Nucleoside from the Urines of Chronic Myelogenous Leukemia Patients	Girish B. Chhed; Helen B. Patrzyc; Arvind K. Bhargava; Pamela F. Crain; Satinder K. Sethi; James A. McCloskey; Shib P. Dutta
613-620	Structures of two Seven-Membered Ring Pyrimidine Nucleoside Derivatives	Paul A. Sutton; Vivian Cody; Victor E. Marquez
621-630	Nucleosides. 140. Stereoselectivity of the Reaction of 1-(2,3-Anhydro-5-O-Benzoyl-β-D-Lyxofuranosyl) Uracil with Ammonium Azide. Isolation and Characterization of 2-Azido-Xylo-Nucleoside Derivatives	Michael E. Perlman; Kyoichi A. Watanabe
631-642	Synthesis of 2S-Dioxo Isosteres of Purine and Pyrimidine Nucleosides IV. Selective Glycosylation of 4-Amino-5H-Imidazo [4, 5-c]-1, 2, 6-Thiadiazine 2, 2-Dioxide	P. Goya; A. Martínez; C. Ochoa
643-653	Propeller Twisting in Single Crystals of Nucleosides	C. C. Wilson; P. Tollin
655-662	Nucleoside H-Phosphonates. V. The Mechanism of Hydrogenphosphonate Diester Formation Using Acyl Chlorides as Coupling Agents in Oligonucleotide Synthesis by the Hydrogenphosphonate Approach	Per J. Garegg; Tor Regberg; Jacek Stawinski; Roger Strömberg

Volume 6, Issue 1-2 (1987)

xiii-xiv	Foreword
a	Editorial board page for “Nucleosides & Nucleotides”, Volume 6, Number 1-2
3-9	The Introduction of C-Substitutents into Pyrimidine- and Purine-Nucleosides	Helmut Vorbrüggen; Konrad Krolikiewicz
11-23	Synthesis and Application of Isosteric Purine 2′-Deoxyribofuranosides	Frank Seela; Uwe Bindig; Hansjürgen Driller; Wilhelm Herdering; Klaus Kaiser; Andreas Kehne; Helmut Rosemeyer; Herbert Steker
25-42	Electrochemical Oxidations of Some Purine Nucleosides. Formation of Some Novel Purine Oligonucleosides	P. Subramanian; S. K. Tyagi; Glenn Dryhurst
43-51	Anomalously Coupled Nucleosides	Erik B. Pedersen
53-63	Fluorine Substituted Analogs of Nucleosides and Nucleotides	Don Bergstrom; Eric Romo; Patrick Shum
65-72	Systematic Synthesis and Biological Evaluation of α - and β-D-Xylo- and Lyxofuranonucleosides of the Five Naturally Occurring Nucleic Acid Bases	G. Gosselin; M. C. Bergogne; J. L. Imbach; J. De Rudder; E. De Clercq
73-83	New Substrate Analogues as Inhibitors of S-Adenosylmetfflonine Decarboxylase	John A. Secrist
85-94	The Synthesis, Mutagenic and Pharmacological Activities of 2-Carbon-Substituted Adenosines	Akira Matsuda; Tohru Ueda
95-109	Triciribine (TCN), A Novel Tricyclic Adenosine Analog with Anticancer Activity	Linda L. Wotring; Joseph L. Roti; Jerry L. Hudson; Joan E. Passiatore; Katherine Z. Borysko; Richard D. Newcomb; Leroy B. Townsend
111-119	DNA-Triesters - The Synthesis and Absolute Configuration Assignments at P-Stereogenic Centres	Piotr Guga; Maria Koziołkiewicz; Andrzej Okruszek; Bogdan Uznański; Wojciech J. Stec
121-129	The Problem of 2′-Protection in Rapid Oligoribonucleotide Synthesis	Colin B. Reese
131-136	The Chemistry of Eukaryotic Messenger RNA	Tsujiaki Hata; Mitsuo Sekine; Kin-Ichiro Miura
137-146	Semi-Mechanized Simultaneous Synthesis of Multiple Oligonucleotide Fragments	H. Seliger; A. Herold; U. Kotschi; J. Lyons; G. Schmidt; F. Eisenbeiß
147-155	Phosphonylmethyl Analogs of Nucleotides and Their Derivatives: Chemistry and Biology	Antonin Holy
157-172	Versatile Oligonucleotides: B DNA, Z DNA, and DNA Hairpins as Seen in Aqueous Solution by Two-Dimensional NMR	Cornells Altona
173-184	Phosphorothioate Analogs of 2–5A: Elucidation of the Stereochemical Course of the Enzymes of the 2–5A Synthetase/RNase L System	Katalin Karikó; Shu Wu Li; Robert W. Sobol Jr.; Lorraine Suhadolnik; Nancy L. Reichenbach; Robert J. Suhadolnik; Ramamurthy Charubala; Wolfgang Pfleiderer
185-195	Chemoenzymatic Gene Synthesis of A Gene for Human Growth Hormone Releasing Hormone (hGHRH), its Expression in E. Coli and Enzymatic Amidation	Joachim W. Engels; Jan Glauder; Hubert Mülliner; Eugen Uhlmann; Waldemar Wetekam; T. Hashimoto Gotoh; Barbara Scheikl-lenz
197-207	Targets for the Antiviral Activity of Pyrimidine and Purine Nucleoside Analogues	Erik De Clercq
209-226	A Convergent Regiospecific Synthesis of the Lariat-Trinucleotides and A^{2′p 5′G} and A^{2′p 5′G}_{3′p 5′C} from A O⁴-2-Nitrophenyl) -Uridine Building Block	J-M. Vial; N. Balgobin; G. Remaud; A. Nyilas; J. Chattopadhyaya
229-232	Synthetic Approaches to Rare 2-Substituted Purine Nucleosides	Vasu Nair; Stanley D. Chamberlain; Raymond Desilvia; Greg S. Buenger
233-237	A Novel Approach to Khantiokerically Pure Carbocyclic Nucleoside Analogues	Michael Bodenteich; Kurt Faber; Gerhard Penn; Herfried Griengl
239-244	Synthesis of 2′,3′-Dideoxycyclopentenyl Carbocyclic Nucleosides as Potential Drugs for the Treatment of AIDS	Victor E. Marquez; Christopher K. H. Tseng; Susan P. Treanor; John S. Driscoll
245-248	Synthesis and Biological Evaluation of 3-Chloro-4-(D-Ribofuranosyl)-Pyridine and 3-(D-Ribofuranosyl)-2- Pyridone	M. Belmans; I. Vrijens; E. L. Esmans; J. A. Lepoivre; F. C. Alderweireldt; L. L. Wotring; L. B. Townsend
249-256	Synthesis and Antitumor Activities of 5-Fluorouracil Derivatives	S. Ozaki; Y. Watanabe; T. Nagase; T. Ogasawara; S. Ahmad; A. Hoshi; M. Iigo
257-260	Synthesis and Biological Properties of 6-Substituted 5-Fluorouridines	K. Felczak; T. Kulikowski; J. A. Vilpo; J. Giziewicz; D. Shugar
261-264	Direct Synthesis of Pyrrole Nucleosides by the Stereospecific Sodium Salt Glycosylation Procedure	G. R. Revankar; K. Ranasamy; R. K. Robins
265-268	Synthesis of 6β-Hydroxyaristeromycin - A Novel Type of Carbocyclic Nucleoside Analogue	Azzouz Ben Cheikh; Jiří Žmlićka

Volume 6, Issue 1-2 (1987)

269-272	A New Method of Synthesis of 4-N-Alkyl Substituted Cytosine Derivatives Via 4-N-Arylsulfonyl or Alkylsulfonyl Intermediates	W. T. Markiewicz; R. Kierzek; B. Hemes
273-277	O⁶-Protection and Other Transformations at Guanosine and Inosine Lactam Sites with Application of Related Pyridinium Salts	S. Mielewczyk; Z. Gdaniec; G. Bobrowska; R. W. Adamiak
279-282	Phosphotriester Synthesis of Oligonucleotides with the Use of N- and O-Nucleophilic Intramolecular Catalysis	V. A. Efimov; A. A. Buryakova; N. N. Polushin; I. Y. Dubey; O. G. Chakhmakhcheva; Yu. A. Ovchinnikov
283-286	Studies on the Synthesis of Oligonucleotides via the Hydrogenphosphonate Approach	Per J. Garegg; Tor Regberg; Jacek Stawinski; Roger Stromberg
287-291	The Use of Nucleoside H-Phosphonates in the Synthesis of Deoxyoligonucleotides	Brian C. Froehler; Mark D. Matteucci
293-296	Use of the 2-(2-Pyridyl)Ethyl Protecting Group in the Synthesis of DNA Fragments via Phosphoramidite Intermediates	Hiroshi Takaku; Tetsuo Watanabe; Shoji Hamamoto
297-300	Base Modification and the Phosphoramidite Approach	L. J. McBride; J. S. Eadie; J. W. Efcavitch; W. A. Andrus
301-305	Quantitative Measurements of Modified Thymine Residues in DNA Chains Formic Acid Hydrolysis	R. Téoule; A. Guy
307-310	Specific Enzymes Degrading Diadenosine Tetraphosphate (Ap₄ A). Promising Targets for Selective Drugs to be Designed	Andrzej Guranowski; Katedra Biochemii; Akademia Rolnicza
311-315	Biological Activities of Oligonucleotides Linked to Poly(L-Lysine)	M. Lemaltre; C. Bisbal; B. Bayard; B. Lebleu
317-320	Base Analogue Interactions in DNA Duplexes	D. M. Brown; N. N. Anand; S. A. Salisbury
321-325	Versatile Methodology for the Construction of Artificial Genes	O. G. Chakhmakhcheva; V. A. Efimov; Yu. A. Ovchinnikov
327-330	DNA Base Pair Binding Specificity of CC-1065	Nicole Y. Thériault; William C. Krueger; Mark D. Prairie
331-334	Site-Directed Mutagenesis of Stahphylococcal Nuclease: Role of Tyrosine Residues in Substrate Binding and Catalysis	E. Uhlmann; J. A. Smith
335-340	Solid Supported Chemical 5′-Phosphorylation of Oligodeoxy-Ribonucleotides that can be Monitored by Trityl Cation Releasi Application to Gene Synthesis	Thomas Horn; Judith S. Allen; Mickey S. Urdea
341-344	A New 5′-Protecting Group for Use in Solid-Phase Synthesis of Oligoribonucleotides	Chris Christodoulou; Sudhir Agrawal; Michael J. Gait
345-348	New Approach to the Synthesis of 2′(3′)-O-Aminoacyloligoribonucleotides Related to the 3′-Terminus of Aminoacyl Transfer Ribonucleic Acid	C. Scalfi-happ; E. Happ; S. Chladek
349-352	Synthesis Of Oligodeoxyribonucleotides Containing an Aliphatic Amino Linker Arm at Selected Adenine Bases and Derivatization with Biotin	Jean-Paul Roduit; Jeffrey Shaw; Angelika Chollet; André Chollet
353-358	Transition Metal Complexes of 5-Amino-1-β-D-Ribofuranosylimidazole-4-Carboxylic Acid 5′-Phosphate, an Intermediate in the de novo Biosynthesis of Purine Nucleotides: Synthesis and Effects on Enzyme Activity	J. R. Chipperfield; R. W. Humble; G. Iveson; K. Kadir; G. Mackenzie; G. Shaw
359-362	Polyfunctional O-Substituted Hydroxylamines: Modification of Nucleic Acids, Inhibition of Sam-Decarboxylase	A. R. Khomutov; A. M. Kritsky; E. Yu. Artamonova; R. M. Khomutov

Volume 6, Issue 1-2 (1987)

365-368	The Preparation and Utility of 5-β-D-Ribofuranosyl-(2H)-Tetrazole as a Key Synthon for C-Nucleoside Chemistry	Joze Kobe; Marija Prhavc; Marijan Hohnjec; Leroy B. Townsend
369-370	Regiospecipic Synthesis of a New Cross-Linked Dinucleoside : 1-(N⁶-Deoxyadenyl)-2-(o⁴-Thymidyl)-Ethane	M. Nogueras; M. Lucas; J-L. Imbach
371-372	Intramolecular Transformations Related to the Structures of Allyl Derivatives of Hypoxanthine and Uracil	V. Škari; M. Škarić-Mlakar; M. Jokić; D. Škarić
373-374	Synthesis of 7-Glycopyranosyl-5-oxq-pyrrolo[2,3-d]Pyrimidine and 4-Glyco Pyranosylamino-Furo[2,3-d]Pyrimidine Derivatives	M. Nogueras; M. L. Quijano; A. Sénchez; M. Melgarejo
375-377	Glycosides Derived from Pyrazino[2,3-C]-1,2,6-Thiadiazine 2,2-Dioxides	P. Goya; A. Martinez; M. L. Jimeno; W. Pfleiderer
379-380	A New Method for Synthesizing Acyclonucleosioes	H. B. Lazrek; M. L. Taha; J. L. Barascut; J. L. Imbach
381-383	Improved Synthesis and Cytostatic Activity of 1-Deazaadenosine	Gloria Cristalli; Palmarisa Franchetti; Mario Grifantini; Sauro Vittori; Teresa Bordoni; Cristina Geroni
385-386	Transglycosylation of Guanine Nucleosides	Jeratzy Boryski; Bozenna Golankiewicz
387-388	Synthesis of Some Quinolinium Nucleosides	L. Kemps; E. L. Esmans; R. Dommisse; J. A. Lepoivre; F. C. Alderweireldt
389-390	One-Step Protection of the Guanine Moiety in 2′-Deoxyguanosine and Guanosine	A. M. A. Pistorius; C. A. A. Claesen; F. J. B. Kremer; E. A. V. Rijk; G. I. Tesser
391-392	Novel Acyclic Analogues of Purine Nucleosides: 2,3-Dihydroxy-1-Methoxypropyl and 3-Hydroxy-1-Methoxypropyl Derivatives	S. Bailey; M. R. Harnden
393-394	Facile Synthesis of Base-Labile 2′-Deoxyribonucleosides: An Improved Synthesis of 2′-Deoxy-5-aza-Cytidine	Jean Ben-hattar; Josef Jiricny
395-396	Deuteration and Tritiation of 2′-Deoxyribonucleosides in the 5′ and 4′ Positions	M. Berger; A. Shaw; J. Cadet; J. R. Jones
397-398	Reactions of Purine Nucleosides with Aqueous Alkalies: The Effect of the C6 Substituent on the Kinetics of the Multistage Pathway	Marri Lönnberg; Pertti Lehikoinen; Rainer Käppi
399-400	Amination of Ethyl 5-Amino-1-Qlycofuranosylimidazole-4-Carboxylates Using Trimethylaluminium	A. Grouiller; R. W. Humble; G. Iveson; G. Mackenzie; B. Najib; H. Pacheco; G. Shaw
401-402	Arylamidation of Purine Nucleosides by 2-Acetylalkoxy- Aminofluorene - an Intramolecular Approach to the Synthesis of Nucleoside - Carcinogen Adducts	A. Leterme; M. F. Lhomme; J. Lhomme
403-405	Synthesis of 5′-O-Dimeth0Xytrityl-4-N-/6-Trifluoroacetamidohexyl/-2′-Deoxycytidine and its Application in the Synthesis of Biotin-Labeled Oligonucleotides	Ryszard Kierzek; Wojciech T. Markiewicz
407-408	Preparative Syntheses of Guanylate-Rich Oligonucleotides Using the Phosphotriester Method in Solution	H. Schott; R. Semmler; K. Cloß
409-411	Oligonucleotide Mediated Mutational Analysis of Recognition Sequence Effects on Lariat Formation During Messenger RNA Splicing in Yeast	Eduard Felder; Alessandra Cellini; John Rossi
413-414	Synthesis and Cloning of a Gene Encoding Human Interleukin-1β (IL-1β)	David C. Humber; Michelle Allsopp; Barry A. Coomber; Lucia G. D'urso; Colin W. Dykes; Adrian N. Hobden; Melville Mitchell; Stewart A. Noble

Volume 6, Issue 1-2 (1987)

415-417	5-Hydroxymethyl-2′-Deoxyuridine: Studies of Antileukemic Properties in Vitro and in Vivo	J. A. Vilpo; D. Bergstrom; L. Kangas; E. Suvanto
419-420	Sequencing of Synthetic DNA Fragments Containing Various 5-Substituted Pyrimidines by Solid-Phase Chemical Degradation Using CCS Paper	Andre Rosenthal
421-422	Mechanism of Antiviral Activity of 5-Ethyl-2′-Deoxyuridine	Ria Bernaerts; Erik De Clercq
423-424	Role of Adenosine Kinase in the Biological (Antiviral and Anticellular) Activities of Adenosine Analogues	Marina Cools; Erik De Clercq; John C. Drach
425-427	Activation of Nucleoside Hydrogenphosphonates by Use of Aryl Sulfonyl Chlorides	Per J. Garegg; Jacek Stawinski; Roger Strömberg
429-432	Studies on the Oxidation of Nucleoside Hydrogenphosphonates	Par J. Garegg; Tor Regberg; Jacek Stawinski; Roger Strömberg
433-435	Synthesis and ¹⁵N NMR of d[CGT(¹⁵N⁶)ACG] and d[CGT(CGT)(15N1)ACG]	Xiolian Gao; Roger A. Jones
437-439	Hybridization Probes with Deoxyinosine, Deoxyxanthosine or Deoxynebularine at Ambiguous Codon Positions	A. Van Aerschot; B. Peeters; H. Vanderhaeghe
441-442	Synthesis and Activity of Oligonucleotides Containing a Biologically Active Nucleoside at the 2′End	P. Herdewijn; R. Charubala; R. Pauwels; E. De Clercq; W. Pfleiderer
443-444	Synthesis and Biological Activity of 3′-Modified 2′-5′ Adenylate Trimers	P. Herdewijn; R. Charubala; R. Pauwels; E. De Clercq; W. Pfleiderer
445-446	Easily Available Column Device for Manual Oligonucleotide Synthesis on Solid Support by P(III) Methodology	R. W. Adamiak; F. Cramer
447-449	Oligomers Containing 2′-Deoxyinosine Isosteres as Ambiguous Nucleoside or 1,3-Propanediol as Nucleoside Substitute	Frank Seela; Klaus Kaiser
451-456	Phosphoramidites of [180] Chiral (Rp)- and (Sp)-Configurated Dimer-Blocks and their Use in Automated Oligonucleotide Synthesis	F. Seela; A. Kehne; W. Herdering; U. Kretschmer
457-460	Substituent Influence on the Reaction Rate of Deoxyribonucleoside Phosphoramidites with Deoxyribonucleosides Catalysed by Tetrazole	Bjarne H. Dahl; John Nielsen; Otto Dahl
461-463	Solid Phase Synthesis of DNA Under a Non-Depurinating Condition with a Base Labile 5′-Protecting Group (Fmoc) Using Phosphiteamidite Approach	N. Balgobin; J. Chattopadhyaya
465-466	Anomeric Mixtures of D-Xylo-and D-Lyxo-Furanonucleosides: Correlations between their Structures and their Retention Times in HPLC Analysis	A. Pompon; G. Gosselin; M. C. Bergogne; J. L. Imbach
467-468	DNA Apurinic Sites: Synthesis of a Model Compound and Study of its Reactivity with 3-Aminocarbazole	J. -J. Vasseur; B. Rayner; J. -L. Imbach; S. Verla; J. A. McCloskey; J. W. Lown; D. K. Chang
469-470	Unexpected Transposition of a Deoxyguanosine Derivative	A. -F. Maggio; M. Lucas; J. -L. Barascut; J. -L. Imbach
471-472	α-DNA. Synthesis, Characterization and Base-Pairing Properties of Unnatural α-Oligodeoxyribonucleotides	P. Morvan; B. Rayner; J. -L. Imbach; D. -K. Chang; J. W. Lown
473-475	Amide Protection in Oligodeoxynucleotide Synthesis	Joachim W. Engels; Matthias Mag

Volume 6, Issue 1-2 (1987)

477-481	Preparation of ¹⁵N Labeled Nucleosides and Large Scale Synthesis of Labeled Oligonucleotides with a New Type DNA-Synthesizer	B. Fera; B. Singrün; G. Kupferschmitt; J. Schmidt; F. Buck; H. Ruterjans
483-484	Oligonucleotide Analogues with Dialkyl Silyl Internucleoside Linkages	Hartmut Seliger; Georg Feger
485-488	Automated Preparation of DNA-RNA Hybrids and their Joining with RNA Ligase; An Approach to Single-Strand Gene Synthesis	D. Zeh; H. Seliger
489-490	Use of Long Oligonucleotides in Gene Synthesis: Chemical Synthesis and Cloning of a Gene for Salmon Calcitonin	F. Hein; H. W. Jansen; E. Uhlmann
491-493	The 9-Fluorenylmethyloxycarbonyl (Fmoc) Group as a 5′-O Base Labile Protecting Group in Solid Supported Oligonucleotide Synthesis	Yunxi; Etienne Sonveaux
495-496	2′-Deoxycoformycin: Biosynthesis and Enzymatic Conversion of 8-Keto-Deoxycoformycin to 2′-Deoxycoformycin by Streptomyces Antibioticus	Jeffery C. Hanvey; Elma Smal; Robert J. Suhadolnik; David C. Baker
497-500	Cordycepin Analogs of 2–5 a as Activators of RNase L: Study of the Structural Requirements for RNase L Activation	Katalin Kariko; Nancy L. Reichenbach; Robert J. Suhadolnik; Ramamurthy Charubala; Wolfgang Pfleiderer
501-503	Base Labile Protecting Groups for Hydroxyl Functions in Ribonucleosides and Deoxyribonucleosides	H. Schirmeister; W. Pfleiderer
505-507	Synthesis of 2′-O-p-Nitrophenylethylsulfonyl-Ribonucleosides	M. Pfister; W. Pfleiderer
509-511	Synthesis of Modified Thymidine Dimers	S. Farkas; W. Pfleiderer
513-516	Synthesis of P-Thioadenylyl (2′-5′) Adenosine and P-Thioadenylyl (2′-5′)-P-Thioadenylyl-(2′-5′)-Adenosine	R. Charubala; W. Pfleiderer
517-520	2′-OH Protection by the p-Nitrophenylethylsulfonyl (NPES) Group in Oligoribonucleotide Synthesis	R. Charubala; W. Pfleiderer
521-522	2′5′-Phosphodiesterase Activity Studies with Xyloadenosine Analogs of 2–5A Cores	P. P. Torrence; D. Alster; S. Huss; G. Gosaelin; J. -L. Imbach
523-524	Only One 3′-Hydroxyl Group Of ppp 5′A 2′p 5′A 2′p 5′A(2–5A) is Required for Activation of the Mouse 2–5A-Dependent Endonuclease	P. F. Torrence; D. Alster; R. Charubala; W. Pfleiderer; D. Brozda
525-526	2′,5′-Phosphodiesterase Activity Depends Upon the Presence of a 3-Hydroxyl Moiety in the Penultimate Position of the Oligonucleotide Substrate	David Alster; Danuta Brozda; Yukio Kitade; Alice Wong; Ramamurthy Charubala; Wolfgang Pfleiderer; Paul Torrence
527-528	Synthesis of 2′-5′ Adenylate Trimers Containing 3′-Modified β-D-Xylofuranosyl-Adenine Derivatives at the 2′-End	K. Ruf; P. Herdewijn; W. Pfleiderer
529-531	Synthesis of 0⁶-Alkylated Guanosine and Deoxyguanosinephosphoramidites	B. S. Schulz; W. Pfleiderer
533-535	5-Substituted 2-(Pyrimidin-2-yl)-Ethanols as New Phosphate Protecting Groups	T. Reiner; W. Pfleiderer
537-539	Synthesis of Terminal Nucleoside Phosphates and Thiophosphates via Phosphoramidite Chemistry	M. W. Schwarz; W. Pfleiderer
541-542	Synthesis and Hybridization Characteristics of Oligodeoxynucleotide-Alkaline Phosphatase Conjugates	Jerry L. Ruth; Edward Jablonski

Volume 5, Issue 5 (1986)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 5, Number 5
461-469	Photochemical Synthesis of 6-Aryluridines¹⁾	Kazue Satoh; Hiromichi Tanaka; Atsuko Andoh; Tadashi Miyasaka
471-480	Restricted Joining of a Decadeoxyribonucleotide for Preparation of an Eicosadeoxyribonucleotide Duplex Containing Recognition Sites for Restriction Enzymes	Y. Ishino; S. Shibahara; E. Ohtsuka; M. Ikehara
481-491	NMR Investigations of the Solution Conformations of Deoxynucleotidyl (3′-5′) Arabinonucleosides	S. H. Gray; C. F. Ainsworth; C. L. Bell; S. S. Danyluk; M. Maccoss
493-501	Negative Chronotropic Action of Adenosine in Rat Atria: Evidence for Action at A₁ Receptors	K. Kurahashi; David M. Paton
503-509	Increased Nucleoside Concentrations in Tumors as Markers of Tiazofurin Action	Hiremagalur N. Jayaram; Konrad Pillwein; George Weber
511-516	Synthesis of the Selenium Analog of the Cytokinin 6-(3-Methyl-2-Butenylamino)-2-Methylthio-9-(β-D-Ribofuranosyl)Purine	Dean S. Wise Jr.; Leroy B. Townsend
517-527	Nucleosides, XLIII¹⁾ Synthesis and Properties of 0⁴-Alkylthymidines	Leonidas Kiriasis; Silke Farkas; Wolfgang Pfleiderer
529-537	Nucleosides, III¹ Synthesis and Properties of 2-Trifluoromethyl-Naphthimidazole-Ribonucleoside	Abdullah Hijazi
539-569	Nucleosides 137. Synthetic Modifications at the 2′Position of Pyrrolo[3,2-D]Pyrimidine and Thieno[3,2-D]Pyrimidine C-Nucleosides, Synthesis of “2′-Deoxy-9-Deazzadenosine” and of “9-Deaza ARA-A”	Kambhampati V. B. Rao; Wa-Yun Ren; Joseph H. Burchenal; Robert S. Klein
571-578	The Carbocyclic Analogue of 5-(1-Propenyl)-2′-Deoxyuridine; Synthesis and Anti-Herpes Activity	John Goodchild; Harry J. Wadsworth; Iain S. Sim

Volume 5, Issue 4 (1986)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 5, Number 4
343-362	Synthesis of Certain 5′-Substituted Derivatives of Ribavirin and Tiazofurin	Naeem B. Hanna; Krishna G. Upadhya; Charles R. Petrie; Roland K. Robins; Ganapathi R. Revankar
363-383	Chemical Synthesis of RNA Fragments Related to the C4N Hypothesis	Hiroshi Tanimura; Mitsuo Sekine; Tsujiaki Hata
385-397	Studies on the Chemistry of 5-Acetoxy-6-(Acetoxymethyl)-Uridines: Synthesis of a New type of 5′-Cyclonucleoside¹	Rama S. Sodum; Brian A. Otter
399-411	Synthetic Studies with Thiosugar Nucleosides¹	G. Wayne Craig; John G. Moffatt
413-421	Uridine-5′-Diphosphate Glucose Analogues. 2¹. Nucleoside Modified Analogues of Antiviral 5′-O-[[[[(α-D-Glucopyranosyl)Oxy Carbonyl]Amino]Sulfonyl]Uridine Derivatives	Ma José Camarasa; Piedad Fernández-Resa; Ma Teresa García-López; Federico G. de las Heras; Paloma P. Méndez-Castrillón
423-429	Synthesis of 2-(β-D-Ribofuranosyl)Thiazole-4-Carboxamide 5′-Phosphate Isosteres	J. Ignacio Andrés; Ma Teresa García-López; Federico G. De las Heras; Paloma P. Méndez-Castrillón
431-439	The Synthesis of Coformycin from 5-Amino-1-β-D-ribofuranosylimidazole-4-carboxamide	H. Jeanette Thomas; James M. Riordan; John A. Montgomery
441-455	Synthests and Biological Evaluation of a Series of Substituted-2-Pyridine-C-Nucleosides. Part II	M. Belmans; I. Vrijens; E. Esmans; R. Dommisse; J. Lepoivre; F. Alderweireldt; L. Townsend; L. Wotring; J. Balzarini; E. De Clercq
457-460	Nucleosides/Tides Abstracts	Marshall W. Logue

Volume 5, Issue 3 (1986)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 5, Number 3
233-241	A Convenient Preparation of a New C-5 Biotinylated dUTP Derivative	Paul S. Nelson; Chander Bahl; Ian Gibbons
243-252	Nucleosides, XLII. Synthesis and Properties of Lin-Naphthotriazole-Ribosides	Abdullah Hijazi; Wolfgang Pfleiderer
253-263	Isolation and Characterization of a Novel Nucleoside from Human Cancer Urine	Henry A. Tworek; Wanda Bolanowska; Arvind K. Bhargava; Elliot M. Rachlin; Girish B. Chheda
265-273	Synthesis of Radio-Labelled and Unlabelled O⁴-Ethylthymidine 5′-Triphosphate	A. Bhattacharyya; B. C. Pal
275-300	Chemical Synthesis of Fully and Partially Xyloadenosine-Substituted 2′, 5′-Oligoadenylates Designed as New Potential Antiviral and Antitumor Agents	Sophie Huss; Gilles Gosselin; Alain Pompon; Jean-Louis Imbach
301-312	Aminopyrimidines and Derivatives. 19 ¹. Reaction of 1, 6-Dihydro-4-Beta; D (2, 3, 4, 6-Tetra-0-Acetyl)Glucopyranosylamino-1-Methyl-Z-Methoxy-6-Oxo Pyrimidine with Choracetyl Chloride	Manuel Nogueras; Luisa Quijano; Miguel Melgarejo; Adolfo Sqnchez
313-323	Approaches to the Synthesis of Sinefungin Via Nitroaldol Reactions	J. Grant Buchanan; Anthony Flinn; Paul H. C. Mundill; Richard H. Wightman
325-330	A Simple and Stable Silica Gel Support for the Oligodeoxyribonucleotide Synthesis	Joseph Deutsch; Sason Cohen; Moshe Weisz; Jehoshua Katzhendler
331-342	Synthesis of 6-Substituted Purine 2′-Azido- and 3′-Azido-Deoxypentopyranoses	Genevieve Carret; Annie Grouiller; Bernard Chabannes; Henri Pacheco

Volume 5, Issue 2 (1986)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 5, Number 2
117-124	Commentary: Metabolic Impediments to the use of Nucleotide Derivatives to Circumvent Resistance to Purine and Pyrimidine Analogs	L. Lee Bennett Jr.; R. W. Brockman; John A. Montgomery
125-134	Synthesis and Biological Evaluation of 3-Deazacytidine and 3-Deazauridine Derivatives	Michel Legraverend; Chi Hung Nguyen; Aurelio Zerial; Emile Bisagni
135-151	Formycin Analogs II. Antiviral and Cytotoxic s-Triazolo [4, 3-a] - and [1, 5-a] Pyridine Derivatives	J. Kobe; B. Brdar; J. Sorič
153-157	Amino-4 Dihydroxy-2, 6 (Desoxy-2-D-ribofurannosyl)-1-s-Triazines	Sylvie Pochet; Tam Huynh-dinh
159-168	Partial Protection of Carbohydrate Derivatives. Part 19. Highly Regioselective 5′-O-Aroylation of 2′-Deoxyribonucleosides in Terms of Dilution - Drop-by-Drop - Addition Procedure	Shigeyoshi Nishino; Hisanao Yamamoto; Yasuhiro Nagato; Yoshiharu Ishido
169-183	Acyclic Nucleosides Containing Two Heterocyclic Bases	Kelvin K. Ogilvie; H. R. Hanna; Zbigniew Proba
185-200	5′-Halogenated Formycins as Inhibitors of 5′-Deoxy-5′-methylthioadenosine Phosphorylase: Protection of Cells Against the Growth-Inhibitory Activity of 5′-Halogenated Adenosines	Shih Hsi Chu; Lynn Ho; Edward Chu; Todd Savarese; Zhi Hao Chen; Elizabeth Claflin Rowe; Ming Yu Wang Chu
201-212	Studies on the Preparation, Isolation, and Reactions of Adenosine Schiff Bases	Edward W. Badger; Deedee S. Szotek; Walter H. Moos
213-222	Synthesis of 2-Azido-(R)-N⁶-p-hydroxyphenylisopropyladenosine (R-AHPIA) as Potential Photoaffinity Probe for A₁ Adenosine Receptors	Gloria Cristalli; Mario Grifantini; Sauro Vittori; Karl-Norbert Klotz; Martin J. Lohse
223-228	Synthesis of 1-(4-Keto-2, 3-O-isopropylidene-α-L-rhamnopyranosyl) uracil	Vera Cheng; Lawrence Hughes; Vivian B. Griffin; Roland Montserret; Abraham P. Ollapally
229-232	Nucelosides/Tides Abstracts

Volume 5, Issue 1 (1986)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 5, Number 1
1-13	Alkaline Degradation of 1,3-Di-(2-Hydroxyethyl)adenosine 3′,5′-cyclic Phosphate. Studies on the Reaction Products	JÓZsef Béres; Yang-Chih Lee; Diana I. Brixner; Jay I. Olsen; Martin P. Schweizer
15-32	Synthesis of a Gene Coding for Human Vasoactive Intestinal Peptide (VIP)	Nicole Y. Theriault; Che-Shen C. Tomich; Wendell Wierenga
33-43	Oligodeoxyribonuclsotide-3′-phosphate Synthesis by Selective Cleavage of 3′-Terminal Uridine	N. F. Krynetskaya; G. V. Zayakina; T. S. Oretskaya; E. M. Volkov; Z. A. Shabarova
45-63	Oligothymidylates Substitubs en Position 3’ Par un Derive De L'Acridine	U. Asseline; N. T. Thuong; C. Hélène
65-77	Polymer Support Oligonucleotide Synthesis XX: Synthesis of a Henhectacosa Deoxynucleotide by Use of a Dimeric Phosphoramidite Synthon	A. Wolter; J. Biernat; H. Köster
79-93	Synthesis And Spectral Properties of Uric Acid Ribosides	Juris A. Maurinš; Ruta A. Paegle; Margeris J. Līdaks; Evgeny I. Kvasyuk; Pjotr V. Kuzmichkin; Igor A. Mikhailopulo
95-112	Structure and Conformation of the Antiviral Agent 5-Methoxymethyl-2′-deoxyuridine	Ossama A. L. El-kabbanit; Irena Ekiel; Louis T. J. Delbaere; Guy Tourigny; Allan L. Stuart; Sagar V. Gupta

Volume 4, Issue 5 (1985)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 4, Number 5
545-564	Synthesis and biological activities of 2-Pyrimidinone Nucleosides. III.^1,2 5-Alkynyl-2-Pyrimidinone 2′-Deoxyribosides	Simon M. N. Efange; Yung-Chi Cheng; Thomas J. Bardos
565-585	Novel Acyclonucleosides. Part I. 2,3-Dihydroxy-1-Methoxypropyl-and 3-Hydroxy-1-Methoxypropyl-Substituted Pyrimidines	Stuart Bailey; Colin T. Shanks; Michael R. Harnden
587-594	Conformational Analysis of 6-Substituted Uridine Analogues: Crystal Structures of Uridine-6-Thiocarboxamide and 6-Cyanouridine	Vivian Cody; Thomas I. Kalman
595-606	A New Simple Synthesis of N-2-Methylguanosine and Its Analogues Via Derivatives of 4-Desmethylwyosine (Nucleosides and Nucleotides. Part 63¹)	Jerzy Boryski; Tohru Ueda
607-612	Introduction of an Azido Group to the C-6 Position of Uridine by the Use of a 6-Iodouridine Derivative	Hiromichi Tanaka; Hiroyuki Hayakawa; Kazuhiro Haraguchi; Tadashi Miyasaka
613-624	Nucleosides. 131. The Synthesis of 5-(2-Chloro-2-Deoxy-β-D-arabino-Furanosyl)Uracil. Reinterpretation of Reaction of ψ-Uridine With α-Acetoxyisobutyryl Chloride. Studies Directed Toward the Synthesis of 2′-Deoxy-2′-Substituted Arabino-Nucleosides. 2	Krzysztof W. Pankiewicz; Kyoichi A. Watanabe
625-639	Adenosine and 2-Chloroadenosine Deaza-Analogues as Adenosine Receptor Agonists¹	Gloria Cristalli; Mario Grifantini; Sauro Vittori; Walter Balduini; Flaminio Cattabeni
641-649	The Synthesis of 5′-O-Dimethoxytrityl-N-Acyl-2′-Deoxynucleosides. Improved ‘‘Transient Protection'’ Approach¹	Ryszard Kierzek
651-659	Synthesis and X-Ray Crystal Structure of 2-β-D-Ribofuranosylthiazole-4-Carboxamide-N₃-Oxide	N. Kent Dalley; Charles R. Petrie III; Ganapathi R. Revankar; Roland K. Robins
661-668	The Structure of Neplanocin C	Kenji Kinoshita; Satoshi Yaginuma; Mitsuo Hayashi; Kazumi Nakatsu
669-679	A New Phosphorylating Agent, Di(2,2,2-Trifluoroethyl) Trimethylsilyl Phosphite. Its Application in Dna Synthesis by The Phosphotriester Approach	Kazuaki Imai; Tsunehiko Ito; Susumu Kondo; Hiroshi Takaku
681-694	Nucleosides. Part 3.¹ Synthesis of 2-N-Substituted 1-β-D-Arabinofuranosylisocytosine Derivatives by The Reaction of 2′,5′-Dichloro-2′,5′-Dideoxyuridine with Amines	Kosaku Hirota; Yukio Kitade; Tetsuo Tomishi; Yoshifumi Maki

Volume 4, Issue 4 (1985)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 4, Number 4
429-445	Syntheses, Activites Biologiques et Etude Conformationnelle D'Alcynyl-5 Desoxy-2′ Uridines	Patrice Vincent; Jean-Pierre Beaucourt; Louis Pichat; Jan Balzarini; Erik De Clercq
447-462	Syntheses et Activites Biologiques de Nouvelles (E)-Alcenyl-5 Desoxy-2′ Uridines	Patrice Vincent; Jean-Pierre Beaucourt; Louis Pichat; Jan Balzarini; Erik De Clercq
465-476	Synthesis of Analogues of Ribosylbarbituric Acid	M. R. Harnden; R. L. Jarvest
477-486	Synthesis of An Acid-Stable 2,5′-Cyclo-2-oxo Analogue of Wyosine (Nucleosides and Nucleotides. Part 61¹)	Jerzy Boryski; Tohru Ueda
487-506	Synthesis and Perkow Reaction of Uridine Derivatives	Joachim Thiem; Dieter Rasch
507-513	N-Substituted Acyclopurinenucleosides with Antiviral Activity	Kelvin K. Ogilvie; H. R. Hanna; Nghe Nguyen-ba; Kendall O. Smith
515-521	Synthesis of 1-(2-Deoxy-β-D-ribofuranosyl)benzimidazole via Cyclonucleosides	Morio Ikehara; Tetsuya Inaoka
523-538	Synthesis and Biological Evaluation of a Series of Substituted 2-Pyridine C-Nucleosides I. Coupling reaction of organo-metallic pyridine compounds with 2,4:3,5-di-O-benzylidene-aldehydo-D-ribose.	Marc Belmans; Eddy Esmans; Roger Dommisse; Jozef Lepoivre; Frank Alderweireldt; Jan Balzarini; Erik De Clercq
539-543	Nucleosides/Tides Abstracts	Marshall W. Logue

Volume 4, Issue 3 (1985)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 4, Number 3
309-345	Fast atom Bombardment Mass Spectrometry of Nucleosides, Nucleotides and Oligonucleotides	Debra L. Slowikowski; Karl H. Schram
347-376	Fast ATOM Bombardment Mass Spectra of Nucleosides. Comparison with Electron Impact and Chemical Ionization Mass Spectra	Debra L. Slowikowski; Karl H. Schram
377-389	Synthesis and Physical Characterization of Bis 3′→5′ Cyclic Dinucleotides (NpNp): RNA Polymerase Inhibitors	Hsu Chin-Yi Jenny; Dennis Don; Jones Oger
391-394	Assignment of ¹³C Chemical Shifts of α-D-Ribonucleoside Sugar Carbons by ¹J(CH) Coupling Constants	Frank Seela; Werner Bussmann
395-400	Synthesis of 5′-O-Aminothymidine and 5′-Deoxy-5′-Hydrazinothymidine, Novel Nucleoside Derivatives	Lawrence C. Davies
401-409	Synthesis of 2′-Deoxy-6,2′-Ethano-Cyclouridine¹ (Nucleosides and Nucleotides. Part 57)	Tohru Ueda; Satoshi Shuto; Miyuki Satoh; Hideo Inoue
411-427	Acyclic Nucleosides other than Acyclovir as Potential Antiviral Agents	Richard J. Remy; John A. Secrist

Volume 4, Issue 1-2 (1985)

a	Editorial board page for “Nucleosides, Nucleotides & Nucleic Acids”, Volume 4, Number 1-2
3-11	Targets for the Antiviral and Antitumor Activities of Nucleoside, Nucleotide and Oligonucleotide Analogues	Erik De Clercq
13-19	Studies in the Synthesis and Biosynthesis of C-Nucleosides	J. G. Buchanan
21-28	Enantioselective Synthesis of Carbocyclic Nucleosides by Enzymatic Approach and the Anticancer Activities	Masaji Ohno
29-66	Synthesis, Biochemical and Chemotherapeutic Activity of Some Azolo[1,3]Oxazine Nucleosides	Leroy B. Townsend; Vladimir G. Beylin; Linda L. Wotring
67-75	Synthesis and Some Biological Properties of Carbon-Bridged Cyclonucleosides and Their Phosphates	Tohru Ueda
77-79	Stabilisation of DNA by Incorporation of Phosphothioate Groups	F. Eckstein
81-94	The p-Nitrophenylethyl Group - An Universal Blocking Group in Nucleoside and Nucleotide Chemistry	W. Pfleiderer; F. Himmelsbach; R. Charubala; H. Schirmeister; A. Beiter; B. Schulz; T. Trichtinger
95-105	Studies on Nucleotide Chemistry 15. Synthesis of Oligodeoxynucleotides Using Amidine Protected Nucleosides	Marvin H. Caruthers; Lincoln J. Mcbride; Laurent P. Bracco; John W. Dubendorff
107-116	Metabolism and Metabolic Effects of Halopurine Nucleosides in Tumor Cells in Culture	L. L. Bennett Jr; C. -H. Chang; P. W. Allan; D. J. Adamson; L. M. Rose; R. W. Brockman; J. A. Secrist III; A. Shortnacy; J. A. Montgomery
117-127	Some Aspects of the Chemical Synthesis of Oligoribonucleotides	Colin B. Reese
131-133	Oxygen Chiral Phosphate in Ribo- and 2′-Deoxyribodinucleoside Monophosphates by Oxidation of Phosphite Intermediates	Frank Seela; Johann Ott; Barry V. L. Potter; Wilhelm Herdering
135-137	HPLC and LC-MS of Nucleosides	F. C. Alderweireldt; E. L. Esmans; P. Geboes
139-142	Rapid Synthesis of Oligodeoxyribonucleotides VIII.¹ An Improved Procedure for Solid-Phase Oligodeoxyribonucleotide Synthesis Using a Controlled Pore Glass Support and Phosphotriester Chemistry	B. S. Sproat; C. Minganti; M. J. Gait
143-146	Regioselective 2′-O Sugar Arylation in Adenine Nucleosides by The Elliptinium Agetate, An Antitumor Agent	G. Pratviel; J. Bernadou; B. Meunier; C. Paoletti
147	l-Methyl-Z-(2′-Hydroxyphenyl)Imidazole–A Catalytic Phosphate protecting group in deoxyoligonucleotide synthesis	Brian C. Froehler; Mark D. Matteucci
149-151	Analogues of Uridinediphosphatehexoses. A New Type of Protein Glycosylation Inhibitors That Show Antiviral Activity	M. J. Camarasa; P. Fernández-resa; M. T. García-lópez; F. G. de las Heras; P. P. Méndez-castrillónt; B. Alarcón; L. Carrasco
153-155	The p-Phenylazophenyloxycarbonyl Protecting Group: Selective Deblocking and Oligonucleotide Synthesis Avoiding Acid Steps	Hartmut Seliger; Udo Kotschi
157-160	Synthesis, Specific Intracellular Delivery and Biological Activity of Novel Stabilized (2′-5′)(A)_n Analogues	B. Bayard; L. D. Leserman; C. Bisbal; G. Huez; M. Silhol; B. Lebleu

Volume 4, Issue 1-2 (1985)

161-163	Reaction of Acetylenic Compounds With Nucleobases in Nucleosides, Nucleotides and Poly(A)	M. Olomucki; J. Y. Le Gall; P. Roques; F. Blois; S. Colinart
165-167	Isopolar vs Isosteric Phosphonate Analogues of Nucleotides	G. Michael Blackburn; Fritz Eckstein; David E. Kent; Timothy D. Perrée
169-171	Preparation and Properties of Chloro-N, N-dialkylamino-2,2,2-trichloroethoxy- and Chloro-N, N-dialkylamino-2,2,2-trichloro-1,1-dimethylethoxyphosphines and their Deoxynucleoside Phosphiteamidates	G. Hering; R. Stöcklein-schneiderwind; I. Ugi; T. Pathak; N. Balgobin; J. Chattopadhyaya
173-175	Synthesis and Antiviral Activity of 5-Halovinyl-6-Aza-2′-Deoxyuridines	W. L. Mitchell; P. Ravenscroft; M. L. Hill; L. J. S. Knutsen; R. F. Newton; D. I. C. Scopes
177-181	The Protection of The 2′-Hydroxyl Function in Oligoribonucleotide Synthesis	A. Sandström; M. Kwiatkowski; J. Chattopadhyaya
183-185	Chemoenzymatic Synthesis of a Gene Control Region	J. Engels; M. Leineweber; E. Uhlmann
187-189	Some Aspects of Ribonucleoside Chemistry	S. Juntunen; H. Essadiq; A. Grouiller; J. Chattopadhyaya
191-193	¹H-NMR Assignment of Single Strand and Duplex Splice Domain of the Consensus Donor Exon:Intron Junction	J. W. Lown; C. C. Hanstock; R. C. Bleackley; J. -L. Imbach; B. Rayner; J. J. Vasseur
195-198	Synthesis of 3′-Deoxyadenylate Trimer	F. Himmelsbach; E. Uhlmann; R. Charubala; W. Pfleiderer
199-200	Glycosylation of 5-Hydroxy-4-cyanoimidazole	Fatma Ibrahim-lodgemann; Grahame Mackenzie; Gordon Shaw
201-203	Synthesis of Oligodeoxynucleotides Containing 5-Bromouracil and N6-Methyladenine	A. M. Delort; A. Guy; D. Molko; R. Teöule
205-207	The Role of Glycosylases in Mismatch Repair: The Use of 7-Deazapurines as Repair-Resistant Lesions in Oligonucl, Eotide-Directed Mutagenesis	Josef Jiricny; Aiko Ubasawa; Steven Wood
211-212	Therapeutic Implications of The Unusually Long Half-Life of (E)-5–(2–bromovinyl)uracil (Bvura) In Vivo	C. Desgranges; G. Razaka; E. De Clercq; H. Bricaud
213-214	Preparation of Guanosines Modified by Carcinogenic Aromatic Amines	B. Robillard; M. F. Lhomme; J. Lhomme
215-216	Non-Glycosidic Derivatives of 5-Fluorouracil	G. J. Koomen; J. B. M. Van Rhijn; U. K. Pandit
217	Approach to the Synthesis of 2-(D-Ribofuranosyl)-Pyridine Compounds	E. L. Esmans; M. Belmans; I. Vryens; R. Dommisse; J. A. Lepoivre; F. C. Alderweireldt
219	A Rapid Protocol For Site-directed Mutagenesis and Gene Synthesis Using Synthetic Oligonucleotides	M. Wintzerith; M. Zenke; T. Grundström; H. Matthes; C. Schatz; A. Staub; P. Chambon
221-223	D-xylo and Lyxofuranonucleosides Reviewed: Some Suggestions on The Mechanism of Activity of Antiviral Nucleosides	J. De Rudder; J. Leclerc; M. Mercier; G. Gosselin; J. L. Imbach
225-226	Corneal Permeability of 5-Iodo-2′-deoxycytidine	V. Sincholle; J. P. Conduzorgues; B. Mbatchi; J. P. Masse
227	Metabolisme Cutane de la Iodo-5-desoxy-2′-cytidine (IDC)	B. Mbatchi; V. Sincholle

Volume 4, Issue 1-2 (1985)

229	Synthesis of a Gene Coding for Vasoactive intestinal Peptide (VIP)	Nicole Y. Theriault; Wendell Wierenga
231-232	Synthesis of Imidazo[1, 2-a]pyrazine Nucleoside Analogues	P. Verschave; G. Hoornaert
233	Oligonucleotide-Intercalant: Substances à Forte Affinité Spécifique pour les Séquences d'Acides Nucléiques Effets de I'Estérification des phosphates	U. Asseline; N. T. Thuong; C. Helene
235	Novel Acyclic Analogues of Pyrimidine Nucleosides: 1-Methoxy-2, 3-Dihydroxypropyl and 1-Methoxy-3-hydroxypropyl Derivatives	S. Bailey; C. T. Shanks; M. R. Harnden
237	Deaza-analogues of Adenosine and 2-Chloroadenosine as Agonists of Adenosine Receptors	G. Cristalli; M. Grifantini; S. Vittori; W. Balduini; F. Cattabeni
239-240	Synthese Regiospecifique d'Un Dinucleoside Ponte: (O⁶ Desoxyguanosnyl)-1(N⁴-desoxycytidyl)-2 Ethane	Annie-Franyoiae Maggio; Marc Lucas; Jean-Louis Barascut; Jean-Louis Imbach
241	5-Haloethyl-deoxyuridine Analogues: Synthesis and Antiviral Activity	Herfried Griengl; Walter Hayden; Erich H'anek
243	A Rational Methodology for Rapid Chemical And Enzymic Synthesis of Long Double Stranded DNA: A Human β-Interferon Gene	R. Frank; G. Gross; G. Heisterberg-moutsis; D. Jentsch; D. Lincoln; U. Leuner; A. Meyerhans; L. Monaco; M. Rieger; H. Blbcker
245	Rapid Purification of Chemically Synthesized Oligodeoxy-Nucleotides	A. Meyerhans; G. Heisterberg-moutsis; G. Kurth; H. Blöcker; R. Frank
247-248	Trichloro-tert.-butyl-cyclic-enediol-phosphate (TCB-CEP), Proposed Reagent for the Syntheses of Oligonucleotides Using the Triester Approach	Peter Lemmen
249	Three-phase - Synthesis of Oligonucleotides	Hartmut Seliger; Kailash Chand Gupta
251	An Unusual Demethylation of 3-Methylguanine	Jerzy Boryski; Bozenna Golankiewicz
253	Anticancer Activities of 7-, and 9-Substituted 3-Deazaguanine Derivatives	Tasneem A. Khwaja; Sumitra Roy-burman; Stephanie Pentecost
255	Base-Pair Mismatch in DNA at 2.3A Resolution	Tom Brown; Olga Kennard; Geoff Kneale
257-258	Synthesis and Properties of Symmetrically Linked Diribonucleotides	M. Nemer; N. Thëriault; A. Schifman; K. K. Ogilvie
259-260	Signal Sequence: Application of Chemical DNA Synthesis to Studies of Studies of Translocation of Expressed Proteins	E. Uhlmann; J. Engels; W. Wetekam
261	Detection of Neuropeptide mRNA in Rat Brain byIn SituHybridization with Radiolabeled Synthetic Oligonucleotide Probes	R. Arentzen; R. W. Manning; B. Wolfson; L. G. Davis; G. A. Higgins; Y. Lin; F. Baldino Jr
263	Convenient Procedure for Oligonucleotide-Directed in vitro Mutagenesis of Cloned DNA	O. Chakhmakhcheva; O. Mirskikh; V. Efimov; Yu. Ovchinnikov
265	Rapid Chemical Synthesis of Oligodeoxyribonucleotides by the Improved Phosphotriester Method	V. A. Efimov; O. G. Chakhmakhcheva
267	Depurination As a Yield Decreasing Mechanism in Oligodeoxynucleotide Synthesis	J. William Efcavitch; Cheryl Heiner

Volume 4, Issue 1-2 (1985)

269	A Large Fragment Approach to Gene Synthesis	H. Rink; M. Liersch; P. Sieber; W. Märki; P. Meyer
271-272	Oligoribonucleotide Synthesis by the Phosphite Procedure from 2′-Dimethoxytritylated Nucleosides	Jean-Luc Decout; Kelvin K. Ogilvie
273	The Synthesis and Base-Pairing Properties of 2-Deoxy-7-deazanebularine	J. Jiricny; A. Ubasawa; S. Wood
275-277	Synthese de la Desamino 9’ Sinefungine	N. Dodic; M. Gèze; P. Blanchard; J. L. Fourrey; Robert Géro
279	As-Triazine-3, 5-Dione Acyclic Nucleosides	Bihi H. Lazrek; Raymond P. Panzica
281	Enzymic Phosphorylation of Some 5-Aminoimidazole Nucleosides to the 5′-Phosphates	Robert W. Humble; Grahame Mackenzie; Gordon Shaw
283	Thymidylate Synthetase-Positive and -Negative Mouse Mammary Carcinoma Cell Lines: Useful Model for Monitoring the Incorporation of Pyrimidine Nucleoside Analogues into Host Cell DNA and for Detecting Thymidylate Synthetase Inhibitors	J. Balzarini; E. De Clercq; D. Ayusawa; T. Seno
285	Two-Dimensional ¹H-N.M.R. Assignment of Short Duplex Oligodeoxyribo-Nucleotides Which May Be Used as Potential Targets for Anticancer Drugs	J. W. Lown; C. C. Hanstock; R. C. Bleackley; J. -L. Imbach; B. Rayner; J. J. Vasseur
287	Selective Deuteration Labelling of 2′-Deoxyguanosine at the Carbon C-4’ Position	M. Berger; J. Cadet
289-290	Synthesis of 5, 6-Dichloro-Benzimidazole-(2′, 5′)-Nucleotide Trimer	K. Ruf; W. Pfleiderer
291-292	p-Nitrophenylethyl-Phosphoramidites	M. W. Schwarz; W. Pfleiderer
293	Acyclonucleoside Inhibitors of Uridine Phosphorylase	M. Draminski; A. Zgit-wroblewska; A. Drabikowska; D. Shugar
295	Biotin-Labeled Synthetic Oligodeoxyribonucleotides: Chemical Synthesis and Uses as Hybridization Probes	André Chollet; Eric H. Kawashima
297	A Rapid Method for Simultaneous Chemical Synthesis of Oligonucleotides in Large Nufiber	H. Ilatthes; T. Grundstrom; M. Zenke; M. Wintzerith; A. Staub; P. Chambon
299	Monothiophosphate Analogs of Dinucleoside Tetraphosphate	A. F. Haikal; C. Chavis; J. L. Imbach
301-302	Raccourci Pour la Synthese de la S-(Amino-3-propyll-5′-thio-5′-aoenosine	P. Dewévre; C. Tapiero; J. L. Irnbach
303	The Synthesis and Antiherpetic Activity of DHBG and Some Analogs	Karin Eklind; Roelf Datema; Ann-Christin Ericson; Curt-Eric Hagberg; Nils-Gunnar Johansson; Susanna Kovacs; Alf Larsson; BjÖRn Lindborg; GÖRan Stening; Bo öberg
305	A Rapid Deprotection Procedure for Phosphotriester DNA Synthesis	T. P. Patel; M. A. Chauncey; T. A. Millican; M. A. W. Eaton
307	Chemical Synthesis and Cloning of a Gene Fragment Designed to Aid Polypeptide Purification	L. D. Bell; J. C. Smith; R. B. Derbyshire; E. Cook; L. Dunthorne; J. Viney; S. Brewer; H. Sassenfeld

Volume 3, Issue 5 (1984)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 3, Number 5
445-483	Covalent Interaction of Proteins and Nucleic Acids. Synthetic and Natural Nucleotide-Peptides	B. A. Juodka
485-498	Automated Solid Phase Synthesis of Oligoribonucleotides. The Synthesis of a tRNA Anticodon Loop from Nucleoside-3'-chlorophosphite Derivatives.	Richard T. Pon; Kelvin K. Ogilvie
499-512	Preparation and Characterization of Oligonucleotides of D- and L-2’ Deoxyuridine	David J. Anderson; Robert J. Reischer; Arlen J. Taylor; William J. Wechter
513-524	Nucleosides. 127. Synthesis of Pyrido[2,3-d]pyrimidine Nucleosides from 5-Cyanouridine	Tsann-Long Su; Kazuho Harada; Kyoichi A. Watanabe
525-535	Antiherpes Simplex Virus Activity of 9-[4-Hydroxy-3-(hydroxymethyl)-1-butyl] guanine	Michael A. Tippie; John C. Martin; Donald F. Smee; Thomas R. Matthews; Julien P. M. Verheyden
537-547	Synthesis of Purine and Pyrimidine Trihydroxyacyclonucleosides	Kelvin K. Ogilvie; Zbigniew A. Proba
549-557	Nucleosides, XL¹ Synthesis and Properties of lin-Naphthamidazole-Ribonucleosides	Abdullah Hijazi; Wolfgang Pfleiderer

Volume 3, Issue 4 (1984)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 3, Number 4
325-337	Synthesis of 2-S-dioxo Isosteres of Purine and Pyrimidine Nucleosides. III. Alkyl And Glycosyl Derivatives of Triazolo-and Thiadiazolothiadiazines.	B. Azmy; P. Fernández-resa; P. Goya; R. Nieves; C. Ochoa; M. Stud; M. L. Jimeno
339-343	Novel Synthesis of a 2, 5'-O-Cycloimidazole Nucleoside	Graham Mackenzie; Gordon Shaw; Hilary A. Wilson
345-351	Studies on the Chemical Synthesis of Potential Antimetabolites. 36. Synthesis and Some Biochemical Properties of (±)1-Deazaaristeromycin	Hiroaki Ohno; Tokuo Itoh; Akihiko Nomura; Yoshihisa Mizuno
353-361	Synthesis of O²- and O⁴-Ethylthymidine 5'-Triphosphates	A. Bhattacharyya; S. Mitra; B. C. Pal
363-367	Phosphorylation of Some 5-Aminoimidazole Nucleosides to the 5’ -Phosphates Using a Phosphotransferase from Wheat	Robert W. Humble; Graham Mackenzie; Gordon Shaw
369-388	New Methods for the Synthesis of Base Sensitive Cyanopyrimidine and Cyanopyridine Nucleosides	Celeste A. Schlieper; James Wemple
389-399	Mesoionic Nucleosides 3: Studies on Mesoionic Imidazo [2,1-b]-1/3-thiazine Derivatives	Richard A. Glennon; Shanaz M. Tejani
401-411	Synthesis of the Natural Product 5'-Deoxy-5-iodotubercidin and Related Halogenated Analogs	Alan F. Cook; Michael J. Holman
413-422	Studies on the Chemical Synthesis of Potential Antimetabolites. 371. Synthesis of 3-Deazaadenine Nucleosides Modified at the Sugar Moiety	Toyoaki Ishikura; Sumiyo Oue; Tokuo Itoh; Akihiko Nomura; Tohru Ueda; Yoshihisa Mizuno
423-439	Sur l'Obtention d'Oligonucleotides en Serie Ara-A	J. L. Barascut; H. B. Lazrek; J. L. Imbach
441-443	Nuclbosidest/tides Abstracts	Marshall W. Logue

Volume 3, Issue 3 (1984)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 3, Number 3
221-232	A Detailed Investigation of The Methylation Reaction of A 5-Bromopyrimidine Nucleoside	M. Márton-Merész; J. Kuszmann; J. Langò; L. Párkányi; A. Kálmán
233-244	Synthesis of 1-methyl-3-β-d-ribofuranosylpyrazolo[4, 3,-D]-pyrimidin-7(6h)-selone and Certain Related Nucleosides and Nucleotides	Bheemarao G. Ugarkar; Roland K. Robins; Ganapathi R. Revankar
245-264	Synthesis and Biological Properties of 9-(2, 4-Dihydroxybutyl) Adenine and Guanine: New Analogues Of 9-(2, 3-Dihydroxyprqpyl)adenine (Dhpa) and 9-(2-Hydroxyethoxymethyl)guanine (Acyclovir)	Jiří žemlička
265-275	Detention D′arabinofuranncwuclbdsides Par Transpdrmation Chemique De Certains Xylofurannonuclesosides	Gilles Gosselin; Maric-Christine Bergogne et Jean-Louis Imbach
277-286	Synthesis of 3′-Amino-3′-deoxyguanosine 5′-Triphosphate	G. M. Visser; R. Keemink; Cecile Schattenkerk; B. Kraal; J. H. Van Boom
287-294	Methylation of a Mesoionic Tricyclic Nucleoside Related to Wyosine	Jerzy Boryski; Bozenna Golankiewicz
295-302	Synthesis of 2′, 3′ -Dideoxy-6, 3′-Methano-cyclouridine and a Furanosyl To Pyranosyl Ring-isomerization In The C-cyclo-nucleoside (Nucleosides and Nucleotides. 53¹)	Tohru Ueda; Satoshi Shuto
303-311	Synthesis And Biological Activity Op Hydpdxymetflyl Analogs op 5-Benzylacyclouridine and 5-Benzyloxybenzylacycloaridine	Shih Hsi Chu; Zhi Hao Chen; Elizabeth C. Rowe; Fardos N. M. Naguib; Hahmoud H. el Kouni; Ming Y. Chu
313-318	Synthesis of 5-Chloro-l-(2, 3-Orisopropylidene-4-keto Rhamnopyranosyl)-uracil	Richard A. Ford; Mitchell Gibson; Hussain Rawji; Lawrence Hughes; Roland Montserret; Abraham P. Ollapally
319-323	Nucleosidesfi/Ides Abstracts	Marshall W. Logue

Volume 3, Issue 2 (1984)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 3, Number 2
115-121	New Acyclic C-Nucleosides of the Imidazole	J. Fuentes Mota; P. Areces Bravo; F. Rebolledo Vicente; J. I. Fernández García-Hierro; J. A. Galbis Pérez
123-146	Synthesis and Stereochemical Assignments for 2-(α- and β-D-Arabinofuranosyl)Thiazole-4-Carboxamides	Cong Jiang; Ralph H. Baur; James J. Dechter; David C. Baker
147-155	Synthesis of 1-(6-Mercaptopurinyl-9)-and 1-(6-Methylmercaptopurinyl-9)-β-D-glucofuranuronosides	Juris A. Maurinš; Ruta A. Paegle; Aina A. Zidermane; Margeris J. Lidaks; Evgeny I. Kvasyuk; Igor A. Mikhailopulo
157-171	Polymer Support Oligonucleotide Synthesis XVI: Synthesis of Oligonucleotides Using Suitably Protected Deoxynucleoside-N-morpholinophosphoramidites on Porous Glass Beads	N. D. Sinha; J. Biernat; H. Köster
173-182	Synthesis of 2′-C-Nitromethyl Derivatives of Uridine and the Structure of a Carbon-Bridged Cyclonucleoside Derived Therefrom (Nucleosides and Nucleotides 51)	Tohru Ueda; Satoshi Shuto; Hideo Inoue
183-186	The Structure of “N¹, N⁶-Carbonyladenosine”	Jiří Žemlička
187-194	Synthesis and X-Ray Crystal Structure of 3-Amino-1-β-D-Ribofuranosyl-s-Triazolo[5, 1-c]-s-Triazole	Steven G. Wood; N. Kent Dalley; Rose D. George; Roland K. Robins; Ganapathi R. Revankar
195-206	Synthesis of 7-Deazatriacanthine and Restricted Rotation of Amino Groups in Pyrrolo[2,3-d]Pyrimidines	Frank Seela; Werner Bussmann
207-219	Aminopyrimidines and Derivatives. 15¹. Synthesis of 3-Glycosyl-vic-Triazolo-(4,5-d) Pyrimidines²	R. Asenjo Asenjo; M. Melgarejo Sampedro; M. No-gueras Montiel; M. Rodríguez Alonso; C. Rodrí-guez Melgarejo; A. Sánchez Rodrigo

Volume 3, Issue 1 (1984)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 3, Number 1
1-31	Determination of the Anomeric Configuration of C-Nucleosides by ¹H and ¹³C NMR Spectroscopy	C. K. Chu; F. M. El-kabbani; B. B. Thompson
33-44	A Simple One-Pot Method for 6-Oxopurine Ribonucleoside Synthesis: Control and Mechanism of Isomer Distribution	Lech W. Dudycz; George E. Wright
45-60	Instability of the Phosphodiester-Amide Interribonucleotide Bond in Neutral Aqueous Solution	J. Tomasz; J. Ludwig
61-67	Chemical Synthesis of Cap Analogues: P¹,P²-Dinucleoside-5′-diphosphates	Wolfgang Goemann; Joachim Kruppa
69-76	Synthesis of Guanylyl (3′→5′)-5-methylcytidine (Gpm⁵C), a Dinucleoside Monophosphate which is Unable to Function as a Primer in the Synthesis of RNA by the Influenza A Virus RNA Polymerase	Zainub Khan; Mario Ariatti; Arthur Hawtrey
77-89	Synthesis of 2-(3-Deoxy-β-D-erythropentofuranosyl)-thiazole-4-carboxamide (3′-Deoxytiazofurin)	Ralph H. Baur; David C. Baker

Volume 2, Issue 5 (1983)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 2, Number 5
399-418	Preparation, Characterization and Reactivity of Diastereomeric Sulfoxides of 8,2′-S-Anhydroadenosine	Aria L. Schifman; Kelvin K. Ogilvie
419-434	Synthesis of 5-Mercaptocytosine Nucleosides and Nucleotides	V. C. Solan; G. L. Szekeres; E. K. Ryu; H. Kung; Y. K. Ho; T. J. Bardos
435-452	Synthesis of Deoxyribonucleotidyl (3′-5′) Arabinonucleosides	S. H. Gray; C. F. Ainsworth; C. L. Bell; S. S. Danyluk; M. Maccoss
453-458	Acetylation of Nucleosides by Acetylsalicylic Acid (Aspirin)¹	Chung K. Chu
459-464	A One Step Synthesis of O⁶-Methyl-2′-deoxyguanosine	Jean Bernadou; Michel Blandin; Bernard Meunier
465-478	Isolation and Identification of 5′-Methylthioadenosine Sulfoxide from Human Urine	John S. Mills; Gordon C. Mills; David J. Mcadoo
479-494	Inhibitors of Adenosine Deaminase: Synthesis of Coformycin and 3′-Deoxycoformycin	L. D. Hawkins; J. C. Hanvey; F. L. Boyd Jr.; David C. Baker; H. Hollis Showalter
495	Erratum

Volume 2, Issue 4 (1983)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 2, Number 4
295-318	Nucleosides Containing Selenium¹ II	Zbigniew J. Witczak
319-325	The Structure of 2′ (R)-Mercapto-2′-deoxyneplanocin A (Nucleosides and Nucleotides 48.)	Kenji Kinoshita; Mitsuo Hayashi; Takao Hirano; Kazumi Nakatsu; Kiyofumi Fukukawa; Tohru Ueda
327-334	Structure of 2′,3′-0-Isopropylidene-5-Bromouridine	Yuriko Yamagata; Yukari Kobayashi; Nobuo Okabe; Ken-Ichi Tomita; Tohru Ueda
335-343	Structure of 2′,3′-0-Isopropylidene-6-cyanouridine	Yuriko Yamagata; Yukari Kobayashi; Nobuo Okabe; Ken-Ichi Tomita; Tomoharu Sano; Hideo Inoue; Tohru Ueda
345-350	Synthesis of 3, N⁴-Dimethylcytidine	Kelvin K. Ogilvie; Harvey A. Kader
351-366	2′,5′-Adenylate and Cordycepin Trimer Cores: Metabolic Stability and Evidence for Antimitogenesis without 5′-Rephosphorylation	Robert J. Suhadolnik; Paul W. Doetsch; Yair Devash; Earl E. Henderson; Ramamurthy Charubala; Wolfgang Pfleiderer
367-372	Stereochemistry at the Benzylic Centre in Hydroxyglycitylanthraquinones	Owen Johnson; Derry W. Jones; David J. Mincher; Gordon Shaw
373-385	Improved Synthesis of 2′-Fluoro-2′-Deoxyadenosine and Synthesis and Carbon-13 NMR Spectrum of Its 3′,5′-Cyclic Phosphate Derivative¹	Seiichi Uesugi; Toshinori Kaneyasu; Jitsuhiro Matsugi; Morio Ikehara
387-397	Studies on the Chemical Synthesis of Potential Antimetabolites. 35.¹ Synthesis of 2-Chloro-1-deazaadenosine and 2-Chloro-1-deazainosine as Candidate Inhibitors for S-Adenosylhomocysteinases and Methyltransferases	Tokuo Itoh; Tomokazu Sugawara; Akihiko Nomura; Yoshihisa Mizuno

Volume 2, Issue 3 (1983)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 2, Number 3
193-202	Utilisation d'Un Nouveau Type de Support Pour la Synthese d'Oligonucleotides en Phase Solide	J. -L. Barascut; J. Cuartero; J. -L. Imbach
203-219	Synthesis and Properties of Mixed Anhydrides of AMP, ADP and ATP with Mesitoic Acid	N. I. Sokolova; S. S. Tretyakova; Z. A. Shabarova
221-229	Chemical Conversion of Some Ribonucleosides into the Corresponding β-D-Arabinofuranosyl Derivatives¹	Nobuo Sakairi; Ichiro Hirao; Yoshiaki Zama; Yoshiharu Ishido
231-242	Tauto Merism and Ionization of Xanthosine	Kunal B. Roy; H. Todd Miles
243-248	Aromatic Photosubstitution Reactions for the Synthesis of 5-Aryl-2′-Deoxyuridines	Laman Al-razzak; Mohamed E. Hassan; Mathias P. Mertes
249-255	Reaction of Azide Ion with 1-(2,3-Anhydrolyxofuranosyl)Uracil. Isolation of 1-(2-Amino-2-deoxy-β-D-Xylo-Furanosyl)uracil and 1-(3-Amino-3-deoxy-β-D-arabinofuranosyl)uracil	Charles F. Hummel; Robert P. Carty
257-274	Induction of Bacterial Differentiation by Adenine- and Adenosine-Analogs and Inhibitors of Nucleic Acid Synthesis	Zain-ul-abedin; Juan M. Lopez; Ernst Freese
275-289	Synthesis of 2′- and 3′-Ketoadenosines	Richard P. Crews; David C. Baker
291-294	A Simple Synthesis of 5-Amino-4-imidazolecarboxamide Riboside-5′-Tri-Phosphate: The Proposed Alarmone for 10-Formyl-tetrahydrofolate Deficiency	Thomas R. Webb

Volume 2, Issue 2 (1983)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 2, Number 2
99-112	Regiochemical Aspects in Reactions of 6-Azauridine Dialdehyde	Josef Nemec; Jerry M. Rhoades
113-125	Conversion of Tubercidin to Toyocamycin: Some Properties of Tubercidin Derivatives (Nucleosides and Nucleotides. 47)¹	Shin-Ichi Watanabe; Tohru Ueda
127-146	Synthesis of Mesoionic Xanthine Nucleosides	Ernst M. Schubert; Robert G. Bass; Richard A. Glennon
147-154	Synthesis of 5-Substituted-1-[[2-Hydroxy-1-(hydroxymethyl)ethoxy]methyl]cytosines	Kelvin K. Ogilvie; Dilip M. Dixit; Bruno K. Radatus; Kendall O. Smith; K. S. Galloway
155-173	The Reaction of D-Arabinopyranosylurea with Malononitrile and Triethyl Orthoformate	E. Stankevich; A. Dreimane; E. Liepinš; A. Kemme; J. Bleidelis
175-187	Formation of 5- and 6-Aminocytosine Nucleosides and Nucleotides from the Corresponding 5-Bromocytosine Derivatives: Synthesis and Reaction Mechanism	David Goldman; Thomas I. Kalman
189-191	Facile Synthesis of 5-Fluorocytidine	Minoti Sharma; James L. Alderfer

Volume 2, Issue 1 (1983)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 2, Number 1
1-20	Queuine, The Q-Containing tRNAs and the Enzymes Responsible for Their Formation	Walter R. Farkas
21-31	Synthesis and Biological Activities of Some New 5′-Substituted S-Adenosylhomocysteine Analogues*	David Shire; Pierre Blanchard; Aly Raies; Françhise Lawrence; Malka Robert-Géro; Edgar Lederer
33-40	Oligonucleotides and Nucleotidepeptides. XLIII. Inhibition of Lipoamide Dehydrogenase by Nucleotidyl-(�N)-amino Acids and Their Ethyl Esters¹	A. Glemzha; B. Juodka
41-49	Synthesis and Properties of 7-Acetyl-1, N⁶-etheno-AMP and 7-Acetyl-1, N⁶-etheno-NAD	Hermann H. Dieter; Rudolf Koberstein
51-61	3′-3′,3′-5′ and 5′-5′ TpT-Amides: Synthesis, Characterization and Alkaline Hydrolysis	J. Tomasz
63-79	P¹-(Thymidine 5′-)P¹-amino-triphosphate: Synthesis, Hydrolysis and Reaction with Cytidine in Alkali¹	J. Tomasz
81-90	Mechanisms of Formation of Cyclic Urea Nucleosides. 2. Direct N-Glycosylation Versus O- to N-Transglycosylation	Victor E. Marquez
91-98	Synthesis of Some Nucleoside Cyclic Ethylene Phosphothionates	S. Parekh; A. Patel; C. J. McNeal; J. Nagyvary

Volume 1, Issue 3 (1982)

a-b	Editorial board page for “Nucleosides & Nucleotides”, Volume 1, Number 3
205-231	Purine Nucleoside 3′,5′-Cyclic Monophosphates as Hormonal Modulators of Cellular Proliferation, Metastases and Lymphocyte Response	Roland K. Robins
233-237	Preparation of 9-β-D-Arabinofuranosylguanine (araG)	Ukken O. Cheriyan; Kelvin K. Ogilvie
239-251	Studies on the Chemical Synthesis of Potential Antimetabolites. 32.¹ Synthesis of β-D-Pentofuranosyldeazaadenines as Candidate Inhibitors for S-Adenosylhomocysteinases and Methyltransferases	Tomokazu Sugawara; Toyoaki Ishikura; Tokuo Itoh; Yoshihisa Mizuno
253-261	N⁴-(3-Methyl-2-Butenyl)-2-(Methylthio)Tubercidin and Its α-Anomer - 7-Deazapurine Nucleosides with Potential Anticytokinin Activity	Frank Seela; Werner Bussmann
263-273	Chemical Conversion of Uridine to 3′-Branched Sugar Nucleosides (Nucleosides and Nucleotides. 42¹.)	Satoshi Shuto; Tatsuyoshi Iwano; Hideo Inoue; Tohru Ueda
275-287	Synthesis of, and Conformational Studies on, 2-Trifluoromethyl, Substituted Benzimidazole Ribofuranosides	Zygmunt Kazimierczuk; Ryszard Stolarski; Lech Dudycz; David Shugar
289-295	Synthese d'Oligodesoxyribonucleotides sur Support de Gel de Silice par la Methode au Phosphotriester	J. Ben Hattar; B. Rayner; J. -L. Imbach
297-313	6,7-Dimethyl-3-β-D-Erythrofuranosyl-1-Phenyl- and 1-p-Fluorophenyl-Pyrazolo[3,4-b]QUINOXALINE*	Mohammed A. E. Sallam

Volume 1, Issue 2 (1982)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 1, Number 2
99-110	Partial Protection of Carbohydrate Derivatives. Part 9¹. Equilibration between 2′, 5′- and 3′, 5′-DI-O-Benzoyladenosine Derivatives Substituted at the N⁶-Position, on Silica Gel	Nobuo Sakairi; Dalilur Rahman; Kazuaki Tamaki; Yoshiharu Ishido
111-125	Oligonucleotides and Nucleotide-Peptides. XXXIX. Synthesis and Properties of the Simplest Models of Covalent Nucleic Acid (Nucleotide)-protein Complexes With The Phosphodiester Bond Between The Components^I	B. Juodka; V. Kirvelienè; P. Povilionis
127-138	Synthesis and Cytostatic Activity of Halomethylthiazole C-Nucleosides and Analogues¹	M. Teresa García-López; Rosario Herranz; Paloma P. Méndez-Castrillón
139-146	Synthetic Nucleosides and Nucleotides. XX¹. Synthesis of Various 1-β-D-Xylofuranosyl-5-Alkyluracils and Related Nucleosides	Chikao Nakayama; Mineo Saneyoshi
147-154	Studies on Nucleoside Analogs. XXV.¹) Synthesis of 5, 7-Dioxopyrimido[5,4-e]-AS-Triazine Glycosides	Haruo Ogura; Hiroshi Takahashi; Kikuko Ohokubo
155-161	Synthesis of Acetylated α-and β-L-Fucosyl Esters of Nucleoside 5′-Monophosphates by the Orthoester Route	Mohammed A. Salam; Edward J. Behrman
163-171	Polyribonucleotides. The Role of Acid/Base Properties in Hydrogen Bond Interactions	Venkataraman Amarnath; Arthur D. Broom
173-178	Nucleosides. 124. 3-Amino-3-deoxyhexopyranosyl Nucleosides. 7. 1-(3-Deoxy-3-Nitro-β-D-glucopyranosyl) Uracil and Its Galactopyranosyl Isomer¹	Akira Matsuda; Moon Woo Chun; Kyoichi A. Watanabe
179-190	Studies on the Chemical Synthesis of Potential Antimetabolites. 31.¹ A Novel Synthesis of 1-Deazaadenosine and Its Conversion to 5′-Deoxy-5′-Isobutylthio-1-Deazaadenosine (1-Deaza-Siba) and S-(1-Deazaadenosyl)-Homocysteine (1-DEAZA-SAH)	Tokuo Itoh; Tomokazu Sugawara; Yoshihisa Mizuno
191-203	Thiocyanation of Tubercidin and Its Derivatization to 6-Propyl-and 6-Cyano Derivatives (Nucleosides and Nucleotides. 41¹.)	Shin-Ichi Watanabe; Tohru Ueda

Volume 1, Issue 1 (1982)

a	Editorial board page for “Nucleosides & Nucleotides”, Volume 1, Number 1
iii-iv	Preface
1-34	Organometallic Intermediates in the Synthesis of Nucleoside Analogs	Donald E. Bergstrom
35-44	Nucleoside and Nucleotide Inhibitors of Inosine Monophosphate (IMP) Dehydrogenase as Potential Antitumor Inhibitors	Roland K. Robins
45-56	Synthesis of Alkylating 1-Glycosyl-5-substituted 1,2,4-Triazoles¹	Federico G. De las Heras; María-José Camarasa
57-64	¹⁸O Labeled Nucleosides. 2. A General Method for the Synthesis of Specifically Labeled Pyrimidine Ribonucleosides¹	R. Thomas Solsten; James A. Mccloskey; Karl H. Schram
65-80	Etude des Parametres Experimentax Influencant la Formation de la Liaison Phosphotriester Activee par le BOP. Application en Synthese Oligodesoxyribonucleotidique	D. Molko; A. Guy; R. Téoule
81-87	Bromine-Induced Selective N-Monodemethylation of N⁶, N⁶-Dimethyl-2′,3′-O-isopropylideneadenosine	Tetsuo Kato; Takeshi Endo; Ji�í �emli�ka
89-98	C-Nucleosides via Glycosyl Alkynyl Ketones. Synthesis of 5(3)-Phenyl-3(5)-(β-D-ribofuranosyl) Pyrazole	Marshall W. Logue; S. Sarangan